EA200400254A1 - Трициклические имидазопиридины - Google Patents
Трициклические имидазопиридиныInfo
- Publication number
- EA200400254A1 EA200400254A1 EA200400254A EA200400254A EA200400254A1 EA 200400254 A1 EA200400254 A1 EA 200400254A1 EA 200400254 A EA200400254 A EA 200400254A EA 200400254 A EA200400254 A EA 200400254A EA 200400254 A1 EA200400254 A1 EA 200400254A1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- imidazopiridines
- tricyclic
- international
- compounds
- application
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 abstract 2
- 210000004051 gastric juice Anatomy 0.000 abstract 1
- 230000028327 secretion Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
- C07D491/14—Ortho-condensed systems
- C07D491/147—Ortho-condensed systems the condensed system containing one ring with oxygen as ring hetero atom and two rings with nitrogen as ring hetero atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
- C07D491/14—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
В заявке описаны соединения формулы 1, в которой заместители и символы имеют значения, указанные в описании. Эти соединения ингибируют выделение желудочного сока.Международная заявка была опубликована вместе с отчетом о международном поиске.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP01119321 | 2001-08-10 | ||
PCT/EP2002/008505 WO2003014123A1 (en) | 2001-08-10 | 2002-07-31 | Tricyclic imidazopyridines |
Publications (2)
Publication Number | Publication Date |
---|---|
EA200400254A1 true EA200400254A1 (ru) | 2004-08-26 |
EA007683B1 EA007683B1 (ru) | 2006-12-29 |
Family
ID=8178292
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EA200400254A EA007683B1 (ru) | 2001-08-10 | 2002-07-31 | Трициклические имидазопиридины |
Country Status (24)
Country | Link |
---|---|
US (1) | US7223771B2 (ru) |
EP (1) | EP1419163B9 (ru) |
JP (1) | JP2005504761A (ru) |
KR (1) | KR20040023739A (ru) |
CN (1) | CN1329395C (ru) |
AT (1) | ATE297931T1 (ru) |
BR (1) | BR0211826A (ru) |
CA (1) | CA2452803A1 (ru) |
DE (1) | DE60204701T2 (ru) |
DK (1) | DK1419163T5 (ru) |
EA (1) | EA007683B1 (ru) |
ES (1) | ES2243788T3 (ru) |
HK (1) | HK1066213A1 (ru) |
HR (1) | HRP20040229A2 (ru) |
HU (1) | HUP0500330A3 (ru) |
IL (1) | IL159554A0 (ru) |
MX (1) | MXPA04001277A (ru) |
NO (1) | NO20040604L (ru) |
NZ (1) | NZ531520A (ru) |
PL (1) | PL368195A1 (ru) |
PT (1) | PT1419163E (ru) |
SI (1) | SI1419163T1 (ru) |
WO (1) | WO2003014123A1 (ru) |
ZA (1) | ZA200400918B (ru) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NZ542177A (en) * | 2003-04-04 | 2009-02-28 | Altana Pharma Ag | Cyclic benzimidazoles for use against gastrointestinal disorders |
AR044129A1 (es) | 2003-05-06 | 2005-08-24 | Altana Pharma Ag | Compuestos intermedios de imidazopiridina. proceso de preparacion. |
CA2526566A1 (en) * | 2003-05-27 | 2004-12-09 | Altana Pharma Ag | Pharmaceutical combinations of a proton pump inhibitor and a compound which modifies gastrointestinal motility |
AR046941A1 (es) * | 2003-12-19 | 2006-01-04 | Altana Pharma Ag | Imidazopiridinas triciclicas y su uso como inhibidores de secrecion de acido gastrico |
WO2005058894A1 (en) * | 2003-12-19 | 2005-06-30 | Altana Pharma Ag | Intermediates for the preparation of tricyclic dihydropyrano -imidazo -pyridines derivatives |
NZ549011A (en) * | 2004-02-17 | 2009-04-30 | Altana Pharma Ag | Tricyclic imidazopyridines and intermediates for the synthesis thereof |
JP2007529472A (ja) * | 2004-03-17 | 2007-10-25 | アルタナ ファルマ アクチエンゲゼルシャフト | 三環式のイミダゾピリジン |
EP1805173A2 (en) * | 2004-03-22 | 2007-07-11 | Altana Pharma AG | 7, 8, 9, 10- tetrahydro-imidazo [2,1-a] isoquinoline derivatives and their use as gastric acid secretion inhibitors |
AR048869A1 (es) * | 2004-04-26 | 2006-06-07 | Altana Pharma Ag | Bencimidazoles triciclicos |
JP2008501766A (ja) * | 2004-06-09 | 2008-01-24 | ニコメッド ゲゼルシャフト ミット ベシュレンクテル ハフツング | 置換された三環式のベンゾイミダゾール |
AR051041A1 (es) * | 2004-10-04 | 2006-12-13 | Altana Pharma Ag | Bencimidazoles triciclicos condensados |
AR054772A1 (es) * | 2005-06-16 | 2007-07-18 | Altana Pharma Ag | Espiro- imidazopiridinas como inhibidores de la secrecion de acido gastrico |
BRPI0710110A2 (pt) * | 2006-03-31 | 2011-08-02 | Novartis Ag | compostos orgánicos |
