CN102119143A - Amide derivative, pest control agent containing the amide derivative and use of the pest control agent - Google Patents

Abstract

Disclosed is an amide derivative having excellent pest control effect, which is represented by general formula (1). In general formula (1), A represents a carbon atom, a nitrogen atom or the like; K represents a non-metal atomic group necessary for forming a cyclic linking group derived from benzene or a heterocyclic ring; X represents a halogen atom or the like; n represents an integer of 0-4; R1 and R2 each represents a hydrogen atom, an alkyl group or the like; T represents -C(=G1)-Q1 or -C(=G1)-G2Q2; G1-G3 each represents an oxygen atom or the like; Q1 and Q2 each represents a hydrogen atom, an alkyl group, an aryl group or the like; Y1 and Y5 each represents a halogen atom or the like; Y2 and Y4 each represents a hydrogen atom or the like; and Y3 represents a C2-C5 haloalkyl group.

Description

Amide derivatives, the noxious organism control agent that contains this amide derivatives and using method thereof

Technical field

The present invention relates to the amide derivatives that contains in noxious organism control agent and this noxious organism control agent and the using method of this amide derivatives.

Background technology

No. 2005/21488 specification sheets disclosed in the world, international disclosing in No. 2005/73165 specification sheets, No. 2006/137376 specification sheets of international publication, No. 2006/137395 specification sheets of international publication discloses multiple amide derivatives.

Summary of the invention

In the crop production of agricultural and gardening etc., the infringement that causes owing to insect etc. still significantly, produce the reasons such as insect that existing medicine had resistance, people expect development of new agricultural or horticultural use noxious organism control agent.

Problem of the present invention is to be provided at that available shows the amide derivatives of insecticidal effect and contains this amide derivatives as the noxious organism control agent of effective constituent and the method for control of harmful organism insect in the agricultural gardening field of wider range.

For the development of new noxious organism control agent, the inventor etc. found that through concentrating on studies, the aromatic carboxylic acid amide derivatives of general formula of the present invention (1) expression is the novel cpd that document is not put down in writing, be noxious organism control agent, particularly the agricultural or horticultural use noxious organism control agent that shows superior efficacy, thereby finished the present invention.

In addition, found to prepare the novel preparation method and the useful intermediates of compound of the present invention, thereby finished the present invention.

That is, the present invention is as described below.

＜1〉amide derivatives of following general formula (1) expression.

{ in the general formula (1), A represents carbon atom, Sauerstoffatom, nitrogen-atoms, oxidized nitrogen-atoms or sulphur atom.Necessary non-metallic atom group when K is illustrated in 2 carbon atoms with A and A bonding and forms cyclic linker group, described cyclic linker group is from benzene, pyridine, N-pyridine oxide, pyrimidine, pyrazine, pyridazine, triazine, pyrroles, pyrazoles, imidazoles, oxazole, isoxazole, thiazole, isothiazole, furans, thiophene, oxadiazole, thiadiazoles or triazole.

X represents hydrogen atom; halogen atom; the C1-C6 alkyl; the C1-C6 haloalkyl; the C3-C9 cycloalkyl; the C3-C9 halogenated cycloalkyl; the C2-C6 alkenyl; the C2-C6 halogenated alkenyl; the C2-C6 alkynyl; C2-C6 halo alkynyl; the C1-C6 alkoxyl group; the C1-C6 halogenated alkoxy; the C2-C6 alkenyl oxy; the C2-C6 halogenated alkenyl oxy; C2-C6 alkynyloxy base; C2-C6 halo alkynyloxy base; the C3-C9 cycloalkyloxy; C3-C9 halo cycloalkyloxy; C1-C6 alkyl sulfenyl; C1-C6 haloalkyl sulfenyl; the C1-C6 alkyl sulphinyl; C1-C6 haloalkyl sulfinyl; the C1-C6 alkyl sulphonyl; the C1-C6 halogenated alkyl sulfonyl; C1-C6 alkyl sulphonyl oxygen base; C1-C6 halogenated alkyl sulfonyl oxygen base; the C2-C7 alkyl-carbonyl; the C2-C7 halogenated alkyl carbonyl; the C3-C7 alkenyl carbonyl; C3-C7 halogenated alkenyl carbonyl; C3-C7 alkynyl carbonyl; C3-C7 halo alkynyl carbonyl; the C4-C10 naphthene base carbonyl; C4-C10 halogenated cycloalkyl carbonyl; C2-C7 alkyl-carbonyl oxygen base; C2-C7 halogenated alkyl carbonyl oxygen base; aryl carbonyl oxygen base; the C2-C7 alkoxy carbonyl; the C2-C7 halo alkoxy carbonyl; C3-C7 alkenyl oxy carbonyl; C3-C7 halogenated alkenyl oxy carbonyl; C3-C7 alkynyloxy base carbonyl; C3-C7 halo alkynyloxy base carbonyl; C4-C10 cycloalkyl oxy carbonyl; C4-C10 halogenated cycloalkyl oxygen base carbonyl; the C2-C7 alkyl-carbonyl-amino; C2-C7 halogenated alkyl carbonyl amino; the C2-C7 alkoxycarbonyl amino; C2-C7 halo alkoxy carbonyl amino; the C2-C7 alkoxy-carbonyl oxy; C2-C7 halo alkoxy carbonyl oxygen base; aryl-amino-carbonyl; amino; formamyl; cyano group; hydroxyl; Pentafluorosulfanyl (pentafluorosulfanyl group); the C1-C6 alkylamino; C1-C6 haloalkyl amino; the C2-C6 alkenyl amino; C2-C6 halogenated alkenyl amino; C2-C6 alkynyl amino; C2-C6 halo alkynyl amino; the C3-C9 cycloalkyl amino; C3-C9 halogenated cycloalkyl amino; the C2-C7 alkyl amino-carbonyl; C2-C7 haloalkyl aminocarboxyl; C3-C7 alkenyl amino carbonyl; C3-C7 halogenated alkenyl aminocarboxyl; C3-C7 alkynyl aminocarboxyl; C3-C7 halo alkynyl aminocarboxyl; C4-C10 cycloalkyl amino carbonyl; C4-C10 halogenated cycloalkyl aminocarboxyl; phenyl; or heterocyclic radical; when having a plurality of X, each X can be same to each other or different to each other.

