DE60200041D1 - Indenoindolon-Derivate, Verfahren zu ihrer Herstellung und die enthaltenden pharmazeutischen Zusammensetzungen - Google Patents

Indenoindolon-Derivate, Verfahren zu ihrer Herstellung und die enthaltenden pharmazeutischen Zusammensetzungen

Info

Publication number: DE60200041D1
Authority: DE; Germany
Prior art keywords: preparation; pharmaceutical compositions; compositions containing; indenoindolone; derivatives
Prior art date: 2001-03-19
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired - Fee Related

Application number

DE60200041T

Other languages

English (en)

Other versions

DE60200041T2 (de

Inventor

Michel Wierzbicki

Marie-Francoise Boussard

Anne Rousseau

Jean-Albert Boutin

Philippe Delagrange

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Laboratoires Servier SAS

Original Assignee

Laboratoires Servier SAS

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-03-19

Filing date

2002-03-18

Publication date

2003-10-30

2002-03-18 Application filed by Laboratoires Servier SAS filed Critical Laboratoires Servier SAS

2003-10-30 Application granted granted Critical

2003-10-30 Publication of DE60200041D1 publication Critical patent/DE60200041D1/de

2004-06-09 Publication of DE60200041T2 publication Critical patent/DE60200041T2/de

2022-03-19 Anticipated expiration legal-status Critical

Status Expired - Fee Related legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/56—Ring systems containing three or more rings
- C07D209/80—[b, c]- or [b, d]-condensed
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Veterinary Medicine (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Diabetes (AREA)
Endocrinology (AREA)
Pain & Pain Management (AREA)
Reproductive Health (AREA)
Epidemiology (AREA)
Psychiatry (AREA)
Hematology (AREA)
Obesity (AREA)
Hospice & Palliative Care (AREA)
Anesthesiology (AREA)
Emergency Medicine (AREA)
Child & Adolescent Psychology (AREA)
Gynecology & Obstetrics (AREA)
Pregnancy & Childbirth (AREA)
Heart & Thoracic Surgery (AREA)
Psychology (AREA)
Cardiology (AREA)
Indole Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

DE60200041T 2001-03-19 2002-03-18 Indenoindolon-Derivate, Verfahren zu ihrer Herstellung und die enthaltenden pharmazeutischen Zusammensetzungen Expired - Fee Related DE60200041T2 (de)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR0103667		2001-03-19
FR0103667A FR2822153B1 (fr)	2001-03-19	2001-03-19	Nouveaux derives d'indenoindolones, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Publications (2)

Publication Number	Publication Date
DE60200041D1 true DE60200041D1 (de)	2003-10-30
DE60200041T2 DE60200041T2 (de)	2004-06-09

Family

ID=8861264

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DE60200041T Expired - Fee Related DE60200041T2 (de)	2001-03-19	2002-03-18	Indenoindolon-Derivate, Verfahren zu ihrer Herstellung und die enthaltenden pharmazeutischen Zusammensetzungen

Country Status (24)

Country	Link
US (1)	US6844445B2 (de)
EP (1)	EP1245565B1 (de)
JP (1)	JP3886829B2 (de)
KR (1)	KR100453979B1 (de)
CN (1)	CN1185214C (de)
AR (1)	AR034861A1 (de)
AT (1)	ATE250578T1 (de)
AU (1)	AU780027B2 (de)
BR (1)	BR0200871A (de)
CA (1)	CA2378628C (de)
DE (1)	DE60200041T2 (de)
DK (1)	DK1245565T3 (de)
EA (1)	EA004711B1 (de)
ES (1)	ES2207629T3 (de)
FR (1)	FR2822153B1 (de)
HK (1)	HK1049159B (de)
HU (1)	HU226674B1 (de)
MX (1)	MXPA02002816A (de)
NO (1)	NO321890B1 (de)
NZ (1)	NZ517855A (de)
PL (1)	PL352866A1 (de)
PT (1)	PT1245565E (de)
SI (1)	SI1245565T1 (de)
ZA (1)	ZA200202220B (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE102006047231B4 (de) *	2006-10-04	2009-02-12	Hemmerling, Hans-Jörg, Dr.	Substituierte Indeno[1,2-b]indolderivate als neue Hemmstoffe der Protein Kinase CK2 und ihre Verwendung als Tumor Therapeutika, Cytostatika und Diagnostika
JP4831077B2 (ja) *	2008-01-15	2011-12-07	三菱電機株式会社	燃料圧力調整器およびそれを用いた燃料供給装置
ES2580702B1 (es)	2015-02-25	2017-06-08	Palobiofarma, S.L.	Derivados de 2-aminopiridina como antagonistas del receptor A2b de adenosina y ligandos del receptor MT3 de melatonina
WO2019058393A1 (en)	2017-09-22	2019-03-28	Jubilant Biosys Limited	HETEROCYCLIC COMPOUNDS AS INHIBITORS OF PAD
FI3697785T3 (fi)	2017-10-18	2023-04-03	Jubilant Epipad LLC	Imidatsopyridiiniyhdisteitä pad:n estäjinä
US11629135B2 (en)	2017-11-06	2023-04-18	Jubilant Prodell Llc	Pyrimidine derivatives as inhibitors of PD1/PD-L1 activation
WO2019102494A1 (en)	2017-11-24	2019-05-31	Jubilant Biosys Limited	Heterocyclic compounds as prmt5 inhibitors
SG11202008950PA (en)	2018-03-13	2020-10-29	Jubilant Prodel LLC	Bicyclic compounds as inhibitors of pd1/pd-l1 interaction/activation

