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ES8604589A1 - Procedimiento para preparar nuevos derivados de imidazo (1,5-a) pirimidina - Google Patents

Procedimiento para preparar nuevos derivados de imidazo (1,5-a) pirimidina

Info

Publication number
ES8604589A1
ES8604589A1 ES534259A ES534259A ES8604589A1 ES 8604589 A1 ES8604589 A1 ES 8604589A1 ES 534259 A ES534259 A ES 534259A ES 534259 A ES534259 A ES 534259A ES 8604589 A1 ES8604589 A1 ES 8604589A1
Authority
ES
Spain
Prior art keywords
preparation
pyrimidine derivatives
imidazo
relates
novel imidazo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES534259A
Other languages
English (en)
Other versions
ES534259A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Kyorin Pharmaceutical Co Ltd
Original Assignee
Kyorin Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kyorin Pharmaceutical Co Ltd filed Critical Kyorin Pharmaceutical Co Ltd
Publication of ES8604589A1 publication Critical patent/ES8604589A1/es
Publication of ES534259A0 publication Critical patent/ES534259A0/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52—Two oxygen atoms
    • C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

PROCEDIMIENTO PARA LA PREPARACION DE DERIVADOS DE IMIDAZO1,5-APIRIMIDINA, DE FORMULA GENERAL (I), EN LA QUE R1, R2 Y R3 SIGNIFICAN UN ATOMO DE ACIDO FARMACEUTICAMENTE ACEPTABLES. CONSISTE EN HACER REACCIONAR UN COMPUESTO DE FORMULA GENERAL (II) CON UN AGENTE DE CONDENSACION, TAL COMO UN CLORURO DE FOSFORILO O UN CLORURO DE TIONILO. DE APLICACION EN TERAPEUTICA EN EL TRATAMIENTO DE ENFERMEDADES FUNGALES, Y TAMBIEN COMO AGENTES ANTISEPTICOS PARA ALIMENTOS EN DIVERSAS FORMAS.
ES534259A 1983-07-12 1984-07-12 Procedimiento para preparar nuevos derivados de imidazo (1,5-a) pirimidina Expired ES8604589A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP58126697A JPS6019789A (ja) 1983-07-12 1983-07-12 イミダゾ〔１，５−ａ〕ピリミジン誘導体

Publications (2)

Publication Number Publication Date
ES8604589A1 true ES8604589A1 (es) 1986-02-01
ES534259A0 ES534259A0 (es) 1986-02-01

Family

ID=14941605

Family Applications (1)

Application Number Title Priority Date Filing Date
ES534259A Expired ES8604589A1 (es) 1983-07-12 1984-07-12 Procedimiento para preparar nuevos derivados de imidazo (1,5-a) pirimidina

Country Status (9)

Country Link
US (1) US4649198A (es)
EP (1) EP0134928B1 (es)
JP (1) JPS6019789A (es)
KR (1) KR910005850B1 (es)
AU (1) AU563849B2 (es)
CA (1) CA1238045A (es)
DE (1) DE3469177D1 (es)
DK (1) DK339584A (es)
ES (1) ES8604589A1 (es)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6143191A (ja) * 1984-08-07 1986-03-01 Kyorin Pharmaceut Co Ltd イミダゾ〔１，５−ａ〕ピリミジン誘導体
HU215433B (hu) * 1986-04-29 2000-05-28 Pfizer Inc. Eljárás új 2-oxo-5-fenil-pirimidin-származékok előállítására
US5395935A (en) * 1992-05-08 1995-03-07 Pfizer Inc. Endo-bicyclo[2.2.1]heptan-2-ol and derived pharmaceutical agents
US7166595B2 (en) * 2002-05-09 2007-01-23 Cytokinetics, Inc. Compounds, methods and compositions
AU2003231799A1 (en) * 2002-05-23 2003-12-12 Merck & Co., Inc. Mitotic kinesin inhibitors
DK1509256T3 (da) * 2002-05-24 2009-11-23 Angiotech Int Ag Præparater og fremgangsmåde til coating af medicinske implantater
US8313760B2 (en) 2002-05-24 2012-11-20 Angiotech International Ag Compositions and methods for coating medical implants
WO2004114655A1 (en) * 2003-06-18 2004-12-29 Thomson Licensing S.A. Apparatus for recording data on motion picture film
CN1898215A (zh) 2003-12-19 2007-01-17 默克公司 有丝分裂驱动蛋白抑制剂
TW202214642A (zh) * 2020-07-02 2022-04-16 大陸商江蘇恆瑞醫藥股份有限公司 咪唑并嘧啶類衍生物、其製備方法及其在醫藥上的應用

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2160020A1 (de) * 1971-12-03 1973-06-07 Bayer Ag Perchlor-imidazo-pyrimidin, verfahren zu seiner herstellung, sowie seine verwendung als fungizid
US3923808A (en) * 1972-12-08 1975-12-02 Janssen Pharmaceutica Nv Bicyclic imidazoles and pyrimidines
US4178449A (en) * 1978-04-17 1979-12-11 American Cyanamid Company Pyrazolo[1,5-a]pyrimidines and imidazo-[1,5-a]pyrimidines
US4236005A (en) * 1979-07-02 1980-11-25 American Cyanamid Company Imidazo[1,5-a]pyrimidines
US4408047A (en) * 1980-03-28 1983-10-04 Merck & Co., Inc. Imidazodiazines

Also Published As

Publication number Publication date
DK339584D0 (da) 1984-07-11
DE3469177D1 (en) 1988-03-10
DK339584A (da) 1985-01-13
US4649198A (en) 1987-03-10
JPS6019789A (ja) 1985-01-31
CA1238045A (en) 1988-06-14
EP0134928A1 (en) 1985-03-27
KR850001213A (ko) 1985-03-16
AU2937184A (en) 1985-01-17
AU563849B2 (en) 1987-07-23
ES534259A0 (es) 1986-02-01
EP0134928B1 (en) 1988-02-03
KR910005850B1 (ko) 1991-08-05
JPH0450315B2 (es) 1992-08-13

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19970401