N represents 0～4 integer.

T represents-C (=G ₁)-Q ₁, or-C (=G ₁)-G ₂Q ₂

G ₁And G ₂Represent Sauerstoffatom or sulphur atom respectively independently.

Q ₁And Q ₂Represent hydrogen atom, C1-C6 alkyl, C1-C6 haloalkyl, C2-C6 alkenyl, C2-C6 halogenated alkenyl, C2-C6 alkynyl, C2-C6 halo alkynyl, C3-C9 cycloalkyl, C3-C9 halogenated cycloalkyl, benzyl, can have substituent phenyl, naphthyl, maybe can have substituent heterocyclic radical.

Y ₁And Y ₅Represent halogen atom, C1-C6 halogenated alkoxy or C1-C3 haloalkyl respectively independently, Y ₂, Y ₄Represent hydrogen atom, halogen atom or C1-C4 alkyl respectively independently, Y ₃Expression C2-C5 haloalkyl.

Need to prove Q ₁And Q ₂In; the substituting group that can have substituent phenyl and can have a substituent heterocyclic radical represents to be selected from the substituting group more than 1 in the following radicals; described group is: halogen atom; the C1-C6 alkyl; the C1-C6 haloalkyl; the C3-C9 cycloalkyl; the C3-C9 halogenated cycloalkyl; the C2-C6 alkenyl; the C2-C6 halogenated alkenyl; the C2-C6 alkynyl; C2-C6 halo alkynyl; the C1-C6 alkoxyl group; the C1-C6 halogenated alkoxy; the C2-C6 alkenyl oxy; the C2-C6 halogenated alkenyl oxy; C2-C6 alkynyloxy base; C2-C6 halo alkynyloxy base; the C3-C9 cycloalkyloxy; C3-C9 halo cycloalkyloxy; C1-C6 alkyl sulfenyl; C1-C6 haloalkyl sulfenyl; the C1-C6 alkyl sulphinyl; C1-C6 haloalkyl sulfinyl; the C1-C6 alkyl sulphonyl; the C1-C6 halogenated alkyl sulfonyl; the C2-C7 alkyl-carbonyl; the C2-C7 halogenated alkyl carbonyl; the C3-C7 alkenyl carbonyl; C3-C7 halogenated alkenyl carbonyl; C3-C7 alkynyl carbonyl; C3-C7 halo alkynyl carbonyl; the C4-C10 naphthene base carbonyl; C4-C10 halogenated cycloalkyl carbonyl; C2-C7 alkyl-carbonyl oxygen base; C2-C7 halogenated alkyl carbonyl oxygen base; C1-C6 alkyl sulphonyl oxygen base; C1-C6 halogenated alkyl sulfonyl oxygen base; the C2-C7 alkoxy carbonyl; the C2-C7 halo alkoxy carbonyl; C3-C7 alkenyl oxy carbonyl; C3-C7 halogenated alkenyl oxy carbonyl; C3-C7 alkynyloxy base carbonyl; C3-C7 halo alkynyloxy base carbonyl; C4-C10 cycloalkyl oxy carbonyl; C4-C10 halogenated cycloalkyl oxygen base carbonyl; the C2-C7 alkyl-carbonyl-amino; C2-C7 halogenated alkyl carbonyl amino; the C2-C7 alkoxycarbonyl amino; C2-C7 halo alkoxy carbonyl amino; the C1-C6 alkylamino; C1-C6 haloalkyl amino; the C2-C6 alkenyl amino; C2-C6 halogenated alkenyl amino; C2-C6 alkynyl amino; C2-C6 halo alkynyl amino; the C3-C9 cycloalkyl amino; C3-C9 halogenated cycloalkyl amino; the C2-C7 alkyl amino-carbonyl; C2-C7 haloalkyl aminocarboxyl; C3-C7 alkenyl amino carbonyl; C3-C7 halogenated alkenyl aminocarboxyl; C3-C7 alkynyl aminocarboxyl; C3-C7 halo alkynyl aminocarboxyl; C4-C10 cycloalkyl amino carbonyl; C4-C10 halogenated cycloalkyl aminocarboxyl; amino; formamyl; cyano group; nitro; hydroxyl; Pentafluorosulfanyl; can have substituent phenyl; and can have substituent heterocyclic radical; when having 2 above substituting groups, each substituting group can be the same or different.

And then, X, Q ₁, and Q ₂In heterocyclic radical represent pyridyl, N-pyridine oxide base, pyrimidyl, pyrazinyl, pyridazinyl, furyl, thienyl, oxazolyl, isoxazolyl, oxadiazole base, thiazolyl, isothiazolyl, thiadiazolyl group, pyrryl, imidazolyl, triazolyl, pyrazolyl or tetrazyl.

G ₃Expression Sauerstoffatom or sulphur atom.

