ES8601229A1 - Procedimiento para la obtencion de o-glicosilamidas sustituidas - Google Patents
Procedimiento para la obtencion de o-glicosilamidas sustituidasInfo
- Publication number
- ES8601229A1 ES8601229A1 ES538339A ES538339A ES8601229A1 ES 8601229 A1 ES8601229 A1 ES 8601229A1 ES 538339 A ES538339 A ES 538339A ES 538339 A ES538339 A ES 538339A ES 8601229 A1 ES8601229 A1 ES 8601229A1
- Authority
- ES
- Spain
- Prior art keywords
- glycosylamides
- acyl
- substituted
- preparation
- methods
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H13/00—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids
- C07H13/12—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids by acids having the group -X-C(=X)-X-, or halides thereof, in which each X means nitrogen, oxygen, sulfur, selenium or tellurium, e.g. carbonic acid, carbamic acid
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/02—Acyclic radicals, not substituted by cyclic structures
- C07H15/04—Acyclic radicals, not substituted by cyclic structures attached to an oxygen atom of the saccharide radical
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biotechnology (AREA)
- Biochemistry (AREA)
- Crystallography & Structural Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Immunology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Saccharide Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Abstract
PROCEDIMIENTO DE OBTENCION DE 0-ACILGLICOSILAMIDAS SUSTITUIDAS DE FORMULA (I). CONSISTENTE EN HACER REACCIONAR UN COMPUESTO DE FORMULA (II) CON UN COMPUESTO AMINO BIEN EN FORMA LIBRE O EN FORMA DE SAL DE ADICION DE ACIDO Y POSTERIORMENTE LA GLICOSILAMINA ASI OBTENIDA ES ACILADA EN EL ATOMO DE NITROGENO CON UN DERIVADO DE ACIDO CARBOXILICO ACIDO CARBONICO ACIDO TIOCARBONICO O ISOCIANATO. EL PRODUCTO INTERMEDIO SE HACE REACCIONAR CON UN DERIVADO DE ACIDO CARBOXILICO ACIDO CARBONICO ACIDO TIOCARBONICO O ISOCIANATO. LAS REACCIONES SE REALIZAN A TEMPERATURAS COMPRENDIDAS ENTRE C30 Y 80JC Y OPCIONALMENTE EN PRESENCIA DE AGENTES AUXILIARES BASICOS. DE APLICACION COMO ACTIVADORES DEL SISTEMA INMUNOLOGICO.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19833344257 DE3344257A1 (de) | 1983-12-07 | 1983-12-07 | Substituierte o-acyl-glycosylamide, verfahren zu iherer herstellung sowie ihre verwendung |
Publications (2)
Publication Number | Publication Date |
---|---|
ES8601229A1 true ES8601229A1 (es) | 1985-11-01 |
ES538339A0 ES538339A0 (es) | 1985-11-01 |
Family
ID=6216279
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES538339A Granted ES538339A0 (es) | 1983-12-07 | 1984-12-06 | Procedimiento para la obtencion de o-glicosilamidas sustituidas |
Country Status (12)
Country | Link |
---|---|
US (1) | US4574122A (es) |
EP (1) | EP0149760B1 (es) |
JP (1) | JPS60155188A (es) |
KR (1) | KR860002110B1 (es) |
AT (1) | ATE45746T1 (es) |
CA (1) | CA1234109A (es) |
DE (2) | DE3344257A1 (es) |
DK (1) | DK583184A (es) |
ES (1) | ES538339A0 (es) |
GR (1) | GR81181B (es) |
IL (1) | IL73721A (es) |
ZA (1) | ZA849504B (es) |
Families Citing this family (10)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE3403495A1 (de) * | 1983-11-23 | 1985-05-30 | Bayer Ag, 5090 Leverkusen | Phosphorylierte glycosylamide, -harnstoffe, -carbamate und -thiocarbamate, verfahren zu ihrer herstellung sowie ihre verwendung |
DE3346623A1 (de) * | 1983-12-14 | 1985-07-04 | Bayer Ag, 5090 Leverkusen | N-glycosylierte harnstoffe, carbamate und thiocarbamate, verfahren zu ihrer herstellung sowie ihre verwendung |
JPS60149597A (ja) * | 1983-12-14 | 1985-08-07 | バイエル・アクチエンゲゼルシヤフト | N‐グリコシル化ウレア類、カルバメート類及びチオカルバメート類 |
