DK304686A - Pyridoncarboxylsyrederivater, fremgangsmaade til fremstilling af samme samt antimikrobielt middel indeholdende derivaterne - Google Patents

Pyridoncarboxylsyrederivater, fremgangsmaade til fremstilling af samme samt antimikrobielt middel indeholdende derivaterne Download PDF

Info

Publication number: DK304686A
Authority: DK; Denmark
Prior art keywords: sup; derivatives; pyridon; preparing; procedure
Prior art date: 1985-06-26

Application number

DK304686A

Other languages

English (en)

Other versions

DK304686D0 (da

DK170641B1 (da

Inventor

Isao Hayakawa

Shohgo Atarashi

Original Assignee

Daiichi Seiyaku Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1985-06-26

Filing date

1986-06-26

Publication date

1987-02-23

1986-06-26 Application filed by Daiichi Seiyaku Co filed Critical Daiichi Seiyaku Co

1986-06-26 Publication of DK304686D0 publication Critical patent/DK304686D0/da

1987-02-23 Publication of DK304686A publication Critical patent/DK304686A/da

1995-11-20 Application granted granted Critical

1995-11-20 Publication of DK170641B1 publication Critical patent/DK170641B1/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Communicable Diseases (AREA)
Public Health (AREA)
Oncology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Pyridine Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Pyrrole Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Table Devices Or Equipment (AREA)
Stringed Musical Instruments (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

DK304686A 1985-06-26 1986-06-26 Pyrrolidinyl-oxoquinolincarboxylsyrederivater, fremgangsmåde til fremstilling af samme samt antimikrobielt middel indeholdende derivaterne DK170641B1 (da)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
JP13983085		1985-06-26
JP13983085		1985-06-26
JP27999185		1985-12-12
JP27999185		1985-12-12

Publications (3)

Publication Number	Publication Date
DK304686D0 DK304686D0 (da)	1986-06-26
DK304686A true DK304686A (da)	1987-02-23
DK170641B1 DK170641B1 (da)	1995-11-20

Family

ID=26472527

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK304686A DK170641B1 (da)	1985-06-26	1986-06-26	Pyrrolidinyl-oxoquinolincarboxylsyrederivater, fremgangsmåde til fremstilling af samme samt antimikrobielt middel indeholdende derivaterne

Country Status (18)