R ₁And R ₂Represent hydrogen atom respectively independently; Sauerstoffatom; halogen atom; hydroxyl; nitro; nitroso-group; trimethyl silyl; t-butyldimethylsilyl; cyano group; amino; can have substituent C1-C6 alkyl; can have substituent C1-C6 haloalkyl; the C2-C7 alkyl-carbonyl; the C2-C7 halogenated alkyl carbonyl; can have substituent C2-C6 alkenyl; can have substituent C2-C6 halogenated alkenyl; can have substituent C2-C6 alkynyl; can have substituent C2-C6 halo alkynyl; the C2-C7 alkoxy carbonyl; the C2-C7 halo alkoxy carbonyl; C3-C7 alkenyl oxy carbonyl; C3-C7 halogenated alkenyl oxy carbonyl; C3-C7 alkynyloxy base carbonyl; C3-C7 halo alkynyloxy base carbonyl; phenyloxycarbonyl; the C2-C7 alkyl amino-carbonyl; C2-C7 haloalkyl aminocarboxyl; C2-C7 alkyl-carbonyl oxygen base; C2-C7 halogenated alkyl carbonyl oxygen base; benzoyl; the C1-C6 alkoxyl group; the C1-C6 halogenated alkoxy; C1-C6 alkyl sulfenyl; C1-C6 haloalkyl sulfenyl; the C1-C6 alkyl sulphinyl; C1-C6 haloalkyl sulfinyl; the C1-C6 alkyl sulphonyl; the C1-C6 halogenated alkyl sulfonyl; benzenesulfonyl; the benzyl alkylsulfonyl; benzyl; or-C (=O) C (=O) R ₇(in the formula, R ₇Expression C1-C6 alkyl, C1-C6 haloalkyl, C1-C6 alkoxyl group or C1-C6 halogenated alkoxy.)。}

But the amide derivatives that does not comprise above-mentioned general formula (1) expression is any one the situation in following (A)～(I).

(A) in the above-mentioned general formula (1), K necessary non-metallic atom group when forming the cyclic linker group from pyridine at 2 carbon atoms, Y with A and A bonding ₁Be halogen atom, Y ₅Be the C1-C6 halogenated alkoxy, T is-C (=G ₁)-Q ₁

(B) in the above-mentioned general formula (1), K is necessary non-metallic atom group when 2 carbon atoms with A and A bonding form cyclic linker group, described cyclic linker group is from pyrroles, pyrazoles, imidazoles, oxazole, isoxazole, thiazole, isothiazole, furans, thiophene, oxadiazole, thiadiazoles or triazole, Y ₁And Y ₅Be halogen atom independently respectively, T is-C (=G ₁)-G ₂Q ₂

(C) in the above-mentioned general formula (1), K is necessary non-metallic atom group when 2 carbon atoms with A and A bonding form cyclic linker group, described cyclic linker group is from pyrroles, pyrazoles, imidazoles, oxazole, isoxazole, thiazole, isothiazole, furans, thiophene, oxadiazole, thiadiazoles or triazole, and T is-C (=G ₁)-Q ₁, Y ₁Be halogen atom, Y ₅Be halogen atom or halogenated alkoxy.

(D) amide compound of following general formula (2) expression.

In the general formula (2), Y ₂～Y ₄, Q ₁, G ₁, G ₃, R ₁, and R ₂With the Y in the general formula (1) ₂～Y ₄, Q ₁, G ₁, G ₃, R ₁, and R ₂The difference synonym.Y ₁Be halogen atom, Y ₅Be the C1-C2 halogenated alkoxy.}

(E) in the above-mentioned general formula (2), Y ₁And Y ₅Be halogen atom independently respectively, X is hydrogen atom, Y ₃Be the C2-C3 haloalkyl.

(F) amide derivatives of following general formula (3) expression.

In the general formula (3), Y ₁And Y ₅Be halogen atom independently respectively, X ₁, X ₃Be hydrogen atom or fluorine atom, Q ₁With the Q in the general formula (1) ₁Synonym, R ₁Be hydrogen atom or methyl, Y ₃Be the C3-C4 perfluoroalkyl.}

(G) amide derivatives of following general formula (4) expression.

In the general formula (4), X ₁Be fluorine atom, X ₂, X ₃And X ₄Be hydrogen atom, Y ₁And Y ₅Differ from one another, be bromine atoms or trifluoromethoxy, Y ₂And Y ₄Be hydrogen atom, Y ₃Be seven fluorine sec.-propyls, Q ₁Be phenyl or 2-chloropyridine-3-base, R ₁And R ₂Differ from one another, be hydrogen atom or methyl.

Perhaps, X ₁Be fluorine atom, X ₂, X ₃And X ₄Be hydrogen atom, Y ₁And Y ₅Be bromine atoms, Y ₂And Y ₄Be hydrogen atom, Y ₃Be pentafluoroethyl group, Q ₁Be 2-fluorophenyl, R ₁And R ₂Be hydrogen atom or methyl independently respectively.}

(H) amide derivatives of following general formula (5) expression.

In the general formula (5), Y ₁And Y ₅Be halogen atom independently respectively, X ₁Be hydrogen atom or fluorine atom, Q ₂Be 2,2,2-three chloroethyls and 3,3,3-three fluoro-n-propyl group, Y ₃Be the C2-C4 haloalkyl.}

(I) amide derivatives of following general formula (6) expression.

In the general formula (6), Y ₁And Y ₅Be halogen atom independently respectively, Q ₂With the Q in the general formula (1) ₂Synonym, R ₁Be hydrogen atom or methyl, Y ₃Be the C3-C4 haloalkyl.}

＜2〉as above-mentioned＜1〉described amide compound, represent with following general formula (7).

