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DK134602B - Analogifremgangsmåde til fremstilling af benzimidazolderivater. - Google Patents

Analogifremgangsmåde til fremstilling af benzimidazolderivater.

Info

Publication number
DK134602B
DK134602B DK321770AA DK321770A DK134602B DK 134602 B DK134602 B DK 134602B DK 321770A A DK321770A A DK 321770AA DK 321770 A DK321770 A DK 321770A DK 134602 B DK134602 B DK 134602B
Authority
DK
Denmark
Prior art keywords
preparation
benzimidazole derivatives
analogous process
analogous
benzimidazole
Prior art date
Application number
DK321770AA
Other languages
Danish (da)
English (en)
Other versions
DK134602C (fi
Inventor
Josephus Ludovicus Hube Gelder
Leopold Frans Corneel Roevens
Alfons Herman Marg Raeymaekers
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of DK134602B publication Critical patent/DK134602B/da
Application granted granted Critical
Publication of DK134602C publication Critical patent/DK134602C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/22—Radicals substituted by doubly bound hetero atoms, or by two hetero atoms other than halogen singly bound to the same carbon atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C205/00—Compounds containing nitro groups bound to a carbon skeleton
    • C07C205/45—Compounds containing nitro groups bound to a carbon skeleton the carbon skeleton being further substituted by at least one doubly—bound oxygen atom, not being part of a —CHO group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/76—Ketones containing a keto group bound to a six-membered aromatic ring
    • C07C49/80—Ketones containing a keto group bound to a six-membered aromatic ring containing halogen
    • C07C49/813—Ketones containing a keto group bound to a six-membered aromatic ring containing halogen polycyclic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/30—Nitrogen atoms not forming part of a nitro radical
    • C07D235/32—Benzimidazole-2-carbamic acids, unsubstituted or substituted; Esters thereof; Thio-analogues thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Fodder In General (AREA)
DK321770AA 1969-06-20 1970-06-22 Analogifremgangsmåde til fremstilling af benzimidazolderivater. DK134602B (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US83524669A 1969-06-20 1969-06-20

Publications (2)

Publication Number Publication Date
DK134602B true DK134602B (da) 1976-12-06
DK134602C DK134602C (fi) 1977-06-27

Family

ID=25269027

Family Applications (2)

Application Number Title Priority Date Filing Date
DK321770AA DK134602B (da) 1969-06-20 1970-06-22 Analogifremgangsmåde til fremstilling af benzimidazolderivater.
DK580275A DK580275A (da) 1969-06-20 1975-12-19 Benzimidazolcarbamater

Family Applications After (1)

Application Number Title Priority Date Filing Date
DK580275A DK580275A (da) 1969-06-20 1975-12-19 Benzimidazolcarbamater

Country Status (20)

