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ES2185412T3 - Composiciones de celecoxib. - Google Patents

Composiciones de celecoxib.

Info

Publication number
ES2185412T3
ES2185412T3 ES99961890T ES99961890T ES2185412T3 ES 2185412 T3 ES2185412 T3 ES 2185412T3 ES 99961890 T ES99961890 T ES 99961890T ES 99961890 T ES99961890 T ES 99961890T ES 2185412 T3 ES2185412 T3 ES 2185412T3
Authority
ES
Spain
Prior art keywords
microns
particles
preferably less
celecoxib
celecoxib compositions
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES99961890T
Other languages
English (en)
Inventor
Danchen Gao
Anthony J Hlinak
Ahmad M Mazhary
James E Truelove
Margaret B Vaughn
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
GD Searle LLC
Original Assignee
GD Searle LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22332446&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ES2185412(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by GD Searle LLC filed Critical GD Searle LLC
Application granted granted Critical
Publication of ES2185412T3 publication Critical patent/ES2185412T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

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    • A61K31/63—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
    • A61K31/635—Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide having a heterocyclic ring, e.g. sulfadiazine
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
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  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
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  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
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  • Dermatology (AREA)
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  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Neurosurgery (AREA)
  • Diabetes (AREA)
  • Biophysics (AREA)
  • Pulmonology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Virology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
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Abstract

Una composición farmacéutica que incluye una o más unidades de dosis individuales sólidas que se pueden administrar por vía oral, comprendiendo cada una celecoxib en partículas en una cantidad de 10 mg a 1.000 mg en mezcla íntima con uno o más excipientes farmacéuticamente aceptables, y que tiene una distribución de tamaños de partículas de celecoxib tal que la D90 de las partículas es inferior a 200 micrasm, preferiblemente inferior a 100 micrasm, más preferiblemente inferior a 40 micrasm, y muy preferiblemente inferior a 25 micrasm, en la mayor dimensión de dichas partículas.
ES99961890T 1998-11-30 1999-11-30 Composiciones de celecoxib. Expired - Lifetime ES2185412T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US11033398P 1998-11-30 1998-11-30

Publications (1)

Publication Number Publication Date
ES2185412T3 true ES2185412T3 (es) 2003-04-16

Family

ID=22332446

Family Applications (1)

Application Number Title Priority Date Filing Date
ES99961890T Expired - Lifetime ES2185412T3 (es) 1998-11-30 1999-11-30 Composiciones de celecoxib.

Country Status (48)

Country Link
US (4) US20050267189A1 (es)
EP (1) EP1049467B1 (es)
JP (1) JP3563036B2 (es)
KR (2) KR20040065307A (es)
CN (2) CN1154490C (es)
AP (1) AP1637A (es)
AR (1) AR020015A1 (es)
AT (1) ATE225650T1 (es)
AU (1) AU748851B2 (es)
BG (1) BG64938B1 (es)
BR (1) BR9908030A (es)
CA (1) CA2319201C (es)
CR (2) CR6210A (es)
CU (1) CU20000176A7 (es)
DE (1) DE69903404T2 (es)
DK (1) DK1049467T3 (es)
EA (1) EA003363B1 (es)
EE (1) EE04834B1 (es)
ES (1) ES2185412T3 (es)
GC (1) GC0000114A (es)
GE (1) GEP20022784B (es)
GT (1) GT199900203A (es)
HK (2) HK1035144A1 (es)
HN (1) HN1999000210A (es)
HR (1) HRP20000434B1 (es)
HU (1) HUP0100867A3 (es)
IL (1) IL136532A (es)
IS (1) IS5555A (es)
MA (1) MA26709A1 (es)
ME (1) ME00416B (es)
NO (1) NO329912B1 (es)
NZ (1) NZ505762A (es)
OA (1) OA11616A (es)
PA (1) PA8486001A1 (es)
PE (1) PE20001349A1 (es)
PL (1) PL200957B1 (es)
PT (1) PT1049467E (es)
RS (1) RS50158B (es)
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EE200000437A (et) 2001-06-15
TNSN99223A1 (fr) 2005-11-10
PE20001349A1 (es) 2000-11-27
NO20003815L (no) 2000-09-29
CR6210A (es) 2004-05-28
CN1537531A (zh) 2004-10-20
SI1049467T1 (en) 2003-04-30
EP1049467A1 (en) 2000-11-08
EP1049467A4 (en) 2001-08-08
HUP0100867A2 (hu) 2002-03-28
IS5555A (is) 2000-06-30
SA99191255B1 (ar) 2006-11-25
AU748851B2 (en) 2002-06-13
KR100501034B1 (ko) 2005-07-18
ATE225650T1 (de) 2002-10-15
IL136532A (en) 2003-01-12
UY26025A1 (es) 2000-08-21
NO329912B1 (no) 2011-01-24
US20120171284A1 (en) 2012-07-05
YU48600A (sh) 2004-07-15
HN1999000210A (es) 2000-08-23
TR200002207T1 (tr) 2000-12-21
CR9842A (es) 2008-05-16
PL200957B1 (pl) 2009-02-27
WO2000032189A1 (en) 2000-06-08
SK283510B6 (sk) 2003-08-05
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JP3563036B2 (ja) 2004-09-08
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EA200000718A1 (ru) 2001-04-23
JP2002531403A (ja) 2002-09-24
KR20010040484A (ko) 2001-05-15
AP2000001874A0 (en) 2000-09-30
UA58576C2 (uk) 2003-08-15
MA26709A1 (fr) 2004-12-20
CN1154490C (zh) 2004-06-23
EP1049467B1 (en) 2002-10-09
BG104680A (en) 2001-02-28
KR20040065307A (ko) 2004-07-21
EA003363B1 (ru) 2003-04-24
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HUP0100867A3 (en) 2002-05-28

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