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EE04343B1 - Pürasoolkarboksüülhappe derivaadid, nende valmistamine ja neid sisaldavad farmatseutilised kompositsioonid - Google Patents

Pürasoolkarboksüülhappe derivaadid, nende valmistamine ja neid sisaldavad farmatseutilised kompositsioonid

Info

Publication number
EE04343B1
EE04343B1 EEP200100399A EEP200100399A EE04343B1 EE 04343 B1 EE04343 B1 EE 04343B1 EE P200100399 A EEP200100399 A EE P200100399A EE P200100399 A EEP200100399 A EE P200100399A EE 04343 B1 EE04343 B1 EE 04343B1
Authority
EE
Estonia
Prior art keywords
preparation
carboxylic acid
pharmaceutical compositions
compositions containing
acid derivatives
Prior art date
Application number
EEP200100399A
Other languages
English (en)
Estonian (et)
Inventor
Barth Francis
Camus Philippe
Martinez Serge
Rinaldi Murielle
Original Assignee
Sanofi-Synthlabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR9901201A external-priority patent/FR2789078B3/fr
Application filed by Sanofi-Synthlabo filed Critical Sanofi-Synthlabo
Publication of EE200100399A publication Critical patent/EE200100399A/xx
Publication of EE04343B1 publication Critical patent/EE04343B1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/32—Alcohol-abuse
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/34—Tobacco-abuse
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C251/72—Hydrazones
    • C07C251/74—Hydrazones having doubly-bound carbon atoms of hydrazone groups bound to hydrogen atoms or to acyclic carbon atoms
    • C07C251/78—Hydrazones having doubly-bound carbon atoms of hydrazone groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of an unsaturated carbon skeleton
    • C07C251/80—Hydrazones having doubly-bound carbon atoms of hydrazone groups bound to hydrogen atoms or to acyclic carbon atoms to carbon atoms of an unsaturated carbon skeleton the carbon skeleton containing rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Obesity (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Hospice & Palliative Care (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicinal Preparation (AREA)
EEP200100399A 1999-02-01 2000-01-28 Pürasoolkarboksüülhappe derivaadid, nende valmistamine ja neid sisaldavad farmatseutilised kompositsioonid EE04343B1 (et)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR9901201A FR2789078B3 (fr) 1999-02-01 1999-02-01 Derives d'acide pyrazolecarboxylique, leur preparation, les compositions pharmaceutiques en contenant
FR9910166A FR2789079B3 (fr) 1999-02-01 1999-08-02 Derive d'acide pyrazolecarboxylique, sa preparation, les compositions pharmaceutiques en contenant
PCT/FR2000/000194 WO2000046209A1 (fr) 1999-02-01 2000-01-28 Derives d'acide pyrazolecarboxylique, leur preparation, les compositions pharmaceutiques en contenant

Publications (2)

Publication Number Publication Date
EE200100399A EE200100399A (et) 2002-10-15
EE04343B1 true EE04343B1 (et) 2004-08-16

Family

ID=26234792

Family Applications (1)

Application Number Title Priority Date Filing Date
EEP200100399A EE04343B1 (et) 1999-02-01 2000-01-28 Pürasoolkarboksüülhappe derivaadid, nende valmistamine ja neid sisaldavad farmatseutilised kompositsioonid

Country Status (37)

Country Link
US (3) US6432984B1 (xx)
EP (1) EP1150961B1 (xx)
JP (1) JP3794925B2 (xx)
KR (1) KR100425405B1 (xx)
CN (1) CN1146544C (xx)
AR (1) AR020558A1 (xx)
AT (1) ATE252562T1 (xx)
AU (1) AU754771B2 (xx)
BG (1) BG65193B1 (xx)
BR (1) BR0007895A (xx)
CA (1) CA2358885C (xx)
CO (1) CO5160257A1 (xx)
CZ (1) CZ297667B6 (xx)
DE (1) DE60006070T2 (xx)
DK (1) DK1150961T3 (xx)
EE (1) EE04343B1 (xx)
ES (1) ES2208267T3 (xx)
FR (1) FR2789079B3 (xx)
HK (1) HK1039329A1 (xx)
HR (1) HRP20010564B1 (xx)
HU (1) HUP0201278A3 (xx)
ID (1) ID29534A (xx)
IL (2) IL144198A0 (xx)
IS (1) IS2448B (xx)
ME (2) ME00052B (xx)
NO (1) NO319824B1 (xx)
NZ (1) NZ512886A (xx)
PE (1) PE20001493A1 (xx)
PL (1) PL198422B1 (xx)
PT (1) PT1150961E (xx)
RS (1) RS50209B (xx)
RU (1) RU2216542C2 (xx)
SK (1) SK284203B6 (xx)
TR (1) TR200102054T2 (xx)
TW (1) TW581764B (xx)
UA (1) UA66900C2 (xx)
WO (1) WO2000046209A1 (xx)

Families Citing this family (128)

* Cited by examiner, † Cited by third party
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FR2882263B1 (fr) * 2005-02-23 2007-04-06 Sanofi Aventis Sa Utilisation d'un derive du pyrazole pour la preparation de medicaments utiles dans la prevention et le traitement des maladies renales
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