DK3429998T3 - Fremgangsmåde til fremstilling af quinolin-2-yl-phenylaminderivater og disses salte - Google Patents
Fremgangsmåde til fremstilling af quinolin-2-yl-phenylaminderivater og disses salte Download PDFInfo
- Publication number
- DK3429998T3 DK3429998T3 DK17710769.5T DK17710769T DK3429998T3 DK 3429998 T3 DK3429998 T3 DK 3429998T3 DK 17710769 T DK17710769 T DK 17710769T DK 3429998 T3 DK3429998 T3 DK 3429998T3
- Authority
- DK
- Denmark
- Prior art keywords
- quinolin
- salts
- preparation
- phenylamine derivatives
- phenylamine
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/38—Nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Virology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Tropical Medicine & Parasitology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- AIDS & HIV (AREA)
- General Chemical & Material Sciences (AREA)
- Molecular Biology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP16000661 | 2016-03-18 | ||
EP16000662 | 2016-03-18 | ||
PCT/EP2017/056544 WO2017158201A1 (en) | 2016-03-18 | 2017-03-20 | Process for preparing quinolin-2-yl-phenylamine derivatives and their salts |
Publications (1)
Publication Number | Publication Date |
---|---|
DK3429998T3 true DK3429998T3 (da) | 2021-11-22 |
Family
ID=58277293
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK17710769.5T DK3429998T3 (da) | 2016-03-18 | 2017-03-20 | Fremgangsmåde til fremstilling af quinolin-2-yl-phenylaminderivater og disses salte |
Country Status (8)
Country | Link |
---|---|
US (2) | US10464903B2 (da) |
EP (1) | EP3429998B1 (da) |
DK (1) | DK3429998T3 (da) |
ES (1) | ES2899926T3 (da) |
HR (1) | HRP20211779T1 (da) |
PL (1) | PL3429998T3 (da) |
PT (1) | PT3429998T (da) |
WO (1) | WO2017158201A1 (da) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2757161A1 (en) | 2013-01-17 | 2014-07-23 | Splicos | miRNA-124 as a biomarker of viral infection |
EP2974729A1 (en) | 2014-07-17 | 2016-01-20 | Abivax | Quinoline derivatives for use in the treatment of inflammatory diseases |
HRP20211779T1 (hr) | 2016-03-18 | 2022-03-04 | Prosynergia S.A.R.L. | Postupak priprave derivata kinolin-2-il-fenilamina i njihovih soli |
EP3594206A1 (en) | 2018-07-09 | 2020-01-15 | Abivax | Phenyl-n-quinoline derivatives for treating a rna virus infection |
EP3669874A1 (en) * | 2018-12-20 | 2020-06-24 | Abivax | Quinoline derivatives for use in the treatment or prevention of cancer |
EP3669873A1 (en) | 2018-12-20 | 2020-06-24 | Abivax | Quinoline derivatives for use ine the traeatment of inflammation diseases |
KR102399037B1 (ko) * | 2020-01-06 | 2022-05-17 | 성균관대학교산학협력단 | 아민화된 아진의 신규한 제조방법 |
EP3858815A1 (en) | 2020-01-31 | 2021-08-04 | Abivax | Co-crystals and salts of 8-chloro-n-(4-(trifluoromethoxy)phenyl)quinolin-2-amine |
EP4063351A1 (en) | 2021-03-26 | 2022-09-28 | Abivax | Preparation method of quinoline derivative compounds |
US20240327388A1 (en) | 2021-05-27 | 2024-10-03 | Jiangsu Hengrui Pharmaceuticals Co., Ltd. | Quinolinamine compound, preparation method therefor and application thereof in pharmaceuticals |
CN118591528A (zh) * | 2022-01-24 | 2024-09-03 | 江苏恒瑞医药股份有限公司 | 喹啉胺类化合物、其制备方法及其在医药上的应用 |
WO2024109936A1 (zh) * | 2022-11-25 | 2024-05-30 | 江苏恒瑞医药股份有限公司 | 一种喹啉胺类化合物晶型及其制备方法 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN104844510B (zh) | 2009-06-12 | 2019-04-23 | Abivax公司 | 用于治疗过早衰老和尤其是早衰的化合物 |
EP2465502A1 (en) * | 2010-12-15 | 2012-06-20 | Société Splicos | Compounds useful for treating AIDS |
HRP20211779T1 (hr) | 2016-03-18 | 2022-03-04 | Prosynergia S.A.R.L. | Postupak priprave derivata kinolin-2-il-fenilamina i njihovih soli |
-
2017
- 2017-03-20 HR HRP20211779TT patent/HRP20211779T1/hr unknown
- 2017-03-20 US US16/084,891 patent/US10464903B2/en active Active
- 2017-03-20 DK DK17710769.5T patent/DK3429998T3/da active
- 2017-03-20 WO PCT/EP2017/056544 patent/WO2017158201A1/en active Application Filing
- 2017-03-20 EP EP17710769.5A patent/EP3429998B1/en active Active
- 2017-03-20 ES ES17710769T patent/ES2899926T3/es active Active
- 2017-03-20 PT PT177107695T patent/PT3429998T/pt unknown
- 2017-03-20 PL PL17710769T patent/PL3429998T3/pl unknown
-
2019
- 2019-11-01 US US16/671,278 patent/US10745357B2/en active Active
Also Published As
Publication number | Publication date |
---|---|
PL3429998T3 (pl) | 2022-03-14 |
EP3429998A1 (en) | 2019-01-23 |
WO2017158201A1 (en) | 2017-09-21 |
US10464903B2 (en) | 2019-11-05 |
US20190077760A1 (en) | 2019-03-14 |
ES2899926T3 (es) | 2022-03-15 |
US10745357B2 (en) | 2020-08-18 |
US20200062713A1 (en) | 2020-02-27 |
PT3429998T (pt) | 2021-11-04 |
HRP20211779T1 (hr) | 2022-03-04 |
EP3429998B1 (en) | 2021-09-01 |
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