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EA201000619A1 - Новые производные имидазола - Google Patents

Новые производные имидазола

Info

Publication number
EA201000619A1
EA201000619A1 EA201000619A EA201000619A EA201000619A1 EA 201000619 A1 EA201000619 A1 EA 201000619A1 EA 201000619 A EA201000619 A EA 201000619A EA 201000619 A EA201000619 A EA 201000619A EA 201000619 A1 EA201000619 A1 EA 201000619A1
Authority
EA
Eurasian Patent Office
Prior art keywords
halogen
haloalkyl
alkyl
group
hydrogen
Prior art date
Application number
EA201000619A
Other languages
English (en)
Inventor
Рафаель Дюмёнье
Клеменс Ламберт
Штефан Трах
Зебастиан Вендеборн
Original Assignee
Зингента Партисипейшнс Аг
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP07020982A external-priority patent/EP2053045A1/en
Application filed by Зингента Партисипейшнс Аг filed Critical Зингента Партисипейшнс Аг
Publication of EA201000619A1 publication Critical patent/EA201000619A1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/50—1,3-Diazoles; Hydrogenated 1,3-diazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Agronomy & Crop Science (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Dentistry (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

В заявке описаны новые производные имидазола формулы I как активные ингредиенты, которые обладают микробиоцидной активностью, в частности фунгицидной активностью,в которой Rобозначает галоген, С-С-алкил или С-С-галогеналкил; Rобозначает необязательно замещенный арил или гетероарил; Rобозначает галоген; Rобозначает водород, галоген, С-С-алкил, С-С-галогеналкил, C-C-алкоксигруппу, С-С-галогеналкоксигруппу или цианогруппу; Rобозначает галоген; Х обозначает N или C(R) и R обозначает водород, галоген, С-С-алкил, С-С-галогеналкил, C-C- алкоксигруппу, С-С-галогеналкоксигруппу или цианогруппу; или их агрохимически приемлемые соли; при условии, что, если Х обозначает C(R), то Rне может обозначать необязательно замещенный арил.
EA201000619A 2007-10-26 2008-10-24 Новые производные имидазола EA201000619A1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP07020982A EP2053045A1 (en) 2007-10-26 2007-10-26 Novel imidazole derivatives
EP07024449 2007-12-17
PCT/EP2008/009043 WO2009053102A1 (en) 2007-10-26 2008-10-24 Novel imidazole derivatives

Publications (1)

Publication Number Publication Date
EA201000619A1 true EA201000619A1 (ru) 2010-10-29

Family

ID=42719243

Family Applications (1)

Application Number Title Priority Date Filing Date
EA201000619A EA201000619A1 (ru) 2007-10-26 2008-10-24 Новые производные имидазола

Country Status (16)

Country Link
US (1) US20110224252A1 (ru)
JP (1) JP2011500750A (ru)
KR (1) KR20100101580A (ru)
CN (1) CN101835773A (ru)
AR (1) AR069037A1 (ru)
AT (1) ATE522517T1 (ru)
BR (1) BRPI0818855A2 (ru)
CL (1) CL2008003178A1 (ru)
CO (1) CO6190578A2 (ru)
EA (1) EA201000619A1 (ru)
GT (1) GT200800229A (ru)
IL (1) IL205148A0 (ru)
MA (1) MA31785B1 (ru)
NZ (1) NZ584387A (ru)
TW (1) TW200926981A (ru)
ZA (1) ZA201002439B (ru)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8877791B2 (en) * 2006-08-04 2014-11-04 Beth Israel Deaconess Medical Center, Inc. Inhibitors of pyruvate kinase and methods of treating disease
CN102448951B (zh) * 2009-04-06 2017-05-10 安吉奥斯医药品有限公司 丙酮酸激酶m2调节剂、治疗组合物和相关使用方法
CA2760929C (en) 2009-05-04 2018-01-02 Agios Pharmaceuticals, Inc. Pkm2 activators for use in the treatment of cancer
IN2012DN00471A (ru) 2009-06-29 2015-06-05 Agios Pharmaceuticals Inc
EP2448581B1 (en) 2009-06-29 2016-12-07 Agios Pharmaceuticals, Inc. Therapeutic compositions and related methods of use
US9221792B2 (en) 2010-12-17 2015-12-29 Agios Pharmaceuticals, Inc N-(4-(azetidine-1-carbonyl) phenyl)-(hetero-) arylsulfonamide derivatives as pyruvate kinase M2 (PMK2) modulators
JP6092118B2 (ja) 2010-12-21 2017-03-08 アジオス ファーマシューティカルズ， インコーポレイテッド ニ環式ｐｋｍ２活性化剤
TWI549947B (zh) 2010-12-29 2016-09-21 阿吉歐斯製藥公司 治療化合物及組成物
ES2970938T3 (es) 2011-05-03 2024-05-31 Agios Pharmaceuticals Inc Activadores de piruvato quinasa para uso en terapia
WO2012151440A1 (en) 2011-05-03 2012-11-08 Agios Pharmaceuticals, Inc. Pyruvate kinase activators for use for increasing lifetime of the red blood cells and treating anemia
WO2014139144A1 (en) 2013-03-15 2014-09-18 Agios Pharmaceuticals, Inc. Therapeutic compounds and compositions
CA2989111C (en) 2015-06-11 2023-10-03 Agios Pharmaceuticals, Inc. Methods of using pyruvate kinase activators
CN109810062B (zh) * 2019-01-24 2022-06-17 云南农业大学 一种苯基咪唑衍生物及其合成方法和在农药中的应用

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL338191A1 (en) * 1997-07-24 2000-10-09 Bayer Ag Nitrophenylsulphonyl imidazoles and their application in fighting against plant and animal pests

Also Published As

Publication number Publication date
KR20100101580A (ko) 2010-09-17
BRPI0818855A2 (pt) 2015-04-14
TW200926981A (en) 2009-07-01
US20110224252A1 (en) 2011-09-15
CN101835773A (zh) 2010-09-15
JP2011500750A (ja) 2011-01-06
ATE522517T1 (de) 2011-09-15
MA31785B1 (fr) 2010-10-01
GT200800229A (es) 2010-04-20
AR069037A1 (es) 2009-12-23
CL2008003178A1 (es) 2009-06-05
ZA201002439B (en) 2011-06-29
CO6190578A2 (es) 2010-08-19
NZ584387A (en) 2011-10-28
IL205148A0 (en) 2010-11-30

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