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DE60204633D1 - Sulfonyl-Heteroaryl-Triazole als entzündungshemmende und analgetische Mittel - Google Patents

Sulfonyl-Heteroaryl-Triazole als entzündungshemmende und analgetische Mittel

Info

Publication number
DE60204633D1
DE60204633D1 DE60204633T DE60204633T DE60204633D1 DE 60204633 D1 DE60204633 D1 DE 60204633D1 DE 60204633 T DE60204633 T DE 60204633T DE 60204633 T DE60204633 T DE 60204633T DE 60204633 D1 DE60204633 D1 DE 60204633D1
Authority
DE
Germany
Prior art keywords
triazoles
sulfonyl
heteroaryl
inflammatory
analgesic agents
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE60204633T
Other languages
English (en)
Other versions
DE60204633T2 (de
Inventor
Subas Man Sakya
Andrei Shavnya
Bryson Rast
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Products Inc
Original Assignee
Pfizer Products Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc filed Critical Pfizer Products Inc
Publication of DE60204633D1 publication Critical patent/DE60204633D1/de
Application granted granted Critical
Publication of DE60204633T2 publication Critical patent/DE60204633T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • A61P29/02—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
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    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

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  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
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  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Diabetes (AREA)
  • Rheumatology (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
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  • Tropical Medicine & Parasitology (AREA)
  • Heart & Thoracic Surgery (AREA)
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DE60204633T 2001-07-05 2002-07-01 Sulfonyl-Heteroaryl-Triazole als entzündungshemmende und analgetische Mittel Expired - Fee Related DE60204633T2 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US30323201P 2001-07-05 2001-07-05

Publications (2)

Publication Number Publication Date
DE60204633D1 true DE60204633D1 (de) 2005-07-21
DE60204633T2 DE60204633T2 (de) 2006-06-14

Family

ID=23171118

Family Applications (1)

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DE60204633T Expired - Fee Related DE60204633T2 (de) 2001-07-05 2002-07-01 Sulfonyl-Heteroaryl-Triazole als entzündungshemmende und analgetische Mittel

Country Status (9)

Country Link
US (2) US6753332B2 (de)
EP (1) EP1273580B1 (de)
JP (1) JP2003040887A (de)
AT (1) ATE297913T1 (de)
BR (1) BR0202546A (de)
CA (1) CA2392271C (de)
DE (1) DE60204633T2 (de)
ES (1) ES2240661T3 (de)
MX (1) MXPA02006723A (de)

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KR100686537B1 (ko) * 2001-12-28 2007-02-27 씨제이 주식회사 사이클로옥시게나제-2 의 저해제로서 선택성이 뛰어난디아릴 1,2,4-트리아졸 유도체
KR100467668B1 (ko) * 2002-08-07 2005-01-24 씨제이 주식회사 1,2,4-트리아졸 유도체, 그 제조방법 및 약제학적 조성물
AU2003264018A1 (en) * 2002-08-09 2004-02-25 Astrazeneca Ab Compounds having an activity at metabotropic glutamate receptors
KR100491317B1 (ko) * 2002-11-26 2005-05-24 씨제이 주식회사 1,2,4-트리아졸 유도체, 그 제조방법 및 약제학적 조성물
EP1673355A1 (de) * 2003-09-22 2006-06-28 Pfizer Limited Substituierte triazolderivate als oxytocinantagonisten
WO2008080938A1 (en) * 2006-12-28 2008-07-10 Basf Se Use 2-substituted pyridines for cancer treatment
JP5719835B2 (ja) 2009-04-27 2015-05-20 ダウ アグロサイエンシィズ エルエルシー 殺虫性ピリジン化合物
EP2527335B1 (de) * 2011-04-26 2013-09-18 King Saud University Triazolderivate als Entzündungshemmer
US8853248B2 (en) * 2012-04-05 2014-10-07 Hubert Maehr (1,2,3-triazolyl)sulfonyl derivatives
CN112142716B (zh) * 2020-10-29 2021-08-31 山东新时代药业有限公司 一种5元杂芳基取代的吡嗪衍生物及其应用

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US4259504A (en) 1979-08-27 1981-03-31 American Cyanamid Company Substituted 1H-1,2,4-triazoles
HU193891B (en) 1984-02-07 1987-12-28 Gyogyszerkutato Intezet Process for production of new derivatives of 1,2,4-triasole
US5256680A (en) 1988-11-29 1993-10-26 Warner-Lambert Company 3,5-di-tertiary-butyl-4-hydroxyphenyl-1,3,4-thiadiazoles, and oxadiazoles and 3,5-di-tertiary-butyl-4-hydroxy-phenyl-1,2,4-thiadazoles, oxadiazoles and triazoles as antiinflammatory agents
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EP1273580B1 (de) 2005-06-15
ATE297913T1 (de) 2005-07-15
DE60204633T2 (de) 2006-06-14
CA2392271A1 (en) 2003-01-05
BR0202546A (pt) 2003-05-13
JP2003040887A (ja) 2003-02-13
CA2392271C (en) 2006-08-29
EP1273580A1 (de) 2003-01-08
MXPA02006723A (es) 2003-01-23
US20030119835A1 (en) 2003-06-26
US6753332B2 (en) 2004-06-22
US20040198735A1 (en) 2004-10-07
ES2240661T3 (es) 2005-10-16

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