DE3508025A1 (de) * | 1985-03-07 | 1986-09-11 | Bayer Ag, 5090 Leverkusen | Substituierte o-sulfonyl-glycosylamide, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel |
DE3521994A1 (de) * | 1985-06-20 | 1987-01-02 | Bayer Ag | N-(2-aminoacylamido-2-desoxy-hexosyl)-amide-, -carbamate und -harnstoffe, verfahren zu ihrer herstellung sowie ihre verwendung in arzneimitteln |
DE3604681A1 (de) * | 1986-02-14 | 1987-08-20 | Bayer Ag | Neue n-glycosylamidderivate, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel |
DE3812681A1 (de) * | 1988-04-16 | 1989-11-02 | Bayer Ag | Substituierte n-glycosylamide, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel |
US5476924A (en) * | 1989-01-27 | 1995-12-19 | Duke University | Protecting group for acetals and methods of using the same in the activation of saccharides |
WO1990014844A2 (en) * | 1989-06-06 | 1990-12-13 | Neorx Corporation | Sugars as cleavable linkers for the delivery and release of agents in native form |
US5872111A (en) * | 1997-05-19 | 1999-02-16 | Lever Brothers Company, Division Of Conopco, Inc. | Compositions comprising glycosylamide surfactants |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2612497A (en) * | 1948-01-24 | 1952-09-30 | Hendrik W Meijer | Process for manufacture of hexose ureides and thioureides |
US3843799A (en) * | 1973-01-26 | 1974-10-22 | Alberta Res Council | Method of feeding ruminants n-glucosyl-n'-ydroxymethylurea |
US4025622A (en) * | 1974-03-06 | 1977-05-24 | Haruo Ogura | Novel sugar ureide and thioureide derivatives |
US4066750A (en) * | 1976-08-02 | 1978-01-03 | Astra Chemical Products Ab | Lactosyl substituted ureides in ruminant feedstuff |
DE3213650A1 (de) * | 1982-04-14 | 1983-10-27 | Bayer Ag, 5090 Leverkusen | N-glycosylierte carbonsaeureamid-derivate, verfahren zu ihrer herstellung sowie ihre verwendung zur beeinflussung der koerpereigenen abwehr |
-
1983
- 1983-12-07 DE DE19833344257 patent/DE3344257A1/de not_active Withdrawn
-
1984
- 1984-11-27 AT AT84114306T patent/ATE45746T1/de not_active IP Right Cessation
- 1984-11-27 EP EP84114306A patent/EP0149760B1/de not_active Expired
- 1984-11-27 DE DE8484114306T patent/DE3479502D1/de not_active Expired
- 1984-11-28 US US06/675,690 patent/US4574122A/en not_active Expired - Fee Related
- 1984-12-04 JP JP59255152A patent/JPS60155188A/ja active Pending
- 1984-12-04 IL IL73721A patent/IL73721A/xx unknown
- 1984-12-04 KR KR1019840007646A patent/KR860002110B1/ko not_active IP Right Cessation
- 1984-12-05 GR GR81181A patent/GR81181B/el unknown
- 1984-12-05 CA CA000469363A patent/CA1234109A/en not_active Expired
- 1984-12-06 DK DK583184A patent/DK583184A/da not_active Application Discontinuation
- 1984-12-06 ES ES538339A patent/ES538339A0/es active Granted
- 1984-12-06 ZA ZA849504A patent/ZA849504B/xx unknown
Also Published As
Publication number | Publication date |
---|---|
DK583184A (da) | 1985-06-08 |
GR81181B (en) | 1985-04-03 |
JPS60155188A (ja) | 1985-08-15 |
KR850004495A (ko) | 1985-07-15 |
US4574122A (en) | 1986-03-04 |
DE3479502D1 (en) | 1989-09-28 |
EP0149760A3 (en) | 1987-04-01 |
EP0149760A2 (de) | 1985-07-31 |
IL73721A (en) | 1990-04-29 |
ZA849504B (en) | 1985-07-31 |
EP0149760B1 (de) | 1989-08-23 |
CA1234109A (en) | 1988-03-15 |
DK583184D0 (da) | 1984-12-06 |
ATE45746T1 (de) | 1989-09-15 |
DE3344257A1 (de) | 1985-06-13 |
IL73721A0 (en) | 1985-03-31 |
KR860002110B1 (ko) | 1986-11-26 |
ES538339A0 (es) | 1985-11-01 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD1A | Patent lapsed |
Effective date: 19970303 |