CS331491A3 - Cyclopeptides, process of their preparation and pharmaceuticals based thereon - Google Patents

Cyclopeptides, process of their preparation and pharmaceuticals based thereon

Info

Publication number: CS331491A3
Authority: CS; Czechoslovakia
Prior art keywords: cyclopeptides; preparation; pharmaceuticals based; pharmaceuticals
Prior art date: 1990-11-02

Application number

CS913314A

Other languages

Czech (cs)

Inventor

Gunter Dr Holzemann

Alfred Dr Jonczyk

Jurgen Harting

Hartmut Greiner

Original Assignee

Merck Patent Gmbh

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1990-11-02

Filing date

1991-11-01

Publication date

1992-05-13

1991-11-01 Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh

1992-05-13 Publication of CS331491A3 publication Critical patent/CS331491A3/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/50—Cyclic peptides containing at least one abnormal peptide link
- C07K7/52—Cyclic peptides containing at least one abnormal peptide link with only normal peptide links in the ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/22—Tachykinins, e.g. Eledoisins, Substance P; Related peptides
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Medicinal Chemistry (AREA)
General Chemical & Material Sciences (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pain & Pain Management (AREA)
Molecular Biology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Genetics & Genomics (AREA)
Biophysics (AREA)
Biochemistry (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Rheumatology (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Pulmonology (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Peptides Or Proteins (AREA)

CS913314A 1990-11-02 1991-11-01 Cyclopeptides, process of their preparation and pharmaceuticals based thereon CS331491A3 (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE4034829A DE4034829A1 (en)	1990-11-02	1990-11-02	CYCLOPEPTIDE

Publications (1)

Publication Number	Publication Date
CS331491A3 true CS331491A3 (en)	1992-05-13

Family

ID=6417499

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
CS913314A CS331491A3 (en)	1990-11-02	1991-11-01	Cyclopeptides, process of their preparation and pharmaceuticals based thereon

Country Status (11)

Country	Link
EP (1)	EP0484719A3 (en)
JP (1)	JPH04300895A (en)
KR (1)	KR920009846A (en)
AU (1)	AU8676291A (en)
CA (1)	CA2054667A1 (en)
CS (1)	CS331491A3 (en)
DE (1)	DE4034829A1 (en)
HU (1)	HUT61582A (en)
IE (1)	IE913831A1 (en)
PT (1)	PT99384A (en)
ZA (1)	ZA918717B (en)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP0916346A3 (en)	1991-09-20	2000-12-06	Glaxo Group Limited	NK-1 receptor antagonists and 5HT3 receptor antagonists for the treatment of emesis
GB9702377D0 (en) *	1996-02-23	1997-03-26	Zeneca Ltd	Peptide derivatives
CA2252417A1 (en)	1996-06-07	1997-12-11	Zeneca Limited	Peptide derivatives
GB9621836D0 (en)	1996-10-19	1996-12-11	Zeneca Ltd	Peptide compounds
GB9624562D0 (en)	1996-11-27	1997-01-15	Zeneca Ltd	Peptide derivatives
KR100408624B1 (en) *	2000-10-06	2003-12-06	엘지전선 주식회사	Poly vinyl chloride insulator composition for wire and cable
JP2010516731A (en)	2007-01-24	2010-05-20	グラクソグループリミテッド	Pharmaceutical composition comprising 2-methoxy-5- (5-trifluoromethyl-tetrazol-1-yl) -benzyl]-(2S-phenyl-piperidin-3S-yl) -amine
UA105182C2 (en)	2008-07-03	2014-04-25	Ньюрексон, Інк.	Benzoxazines, benzothiazines, and related compounds having nos inhibitory activity
US9446029B2 (en)	2010-07-27	2016-09-20	Colorado State University Research Foundation	Use of NK-1 receptor antagonists in management of visceral pain
EP2766347B1 (en)	2011-10-14	2016-05-04	Bristol-Myers Squibb Company	Substituted tetrahydroisoquinoline compounds as factor xia inhibitors
KR101937514B1 (en)	2011-10-14	2019-01-10	브리스톨-마이어스 스큅 컴퍼니	Substituted tetrahydroisoquinoline compounds as factor xia inhibitors
ES2572908T3 (en)	2011-10-14	2016-06-03	Bristol-Myers Squibb Company	Tetrahydroisoquinoline compounds substituted as factor XIa inhibitors
WO2014059202A1 (en)	2012-10-12	2014-04-17	Bristol-Myers Squibb Company	Guanidine substituted tetrahydroisoquinoline compounds as factor xia inhibitors
EP2906551B1 (en)	2012-10-12	2018-02-28	Bristol-Myers Squibb Company	Crystalline forms of a factor xia inhibitor
WO2014059214A1 (en)	2012-10-12	2014-04-17	Bristol-Myers Squibb Company	Guanidine and amine substituted tetrahydroisoquinoline compounds as factor xia inhibitors
JP6479763B2 (en)	2013-03-25	2019-03-06	ブリストル−マイヤーズスクイブカンパニーＢｒｉｓｔｏｌ−ＭｙｅｒｓＳｑｕｉｂｂＣｏｍｐａｎｙ	Substituted azole containing tetrahydroisoquinolines as factor XIA inhibitors
US20170002006A1 (en)	2014-01-31	2017-01-05	Bristol-Myers Squibb Company	Macrocycles with hetrocyclic p2' groups as factor xia inhibitors
NO2760821T3 (en)	2014-01-31	2018-03-10
ES2714283T3 (en)	2014-09-04	2019-05-28	Bristol Myers Squibb Co	Macrocycles of diamide that are inhibitors of FXIa
US9453018B2 (en)	2014-10-01	2016-09-27	Bristol-Myers Squibb Company	Pyrimidinones as factor XIa inhibitors

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB8807246D0 (en) *	1988-03-25	1988-04-27	Merck Sharp & Dohme	Therapeutic agents
ZA906188B (en) *	1989-08-10	1991-06-26	Merrell Dow Pharma	Cyclic neurokinin a antagonists

1990
- 1990-11-02 DE DE4034829A patent/DE4034829A1/en not_active Withdrawn
1991
- 1991-10-19 EP EP19910117864 patent/EP0484719A3/en not_active Withdrawn
- 1991-10-25 AU AU86762/91A patent/AU8676291A/en not_active Abandoned
- 1991-10-29 KR KR1019910019015A patent/KR920009846A/en not_active Application Discontinuation
- 1991-10-30 PT PT99384A patent/PT99384A/en not_active Application Discontinuation
- 1991-10-31 CA CA002054667A patent/CA2054667A1/en not_active Abandoned
- 1991-11-01 JP JP3349287A patent/JPH04300895A/en active Pending
- 1991-11-01 IE IE383191A patent/IE913831A1/en not_active Application Discontinuation
- 1991-11-01 CS CS913314A patent/CS331491A3/en unknown
- 1991-11-01 HU HU913450A patent/HUT61582A/en unknown
- 1991-11-01 ZA ZA918717A patent/ZA918717B/en unknown

Also Published As

Publication number	Publication date
HUT61582A (en)	1993-01-28
AU8676291A (en)	1992-05-07
JPH04300895A (en)	1992-10-23
EP0484719A3 (en)	1993-05-19
HU913450D0 (en)	1992-01-28
DE4034829A1 (en)	1992-05-07
IE913831A1 (en)	1992-05-22
EP0484719A2 (en)	1992-05-13
PT99384A (en)	1992-09-30
CA2054667A1 (en)	1992-05-03
ZA918717B (en)	1992-08-26
KR920009846A (en)	1992-06-25

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