DK1216249T3 - Usubstituerede ethyl- og propylderivater af phenoxythienoisoxazoler som D4-antagonister - Google Patents

Usubstituerede ethyl- og propylderivater af phenoxythienoisoxazoler som D4-antagonister

Info

Publication number: DK1216249T3
Authority: DK; Denmark
Prior art keywords: phenoxythienoisoxazoles; antagonists; unsubstituted ethyl; propyl derivatives; propyl
Prior art date: 1999-09-14

Application number

DK00964967T

Other languages

English (en)

Inventor

George E Lee

John G Jurcak

Timothy A Ayers

Original Assignee

Aventis Pharma Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-09-14

Filing date

2000-09-13

Publication date

2004-03-15

2000-09-13 Application filed by Aventis Pharma Inc filed Critical Aventis Pharma Inc

2004-03-15 Application granted granted Critical

2004-03-15 Publication of DK1216249T3 publication Critical patent/DK1216249T3/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Psychology (AREA)
Psychiatry (AREA)
Addiction (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

DK00964967T 1999-09-14 2000-09-13 Usubstituerede ethyl- og propylderivater af phenoxythienoisoxazoler som D4-antagonister DK1216249T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US39615699A	1999-09-14	1999-09-14
PCT/US2000/024949 WO2001019832A2 (en)	1999-09-14	2000-09-13	Thienoisoxazole phenoxy unsubstituted ethyl and propyl derivatives useful as d4 antagonists

Publications (1)

Publication Number	Publication Date
DK1216249T3 true DK1216249T3 (da)	2004-03-15

Family

ID=23566087

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK00964967T DK1216249T3 (da)	1999-09-14	2000-09-13	Usubstituerede ethyl- og propylderivater af phenoxythienoisoxazoler som D4-antagonister

Country Status (23)

Country	Link
EP (1)	EP1216249B1 (da)
JP (1)	JP4717306B2 (da)
KR (1)	KR20020027644A (da)
AR (1)	AR032135A1 (da)
AT (1)	ATE254620T1 (da)
AU (1)	AU7577200A (da)
BR (1)	BR0014513A (da)
CA (1)	CA2383327C (da)
CZ (1)	CZ2002896A3 (da)
DE (1)	DE60006698T2 (da)
DK (1)	DK1216249T3 (da)
EA (1)	EA004177B1 (da)
EE (1)	EE200200133A (da)
ES (1)	ES2206305T3 (da)
HU (1)	HUP0202712A3 (da)
IL (1)	IL148522A0 (da)
MX (1)	MXPA02002690A (da)
NO (1)	NO20021249L (da)
PL (1)	PL354481A1 (da)
PT (1)	PT1216249E (da)
SK (1)	SK3502002A3 (da)
WO (1)	WO2001019832A2 (da)
ZA (1)	ZA200201760B (da)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB0207449D0 (en) *	2002-03-28	2002-05-08	Glaxo Group Ltd	Novel compounds
WO2018166855A1 (en)	2017-03-16	2018-09-20	Basf Se	Heterobicyclic substituted dihydroisoxazoles

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4728651A (en) *	1985-10-24	1988-03-01	Hoechst-Roussel Pharmaceuticals Inc.	Antihypertensive thieno-isoxazoles and -pyrazoles
US6187774B1 (en) *	1996-03-04	2001-02-13	Yoshitomi Pharmaceutical Industries, Ltd.	Fused heterocyclic compounds and pharmaceutical applications thereof
HUP9603001A3 (en) *	1996-10-30	1999-07-28	Richter Gedeon Vegyeszet	Heterocycle compounds comprising nitrogen, process for producing them and pharmaceutical compositions containing the same
DK1054885T3 (da) *	1998-02-09	2007-10-15	Duphar Int Res	Benzisoxasolderivater med D4-antagonistisk virkning

2000
- 2000-09-13 EE EEP200200133A patent/EE200200133A/xx unknown
- 2000-09-13 WO PCT/US2000/024949 patent/WO2001019832A2/en not_active Application Discontinuation
- 2000-09-13 PL PL00354481A patent/PL354481A1/xx unknown
- 2000-09-13 IL IL14852200A patent/IL148522A0/xx unknown
- 2000-09-13 ES ES00964967T patent/ES2206305T3/es not_active Expired - Lifetime
- 2000-09-13 DE DE60006698T patent/DE60006698T2/de not_active Expired - Lifetime
- 2000-09-13 AR ARP000104794A patent/AR032135A1/es not_active Application Discontinuation
- 2000-09-13 MX MXPA02002690A patent/MXPA02002690A/es active IP Right Grant
- 2000-09-13 CZ CZ2002896A patent/CZ2002896A3/cs unknown
- 2000-09-13 AT AT00964967T patent/ATE254620T1/de not_active IP Right Cessation
- 2000-09-13 PT PT00964967T patent/PT1216249E/pt unknown
- 2000-09-13 DK DK00964967T patent/DK1216249T3/da active
- 2000-09-13 CA CA002383327A patent/CA2383327C/en not_active Expired - Fee Related
- 2000-09-13 HU HU0202712A patent/HUP0202712A3/hu unknown
- 2000-09-13 EP EP00964967A patent/EP1216249B1/en not_active Expired - Lifetime
- 2000-09-13 SK SK350-2002A patent/SK3502002A3/sk unknown
- 2000-09-13 EA EA200200357A patent/EA004177B1/ru not_active IP Right Cessation
- 2000-09-13 KR KR1020027003354A patent/KR20020027644A/ko not_active Application Discontinuation
- 2000-09-13 AU AU75772/00A patent/AU7577200A/en not_active Abandoned
- 2000-09-13 JP JP2001523409A patent/JP4717306B2/ja not_active Expired - Fee Related
- 2000-09-13 BR BR0014513-0A patent/BR0014513A/pt not_active IP Right Cessation
2002
- 2002-03-01 ZA ZA200201760A patent/ZA200201760B/en unknown
- 2002-03-13 NO NO20021249A patent/NO20021249L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
HUP0202712A2 (hu)	2002-12-28
EP1216249A2 (en)	2002-06-26
BR0014513A (pt)	2002-07-02
AR032135A1 (es)	2003-10-29
AU7577200A (en)	2001-04-17
EA200200357A1 (ru)	2002-10-31
CZ2002896A3 (cs)	2002-08-14
ATE254620T1 (de)	2003-12-15
DE60006698D1 (de)	2003-12-24
DE60006698T2 (de)	2004-09-23
NO20021249L (no)	2002-05-10
HUP0202712A3 (en)	2004-12-28
SK3502002A3 (en)	2002-09-10
WO2001019832A3 (en)	2001-10-04
WO2001019832A2 (en)	2001-03-22
JP4717306B2 (ja)	2011-07-06
CA2383327A1 (en)	2001-03-22
EE200200133A (et)	2003-04-15
NO20021249D0 (no)	2002-03-13
JP2003509431A (ja)	2003-03-11
PT1216249E (pt)	2004-04-30
ZA200201760B (en)	2003-08-27
CA2383327C (en)	2009-11-03
IL148522A0 (en)	2002-09-12
PL354481A1 (en)	2004-01-26
EP1216249B1 (en)	2003-11-19
KR20020027644A (ko)	2002-04-13
EA004177B1 (ru)	2004-02-26
ES2206305T3 (es)	2004-05-16
MXPA02002690A (es)	2004-09-10

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DK1216249T3 (da)	2004-03-15	Usubstituerede ethyl- og propylderivater af phenoxythienoisoxazoler som D4-antagonister