{ in the general formula (7), n is 4, X, Y ₁～Y ₅, Q ₁, G ₁, G ₃, R ₁, and R ₂With X, the Y in the general formula (1) ₁～Y ₅, Q ₁, G ₁, G ₃, R ₁, and R ₂The difference synonym.}

＜3〉as above-mentioned＜2〉described amide derivatives, represent with following general formula (8).

In the general formula (8), Q ₁Expression can have substituent phenyl maybe can have substituent pyridyl.X ₁, X ₂, X ₃And X ₄Represent hydrogen atom or fluorine atom respectively independently.R ₁And R ₂Represent hydrogen atom or C1-C3 alkyl respectively independently.Y ₁And Y ₅Represent halogen atom, C1-C3 halogenated alkoxy or C1-C3 haloalkyl respectively independently, Y ₂And Y ₄Represent hydrogen atom, halogen atom or C1-C4 alkyl, Y respectively independently ₃Expression C3-C4 haloalkyl.

Wherein, Y ₁And Y ₅When being halogen atom simultaneously, X ₁And X ₂In at least-side be fluorine atom.In addition, Y ₁Or Y ₅During for the C1-C3 halogenated alkoxy, X ₂Be fluorine atom.}

＜4〉as above-mentioned＜3〉described amide derivatives, in the above-mentioned general formula (8), Y ₃Be the C3-C4 perfluoroalkyl.

＜5〉as above-mentioned＜4〉described amide derivatives, in the above-mentioned general formula (8), Y ₁And Y ₅Be chlorine atom, bromine atoms, iodine atom, trifluoromethoxy, trifluoromethyl or pentafluoroethyl group independently respectively, Y ₂, Y ₄Be hydrogen atom.

＜6〉as above-mentioned＜5〉described amide derivatives, in the above-mentioned general formula (8), X ₁And X ₂Be hydrogen atom or fluorine atom independently respectively, X ₃And X ₄Be hydrogen atom.

＜7〉as above-mentioned＜6〉described amide derivatives, in the above-mentioned general formula (8), R ₁And R ₂Be hydrogen atom or methyl independently respectively.

＜8〉as above-mentioned＜7〉described amide derivatives, in the above-mentioned general formula (8), Q ₁For having substituent phenyl or the pyridyl that is selected from halogen atom, C1 haloalkyl, nitro and the cyano group.

＜9〉as above-mentioned＜8〉described amide derivatives, in the above-mentioned general formula (8), Q ₁In substituent quantity be 1 or 2.

＜10〉as above-mentioned＜9〉described amide derivatives, in the above-mentioned general formula (8), Q ₁Be phenyl, the 2-fluorophenyl, the 3-fluorophenyl, the 4-fluorophenyl, the 2-chloro-phenyl-, the 3-chloro-phenyl-, the 4-chloro-phenyl-, the 2-bromophenyl, the 3-bromophenyl, the 4-bromophenyl, the 2-iodophenyl, the 3-iodophenyl, the 4-iodophenyl, (2-trifluoromethyl) phenyl, (3-trifluoromethyl) phenyl, (4-trifluoromethyl) phenyl, the 2-nitrophenyl, the 3-nitrophenyl, the 4-nitrophenyl, the 2-cyano-phenyl, the 3-cyano-phenyl, the 4-cyano-phenyl, 2, the 6-difluorophenyl, 3, the 4-dichlorophenyl, 2, the 4-dichlorophenyl, 2-chloro-4-fluorophenyl, 2-chloro-4, the 5-difluorophenyl, 4-bromo-2-chloro-phenyl-, 2-bromo-4-chloro-phenyl-, 2-bromo-4-fluorophenyl, 2-chloro-4-nitrophenyl, 3,5-dicyano phenyl, 4-cyano group-2-fluorophenyl, 2-chloro-4-cyano-phenyl, pyridin-3-yl, 2-fluorine pyridin-3-yl, 2-chloropyridine-3-base, 2-bromopyridine-3-base, 2-iodine pyridine-3-base, 2-(trifluoromethyl) pyridin-3-yl, 2-nitropyridine-3-base, 2-cyanopyridine-3-base, 6-fluorine pyridin-3-yl, 6-chloropyridine-3-base, 6-bromopyridine-3-base, 6-iodine pyridine-3-base, 6-(trifluoromethyl) pyridin-3-yl, 6-nitropyridine-3-base, 6-cyanopyridine-3-base, 5-fluorine pyridin-3-yl, 5-chloropyridine-3-base, 5-bromopyridine-3-base, 5-iodine pyridine-3-base, 5-(trifluoromethyl) pyridin-3-yl, 5-nitropyridine-3-base, 5-cyanopyridine-3-base, 4-fluorine pyridin-3-yl, 4-chloropyridine-3-base, 4-bromopyridine-3-base, 4-iodine pyridine-3-base, 4-(trifluoromethyl) pyridin-3-yl, 4-nitropyridine-3-base, 4-cyanopyridine-3-base, 2,6-dichloropyridine-3-base, N-pyridine oxide-3-base, pyridin-4-yl, 2-chloropyridine-4-base, 3-bromopyridine-4-base, 3,5-dichloropyridine-4-base, 3-(trifluoromethyl) pyridin-4-yl, 2,6-dicyanopyridine-4-base, N-pyridine oxide-4-base, pyridine-2-base, 3-chloropyridine-2-base, 4-bromopyridine-2-base, 5-iodine pyridine-2-base, 6-chloropyridine-2-base or 4-cyanopyridine-2-base.