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CZ65393A3 (en) *	1990-10-16	1994-02-16	Univ Bath	Indenoindole derivative, process of its preparation and pharmaceutical preparation in which said derivative is comprised

2001
- 2001-03-19 FR FR0103667A patent/FR2822153B1/fr not_active Expired - Fee Related
2002
- 2002-03-14 MX MXPA02002816A patent/MXPA02002816A/es active IP Right Grant
- 2002-03-18 CN CNB021075778A patent/CN1185214C/zh not_active Expired - Fee Related
- 2002-03-18 DE DE60200041T patent/DE60200041T2/de not_active Expired - Fee Related
- 2002-03-18 NO NO20021330A patent/NO321890B1/no not_active IP Right Cessation
- 2002-03-18 EA EA200200263A patent/EA004711B1/ru unknown
- 2002-03-18 JP JP2002073851A patent/JP3886829B2/ja not_active Expired - Fee Related
- 2002-03-18 PT PT02290668T patent/PT1245565E/pt unknown
- 2002-03-18 SI SI200230003T patent/SI1245565T1/xx unknown
- 2002-03-18 AT AT02290668T patent/ATE250578T1/de not_active IP Right Cessation
- 2002-03-18 AR ARP020100952A patent/AR034861A1/es unknown
- 2002-03-18 ES ES02290668T patent/ES2207629T3/es not_active Expired - Lifetime
- 2002-03-18 NZ NZ517855A patent/NZ517855A/xx unknown
- 2002-03-18 DK DK02290668T patent/DK1245565T3/da active
- 2002-03-18 EP EP02290668A patent/EP1245565B1/de not_active Expired - Lifetime
- 2002-03-19 AU AU27469/02A patent/AU780027B2/en not_active Ceased
- 2002-03-19 CA CA002378628A patent/CA2378628C/fr not_active Expired - Fee Related
- 2002-03-19 BR BR0200871-8A patent/BR0200871A/pt not_active IP Right Cessation
- 2002-03-19 ZA ZA200202220A patent/ZA200202220B/xx unknown
- 2002-03-19 PL PL02352866A patent/PL352866A1/xx not_active IP Right Cessation
- 2002-03-19 HU HU0201024A patent/HU226674B1/hu not_active IP Right Cessation
- 2002-03-19 KR KR10-2002-0014738A patent/KR100453979B1/ko not_active IP Right Cessation
- 2002-03-19 US US10/100,784 patent/US6844445B2/en not_active Expired - Fee Related
2003
- 2003-02-18 HK HK03101148.6A patent/HK1049159B/zh not_active IP Right Cessation

Also Published As

Publication number	Publication date
CA2378628C (fr)	2007-07-10
NO20021330L (no)	2002-09-20
US20020173531A1 (en)	2002-11-21
JP2002322150A (ja)	2002-11-08
MXPA02002816A (es)	2004-11-12
DE60200041T2 (de)	2004-06-09
NZ517855A (en)	2002-10-25
AU2746902A (en)	2002-09-26
ATE250578T1 (de)	2003-10-15
EP1245565B1 (de)	2003-09-24
FR2822153A1 (fr)	2002-09-20
HUP0201024A3 (en)	2003-12-29
HK1049159B (zh)	2005-07-29
EA200200263A3 (ru)	2002-12-26
JP3886829B2 (ja)	2007-02-28
ZA200202220B (en)	2002-10-10
KR100453979B1 (ko)	2004-10-20
EA004711B1 (ru)	2004-06-24
CN1375490A (zh)	2002-10-23
HU0201024D0 (de)	2002-05-29
AR034861A1 (es)	2004-03-24
KR20020074420A (ko)	2002-09-30
HK1049159A1 (en)	2003-05-02
FR2822153B1 (fr)	2003-10-31
HU226674B1 (en)	2009-06-29
DK1245565T3 (da)	2004-01-12
SI1245565T1 (en)	2003-12-31
PL352866A1 (en)	2002-09-23
CA2378628A1 (fr)	2002-09-19
PT1245565E (pt)	2003-12-31
ES2207629T3 (es)	2004-06-01
EA200200263A2 (ru)	2002-10-31
NO321890B1 (no)	2006-07-17
HUP0201024A2 (hu)	2002-11-28
AU780027B2 (en)	2005-02-24
EP1245565A1 (de)	2002-10-02
BR0200871A (pt)	2003-01-07
US6844445B2 (en)	2005-01-18
CN1185214C (zh)	2005-01-19
NO20021330D0 (no)	2002-03-18

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Legal Events

Date	Code	Title	Description
2004-10-21	8364	No opposition during term of opposition
2011-01-20	8339	Ceased/non-payment of the annual fee