WO2008071766A2 (en) * | 2006-12-14 | 2008-06-19 | Nycomed Gmbh | Spiro-indene substituted imidazonaphythyridine and pyranoimidazopyridine derivatives as inhibitors of gastric acid secretion |
KR200452179Y1 (ko) * | 2009-05-20 | 2011-02-10 | 주식회사 신성일렉스 | 항공 장애물 표시 장치 |
EP2452680B1 (en) | 2009-07-09 | 2019-12-18 | RaQualia Pharma Inc. | Acid pump antagonist for the treatment of diseases involved in abnormal gastrointestinal motility |
GB201321730D0 (en) * | 2013-12-09 | 2014-01-22 | Ucb Pharma Sa | Therapeutic agents |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4468400A (en) * | 1982-12-20 | 1984-08-28 | Schering Corporation | Antiulcer tricyclic imidazo [1,2-a]pyridines |
SE9401197D0 (sv) * | 1994-04-11 | 1994-04-11 | Astra Ab | Active compounds |
DK0971922T3 (da) * | 1997-03-24 | 2004-08-16 | Altana Pharma Ag | Tetrahydropyrido-forbindelser |
IL132608A0 (en) * | 1997-05-28 | 2001-03-19 | Byk Gulden Lomberg Chem Fab | Fused dihydropyran compounds medicaments containing the same and the use thereof |
HUP0001555A3 (en) | 1997-10-30 | 2001-01-29 | Altana Pharma Ag | Tetrahydro-imidazo-naphthyridine derivatives, pharmaceutical compositions thereof and process for their preparation |
US6696461B2 (en) * | 2000-03-29 | 2004-02-24 | Altana Pharma Ag | Tricyclic imidazopyridines |
-
2002
- 2002-07-31 EA EA200400254A patent/EA007683B1/ru not_active IP Right Cessation
- 2002-07-31 US US10/485,515 patent/US7223771B2/en not_active Expired - Fee Related
- 2002-07-31 DE DE60204701T patent/DE60204701T2/de not_active Expired - Fee Related
- 2002-07-31 IL IL15955402A patent/IL159554A0/xx unknown
- 2002-07-31 BR BR0211826-2A patent/BR0211826A/pt not_active IP Right Cessation
- 2002-07-31 CN CNB028156013A patent/CN1329395C/zh not_active Expired - Fee Related
- 2002-07-31 SI SI200230179T patent/SI1419163T1/sl unknown
- 2002-07-31 WO PCT/EP2002/008505 patent/WO2003014123A1/en active IP Right Grant
- 2002-07-31 NZ NZ531520A patent/NZ531520A/en unknown
- 2002-07-31 ES ES02794528T patent/ES2243788T3/es not_active Expired - Lifetime
- 2002-07-31 HU HU0500330A patent/HUP0500330A3/hu unknown
- 2002-07-31 MX MXPA04001277A patent/MXPA04001277A/es active IP Right Grant
- 2002-07-31 CA CA002452803A patent/CA2452803A1/en not_active Abandoned
- 2002-07-31 AT AT02794528T patent/ATE297931T1/de not_active IP Right Cessation
- 2002-07-31 PL PL02368195A patent/PL368195A1/xx not_active Application Discontinuation
- 2002-07-31 JP JP2003519072A patent/JP2005504761A/ja not_active Withdrawn
- 2002-07-31 DK DK02794528T patent/DK1419163T5/da active
- 2002-07-31 EP EP02794528A patent/EP1419163B9/en not_active Expired - Lifetime
- 2002-07-31 KR KR10-2004-7001988A patent/KR20040023739A/ko not_active Application Discontinuation
- 2002-07-31 PT PT02794528T patent/PT1419163E/pt unknown
-
2004
- 2004-02-04 ZA ZA200400918A patent/ZA200400918B/en unknown
- 2004-02-10 NO NO20040604A patent/NO20040604L/no not_active Application Discontinuation
- 2004-03-08 HR HR20040229A patent/HRP20040229A2/hr not_active Application Discontinuation
- 2004-11-16 HK HK04109042A patent/HK1066213A1/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
ES2243788T3 (es) | 2005-12-01 |
ATE297931T1 (de) | 2005-07-15 |
HUP0500330A2 (hu) | 2005-07-28 |
ZA200400918B (en) | 2005-04-20 |
CN1329395C (zh) | 2007-08-01 |
PL368195A1 (en) | 2005-03-21 |
WO2003014123A1 (en) | 2003-02-20 |
DK1419163T5 (da) | 2005-12-19 |
MXPA04001277A (es) | 2004-05-27 |
EA007683B1 (ru) | 2006-12-29 |
DE60204701T2 (de) | 2006-08-03 |
US7223771B2 (en) | 2007-05-29 |
CA2452803A1 (en) | 2003-02-20 |
NO20040604L (no) | 2004-02-10 |
EP1419163B9 (en) | 2005-11-09 |
EP1419163B1 (en) | 2005-06-15 |
CN1541219A (zh) | 2004-10-27 |
NZ531520A (en) | 2005-10-28 |
IL159554A0 (en) | 2004-06-01 |
EP1419163A1 (en) | 2004-05-19 |
HK1066213A1 (en) | 2005-03-18 |
JP2005504761A (ja) | 2005-02-17 |
US20050049272A1 (en) | 2005-03-03 |
HUP0500330A3 (en) | 2009-12-28 |
SI1419163T1 (sl) | 2005-12-31 |
HRP20040229A2 (en) | 2005-02-28 |
KR20040023739A (ko) | 2004-03-18 |
BR0211826A (pt) | 2005-06-28 |
DE60204701D1 (de) | 2005-07-21 |
PT1419163E (pt) | 2005-10-31 |
DK1419163T3 (da) | 2005-10-17 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM4A | Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s) |
Designated state(s): BY RU |