＜11〉as above-mentioned＜10〉described amide derivatives; the compound of above-mentioned general formula (8) expression is 3-benzoylamino-N-(2-bromo-6-chloro-4-(perfluoropropane-2-yl) phenyl)-2-fluorobenzamide; (3-(2 for 2-chloro-N-; 6-two bromo-4-(perfluoropropane-2-yl) phenyl amino formyl radical)-and the 2-fluorophenyl) niacinamide; 3-(4-cyano group-N-methyl-benzamide base)-N-(2; 6-two bromo-4-(perfluoropropane-2-yl) phenyl)-the 2-fluorobenzamide; (3-(2 for 2-chloro-N-; 6-two bromo-4-(perfluoropropane-2-yl) phenyl amino formyl radical)-the 2-fluorophenyl)-the N-methylnicotinamide; 3-benzoylamino-N-(2; 6-two iodo-4-(perfluoropropane-2-yl) phenyl)-the 2-fluorobenzamide; 3-benzoylamino-N-(2; 6-two bromo-4-(perfluoropropane-2-yl) phenyl)-the 2-fluorobenzamide; N-(2; 6-two bromo-4-(perfluoropropane-2-yl) phenyl)-2-fluoro-3-(N-methyl-benzamide base) benzamide; (3-(2 for 6-chloro-N-; 6-two bromo-4-(perfluoropropane-2-yl) phenyl amino formyl radical)-the 2-fluorophenyl)-the N-methylnicotinamide; 3-(3-cyano group-N-methyl-benzamide base)-N-(2; 6-two bromo-4-(perfluoropropane-2-yl) phenyl)-the 2-fluorobenzamide; N-(2; 6-two chloro-4-(perfluoropropane-2-yl) phenyl)-2-fluoro-3-(N-methyl-benzamide base) benzamide; 3-(4-cyano group-N-methyl-benzamide base)-N-(2; 6-two chloro-4-(perfluoropropane-2-yl) phenyl)-the 2-fluorobenzamide; (3-(2 for 2-chloro-N-; 6-two chloro-4-(perfluoropropane-2-yl) phenyl amino formyl radical)-the 2-fluorophenyl)-the N-methylnicotinamide; N-(2; 6-two iodo-4-(perfluoropropane-2-yl) phenyl)-2-fluoro-3-(N-methyl-benzamide base) benzamide; 3-(4-cyano group-N-methyl-benzamide base)-N-(2; 6-two iodo-4-(perfluoropropane-2-yl) phenyl)-the 2-fluorobenzamide; 3-benzoylamino-N-(2; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl)-the 2-fluorobenzamide; N-(2; 6-two iodo-4-(perfluoropropane-2-yl) phenyl)-2-fluoro-3-(2-fluorobenzoyl amido) benzamide; N-(2; 6-two iodo-4-(perfluoropropane-2-yl) phenyl)-2-fluoro-3-(4-fluorobenzoyl amido) benzamide; 3-(2; 6-difluorobenzamide base)-N-(2,6-two iodo-4-(perfluoropropane-2-yl) phenyl)-2-fluorobenzamide; N-(2-bromo-6-iodo-4-(perfluoropropane-2-yl) phenyl)-2-fluoro-3-(N-methyl-benzamide base) benzamide; N-(3-(2-bromo-6-iodo-4-(perfluoropropane-2-yl) phenyl amino formyl radical)-2-fluorophenyl)-2-chloro-N-methylnicotinamide;

3-(4-cyano group benzoylamino)-N-(2; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl)-the 2-fluorobenzamide; 3-(3-cyano group benzoylamino)-N-(2; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl)-the 2-fluorobenzamide; N-(2; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl)-2-fluoro-3-(N-methyl-benzamide base) benzamide; 3-(4-cyano group-N-methyl-benzamide base)-N-(2; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl)-the 2-fluorobenzamide; 3-(3-cyano group-N-methyl-benzamide base)-N-(2; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl)-the 2-fluorobenzamide; (3-(2 for 6-chloro-N-; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical)-the 2-fluorophenyl)-the N-methylnicotinamide; 3-benzoylamino-N-(2; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl)-the 2-fluorobenzamide; 3-(3-cyano group benzoylamino)-N-(2; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl)-the 2-fluorobenzamide; 3-(4-cyano group benzoylamino)-N-(2; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl)-the 2-fluorobenzamide; N-(2; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl)-2-fluoro-3-(N-methyl-benzamide base) benzamide; 3-(3-cyano group-N-methyl-benzamide base)-N-(2; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl)-the 2-fluorobenzamide; 3-(4-cyano group-N-methyl-benzamide base)-N-(2; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl)-the 2-fluorobenzamide; 3-benzoylamino-N-(2; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl) benzamide; (3-(2 for 2-chloro-N-; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) niacinamide phenyl); (3-(2 for 6-chloro-N-; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) niacinamide phenyl); (3-(2 for 3-cyano group-N-; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) benzamide phenyl); 3-(4-cyano group benzoylamino)-N-(2; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl) benzamide; (3-(2 for N-; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) phenyl)-the 2-fluorobenzamide; N-(2; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl)-3-(3-fluorobenzoyl amido) benzamide; N-(2,6-two iodo-4-(perfluorinated butane-2-yl) phenyl)-3-(4-fluorobenzoyl amido) benzamide;

