DK158669C - Fremgangsmaade til fremstilling af 6beta-halogensubstituerede penicillansyrederivater. - Google Patents

Fremgangsmaade til fremstilling af 6beta-halogensubstituerede penicillansyrederivater.

Info

Publication number: DK158669C
Authority: DK; Denmark
Prior art keywords: 6beta; halogen; preparing; procedure; acid derivatives
Prior art date: 1979-05-21

Application number

DK218580A

Other languages

English (en)

Other versions

DK158669B (da

DK218580A (da

Inventor

Welf Von Daehne

Original Assignee

Leo Pharm Prod Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1979-05-21

Filing date

1980-05-20

Publication date

1991-01-21

1980-05-20 Application filed by Leo Pharm Prod Ltd filed Critical Leo Pharm Prod Ltd

1980-11-22 Publication of DK218580A publication Critical patent/DK218580A/da

1990-07-02 Publication of DK158669B publication Critical patent/DK158669B/da

1991-01-21 Application granted granted Critical

1991-01-21 Publication of DK158669C publication Critical patent/DK158669C/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

DK218580A 1979-05-21 1980-05-20 Fremgangsmaade til fremstilling af 6beta-halogensubstituerede penicillansyrederivater. DK158669C (da)

Applications Claiming Priority (8)

Application Number	Priority Date	Filing Date	Title
GB7917665		1979-05-21
GB7917665		1979-05-21
GB7930819		1979-09-05
GB7930819		1979-09-05
GB7941252		1979-11-29
GB7941252		1979-11-29
GB8006681		1980-02-27
GB8006681		1980-02-27

Publications (3)

Publication Number	Publication Date
DK218580A DK218580A (da)	1980-11-22
DK158669B DK158669B (da)	1990-07-02
DK158669C true DK158669C (da)	1991-01-21

Family

ID=27449123

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
DK218580A DK158669C (da)	1979-05-21	1980-05-20	Fremgangsmaade til fremstilling af 6beta-halogensubstituerede penicillansyrederivater.
DK562589A DK158670C (da)	1979-05-21	1989-11-10	Fremgangsmaade til fremstilling af 6beta-halogensubstituerede penicillansyrederivater

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
DK562589A DK158670C (da)	1979-05-21	1989-11-10	Fremgangsmaade til fremstilling af 6beta-halogensubstituerede penicillansyrederivater

Country Status (19)

Country	Link
US (3)	US4446144A (da)
JP (1)	JPS55154977A (da)
AU (3)	AU534754B2 (da)
BE (1)	BE883390A (da)
CA (1)	CA1265787A (da)
DE (3)	DE3051037C2 (da)
DK (2)	DK158669C (da)
FI (1)	FI801618A (da)
FR (2)	FR2457294A1 (da)
GR (1)	GR68372B (da)
IE (2)	IE49770B1 (da)
IL (1)	IL59948A0 (da)
IT (1)	IT1133091B (da)
LU (1)	LU82468A1 (da)
NL (1)	NL8002911A (da)
NZ (1)	NZ193597A (da)
PH (2)	PH17959A (da)
PT (1)	PT71273A (da)
SE (3)	SE452465B (da)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4432970A (en) *	1979-11-23	1984-02-21	Pfizer Inc.	6-beta-Halopenicillanic acid 1,1-dioxides as beta-lactamase inhibitors
IE51846B1 (en) *	1980-11-17	1987-04-15	Leo Pharm Prod Ltd	Pharmaceutical preparation for veterinary use and an appliance containing it
US4521533A (en) *	1984-07-12	1985-06-04	Pfizer Inc.	Salts of 6-alpha-(aminomethyl)penicillanic acid 1,1-dioxide esters and beta-lactam antibiotics
GB8522156D0 (en) *	1985-09-06	1985-10-09	Leo Pharm Prod Ltd	Producing chemical compounds
US5589354A (en) *	1994-12-20	1996-12-31	Biopure Corporation	Halogenation of cephalexin with haloperoxidase from Rathayibacter biopuresis
US5695951A (en) *	1994-12-20	1997-12-09	Biopure Corporation	Chlorination of cephalexin with chloroperoxidase from Rathayibacter biopuresis
ES2183223T5 (es)	1996-12-18	2015-05-07	Bimeda Research & Development Limited	Composición intramamaria para uso veterinario que no contiene agentes antiinflamatorios
US20020035107A1 (en) *	2000-06-20	2002-03-21	Stefan Henke	Highly concentrated stable meloxicam solutions
PT1558263E (pt) *	2002-10-25	2006-10-31	Intervet Int Bv	Composicao farmaceutica de libertacao prolongada
EP1568369A1 (en)	2004-02-23	2005-08-31	Boehringer Ingelheim Vetmedica Gmbh	Use of meloxicam for the treatment of respiratory diseases in pigs
DE102004025324A1 (de) *	2004-05-19	2005-12-08	Boehringer Ingelheim Vetmedica Gmbh	Flüssige Zubereitung für die Veterinärmedizin, Verfahren zu deren Herstellung und deren Verwendung
EP2874623B1 (en)	2012-07-17	2018-12-12	Bayer New Zealand Limited	Injectable antibiotic formulations and their methods of use
DK2874624T3 (da) *	2012-07-17	2019-11-11	Bayer New Zealand Ltd	Injicerbare antibiotiske formuleringer og fremgangsmåder til brug af disse
WO2014098624A1 (en) *	2012-12-20	2014-06-26	Alleva Animal Health Limited	Veterinary injectable formulations
EP4265241A1 (en) *	2022-04-20	2023-10-25	Bilim Ilac Sanayii Ve Ticaret A.S.	Tablet formulations for the treatment of urinary system infections and method for the preparation of such formulations

