ES542134A0 - Un procedimiento para la preparacion de un antibiotico de macrolida - Google Patents

Un procedimiento para la preparacion de un antibiotico de macrolida

Info

Publication number: ES542134A0
Authority: ES; Spain
Prior art keywords: macrolida; antibiotic; procedure; preparation
Prior art date: 1984-04-13
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

ES542134A

Other languages

English (en)

Other versions

ES8607335A1 (es

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Pfizer Inc

Original Assignee

Pfizer Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1984-04-13

Filing date

1985-04-11

Publication date

1986-06-16

1984-04-13 Priority claimed from US06/600,252 external-priority patent/US4512982A/en

1985-04-11 Application filed by Pfizer Inc filed Critical Pfizer Inc

1986-06-16 Publication of ES542134A0 publication Critical patent/ES542134A0/es

1986-06-16 Publication of ES8607335A1 publication Critical patent/ES8607335A1/es

Status Expired legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Health & Medical Sciences (AREA)
Biochemistry (AREA)
Biotechnology (AREA)
General Health & Medical Sciences (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Saccharide Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

ES542134A 1984-04-13 1985-04-11 Un procedimiento para la preparacion de un antibiotico de macrolida Expired ES8607335A1 (es)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US06/600,252 US4512982A (en)	1984-04-13	1984-04-13	9α-Aza-9α-homoerythromycin compounds, pharmaceutical composition and therapeutic method
US06/616,529 US4518590A (en)	1984-04-13	1984-06-04	9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method

Publications (2)

Publication Number	Publication Date
ES542134A0 true ES542134A0 (es)	1986-06-16
ES8607335A1 ES8607335A1 (es)	1986-06-16

Family

ID=27083554

Family Applications (3)

Application Number	Title	Priority Date	Filing Date
ES542134A Expired ES8607335A1 (es)	1984-04-13	1985-04-11	Un procedimiento para la preparacion de un antibiotico de macrolida
ES551503A Expired ES8704965A1 (es)	1984-04-13	1986-01-31	Un procedimiento para la preparacion de un antibiotico de macrolida
ES551502A Expired ES8705458A1 (es)	1984-04-13	1986-01-31	Un procedimiento para la preparacion de un antibiotico de macrolida

Family Applications After (2)

Application Number	Title	Priority Date	Filing Date
ES551503A Expired ES8704965A1 (es)	1984-04-13	1986-01-31	Un procedimiento para la preparacion de un antibiotico de macrolida
ES551502A Expired ES8705458A1 (es)	1984-04-13	1986-01-31	Un procedimiento para la preparacion de un antibiotico de macrolida

Country Status (19)