(3-(2 for N-; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) phenyl)-2; the 6-difluorobenzamide; (3-(2 for N-; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide; (3-(2 for 2-chloro-N-; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) phenyl)-the N-methylnicotinamide; (3-(2 for 6-chloro-N-; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) phenyl)-the N-methylnicotinamide; (3-(2 for 3-cyano group-N-; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide; (3-(2 for 4-cyano group-N-; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide; (3-(2 for N-; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) phenyl)-2-fluoro-N-methyl-benzamide; (3-(2 for N-; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) phenyl)-3-fluoro-N-methyl-benzamide; (3-(2 for N-; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) phenyl)-4-fluoro-N-methyl-benzamide; (3-(2 for N-; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) phenyl)-2; 6-two fluoro-N-methyl-benzamides; (3-(2 for 2-chloro-N-; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical)-and the 2-fluorophenyl) niacinamide; (3-(2 for 6-chloro-N-; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical)-and the 2-fluorophenyl) niacinamide; N-(2; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl)-2-fluoro-3-(2-fluorobenzoyl amido) benzamide; N-(2; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl)-2-fluoro-3-(3-fluorobenzoyl amido) benzamide; N-(2; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl)-2-fluoro-3-(4-fluorobenzoyl amido) benzamide; 3-(2; 6-difluorobenzamide base)-N-(2; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl)-the 2-fluorobenzamide; 3-benzoylamino-N-(2; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl) benzamide; (3-(2 for 6-chloro-N-; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) niacinamide phenyl); (3-(2 for N-; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) phenyl)-the 2-fluorobenzamide; 2-chloro-N-(3-(2,6-two bromo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) phenyl) niacinamide;

N-(2; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl)-3-(3-fluorobenzoyl amido) benzamide; N-(2; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl)-3-(4-fluorobenzoyl amido) benzamide; (3-(2 for N-; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) phenyl)-2; the 6-difluorobenzamide; (3-(2 for 3-cyano group-N-; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) benzamide phenyl); 3-(4-cyano group benzoylamino)-N-(2; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl) benzamide; (3-(2 for 2-chloro-N-; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical)-the 2-fluorophenyl)-the N-methylnicotinamide; (3-(2 for 6-chloro-N-; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical)-the 2-fluorophenyl)-the N-methylnicotinamide; (3-(2 for N-; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical)-the 2-fluorophenyl)-2-fluoro-N-methyl-benzamide; N-(2; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl)-2-fluoro-3-(3-fluoro-N-methyl-benzamide base) benzamide; N-(2; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl)-2-fluoro-3-(4-fluoro-N-methyl-benzamide base) benzamide; (3-(2 for N-; 6-two iodo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical)-and the 2-fluorophenyl)-2; 6-two fluoro-N-methyl-benzamides; (3-(2 for N-; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide; (3-(2 for 2-chloro-N-; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) phenyl)-the N-methylnicotinamide; (3-(2 for 6-chloro-N-; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) phenyl)-the N-methylnicotinamide; (3-(2 for 3-cyano group-N-; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide; (3-(2 for 4-cyano group-N-; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide; (3-(2 for N-; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) phenyl)-2-fluoro-N-methyl-benzamide; (3-(2 for N-; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) phenyl)-3-fluoro-N-methyl-benzamide; (3-(2 for N-; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) phenyl)-4-fluoro-N-methyl-benzamide; (3-(2 for N-; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical) phenyl)-2,6-two fluoro-N-methyl-benzamides;

(3-(2 for 2-chloro-N-; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical)-and the 2-fluorophenyl) niacinamide; (3-(2 for 6-chloro-N-; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical)-and the 2-fluorophenyl) niacinamide; N-(2; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl)-2-fluoro-3-(2-fluorobenzoyl amido) benzamide; N-(2; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl)-2-fluoro-3-(3-fluorobenzoyl amido) benzamide; N-(2; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl)-2-fluoro-3-(4-fluorobenzoyl amido) benzamide; N-(2; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl)-3-(2; 6-difluorobenzamide base)-the 2-fluorobenzamide; (3-(2 for 2-chloro-N-; 6-two iodo-4-(perfluoropropane-2-yl) phenyl amino formyl radical)-and the 2-fluorophenyl) niacinamide; (3-(2 for 6-chloro-N-; 6-two iodo-4-(perfluoropropane-2-yl) phenyl amino formyl radical)-and the 2-fluorophenyl) niacinamide; 3-(3-cyano group benzoylamino)-N-(2; 6-two iodo-4-(perfluoropropane-2-yl) phenyl)-the 2-fluorobenzamide; 3-(4-cyano group benzoylamino)-N-(2; 6-two iodo-4-(perfluoropropane-2-yl) phenyl)-the 2-fluorobenzamide; N-(2; 6-two iodo-4-(perfluoropropane-2-yl) phenyl)-2-fluoro-3-(3-fluorobenzoyl amido) benzamide; (3-(2 for 2-chloro-N-; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical)-the 2-fluorophenyl)-the N-methylnicotinamide; (3-(2 for N-; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical)-the 2-fluorophenyl)-2-fluoro-N-methyl-benzamide; N-(2; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl)-2-fluoro-3-(3-fluoro-N-methyl-benzamide base) benzamide; N-(2; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl)-2-fluoro-3-(4-fluoro-N-methyl-benzamide base) benzamide; (3-(2 for N-; 6-two bromo-4-(perfluorinated butane-2-yl) phenyl amino formyl radical)-and the 2-fluorophenyl)-2; 6-two fluoro-N-methyl-benzamides; 3-(3-cyano group-N-methyl-benzamide base)-N-(2; 6-two iodo-4-(perfluoropropane-2-yl) phenyl)-the 2-fluorobenzamide; (3-(2 for N-; 6-two iodo-4-(perfluoropropane-2-yl) phenyl amino formyl radical)-the 2-fluorophenyl)-2-fluoro-N-methyl-benzamide; N-(2; 6-two iodo-4-(perfluoropropane-2-yl) phenyl)-2-fluoro-3-(3-fluoro-N-methyl-benzamide base) benzamide; 6-chloro-N-(3-(2,6-two iodo-4-(perfluoropropane-2-yl) phenyl amino formyl radical)-2-fluorophenyl)-N-methylnicotinamide;

