DE60111228D1 - Heteropolycyclische inhibitoren - Google Patents
Heteropolycyclische inhibitorenInfo
- Publication number
- DE60111228D1 DE60111228D1 DE60111228T DE60111228T DE60111228D1 DE 60111228 D1 DE60111228 D1 DE 60111228D1 DE 60111228 T DE60111228 T DE 60111228T DE 60111228 T DE60111228 T DE 60111228T DE 60111228 D1 DE60111228 D1 DE 60111228D1
- Authority
- DE
- Germany
- Prior art keywords
- heteropolycyclic
- inhibitors
- administering
- compound
- formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Fee Related
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US61103800A | 2000-07-06 | 2000-07-06 | |
US611038 | 2000-07-06 | ||
PCT/IB2001/001519 WO2002002562A2 (en) | 2000-07-06 | 2001-07-06 | Heteropolycyclic inhibitors |
Publications (2)
Publication Number | Publication Date |
---|---|
DE60111228D1 true DE60111228D1 (de) | 2005-07-07 |
DE60111228T2 DE60111228T2 (de) | 2006-03-16 |
Family
ID=24447360
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DE60111228T Expired - Fee Related DE60111228T2 (de) | 2000-07-06 | 2001-07-06 | Heteropolycyclische inhibitoren |
Country Status (8)
Country | Link |
---|---|
US (2) | US6514972B2 (de) |
EP (1) | EP1296985B1 (de) |
AT (1) | ATE296827T1 (de) |
AU (1) | AU2001277659A1 (de) |
CA (1) | CA2414885A1 (de) |
DE (1) | DE60111228T2 (de) |
ES (1) | ES2243527T3 (de) |
WO (1) | WO2002002562A2 (de) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6514972B2 (en) * | 2000-07-06 | 2003-02-04 | Kinetek Pharmaceuticals, Inc. | Heteropolycyclic inhibitors of protein kinases |
US8715708B2 (en) * | 2005-08-31 | 2014-05-06 | University Of Maryland | Cyclic acetal biomaterials |
CA2632635C (en) * | 2005-12-08 | 2014-04-29 | Hybrigenics Sa | Novel inhibitors of cysteine proteases, the pharmaceutical compositions thereof and their therapeutic applications |
US7462615B2 (en) * | 2005-12-08 | 2008-12-09 | Hybrigenics Sa | Inhibitors of cysteine proteases, the pharmaceutical compositions thereof and their therapeutic applications |
EP1798232A1 (de) * | 2005-12-08 | 2007-06-20 | Hybrigenics S.A. | Cysteine Proteasehemmer, deren pharmazeutische Zusammensetzungen und therapeutische Anwendungen |
MX2009004517A (es) * | 2006-10-30 | 2009-05-13 | Hybrigenics Sa | Nuevos inhibidores tetraciclicos de las proteasas de cisteina, las composiciones farmaceuticas de las mismas y sus aplicaciones terapeuticas. |
US7875613B2 (en) * | 2006-10-30 | 2011-01-25 | Hybrigenics Sa | Tetracyclic inhibitors of cysteine proteases, the pharmaceutical compositions thereof and their therapeutic applications |
EP1918292A1 (de) * | 2006-10-30 | 2008-05-07 | Hybrigenics S.A. | Tetrazyklische Inhibitoren für Cysteinproteasen, pharmazeutische Zubereitungen und therapeutische Anwendungen |
WO2012006104A2 (en) * | 2010-06-28 | 2012-01-12 | Academia Sinica, Taiwan | Compounds and methods for treating tuberculosis infection |
CN103520165A (zh) * | 2013-10-31 | 2014-01-22 | 华东理工大学 | 茚并三嗪类化合物作为依赖nad(p)h的醌氧化还原酶底物的用途 |
US10517871B2 (en) | 2015-05-15 | 2019-12-31 | Indiana University Research And Technology Corporation | Survivin-targeting anti-tumor agents and uses thereof |
CN105061360B (zh) * | 2015-07-28 | 2018-06-19 | 首都师范大学 | 一种3,4-二氨基-1,2,5-噻二唑的提纯方法 |
JP2022511371A (ja) | 2018-09-28 | 2022-01-31 | アキュセラ インコーポレイテッド | Vap-1の阻害剤 |
CN113368080B (zh) * | 2020-02-25 | 2023-11-17 | 香港中文大学 | 稳定的、生物粘附的、扩散限制性团聚体 |
WO2022103827A1 (en) * | 2020-11-10 | 2022-05-19 | New Mexico Tech University Research Park Corporation | Kp372-1-induced dna damage as a chemotherapeutic approach to treat cancer |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4159375A (en) * | 1978-08-24 | 1979-06-26 | American Cyanamid Company | 6- AND 7-Aryl-1,2,4-triazolo[4,3-b]-1,2,4-triazines |
US4405619A (en) * | 1981-09-02 | 1983-09-20 | Diamond Shamrock Corporation | Antiinflammatory substituted-1,2,4-triazolo[4,3-b]-1,2,4-triazines |
