EA201790650A1 - DOSAGE FORM AND METHODS OF APPLICATION OF ABIRATERONE ACETATE - Google Patents
DOSAGE FORM AND METHODS OF APPLICATION OF ABIRATERONE ACETATEInfo
- Publication number
- EA201790650A1 EA201790650A1 EA201790650A EA201790650A EA201790650A1 EA 201790650 A1 EA201790650 A1 EA 201790650A1 EA 201790650 A EA201790650 A EA 201790650A EA 201790650 A EA201790650 A EA 201790650A EA 201790650 A1 EA201790650 A1 EA 201790650A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- methods
- application
- abiraterone acetate
- dosage form
- compositions
- Prior art date
Links
- 229960004103 abiraterone acetate Drugs 0.000 title abstract 2
- UVIQSJCZCSLXRZ-UBUQANBQSA-N abiraterone acetate Chemical compound C([C@@H]1[C@]2(C)CC[C@@H]3[C@@]4(C)CC[C@@H](CC4=CC[C@H]31)OC(=O)C)C=C2C1=CC=CN=C1 UVIQSJCZCSLXRZ-UBUQANBQSA-N 0.000 title abstract 2
- 239000002552 dosage form Substances 0.000 title abstract 2
- 239000000203 mixture Substances 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
- A61K31/573—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Urology & Nephrology (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Epoxy Compounds (AREA)
Abstract
Описаны фармацевтические композиции, включая дозированные лекарственные формы, содержащие абиратерона ацетат, и способы получения таких композиций.Pharmaceutical compositions are described, including dosage forms containing abiraterone acetate, and methods for making such compositions.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201462052294P | 2014-09-18 | 2014-09-18 | |
US14/707,922 US20150246060A1 (en) | 2013-03-15 | 2015-05-08 | Abiraterone Acetate Formulation and Methods of Use |
PCT/US2015/050889 WO2016044701A1 (en) | 2014-09-18 | 2015-09-18 | Abiraterone acetate formulation and methods of use |
Publications (1)
Publication Number | Publication Date |
---|---|
EA201790650A1 true EA201790650A1 (en) | 2017-07-31 |
Family
ID=55533897
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA201790650A EA201790650A1 (en) | 2014-09-18 | 2015-09-18 | DOSAGE FORM AND METHODS OF APPLICATION OF ABIRATERONE ACETATE |
Country Status (17)
Country | Link |
---|---|
EP (1) | EP3193857A4 (en) |
JP (1) | JP2017528457A (en) |
KR (2) | KR102491439B1 (en) |
CN (1) | CN106687112A (en) |
AP (1) | AP2017009804A0 (en) |
AU (1) | AU2015317466A1 (en) |
BR (1) | BR112017003219A2 (en) |
CA (1) | CA2958316A1 (en) |
CO (1) | CO2017002472A2 (en) |
EA (1) | EA201790650A1 (en) |
IL (1) | IL250270B (en) |
MD (1) | MD20170048A2 (en) |
MX (1) | MX2017003525A (en) |
PH (1) | PH12017500239A1 (en) |
SG (1) | SG11201701139YA (en) |
TN (2) | TN2018000318A1 (en) |
WO (1) | WO2016044701A1 (en) |
Families Citing this family (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2016162229A1 (en) | 2015-04-10 | 2016-10-13 | Capsugel Belgium N.V. | Abiraterone acetate lipid formulations |
EP3606506A4 (en) * | 2017-04-07 | 2021-01-06 | MAA Laboratories, Inc. | PROCESS FOR IMPROVING THE SOLUBILITY AND BIOAVAILABILITY OF THERAPEUTICS |
EP3914234A4 (en) * | 2019-01-25 | 2022-09-14 | Shenzhen Pharmacin Co., Ltd. | Pharmaceutical compositions |
CA3131034A1 (en) | 2019-03-06 | 2020-09-10 | Matthew J. Sharp | Abiraterone prodrugs |
CN110742870B (en) * | 2019-12-04 | 2021-04-20 | 武汉大学 | Abiraterone acetate preparation and preparation method thereof |
CN111110646A (en) * | 2020-02-19 | 2020-05-08 | 纳兰迦(上海)生物医药科技有限公司 | Prescription and preparation method of low-specification abiraterone acetate oral preparation |
CN113384542B (en) * | 2020-03-14 | 2024-03-29 | 鲁南制药集团股份有限公司 | Tablet of steroid CYP17 inhibitor solid dispersion and preparation method thereof |
BR112022021040A2 (en) * | 2020-04-16 | 2022-12-06 | Tavanta Therapeutics Hungary Incorporated | METHODS AND COMPOSITIONS FOR THE TREATMENT OF PROSTATE CANCER |