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE1089385B (de)	1954-06-21	1960-09-22	Biochemie Gmbh	Verfahren zur Herstellung von in Wasser schwer loeslichen, besonders fuer die Oraltherapie geeigneten Salzen des Penicillins mit organischen Basen
DE1031795B (de)	1955-09-29	1958-06-12	Chimiotherapie Lab Franc	Verfahren zur Herstellung eines Salzes aus Penicillin und einer Piperazinbase
US3206469A (en) *	1961-08-15	1965-09-14	Lepetit Spa	6-halopenicillanic acid
GB1297555A (da) *	1970-09-22	1972-11-22
GB1377817A (en) *	1971-06-09	1974-12-18	Beecham Group Ltd	Penicillins and cephalosporins
US4234579A (en) *	1977-06-07	1980-11-18	Pfizer Inc.	Penicillanic acid 1,1-dioxides as β-lactamase inhibitors
IN149747B (da) *	1977-06-07	1982-04-03	Pfizer
US4180506A (en) *	1978-01-18	1979-12-25	Rex Pratt	6β-Bromo penicillanic acid
US4203992A (en) *	1978-12-11	1980-05-20	E. R. Squibb & Sons, Inc.	β-Bromopenicillanic acid sulfone
CA1158639A (en) *	1978-12-11	1983-12-13	Eric M. Gordon	6-bromopenicillanic acid sulfone
EP0013617B1 (en) *	1979-01-10	1984-07-04	Beecham Group Plc	Penicillin derivatives, process for their preparation and pharmaceutical compositions containing certain of these compounds
IL59081A0 (en) *	1979-01-10	1980-05-30	Schering Corp	2-penem compounds and a method for preparing them
US4518530A (en) *	1979-03-05	1985-05-21	Pfizer Inc.	6-β-Substituted penicillanic acids as β-lactamase inhibitors
US4397783A (en) *	1979-03-05	1983-08-09	Pfizer Inc.	Process for converting 6,6-disubstituted penicillanic acid derivatives to the 6-β-congeners
US4287181A (en) *	1979-10-22	1981-09-01	Pfizer Inc.	Derivatives of 6β-hydroxyalkylpenicillanic acids as β-lactamase inhibitors
US4432970A (en) *	1979-11-23	1984-02-21	Pfizer Inc.	6-beta-Halopenicillanic acid 1,1-dioxides as beta-lactamase inhibitors