N-(2; 6-two iodo-4-(perfluoropropane-2-yl) phenyl)-2-fluoro-3-(4-fluoro-N-methyl-benzamide base) benzamide; (3-(2 for N-; 6-two iodo-4-(perfluoropropane-2-yl) phenyl amino formyl radical)-and the 2-fluorophenyl)-2; 6-two fluoro-N-methyl-benzamides; N-(2; 6-two bromo-4-(perfluoropropane-2-yl) phenyl)-2-fluoro-3-(2-fluorobenzoyl amido) benzamide; N-(2; 6-two bromo-4-(perfluoropropane-2-yl) phenyl)-2-fluoro-3-(3-fluorobenzoyl amido) benzamide; N-(2; 6-two bromo-4-(perfluoropropane-2-yl) phenyl)-2-fluoro-3-(4-fluorobenzoyl amido) benzamide; N-(2; 6-two bromo-4-(perfluoropropane-2-yl) phenyl)-3-(2; 6-difluorobenzamide base)-the 2-fluorobenzamide; (3-(2 for 6-chloro-N-; 6-two bromo-4-(perfluoropropane-2-yl) phenyl amino formyl radical)-and the 2-fluorophenyl) niacinamide; 3-(3-cyano group benzoylamino)-N-(2; 6-two bromo-4-(perfluoropropane-2-yl) phenyl)-the 2-fluorobenzamide; 3-(4-cyano group benzoylamino)-N-(2; 6-two bromo-4-(perfluoropropane-2-yl) phenyl)-the 2-fluorobenzamide; (3-(2 for 2-chloro-N-; 6-two iodo-4-(perfluoropropane-2-yl) phenyl amino formyl radical)-the 2-fluorophenyl)-the N-methylnicotinamide; (3-(2 for N-; 6-two bromo-4-(perfluoropropane-2-yl) phenyl amino formyl radical)-the 2-fluorophenyl)-2-fluoro-N-methyl-benzamide; N-(2; 6-two bromo-4-(perfluoropropane-2-yl) phenyl)-2-fluoro-3-(3-fluoro-N-methyl-benzamide base) benzamide; N-(2; 6-two bromo-4-(perfluoropropane-2-yl) phenyl)-2-fluoro-3-(4-fluoro-N-methyl-benzamide base) benzamide; (3-(2 for N-; 6-two bromo-4-(perfluoropropane-2-yl) phenyl amino formyl radical)-and the 2-fluorophenyl)-2,6-two fluoro-N-methyl-benzamides; 3-benzoylamino-N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethoxy) phenyl)-2-fluorobenzamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethoxy) phenyl amino formyl radical)-2-fluorophenyl)-2-chloro niacinamide; N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethoxy) phenyl)-3-(4-cyano group benzoylamino)-2-fluorobenzamide; 3-benzoylamino-N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-2-chloro niacinamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-2-chloro-N-methylnicotinamide; 3-benzoylamino-N-(2-chloro-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 2-chloro-N-(3-(2-chloro-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) niacinamide; N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-(3-cyano group benzoylamino) benzamide;

N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-(4-cyano group benzoylamino) benzamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-3-cyano group-N-methyl-benzamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-4-cyano group-N-methyl-benzamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-2-fluoro-N-methylnicotinamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methyl-4-nitrobenzamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-6-chloro-N-methylnicotinamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-6-cyano group-N-methylnicotinamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methyl-3-nitro benzamide; N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-N-methyl-3-(N-methyl-benzamide base) benzamide; N-(3-((2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) (methyl) formamyl) phenyl)-2-chloro-N-methylnicotinamide; 2-bromo-N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) niacinamide; 2-chloro-N-(3-(2-chloro-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methylnicotinamide; N-(3-(2-chloro-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-4-cyano group-N-methyl-benzamide; 3-benzoylamino-N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-fluorobenzamide; N-(5-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical)-2-fluorophenyl)-2-chloro niacinamide; N-(3-((2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) (methyl) formamyl) phenyl)-2-chloro niacinamide; N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-fluoro-3-(N-methyl-benzamide base) benzamide; N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-(4-cyano group-N-methyl-benzamide base)-4-fluorobenzamide; N-(5-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical)-2-fluorophenyl)-2-chloro-N-methylnicotinamide; 3-benzoylamino-N-(4-(perfluoropropane-2-yl)-2,6-two (trifluoromethyl) phenyl) benzamide;