TW202207925A (en) * | 2020-05-08 | 2022-03-01 | 比利時商健生藥品公司 | Treatments of prostate cancer with combinations of abiraterone acetate and niraparib |
EP3944860A1 (en) | 2020-07-30 | 2022-02-02 | Galenicum Health S.L.U. | Abiraterone for use in a method of treating cancer |
JP2024506382A (en) | 2021-02-15 | 2024-02-13 | プロペラ セラピューティクス インコーポレイテッド | Abiraterone prodrug |
KR20240044329A (en) | 2022-09-28 | 2024-04-04 | 한미약품 주식회사 | Oral composite tablet comprising abiraterone acetate and prednisolone |
KR20240145412A (en) | 2023-03-27 | 2024-10-07 | 한미약품 주식회사 | Pharmaceutical formulation comprising abiraterone acetate and prednisolone and method for preparing same |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN105919939A (en) * | 2009-04-24 | 2016-09-07 | 伊休蒂卡有限公司 | Production of encapsulated nanoparticles at commercial scale |
GB201207886D0 (en) * | 2012-05-04 | 2012-06-20 | Jagotec Ag | Improvements in or relating to organic compounds |
WO2014009437A1 (en) * | 2012-07-11 | 2014-01-16 | Sandoz Ag | Oxidation stability of abiraterone acetate |
WO2014009436A1 (en) * | 2012-07-11 | 2014-01-16 | Sandoz Ag | Nanosuspension of abiraterone acetate |
WO2014009434A1 (en) * | 2012-07-11 | 2014-01-16 | Sandoz Ag | Self-microemulsifying drug delivery system of abiraterone or abiraterone acetate |
CN102743393A (en) | 2012-07-27 | 2012-10-24 | 海南盛科生命科学研究院 | Medicinal composition containing abiraterone acetate and preparation technology thereof |
KR102121404B1 (en) * | 2013-03-15 | 2020-06-11 | 썬 파마 글로벌 에프제트이 | Abiraterone acetate formulation |
-
2015
- 2015-09-18 CN CN201580050453.8A patent/CN106687112A/en active Pending
- 2015-09-18 EA EA201790650A patent/EA201790650A1/en unknown
- 2015-09-18 CA CA2958316A patent/CA2958316A1/en active Pending
- 2015-09-18 MD MDA20170048A patent/MD20170048A2/en not_active Application Discontinuation
- 2015-09-18 SG SG11201701139YA patent/SG11201701139YA/en unknown
- 2015-09-18 TN TNP/2018/000318A patent/TN2018000318A1/en unknown
- 2015-09-18 AU AU2015317466A patent/AU2015317466A1/en not_active Abandoned
- 2015-09-18 KR KR1020177008938A patent/KR102491439B1/en active Active
- 2015-09-18 BR BR112017003219A patent/BR112017003219A2/en not_active IP Right Cessation
- 2015-09-18 MX MX2017003525A patent/MX2017003525A/en unknown
- 2015-09-18 AP AP2017009804A patent/AP2017009804A0/en unknown
- 2015-09-18 EP EP15842591.8A patent/EP3193857A4/en not_active Withdrawn
- 2015-09-18 JP JP2017512783A patent/JP2017528457A/en active Pending
- 2015-09-18 WO PCT/US2015/050889 patent/WO2016044701A1/en active Application Filing
- 2015-09-18 TN TN2017000098A patent/TN2017000098A1/en unknown
- 2015-09-18 KR KR1020237001893A patent/KR102617537B1/en active Active
-
2017
- 2017-01-25 IL IL250270A patent/IL250270B/en active IP Right Grant
- 2017-02-09 PH PH12017500239A patent/PH12017500239A1/en unknown
- 2017-03-15 CO CONC2017/0002472A patent/CO2017002472A2/en unknown
Also Published As
Publication number | Publication date |
---|---|
TN2017000098A1 (en) | 2018-10-19 |
EP3193857A4 (en) | 2018-04-11 |
IL250270B (en) | 2021-02-28 |
TN2018000318A1 (en) | 2020-01-16 |
CN106687112A (en) | 2017-05-17 |
MD20170048A2 (en) | 2017-08-31 |
JP2017528457A (en) | 2017-09-28 |
KR102491439B1 (en) | 2023-01-25 |
MX2017003525A (en) | 2017-06-21 |
KR102617537B1 (en) | 2023-12-22 |
IL250270A0 (en) | 2017-03-30 |
AP2017009804A0 (en) | 2017-03-31 |
PH12017500239A1 (en) | 2017-07-03 |
CO2017002472A2 (en) | 2017-07-11 |
BR112017003219A2 (en) | 2017-11-28 |
KR20170070025A (en) | 2017-06-21 |
CA2958316A1 (en) | 2016-03-24 |
SG11201701139YA (en) | 2017-03-30 |
WO2016044701A1 (en) | 2016-03-24 |
EP3193857A1 (en) | 2017-07-26 |
AU2015317466A1 (en) | 2017-02-23 |
KR20230014878A (en) | 2023-01-30 |
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