1980
- 1980-04-29 IL IL59948A patent/IL59948A0/xx unknown
- 1980-04-29 IE IE2559/84A patent/IE49770B1/en unknown
- 1980-04-29 IE IE868/80A patent/IE49768B1/en not_active IP Right Cessation
- 1980-05-01 NZ NZ193597A patent/NZ193597A/en unknown
- 1980-05-05 PH PH23982A patent/PH17959A/en unknown
- 1980-05-12 GR GR61906A patent/GR68372B/el unknown
- 1980-05-19 SE SE8003722A patent/SE452465B/sv not_active IP Right Cessation
- 1980-05-20 CA CA000352237A patent/CA1265787A/en not_active Expired - Fee Related
- 1980-05-20 LU LU82468A patent/LU82468A1/fr unknown
- 1980-05-20 JP JP6768580A patent/JPS55154977A/ja active Granted
- 1980-05-20 DK DK218580A patent/DK158669C/da not_active IP Right Cessation
- 1980-05-20 NL NL8002911A patent/NL8002911A/nl not_active Application Discontinuation
- 1980-05-20 FI FI801618A patent/FI801618A/fi not_active Application Discontinuation
- 1980-05-20 DE DE19803051037 patent/DE3051037C2/de not_active Expired
- 1980-05-20 PT PT71273A patent/PT71273A/pt unknown
- 1980-05-20 DE DE19803051038 patent/DE3051038C2/de not_active Expired
- 1980-05-20 FR FR8011263A patent/FR2457294A1/fr active Granted
- 1980-05-20 IT IT67790/80A patent/IT1133091B/it active
- 1980-05-20 AU AU58584/80A patent/AU534754B2/en not_active Ceased
- 1980-05-20 BE BE0/200687A patent/BE883390A/fr not_active IP Right Cessation
- 1980-05-20 DE DE19803019244 patent/DE3019244A1/de active Granted
- 1980-11-17 US US06/207,614 patent/US4446144A/en not_active Expired - Lifetime
1982
- 1982-03-04 FR FR8203636A patent/FR2499575A1/fr active Granted
1983
- 1983-08-26 AU AU18487/83A patent/AU541323B2/en not_active Ceased
- 1983-08-26 PH PH29453A patent/PH19005A/en unknown
- 1983-08-26 AU AU18486/83A patent/AU541322B2/en not_active Ceased
- 1983-12-23 US US06/564,901 patent/US4594246A/en not_active Expired - Fee Related
1984
- 1984-12-06 SE SE8406202A patent/SE462097B/sv not_active IP Right Cessation
- 1984-12-06 SE SE8406201A patent/SE462096B/sv not_active IP Right Cessation
1986
- 1986-03-31 US US06/845,941 patent/US4672114A/en not_active Expired - Fee Related
1989
- 1989-11-10 DK DK562589A patent/DK158670C/da not_active IP Right Cessation

Also Published As

Publication number	Publication date
NZ193597A (en)	1985-04-30
FR2457294A1 (fr)	1980-12-19
DE3019244A1 (de)	1980-12-04
JPH0140837B2 (da)	1989-08-31
DK158669B (da)	1990-07-02
FR2499575B1 (da)	1985-03-01
AU541322B2 (en)	1985-01-03
AU541323B2 (en)	1985-01-03
DE3051038A1 (da)	1986-03-20
DE3019244C2 (da)	1989-04-06
IE800868L (en)	1980-11-21
US4672114A (en)	1987-06-09
IL59948A0 (en)	1980-06-30
US4594246A (en)	1986-06-10
BE883390A (fr)	1980-11-20
DK562589A (da)	1989-11-10
FR2499575A1 (fr)	1982-08-13
SE8406201D0 (sv)	1984-12-06
SE8406202L (sv)	1984-12-06
IE49770B1 (en)	1985-12-11
SE462097B (sv)	1990-05-07
FR2457294B1 (da)	1984-01-13
JPS55154977A (en)	1980-12-02
GR68372B (da)	1981-12-28
AU534754B2 (en)	1984-02-16
US4446144A (en)	1984-05-01
IE842559L (en)	1980-11-21
SE8406202D0 (sv)	1984-12-06
IT8067790A0 (it)	1980-05-20
AU5858480A (en)	1980-11-27
DK158670B (da)	1990-07-02
DK562589D0 (da)	1989-11-10
SE452465B (sv)	1987-11-30
SE462096B (sv)	1990-05-07
NL8002911A (nl)	1980-11-25
DK158670C (da)	1991-01-07
PT71273A (en)	1980-06-01
SE8003722L (sv)	1980-11-22
FI801618A (fi)	1980-11-22
IT1133091B (it)	1986-07-09
PH17959A (en)	1985-02-20
AU1848683A (en)	1983-12-22
DE3051037C2 (da)	1989-03-30
AU1848783A (en)	1983-12-22
PH19005A (en)	1985-12-03
DE3051038C2 (da)	1989-04-13
IE49768B1 (en)	1985-12-11
DK218580A (da)	1980-11-22
LU82468A1 (fr)	1980-12-16
SE8406201L (sv)	1984-12-06
CA1265787A (en)	1990-02-13