Country	Link
US (1)	US4518590A (es)
EP (1)	EP0159856B1 (es)
KR (1)	KR860002111B1 (es)
AU (1)	AU549235B2 (es)
CA (1)	CA1234805A (es)
DE (1)	DE3565267D1 (es)
DK (1)	DK164785A (es)
EG (1)	EG17459A (es)
ES (3)	ES8607335A1 (es)
FI (1)	FI851449L (es)
GR (1)	GR850900B (es)
HU (1)	HU195668B (es)
IE (1)	IE57739B1 (es)
IL (1)	IL74865A (es)
NO (1)	NO161497C (es)
NZ (1)	NZ211769A (es)
PH (1)	PH21185A (es)
PT (1)	PT80270B (es)
YU (3)	YU62385A (es)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5075289A (en) *	1988-06-07	1991-12-24	Abbott Laboratories	9-r-azacyclic erythromycin antibiotics
US4904644A (en) *	1988-08-03	1990-02-27	Schering Corporation	Antimicrobial compound isolated from Actinomadura fulva subsp indica
EP0503932B1 (en)	1991-03-15	1998-12-02	Merck & Co. Inc.	9-Deoxo-9(z)-hydroxy-iminoerythromycin A and O-derivatives thereof
US5912331A (en) *	1991-03-15	1999-06-15	Merck & Co., Inc.	Process for the preparation of 9-deoxo-9(Z)-hydroxyiminoerythromycin A
US5985844A (en) *	1992-03-26	1999-11-16	Merck & Co., Inc.	Homoerythromycin A derivatives modified at the 4"-and 8A-positions
AU663089B2 (en) *	1991-04-09	1995-09-28	Abbott Laboratories	Macrocyclic lactam prokinetic agents
US5189159A (en) *	1992-04-02	1993-02-23	Merck & Co., Inc.	8a-AZA-8a-homoerythromycin cyclic iminoethers
US5523399A (en) *	1991-12-27	1996-06-04	Taisho Pharmaceutical Co., Ltd.	5-O-desosaminylerythronolide derivatives
US5215980A (en) *	1992-01-17	1993-06-01	Merck & Co., Inc.	10-AZA-9-deoxo-11-deoxy-erythromycin A and derivatives thereof
US5210235A (en) *	1992-08-26	1993-05-11	Merck & Co., Inc.	Methods of elaborating erythromycin fragments into amine-containing fragments of azalide antibiotics
US5332807A (en) *	1993-04-14	1994-07-26	Merck & Co., Inc.	Process of producing 8A- and 9A-azalide antibiotics
CA2162401C (en) *	1993-05-19	1998-11-03	Bingwei V. Yang	Intermediate for azithromycin
US5441939A (en) *	1994-03-04	1995-08-15	Pfizer Inc.	3"-desmethoxy derivatives of erythromycin and azithromycin
FR2739620B1 (fr) *	1995-10-09	1997-12-19	Roussel Uclaf	Nouveaux derives de la 5-0-desosaminyl 6-o-methyl erythronolide a, leur procede de preparation et leur application a la preparation de produits biologiquement actifs
USRE38426E1 (en) *	1995-10-09	2004-02-10	Aventis Pharma S.A.	5-O-deosaminyl 6-O-methyl erythronolide A derivatives, preparation method therefor and use thereof for preparing biologically active materials
WO2002015842A2 (en)	2000-08-23	2002-02-28	Wockhardt Limited	Process for preparation of anhydrous azithromycin
RU2263117C2 (ru)	2001-04-27	2005-10-27	Пфайзер Продактс Инк.	Способ получения 4"-замещенных производных 9-деоксо-9а-аза-9а-гомоэритромицина а
EP1482957A4 (en)	2002-02-15	2006-07-19	Merckle Gmbh	ANTIBIOTIC CONJUGATES
US20060099660A1 (en)	2002-02-15	2006-05-11	Synovo Gmbh	Conjugates of biologically active compounds, methods for their preparation and use, formulation and pharmaceutical applications thereof
EP1483277A4 (en)	2002-02-15	2007-10-03	Merckle Gmbh	CONJUGATES OF BIOLOGICALLY ACTIVE COMPOUNDS, METHODS OF PREPARATION AND USE, AND FORMULATION AND PHARMACEUTICAL APPLICATIONS
GB0310992D0 (en) *	2003-05-13	2003-06-18	Glaxo Group Ltd	Novel compounds
US7468428B2 (en) *	2004-03-17	2008-12-23	App Pharmaceuticals, Llc	Lyophilized azithromycin formulation
US20060116336A1 (en) *	2004-03-17	2006-06-01	American Pharmaceutical Partners, Inc.	Lyophilized azithromycin formulation

