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DK0546388T3 - Azaheterocyclylmethyl-chromaner som aktive stoffer til behandling af sygdomme i centralnervesystemet - Google Patents

Azaheterocyclylmethyl-chromaner som aktive stoffer til behandling af sygdomme i centralnervesystemet

Info

Publication number
DK0546388T3
DK0546388T3 DK92120187.7T DK92120187T DK0546388T3 DK 0546388 T3 DK0546388 T3 DK 0546388T3 DK 92120187 T DK92120187 T DK 92120187T DK 0546388 T3 DK0546388 T3 DK 0546388T3
Authority
DK
Denmark
Prior art keywords
treatment
nervous system
central nervous
azaheterocyclylmethyl
chromanes
Prior art date
Application number
DK92120187.7T
Other languages
English (en)
Inventor
Hans-Georg Dr Heine
Jean Marie Viktor Dr De Vry
Wolfgang Dr Dompert
Henning Dr Sommermeyer
Rudolf Dr Schohe-Loop
Thomas Dr Dr Glaser
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Application granted granted Critical
Publication of DK0546388T3 publication Critical patent/DK0546388T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Endocrinology (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Hospice & Palliative Care (AREA)
  • Anesthesiology (AREA)
  • Addiction (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pyrane Compounds (AREA)
  • Cosmetics (AREA)
DK92120187.7T 1991-12-09 1992-11-26 Azaheterocyclylmethyl-chromaner som aktive stoffer til behandling af sygdomme i centralnervesystemet DK0546388T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4140540A DE4140540A1 (de) 1991-12-09 1991-12-09 Neue azaheterocyclylmethyl-chromane

Publications (1)

Publication Number Publication Date
DK0546388T3 true DK0546388T3 (da) 1996-07-29

Family

ID=6446618

Family Applications (1)

Application Number Title Priority Date Filing Date
DK92120187.7T DK0546388T3 (da) 1991-12-09 1992-11-26 Azaheterocyclylmethyl-chromaner som aktive stoffer til behandling af sygdomme i centralnervesystemet

Country Status (22)

Country Link
US (5) US5371094A (da)
EP (1) EP0546388B1 (da)
JP (1) JP3220266B2 (da)
AT (1) ATE136030T1 (da)
AU (1) AU650182B2 (da)
CA (1) CA2084542A1 (da)
CZ (1) CZ283680B6 (da)
DE (2) DE4140540A1 (da)
DK (1) DK0546388T3 (da)
ES (1) ES2086623T3 (da)
FI (1) FI925549A (da)
GR (1) GR3019450T3 (da)
HU (1) HUT65427A (da)
IL (1) IL104006A (da)
MX (1) MX9206817A (da)
NO (1) NO303174B1 (da)
NZ (1) NZ245381A (da)
PH (1) PH31072A (da)
RU (1) RU2089549C1 (da)
SK (1) SK278553B6 (da)
TW (1) TW210339B (da)
ZA (1) ZA929498B (da)

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US5478934A (en) * 1994-11-23 1995-12-26 Yuan; Jun Certain 1-substituted aminomethyl imidazole and pyrrole derivatives: novel dopamine receptor subtype specific ligands
US6096763A (en) * 1995-02-23 2000-08-01 Merck & Co., Inc. α1a adrenergic receptor antagonists
US5541199A (en) * 1995-06-02 1996-07-30 American Home Products Corporation Chroman-2-ylmethylamino derivatives
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US5670667A (en) * 1995-07-25 1997-09-23 American Home Products Corporation Chroman-2-ylmethylamino derivatives
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US6555560B2 (en) 2001-04-30 2003-04-29 Wyeth Antidepressant azaheterocyclylmethyl derivatives of 1,4,5-trioxa-phenanthrene
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Also Published As

Publication number Publication date
NO303174B1 (no) 1998-06-08
FI925549A0 (fi) 1992-12-07
JPH05279357A (ja) 1993-10-26
RU2089549C1 (ru) 1997-09-10
US5371094A (en) 1994-12-06
EP0546388A1 (de) 1993-06-16
JP3220266B2 (ja) 2001-10-22
IL104006A0 (en) 1993-05-13
TW210339B (da) 1993-08-01
EP0546388B1 (de) 1996-03-27
DE59205846D1 (de) 1996-05-02
HUT65427A (en) 1994-06-28
MX9206817A (es) 1994-06-30
PH31072A (en) 1998-02-05
ZA929498B (en) 1993-06-10
CZ361392A3 (en) 1993-10-13
SK361392A3 (en) 1997-09-10
IL104006A (en) 1997-02-18
SK278553B6 (en) 1997-09-10
ES2086623T3 (es) 1996-07-01
NO924546L (no) 1993-06-10
US5545643A (en) 1996-08-13
AU650182B2 (en) 1994-06-09
DE4140540A1 (de) 1993-06-17
CA2084542A1 (en) 1993-06-10
US5696136A (en) 1997-12-09
GR3019450T3 (en) 1996-06-30
ATE136030T1 (de) 1996-04-15
NZ245381A (en) 1995-03-28
US5696137A (en) 1997-12-09
US5693653A (en) 1997-12-02
FI925549A (fi) 1993-06-10
HU9203894D0 (en) 1993-03-29
CZ283680B6 (cs) 1998-06-17
AU2993892A (en) 1993-06-10
NO924546D0 (no) 1992-11-25

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