Publication	Publication Date	Title
DK478980A (da)	1981-05-13	Fremgangsmaade til fremstilling af imidazol-5-eddikesyrederivater
DK363179A (da)	1980-03-02	Fremgangsmaade til fremstilling af tetrazolylalkoxycarbostyrilderivater
DK457779A (da)	1980-05-01	Fremgangsmaade til fremstilling af 4-hydroxy-2-pyronderivater
DK156056C (da)	1989-11-06	Analogifremgangsmaade til fremstilling af 4-amino-3-quinolin-carboxylsyrederivater
DK540080A (da)	1981-06-20	Fremgangsmaade til fremstilling af 2-amino-4-hydroxyquinazolinderivater
NO802546L (no)	1981-03-02	Fremgangsmaate ved fremstilling av beta-carbolin-3-carboxylsyre-derivater.
DK488379A (da)	1980-05-19	Fremgangsmaade til fremstilling af polyetherderivater
DK286777A (da)	1977-12-30	Fremgangsmade til fremstilling af penicillansyrederivater
DK502078A (da)	1979-05-15	Frefmgangsmaade til fremstilling af cephalosporansyrederivater
DK158669C (da)	1991-01-21	Fremgangsmaade til fremstilling af 6beta-halogensubstituerede penicillansyrederivater.
DK396880A (da)	1981-03-21	Fremgangsmaade til fremstilling af cyclohexancarboxylsyrederivater
DK99980A (da)	1980-09-09	Fremgangsmaade til fremstilling af mercaptoacyldihydropyrazolcarboxylsyrederivater
DK455877A (da)	1978-04-15	Fremgangsmaade til fremstilling af phenyleddikesyrederivater
DK138879A (da)	1979-10-06	Fremgangsmaade til fremstilling af lysergolderivater
DK424080A (da)	1981-04-12	Fremgangsmaade til fremstilling af penicillansyrederivater
DK154554C (da)	1989-04-17	Fremgangsmaade til fremstilling af alfa-methyl-carbazol-2-eddikesyrederivater
DK144277C (da)	1982-07-05	Fremgangsmaade til fremstilling af 6-aminopenicillansyre
DK57381A (da)	1981-08-13	Fremgansmaade til fremstilling af bifenyloxypropionsyrederivater
DK394978A (da)	1979-03-08	Fremgangsmaade til fremstilling af bromerede cephalosporansyrederivater
DK12879A (da)	1979-07-21	R fremgangsmaade til fremstilling af ergopeptidalkaloidderivate
DK145741C (da)	1983-08-01	Fremgangsmaade til fremstilling af 6-chlor-alfa-methyl-carbazol-2-eddikesyre
DK149962C (da)	1987-05-04	Fremgangsmaade til fremstilling af 2,5-diketogluconsyre
DK260079A (da)	1979-12-23	Fremgangsmaade til fremstilling af phenoxyalkylamid-derivater
DK362379A (da)	1980-03-07	Fremgangsmaade til fremstilling af alfa-alkyl-o-oxybenzylaminderivater
DK149197C (da)	1986-08-11	Fremgangsmaade til fremstilling af d,1-beta-benzoylamido-isosmoersyre

Legal Events

Date	Code	Title	Description
1996-01-22	PBP	Patent lapsed