Country	Link
US (4)	US5098912A (da)
EP (1)	EP0207420B1 (da)
JP (2)	JPH0745491B2 (da)
KR (1)	KR930005001B1 (da)
AT (1)	ATE75740T1 (da)
AU (1)	AU589978B2 (da)
CA (1)	CA1301760C (da)
DE (1)	DE3685157D1 (da)
DK (1)	DK170641B1 (da)
ES (1)	ES8707520A1 (da)
FI (1)	FI87071C (da)
GR (1)	GR861649B (da)
IE (1)	IE59188B1 (da)
IL (1)	IL79189A (da)
NO (1)	NO167090C (da)
PH (1)	PH24886A (da)
PT (1)	PT82839B (da)
YU (1)	YU46526B (da)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE3508816A1 (de) *	1985-01-10	1986-07-10	Bayer Ag, 5090 Leverkusen	6,7-disubstituierte 1-cyclopropyl-1,4-dihydro-4-oxo-1,8-naphtyridin-3-carbonsaeuren
US4920120A (en) *	1988-01-25	1990-04-24	Warner-Lambert Company	Antibacterial agents
US5585491A (en) *	1988-01-25	1996-12-17	Otsuka Pharmaceutical Co., Ltd.	Antibacterial agents
CA1332605C (en) *	1988-10-03	1994-10-18	Yasuhiro Nishitani	Pyridonecarboxylic acids
US5258528A (en) *	1990-11-30	1993-11-02	Warner-Lambert Company	Individual stereoisomers of pyrrolidine methanamines substituted on the ring nitrogen by a 1-phenylethyl group
US5157128A (en) *	1990-11-30	1992-10-20	Warner-Lambert Company	Certain optically active substituted α,α-dialkyl-pyrrolidine-3-methamines useful as intermediates
ATE181915T1 (de) *	1990-11-30	1999-07-15	Warner Lambert Co	Individuelle stereoisomere von 7-(3-(aminoalkyl)- 1-pyrrolidinyl>-quinolone und naphthyridone als antibakterielle wirkstoffe
US5364861A (en) *	1990-11-30	1994-11-15	Warner-Lambert Company	Optical isomers of 7-[3-(1,1-dialkylmethyl-1-amino-1-pyrrolidinyl]-quinolones and naphthyridones as antibacterial agents
EP0550016A1 (en) *	1991-12-31	1993-07-07	Korea Research Institute Of Chemical Technology	Novel quinolone carboxylic acid derivatives and processes for preparing same
DE69627985T2 (de) *	1995-02-02	2004-02-19	Daiichi Pharmaceutical Co., Ltd.	Heterozyklische verbindungen
EA003321B1 (ru) *	1995-11-22	2003-04-24	Дайити Фармасьютикал Ко., Лтд.	Производные аминоциклоалкилпирролидона и антибактериальное лекарственное средство на их основе
US6121285A (en) *	1995-11-22	2000-09-19	Daiichi Pharmaceutical Co., Ltd.	Substituted aminocycloalkylpyrrolidine derivatives and cis-substituted aminocycloalkylpyrrolidine derivatives
JP4094061B2 (ja)	1996-07-12	2008-06-04	第一三共株式会社	シス置換アミノシクロプロパン誘導体
WO1998052939A1 (fr) *	1997-05-21	1998-11-26	Daiichi Pharmaceutical Co., Ltd.	Derives d'aminocycloalkyle-pyrrolidine cis-disubstitues
ZA984527B (en) *	1997-05-30	1998-12-03	Daiichi Seiyaku Co	Substituted cyclobutylamine derivative
RU2193558C2 (ru) *	1997-09-15	2002-11-27	Дзе Проктер Энд Гэмбл Компани	Производные хинолона и фармацевтическая композиция на их основе
US6387928B1 (en)	1997-09-15	2002-05-14	The Procter & Gamble Co.	Antimicrobial quinolones, their compositions and uses
ATE249432T1 (de) *	1998-05-29	2003-09-15	Upjohn Co	3-((1'-n-methylamino)ethyl-n-benzyl)pyrrolidin- monomethanesulfonat
DE60011264T2 (de) *	1999-03-10	2005-07-14	Daiichi Pharmaceutical Co., Ltd.	Aminomethylpyrrolidin-derivate mit aromatischen substituenten
JP2003521686A (ja) *	2000-01-28	2003-07-15	ピオン，インコーポレイテッド	溶解度−ｐＨプロフィールの測定
CN1269817C (zh) *	2000-11-20	2006-08-16	第一制药株式会社	脱卤代化合物
PL1666477T3 (pl) *	2003-09-10	2013-11-29	Kyorin Seiyaku Kk	Pochodna kwasu 7-(4-podstawionego-3-cyklopropyloaminometylo-1- pirolidynylo)chinolonokarboksylowego
WO2005030752A1 (ja) *	2003-09-29	2005-04-07	Daiichi Pharmaceutical Co., Ltd.	８−シアノキノロンカルボン酸誘導体
MX2008012327A (es) *	2006-03-28	2008-10-09	Procter & Gamble	Un proceso de reduccion con hidruro para preparar intermedios de quinolona.
JP2009531418A (ja) *	2006-03-28	2009-09-03	ザプロクターアンドギャンブルカンパニー	キノロン中間体調製のためのカップリング方法
CA2647346C (en) *	2006-03-28	2011-07-19	The Procter & Gamble Company	Malate salts, and polymorphs of (3s,5s)-7-[3-amino-5-methyl-piperidinyl]-1-cyclopropyl-1,4-dihydro-8-methoxy-4-oxo-3-quinolinecarboxylic acid
EP2149571A4 (en) *	2007-05-24	2010-09-01	Kyorin Seiyaku Kk	MUTILINE DERIVATIVE WITH A RINGED, HETEROCYCLIC AND AROMATIC CARBOXYLIC ACID STRUCTURE IN A SUBSTITUTE AT POSITION 14
CN116606280A (zh) *	2023-03-13	2023-08-18	广东工业大学	一种氟喹诺酮类化合物及其在制备抗菌药物中的应用