Country Link
US (1) US3657267A (fi)
JP (1) JPS501272B1 (fi)
AT (2) AT302358B (fi)
BE (1) BE752089A (fi)
CH (1) CH520684A (fi)
CS (1) CS201522B2 (fi)
DK (2) DK134602B (fi)
ES (1) ES380579A1 (fi)
FI (1) FI52719C (fi)
FR (1) FR2052988B1 (fi)
GB (1) GB1307306A (fi)
HK (1) HK77976A (fi)
IL (1) IL34746A (fi)
IT (1) IT1035027B (fi)
MY (1) MY7300477A (fi)
NL (1) NL147139B (fi)
PL (1) PL72724B1 (fi)
SE (1) SE366045B (fi)
YU (1) YU34195B (fi)
ZA (1) ZA704191B (fi)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2201208A1 (de) * 1972-01-12 1973-08-02 Basf Ag Verfahren zur herstellung von aromatischen ketonen
US3929821A (en) * 1972-12-29 1975-12-30 Syntex Inc 5 (6)-Benzene ring substituted benzimidazole-2-carbamate derivatives
US4258198A (en) * 1973-05-29 1981-03-24 Smithkline Corporation 5-Cycloalkyl thio- and oxy-2-carbalkoxyaminobenzimidazoles
US3969526A (en) * 1973-05-29 1976-07-13 Smithkline Corporation Anthelmintic 5-heterocycliothio and oxy-2-carbalkoxyaminobenzimidazles
DE2443297A1 (de) * 1974-09-10 1976-03-18 Hoechst Ag Anthelminthisch wirksame basisch substituierte 2-carbalkoxy-amino-benzimidazolyl-5(6)-phenylaether und -ketone sowie verfahren zu ihrer herstellung
US4026936A (en) * 1975-08-07 1977-05-31 Hoffmann-La Roche Inc. Anthelmintic pyridine and thiazole substituted benzimidazole carbamates
US4031234A (en) * 1975-08-18 1977-06-21 Syntex (U.S.A.) Inc. 1,5(6)-Disubstituted benzimidazole-2-carbamate derivatives having anthelmintic activity
US4032536A (en) * 1976-07-22 1977-06-28 Janssen Pharmaceutica N.V. (1h-benzimidazol-2-yl)carbamates
IT1076022B (it) * 1977-04-20 1985-04-22 Montedison Spa Benzimidazolcarbammati antielmintici
JPS5535611A (en) * 1978-08-31 1980-03-12 Matsushita Electric Works Ltd Instrument with mouth washing instrument
US4299837A (en) 1979-12-05 1981-11-10 Montedison S.P.A. Anthelmintic benzimidazole-carbamates
US4435418A (en) 1982-12-13 1984-03-06 Smithkline Beckman Corporation 5-Phenylethenylbenzimidazoles
US4438135A (en) 1983-01-07 1984-03-20 Smithkline Beckman Corporation 1-(3,4-Bis-(3-(lower alkoxycarbonyl)-2-thioureido)-phenyl-1-phenylthylenes
WO1990010630A1 (en) * 1989-03-15 1990-09-20 Janssen Pharmaceutica N.V. [5(6)-(benzisoxa-, benzisothia- or indazol-3-yl)-1h-benzimidazol-2-yl] carbamates
NZ232785A (en) * 1989-03-15 1991-03-26 Janssen Pharmaceutica Nv 5-(1,2 benzisoxazol-, benzimidazol and benzisothiazol-3- yl)-1h-benzimadazol-2-yl carbamic acid ester derivatives preparatory processes, intermediates and anthelmintic compositions
US5256681A (en) * 1989-03-15 1993-10-26 Janssen Pharmaceutica N.V. [5(6)-(benzisoxa-,benzisothia-or indazol-3-yl)-1H-benzimidazol-2-yl]carbamates
US5278181A (en) * 1992-05-12 1994-01-11 Board Of Regents Acting On Behalf Of The University Of Michigan Soluble alkyl[5-[amino (phenyl)methyl]-1H-benzimidazol-2-yl] carbamate anthelmintics
JP5227795B2 (ja) * 2005-07-28 2013-07-03 インターベツト・インターナシヨナル・ベー・ベー 抗寄生虫活性を有する新規ベンゾイミダゾール（チオ）カルバメートおよびその合成
WO2008091358A1 (en) * 2006-06-12 2008-07-31 Smith And Nephew Inc Systems, methods and devices for tibial resection
PL2037914T3 (pl) 2006-06-14 2014-04-30 Intervet Int Bv Zawiesina zawierająca karbaminian benzoimidazolu i polisorbat
WO2013110975A1 (es) 2012-01-27 2013-08-01 Siegfried Rhein S.A. De C.V. Composición de nitazoxanida mejorada y proceso para prepararla
EP2902024B1 (en) 2012-09-27 2017-11-29 Siegfried Rhein S.A. De C.V. Synergic composition of nitazoxanide and mebendazole, methods for the preparation thereof, and use of said composition for the treatment of human parasitosis
CN108884054B (zh) 2015-11-30 2022-08-02 儿童医学中心公司 用于治疗增殖性疾病的化合物
CN117899079A (zh) 2017-06-22 2024-04-19 希普拉有限公司 癌症的治疗方法
CN109467512B (zh) * 2018-12-18 2021-06-08 苏州开元民生科技股份有限公司 一种3,4-二氨基-二苯甲酮的合成方法
CN113979949A (zh) * 2021-12-17 2022-01-28 山东国邦药业有限公司 一种氟苯咪唑的制备方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1111957A (en) * 1966-05-20 1968-05-01 Smith Kline French Lab Improvements in or relating to anthelmintic compositions

Also Published As

Publication number Publication date
ES380579A1 (es) 1973-04-01
IT1035027B (it) 1979-10-20
SE366045B (fi) 1974-04-08
FI52719B (fi) 1977-08-01
HK77976A (en) 1976-12-17
DK134602C (fi) 1977-06-27
CH520684A (fr) 1972-03-31
FI52719C (fi) 1977-11-10
MY7300477A (en) 1973-12-31
GB1307306A (en) 1973-02-21
NL7009024A (fi) 1970-12-22
BE752089A (fr) 1970-12-17
CS201522B2 (en) 1980-11-28
PL72724B1 (fi) 1974-08-30
YU154470A (en) 1978-09-18
AT307798B (de) 1973-06-12
DE2029637B2 (de) 1976-09-23
DE2029637A1 (de) 1971-02-18
AT302358B (de) 1972-10-10
YU34195B (en) 1979-02-28
IL34746A0 (en) 1970-08-19
JPS501272B1 (fi) 1975-01-16
NL147139B (nl) 1975-09-15
IL34746A (en) 1973-01-30
FR2052988A1 (fi) 1971-04-16
FR2052988B1 (fi) 1973-08-10
US3657267A (en) 1972-04-18
ZA704191B (en) 1972-02-23
DK580275A (da) 1975-12-19

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