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
SE445223B (sv) *	1977-02-04	1986-06-09	Pfizer	Sett att framstella 4"-amino-erytomylin-a-derivat
US4150220A (en) *	1977-02-04	1979-04-17	Pfizer Inc.	Semi-synthetic 4"-erythromycin A derivatives
US4180654A (en) *	1978-01-03	1979-12-25	Pfizer Inc.	4"-Deoxy-4"-acylamido derivatives of oleandomycin, erythromycin and erythromycin carbonate
SI7910768A8 (en) *	1979-04-02	1996-06-30	Pliva Pharm & Chem Works	Process for pripering 11-aza-4-0-cladinosyl-6-0-desosaminyl-15-ethyl- 7,13,14-trihydroxy-3,5,7,9,12,14-hexamethyl- oxacyclopentadecane-2-one and their derivatives
YU43006B (en) *	1981-03-06	1989-02-28	Pliva Pharm & Chem Works	Process for preparing n-methyl-11-aza-10-deoxo-10-dihydro erythromycin and derivatives thereof
US4474768A (en) *	1982-07-19	1984-10-02	Pfizer Inc.	N-Methyl 11-aza-10-deoxo-10-dihydro-erytromycin A, intermediates therefor
US4465674A (en) *	1983-09-06	1984-08-14	Pfizer Inc.	Azahomoerythromycin D derivative and intermediates therefor

1984
- 1984-06-04 US US06/616,529 patent/US4518590A/en not_active Expired - Lifetime
1985
- 1985-04-09 GR GR850900A patent/GR850900B/el not_active IP Right Cessation
- 1985-04-10 EP EP85302507A patent/EP0159856B1/en not_active Expired
- 1985-04-10 IL IL74865A patent/IL74865A/xx not_active IP Right Cessation
- 1985-04-10 DE DE8585302507T patent/DE3565267D1/de not_active Expired
- 1985-04-11 EG EG239/85A patent/EG17459A/xx active
- 1985-04-11 PT PT80270A patent/PT80270B/pt not_active IP Right Cessation
- 1985-04-11 ES ES542134A patent/ES8607335A1/es not_active Expired
- 1985-04-11 FI FI851449A patent/FI851449L/fi not_active Application Discontinuation
- 1985-04-11 CA CA000478792A patent/CA1234805A/en not_active Expired
- 1985-04-11 IE IE912/85A patent/IE57739B1/en not_active IP Right Cessation
- 1985-04-11 PH PH32123A patent/PH21185A/en unknown
- 1985-04-12 YU YU00623/85A patent/YU62385A/xx unknown
- 1985-04-12 NZ NZ211769A patent/NZ211769A/en unknown
- 1985-04-12 HU HU851370A patent/HU195668B/hu not_active IP Right Cessation
- 1985-04-12 DK DK164785A patent/DK164785A/da not_active IP Right Cessation
- 1985-04-12 NO NO851466A patent/NO161497C/no not_active IP Right Cessation
- 1985-04-12 AU AU41070/85A patent/AU549235B2/en not_active Ceased
- 1985-04-12 KR KR1019850002453A patent/KR860002111B1/ko not_active IP Right Cessation
1986
- 1986-01-31 ES ES551503A patent/ES8704965A1/es not_active Expired
- 1986-01-31 ES ES551502A patent/ES8705458A1/es not_active Expired
1987
- 1987-07-06 YU YU01267/87A patent/YU126787A/xx unknown
- 1987-07-06 YU YU01268/87A patent/YU126887A/xx unknown

Also Published As

Publication number	Publication date
AU4107085A (en)	1985-10-17
EP0159856B1 (en)	1988-09-28
KR850007435A (ko)	1985-12-04
NO851466L (no)	1985-10-14
AU549235B2 (en)	1986-01-23
FI851449A0 (fi)	1985-04-11
IL74865A (en)	1987-12-31
HUT37629A (en)	1986-01-23
NO161497B (no)	1989-05-16
PT80270B (pt)	1987-10-20
EG17459A (en)	1992-12-30
EP0159856A3 (en)	1986-03-19
ES551502A0 (es)	1987-05-01
IE850912L (en)	1985-10-13
YU126887A (en)	1988-02-29
YU126787A (en)	1988-02-29
NZ211769A (en)	1987-10-30
FI851449L (fi)	1985-10-14
PT80270A (en)	1985-05-01
GR850900B (es)	1985-11-25
YU62385A (en)	1988-02-29
NO161497C (no)	1989-08-23
CA1234805A (en)	1988-04-05
DK164785A (da)	1985-12-10
HU195668B (en)	1988-06-28
DK164785D0 (da)	1985-04-12
KR860002111B1 (ko)	1986-11-26
ES8705458A1 (es)	1987-05-01
IL74865A0 (en)	1985-07-31
IE57739B1 (en)	1993-03-24
ES8704965A1 (es)	1987-04-16
ES8607335A1 (es)	1986-06-16
ES551503A0 (es)	1987-04-16
US4518590A (en)	1985-05-21
DE3565267D1 (en)	1988-11-03
EP0159856A2 (en)	1985-10-30
PH21185A (en)	1987-08-12