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IE55898B1 (en) *	1982-09-09	1991-02-14	Warner Lambert Co	Antibacterial agents
US4665079A (en) *	1984-02-17	1987-05-12	Warner-Lambert Company	Antibacterial agents
DE3318145A1 (de) *	1983-05-18	1984-11-22	Bayer Ag, 5090 Leverkusen	7-amino-1-cyclopropyl-6,8-difluor-1,4-dihydro-4-oxo-3-chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel
JPS60228479A (ja) *	1984-04-26	1985-11-13	Toyama Chem Co Ltd	１，４−ジヒドロ−４−オキソナフチリジン誘導体およびその塩
IE58742B1 (en) *	1984-07-20	1993-11-05	Warner Lambert Co	Substituted-9-fluoro-3-methyl-7-oxo-2,3-dihydro-7h-pyrido[1,2,3-de] [1,4]benzoxauine-6-carboxylic acids; sibstituted-5-amino-6-6fluoro-4-oxo.1,4-dihydroquinoline-3 carboxylic acids; substituted-5-amino-6-fluoro-1,4-dihydro-4-oxo-1.8-naphthyridine-3-carboxylic acids; derivatives thereof; pharmaceutical compositions comprising the compounds; and processes for producing the compounds
DE3509546A1 (de) *	1985-03-16	1986-09-25	Bayer Ag, 5090 Leverkusen	7-amino-1-(subst.cyclopropyl)-1,4-dihydro-4-oxo-3-chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel
US4657913A (en) *	1985-04-18	1987-04-14	Warner-Lambert Company	Trifluoro- quinoline -3- carboxylic acids and their use as anti-bacterial agents
EP0242789A3 (en) *	1986-04-25	1990-09-05	Dainippon Pharmaceutical Co., Ltd.	Novel quinoline derivates and processes for preparation thereof
US4851418A (en) *	1987-08-21	1989-07-25	Warner-Lambert Company	Naphthyridine antibacterial agents containing an α-amino acid in the side chain of the 7-substituent
US4920120A (en) *	1988-01-25	1990-04-24	Warner-Lambert Company	Antibacterial agents

