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DE60104340D1 - Verfahren zur Herstellung von wirkstofbeladenen Polymer-Micellen Zusammensetzung - Google Patents

Verfahren zur Herstellung von wirkstofbeladenen Polymer-Micellen Zusammensetzung

Info

Publication number
DE60104340D1
DE60104340D1 DE60104340T DE60104340T DE60104340D1 DE 60104340 D1 DE60104340 D1 DE 60104340D1 DE 60104340 T DE60104340 T DE 60104340T DE 60104340 T DE60104340 T DE 60104340T DE 60104340 D1 DE60104340 D1 DE 60104340D1
Authority
DE
Germany
Prior art keywords
drug
polymeric micelle
preparation
production process
water
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60104340T
Other languages
English (en)
Other versions
DE60104340T2 (de
Inventor
Masayuki Yokoyama
Eiichi Honzawa
Yasuaki Ogawa
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
NanoCarrier Co Ltd
Original Assignee
NanoCarrier Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by NanoCarrier Co Ltd filed Critical NanoCarrier Co Ltd
Publication of DE60104340D1 publication Critical patent/DE60104340D1/de
Application granted granted Critical
Publication of DE60104340T2 publication Critical patent/DE60104340T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/127—Synthetic bilayered vehicles, e.g. liposomes or liposomes with cholesterol as the only non-phosphatidyl surfactant
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
    • A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Dispersion Chemistry (AREA)
  • Epidemiology (AREA)
  • Communicable Diseases (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Oncology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DE60104340T 2000-02-09 2001-02-07 Verfahren zur Herstellung von wirkstoffbeladenen Polymer-Mizellen-Zusammen- setzung Expired - Lifetime DE60104340T2 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2000032156A JP3523821B2 (ja) 2000-02-09 2000-02-09 薬物が封入されたポリマーミセルの製造方法および該ポリマーミセル組成物
JP2000032156 2000-02-09

Publications (2)

Publication Number Publication Date
DE60104340D1 true DE60104340D1 (de) 2004-08-26
DE60104340T2 DE60104340T2 (de) 2004-12-02

Family

ID=18556810

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60104340T Expired - Lifetime DE60104340T2 (de) 2000-02-09 2001-02-07 Verfahren zur Herstellung von wirkstoffbeladenen Polymer-Mizellen-Zusammen- setzung

Country Status (9)

Country Link
US (2) US20010014354A1 (de)
EP (1) EP1127570B1 (de)
JP (1) JP3523821B2 (de)
KR (1) KR100797429B1 (de)
CN (1) CN1188112C (de)
AT (1) ATE271380T1 (de)
CA (1) CA2334615C (de)
DE (1) DE60104340T2 (de)
TW (1) TWI235069B (de)

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JP5249016B2 (ja) 2006-03-28 2013-07-31 日本化薬株式会社 タキサン類の高分子結合体
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US8334364B2 (en) 2006-11-06 2012-12-18 Nipon Kayaku Kabushiki Kaisha High-molecular weight derivative of nucleic acid antimetabolite
JP5548365B2 (ja) 2006-11-08 2014-07-16 日本化薬株式会社 核酸系代謝拮抗剤の高分子誘導体
US20080312581A1 (en) * 2007-06-06 2008-12-18 Biovaluation & Analysis, Inc. Peptosomes for Use in Acoustically Mediated Intracellular Drug Delivery in vivo
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EP2201935B1 (de) * 2008-12-26 2020-07-08 Samyang Biopharmaceuticals Corporation Polymere Mizellenzusammensetzung, die ein schlecht lösliches Arzneimittel enthält, und zugehöriges Herstellungsverfahren
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CN104856949A (zh) * 2014-02-25 2015-08-26 苏州雷纳药物研发有限公司 一种多西他赛胶束载药系统及其制备方法
CN104072706A (zh) * 2014-07-08 2014-10-01 成都市绿科华通科技有限公司 多功能聚乳酸衍生物药物载体材料
CN104086722A (zh) * 2014-07-08 2014-10-08 成都市绿科华通科技有限公司 一种生物多孔材料的制备方法
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Also Published As

Publication number Publication date
US7223419B2 (en) 2007-05-29
US20010014354A1 (en) 2001-08-16
JP3523821B2 (ja) 2004-04-26
TWI235069B (en) 2005-07-01
EP1127570A3 (de) 2001-09-12
JP2001226294A (ja) 2001-08-21
CN1307866A (zh) 2001-08-15
CA2334615C (en) 2010-09-07
US20040056372A1 (en) 2004-03-25
EP1127570A2 (de) 2001-08-29
ATE271380T1 (de) 2004-08-15
KR20010078773A (ko) 2001-08-21
DE60104340T2 (de) 2004-12-02
KR100797429B1 (ko) 2008-01-23
CN1188112C (zh) 2005-02-09
CA2334615A1 (en) 2001-08-09
EP1127570B1 (de) 2004-07-21

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