GB8826237D0 (en) | 1988-11-09 | 1988-12-14 | Univ Belfast | Fingerprint reagent |
WO1995024190A2 (en) | 1994-03-07 | 1995-09-14 | Sugen, Inc. | Receptor tyrosine kinase inhibitors for inhibiting cell proliferative disorders and compositions thereof |
AU2001240021A1 (en) * | 2000-04-13 | 2001-10-30 | Millennium Pharmaceuticals, Inc. | Diazafluorenone il-8 receptor antagonists |
US6514972B2 (en) * | 2000-07-06 | 2003-02-04 | Kinetek Pharmaceuticals, Inc. | Heteropolycyclic inhibitors of protein kinases |
-
2001
- 2001-07-06 US US09/900,073 patent/US6514972B2/en not_active Expired - Fee Related
- 2001-07-06 WO PCT/IB2001/001519 patent/WO2002002562A2/en active IP Right Grant
- 2001-07-06 ES ES01955500T patent/ES2243527T3/es not_active Expired - Lifetime
- 2001-07-06 DE DE60111228T patent/DE60111228T2/de not_active Expired - Fee Related
- 2001-07-06 CA CA002414885A patent/CA2414885A1/en not_active Abandoned
- 2001-07-06 EP EP01955500A patent/EP1296985B1/de not_active Expired - Lifetime
- 2001-07-06 AU AU2001277659A patent/AU2001277659A1/en not_active Abandoned
- 2001-07-06 AT AT01955500T patent/ATE296827T1/de not_active IP Right Cessation
-
2002
- 2002-12-04 US US10/310,600 patent/US7196083B2/en not_active Expired - Fee Related
Also Published As
Publication number | Publication date |
---|---|
US20020035251A1 (en) | 2002-03-21 |
CA2414885A1 (en) | 2002-01-10 |
US20030144294A1 (en) | 2003-07-31 |
WO2002002562A3 (en) | 2002-05-02 |
EP1296985A2 (de) | 2003-04-02 |
AU2001277659A1 (en) | 2002-01-14 |
ATE296827T1 (de) | 2005-06-15 |
WO2002002562A2 (en) | 2002-01-10 |
DE60111228T2 (de) | 2006-03-16 |
US7196083B2 (en) | 2007-03-27 |
US6514972B2 (en) | 2003-02-04 |
EP1296985B1 (de) | 2005-06-01 |
ES2243527T3 (es) | 2005-12-01 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
ATE296827T1 (de) | Heteropolycyclische inhibitoren | |
DK1223980T3 (da) | Anvendelse af CSF-1-inhibitorer | |
CY1108738T1 (el) | Θεραπευτικοι παραγοντες χρησιμοι για την αγωγη του πονου | |
ATE377004T1 (de) | Proteinkinaseinhibitoren | |
DE60331187D1 (de) | Kinaseinhibitoren | |
DOP2001000151A (es) | Derivados de imidazopirimidina y derivados de triazolopimidina. | |
DE60335359D1 (de) | Phthalazinonderivate | |
EA200300906A1 (ru) | Новые спиротрициклические производные и их применение в качестве ингибиторов фосфодиэстеразы-7 | |
BG106585A (en) | Kinase inhibitors as therapeutic agents | |
CY1107634T1 (el) | Φαρμακευτικη συνθεση | |
EA200200769A1 (ru) | Ингибиторы гиразы и их применение | |
HRP20090159T1 (en) | Use of glucosidase inhibitors for therapy of mucovisidosis | |
CY1111396T1 (el) | Ρινικη χορηγηση μετοκλοπραμιδης για την αγωγη της γαστροπαρεσης | |
SE0104248D0 (sv) | Method of treatment | |
EA200101077A1 (ru) | Композиция для профилактики или лечения слабоумия, включающая производное гидроксикоричной кислоты или экстракт растения рода angelicae, содержащий его | |
SE0301232D0 (sv) | Novel use | |
DK1458393T3 (da) | Substituerede diketopiperaziner som oxytocinantagonister | |
GB9903403D0 (en) | Substituted stilbene compounds with vascular damaging activity | |
MY143245A (en) | 4- 2-(cycloalkylamino)pyrimidin-4-yl-(phenyl)-imidazolin-2-one derivatives as p38 map-kinase inhibitors for the treatment of inflammatory diseases | |
MY139228A (en) | Imidazolinylmethyl aralkylsulfonamides | |
SE0004827D0 (sv) | Therapeutic compounds | |
MXPA03000337A (es) | Inhibidores de trombina que comprenden un grupo aminoisoquinolina. | |
MXPA05003909A (es) | Compuestos de benzopiranona, composiciones de los mismos, y metodos para el tratamiento o prevencion del cancer. | |
RS50449B (sr) | Supstituisani bisindolilmaleimidi za inhibiciju proliferacije ćelija | |
DE60108873D1 (de) | Nicht-antibakterielle tetrazykline als anti-pilz medikamente |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
8364 | No opposition during term of opposition | ||
8339 | Ceased/non-payment of the annual fee |