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CY1106980T1 - Παραγωγα ν-(αρυλοσουλφονυλο) βητα-αμινοξεων που φερουν μια ομαδα υποκαταστατου αμινοαιθυλιου, η διαδικασια παρασκευης τους και οι φαρμακευτικες συνθεσεις που τα περιεχουν - Google Patents

Παραγωγα ν-(αρυλοσουλφονυλο) βητα-αμινοξεων που φερουν μια ομαδα υποκαταστατου αμινοαιθυλιου, η διαδικασια παρασκευης τους και οι φαρμακευτικες συνθεσεις που τα περιεχουν

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Publication number
CY1106980T1
CY1106980T1 CY20071101426T CY071101426T CY1106980T1 CY 1106980 T1 CY1106980 T1 CY 1106980T1 CY 20071101426 T CY20071101426 T CY 20071101426T CY 071101426 T CY071101426 T CY 071101426T CY 1106980 T1 CY1106980 T1 CY 1106980T1
Authority
CY
Cyprus
Prior art keywords
arylosulphonylo
aminoythylate
aminoxy
producers
substitute
Prior art date
Application number
CY20071101426T
Other languages
English (en)
Inventor
Bernard Ferrari
Jean Gougat
Yvette Muneaux
Pierre Perreaut
Lionel Sarran
Original Assignee
Sanofi-Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi-Aventis filed Critical Sanofi-Aventis
Publication of CY1106980T1 publication Critical patent/CY1106980T1/el

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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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Abstract

Η εφεύρεση αφορά τις ενώσεις του τύπου (Ι). Οι ενώσεις αυτές παρουσιάσουν μια σχέση για τους υποδοχείς της βραδυκινίνης με μια επιλεκτικότητα για τους υποδοχείς Β1, μπορούν να χρησιμοποιηθούν για την προετοιμασία των φαρμάκων που προορίζονται για τη θεραπεία ή την πρόληψη παθολογιών φλεγμονής και των φλεγμονωδών ασθενειών βαριάς ή χρόνιας μορφής.
CY20071101426T 2001-03-28 2007-11-07 Παραγωγα ν-(αρυλοσουλφονυλο) βητα-αμινοξεων που φερουν μια ομαδα υποκαταστατου αμινοαιθυλιου, η διαδικασια παρασκευης τους και οι φαρμακευτικες συνθεσεις που τα περιεχουν CY1106980T1 (el)

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FR0104315A FR2822827B1 (fr) 2001-03-28 2001-03-28 Nouveaux derives de n-(arylsulfonyl) beta-aminoacides comportant un groupe aminomethyle substitue, leur procede de preparation et les compositions pharmaceutiques en contenant
EP02724383A EP1373233B1 (fr) 2001-03-28 2002-03-27 Derives de n-(arylsulfonyl)beta-aminoacides comportant un groupe aminoethyle substitue, leur procede de preparation et les compositions pharmaceutiques en contenant

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CY1106980T1 true CY1106980T1 (el) 2012-09-26

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IL192233A (en) 2012-07-31
BG108201A (bg) 2004-09-30
US7157454B2 (en) 2007-01-02
CZ301337B6 (cs) 2010-01-20
MA26995A1 (fr) 2004-12-20
EA006430B1 (ru) 2005-12-29
BR0208489A (pt) 2004-03-30
ES2291464T3 (es) 2008-03-01
HRP20030748A2 (en) 2004-12-31
HUP0401538A3 (en) 2008-05-28
IS2582B (is) 2010-02-15
DE60222248D1 (de) 2007-10-18
IL192233A0 (en) 2008-12-29
IS6906A (is) 2003-08-07

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