Publication	Publication Date	Title
ES547840A0 (es)	1986-09-01	Un procedimiento para la preparacion de alquilsulfonamidofe-nilalquilaminas
ES540366A0 (es)	1986-05-16	Un procedimiento para la preparacion de un compuesto
ES551503A0 (es)	1987-04-16	Un procedimiento para la preparacion de un antibiotico de macrolida
ES557126A0 (es)	1987-08-16	Un procedimiento para la preparacion de triazolobenzodiazepinas
ES536455A0 (es)	1985-11-16	Un procedimiento para la preparacion de un antibiotico bbm-2478.
ES554609A0 (es)	1987-08-16	Un procedimiento para la preparacion de derivados de oxindol
ES540200A0 (es)	1986-11-16	Un procedimiento para la preparacion de acidos 7-amino-3-me-til sustituido-3-defem-4-carboxilicos
ES544970A0 (es)	1986-02-01	Un procedimiento para la preparacion de derivados de benzo- tiofeno
ES545298A0 (es)	1986-09-01	Un procedimiento para la preparacion de 4-amino-2-fenilqui- nolinas
ES553602A0 (es)	1987-12-01	Un procedimiento para la preparacion de nuevas quinazolindionas
ES548960A0 (es)	1986-04-16	Un procedimiento para la preparacion de derivados de hidan- toina
ES541373A0 (es)	1985-12-16	Un procedimiento para la preparacion de un compuesto de 2-oxindol-1-carboxamida
ES549601A0 (es)	1987-04-16	Un procedimiento para la preparacion de arilquinolonas 7- sustituidas
ES551508A0 (es)	1987-02-16	Un procedimiento para la preparacion de nuevas sulfonilureas
ES557267A0 (es)	1988-02-16	Un procedimiento para la preparacion de derivados amidinofenilicos
ES542517A0 (es)	1986-01-01	Un procedimiento para la preparacion de monoalquil-polial- quilenpoliaminas
ES552987A0 (es)	1987-10-16	Un procedimiento para la preparacion de piridazinilimidazolidinonas
ES544214A0 (es)	1987-05-01	Un procedimiento para la preparacion de un derivado de n-metil-1-alquiltio-2-nitroetonamina
ES553605A0 (es)	1987-11-01	Un procedimiento para la preparacion de derivados de carbpenem
ES551129A0 (es)	1987-05-01	Un procedimiento para la preparacion de nuevas 3-alcoxi-2-(n-pirrolidino)-n-pirimidinil- o n-pirazinil-propilaminas
ES544397A0 (es)	1986-07-16	Un procedimiento para la preparacion de un compuesto
ES542674A0 (es)	1987-06-01	Un procedimiento para la preparacion de compuestos de cefa- losporina
ES551506A0 (es)	1987-01-16	Un procedimiento para la preparacion de etanodiimidamidas
ES544558A0 (es)	1986-09-01	Un procedimiento para la preparacion de derivados de dihi- dropiridina
ES551275A0 (es)	1987-07-16	Un procedimiento para la preparacion de un compuesto de 2-oxindol-1-carboxamida

Legal Events

Date	Code	Title	Description
2006-11-01	FD1A	Patent lapsed	Effective date: 20040410