1986
- 1986-06-23 AT AT86108547T patent/ATE75740T1/de not_active IP Right Cessation
- 1986-06-23 DE DE8686108547T patent/DE3685157D1/de not_active Expired - Lifetime
- 1986-06-23 IL IL79189A patent/IL79189A/xx not_active IP Right Cessation
- 1986-06-23 EP EP86108547A patent/EP0207420B1/en not_active Expired - Lifetime
- 1986-06-24 FI FI862688A patent/FI87071C/fi not_active IP Right Cessation
- 1986-06-25 GR GR861649A patent/GR861649B/el unknown
- 1986-06-25 PT PT82839A patent/PT82839B/pt unknown
- 1986-06-25 IE IE169686A patent/IE59188B1/en not_active IP Right Cessation
- 1986-06-25 CA CA000512446A patent/CA1301760C/en not_active Expired - Lifetime
- 1986-06-25 NO NO862559A patent/NO167090C/no not_active IP Right Cessation
- 1986-06-25 AU AU59245/86A patent/AU589978B2/en not_active Expired
- 1986-06-25 ES ES556754A patent/ES8707520A1/es not_active Expired
- 1986-06-26 DK DK304686A patent/DK170641B1/da not_active IP Right Cessation
- 1986-06-26 PH PH33956A patent/PH24886A/en unknown
- 1986-06-26 YU YU112086A patent/YU46526B/sh unknown
- 1986-06-26 KR KR1019860005150A patent/KR930005001B1/ko not_active Expired - Lifetime
- 1986-06-26 JP JP61150581A patent/JPH0745491B2/ja not_active Expired - Lifetime
1989
- 1989-12-12 US US07/449,160 patent/US5098912A/en not_active Expired - Lifetime
1991
- 1991-12-24 US US07/812,830 patent/US5416222A/en not_active Expired - Lifetime
1993
- 1993-06-21 JP JP5148887A patent/JP2686705B2/ja not_active Expired - Lifetime
1994
- 1994-03-04 US US08/205,638 patent/US5380874A/en not_active Expired - Lifetime
1995
- 1995-03-20 US US08/406,594 patent/US5476950A/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
JPH0745491B2 (ja)	1995-05-17
ES8707520A1 (es)	1987-08-01
DK304686D0 (da)	1986-06-26
IE861696L (en)	1986-12-26
JP2686705B2 (ja)	1997-12-08
AU589978B2 (en)	1989-10-26
CA1301760C (en)	1992-05-26
FI87071C (fi)	1992-11-25
PT82839B (pt)	1988-04-21
DE3685157D1 (de)	1992-06-11
NO862559D0 (no)	1986-06-25
DK170641B1 (da)	1995-11-20
IE59188B1 (en)	1994-01-26
PH24886A (en)	1990-12-26
YU46526B (sh)	1993-11-16
NO862559L (no)	1986-12-29
EP0207420A2 (en)	1987-01-07
FI862688A0 (fi)	1986-06-24
IL79189A0 (en)	1986-09-30
ES556754A0 (es)	1987-08-01
GR861649B (en)	1986-10-30
IL79189A (en)	1990-07-12
FI87071B (fi)	1992-08-14
NO167090B (no)	1991-06-24
US5416222A (en)	1995-05-16
ATE75740T1 (de)	1992-05-15
AU5924586A (en)	1987-01-08
YU112086A (en)	1991-04-30
US5476950A (en)	1995-12-19
FI862688L (fi)	1986-12-27
EP0207420B1 (en)	1992-05-06
KR870000321A (ko)	1987-02-17
JPS62234082A (ja)	1987-10-14
US5098912A (en)	1992-03-24
PT82839A (en)	1986-07-01
NO167090C (no)	1991-10-02
US5380874A (en)	1995-01-10
JPH09143157A (ja)	1997-06-03
KR930005001B1 (ko)	1993-06-11
EP0207420A3 (en)	1988-04-20

Publication	Publication Date	Title
DK304686D0 (da)	1986-06-26	Pyridoncarboxylsyrederivater, fremgangsmaade til fremstilling af samme samt antimikrobielt middel indeholdende derivaterne
ES8702371A1 (es)	1986-12-16	Un procedimiento para preparar nuevos derivados de 6-(4-fenilo sustituido -3(2h) piradazinona.
ES2001670A6 (es)	1988-06-01	Procedimiento para preparar derivados de fenoxiftalida y composiciones herbicidas que los contienen
UA6332A1 (uk)	1994-12-29	Фунгіцидна композиція
DE3672446D1 (en)	1990-08-09	Pantothenolderivate.
GB2182328B (en)	1989-09-20	Diphenyl ether derivatives
IT7829411A0 (it)	1978-11-03	Contenitore, particolarmente per usi d'ufficio.
GB8625106D0 (en)	1986-11-26	Diphenyl ether herbicides
AU2167588A (en)	1989-03-02	Diphenyl ether herbicides
DE3671895D1 (de)	1990-07-19	Stickstoff enthaltende organosilicium-verbindungen.
NO862839D0 (no)	1986-07-14	Tilkoblingslist for telekommunikasjonsanlegg.
JPS5387380A (en)	1978-08-01	Tris(omega-hydroxy polyether)isocyanurate and its preparation
JPS52131580A (en)	1977-11-04	N-substituted pyridinium-2-sulfonylimines, containing same as active ingredient
JPS5233695A (en)	1977-03-14	Novel antimicrobial materials
SU1162191A1 (ru)	2006-12-27	1,1-Этилиденди-(5-бром-2-фуроиламин), проявляющий противовоспалительную активность
CS185939B1 (en)	1978-10-31	Connection for the protection of the tyrostor regulators for feeding the d.c.electromotors

Legal Events

Date	Code	Title	Description
1995-11-20	B1	Patent granted (law 1993)
2006-07-17	PUP	Patent expired