2-chloro-N-(3-(4-(perfluoropropane-2-yl)-2; 6-two (trifluoromethyl) phenyl amino formyl radical) niacinamide phenyl); N-methyl-N-(3-(4-(perfluoropropane-2-yl)-2; 6-two (trifluoromethyl) phenyl amino formyl radical) benzamide phenyl); 2-chloro-N-methyl-N-(3-(4-(perfluoropropane-2-yl)-2; 6-two (trifluoromethyl) phenyl amino formyl radical) niacinamide phenyl); 3-benzoylamino-N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-N-methyl-benzamide; N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-(3-cyano group benzoylamino)-N-methyl-benzamide; N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-(4-cyano group benzoylamino)-N-methyl-benzamide; N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-(3-cyano group-N-methyl-benzamide base)-N-methyl-benzamide; N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-(4-cyano group-N-methyl-benzamide base)-N-methyl-benzamide; 2-bromo-N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methylnicotinamide; 3-benzoylamino-N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-fluorobenzamide; 2-bromo-N-(3-((2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) (methyl) formamyl) phenyl) niacinamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical)-2-fluorophenyl)-2-chloro niacinamide; 3-benzoylamino-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 2-chloro-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) niacinamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-4-cyano group-2-fluoro-N-methyl-benzamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-4-cyano group-2-fluorobenzamide; 3-cyano group-N-(3-(4-(perfluoropropane-2-yl)-2; 6-two (trifluoromethyl) phenyl amino formyl radical) benzamide phenyl); 3-(4-cyano group benzoylamino)-N-(4-(perfluoropropane-2-yl)-2; 6-two (trifluoromethyl) phenyl) benzamide; 3-cyano group-N-methyl-N-(3-(4-(perfluoropropane-2-yl)-2; 6-two (trifluoromethyl) phenyl amino formyl radical) benzamide phenyl); 4-cyano group-N-methyl-N-(3-(4-(perfluoropropane-2-yl)-2,6-two (trifluoromethyl) phenyl amino formyl radical) phenyl) benzamide;

N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-(4-cyano group benzoylamino)-2-fluorobenzamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical)-2-fluorophenyl)-2-chloro-N-methylnicotinamide; N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-(4-cyano group-N-methyl-benzamide base)-2-fluorobenzamide; N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-fluoro-3-(N-methyl-benzamide base) benzamide; N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-(3-cyano group-N-methyl-benzamide base)-2-fluorobenzamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-2-chloro-4-cyano group-N-methyl-benzamide; 3-benzoylamino-N-methyl-N-(4-(perfluoropropane-2-yl)-2; 6-two (trifluoromethyl) phenyl) benzamide; 2-chloro-N-(3-(methyl (4-(perfluoropropane-2-yl)-2; 6-two (trifluoromethyl) phenyl) niacinamide phenyl formamyl)); 3-(3-cyano group benzoylamino)-N-methyl-N-(4-(perfluoropropane-2-yl)-2; 6-two (trifluoromethyl) phenyl) benzamide; 2-bromo-N-(3-(methyl (4-(perfluoropropane-2-yl)-2; 6-two (trifluoromethyl) phenyl) niacinamide phenyl formamyl)); 2-bromo-N-(3-(4-(perfluoropropane-2-yl)-2; 6-two (trifluoromethyl) phenyl amino formyl radical) niacinamide phenyl); 2-bromo-N-methyl-N-(3-(4-(perfluoropropane-2-yl)-2,6-two (trifluoromethyl) phenyl amino formyl radical) phenyl) niacinamide; 3-(4-cyano group benzoylamino)-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 3-cyano group-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) benzamide; 2-bromo-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) niacinamide; 4-cyano group-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide; 2-chloro-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methylnicotinamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-2-iodo niacinamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical)-2-fluorophenyl)-N-methylnicotinamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical)-2-fluorophenyl)-6-fluoro-N-methylnicotinamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical)-2-fluorophenyl)-4-cyano group-2-fluoro-N-methyl-benzamide;

N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical)-2-fluorophenyl)-6-chloro-N-methylnicotinamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical)-2-fluorophenyl)-3; 5-dicyano-N-methyl-benzamide; 3-benzoylamino-2-fluoro-N-(4-(perfluoropropane-2-yl)-2; 6-two (trifluoromethyl) phenyl) benzamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-3,5-dicyano-N-methyl-benzamide; 3-benzoylamino-2-fluoro-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 2-chloro-N-(2-fluoro-3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) niacinamide; 3-benzoylamino-N-(2-bromo-6-(perfluor ethyl)-4-(perfluoropropane-2-yl) phenyl)-2-fluorobenzamide; 3-benzoylamino-N-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl)-2-fluorobenzamide; N-(3-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical)-2-fluorophenyl)-2-chloro niacinamide; N-(2-bromo-6-(perfluor ethyl)-4-(perfluoropropane-2-yl) phenyl)-3-(4-cyano group benzoylamino)-2-fluorobenzamide; N-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl)-2-fluoro-3-(N-methyl-benzamide base) benzamide; N-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl)-3-(3-cyano group-N-methyl-benzamide base)-2-fluorobenzamide; N-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl)-3-(4-cyano group-N-methyl-benzamide base)-2-fluorobenzamide; 2-fluoro-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-(N-methyl-benzamide base) benzamide; 3-(4-cyano group-N-methyl-benzamide base)-2-fluoro-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; N-(3-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide; 3-benzoylamino-N-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 3-benzoylamino-2-fluoro-N-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 2-fluoro-N-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl)-3-(N-methyl-benzamide base) benzamide; 3-(4-cyano group-N-methyl-benzamide base)-2-fluoro-N-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl) benzamide;

3-(3-cyano group-N-methyl-benzamide base)-2-fluoro-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 2-fluoro-N-(2-fluoro-3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide; 2-fluoro-3-(3-fluoro-N-methyl-benzamide base)-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 2-fluoro-3-(4-fluoro-N-methyl-benzamide base)-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 2; 6-two fluoro-N-(2-fluoro-3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide; 6-chloro-N-(2-fluoro-3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) niacinamide; 3-(3-cyano group benzoylamino)-2-fluoro-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 3-(4-cyano group benzoylamino)-2-fluoro-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 2-fluoro-3-(2-fluorobenzoyl amido)-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 2-fluoro-3-(3-fluorobenzoyl amido)-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical)-2-fluorophenyl)-2-fluoro-N-methyl-benzamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical)-2-fluorophenyl)-2,6-two fluoro-N-methyl-benzamides; N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-fluoro-3-(3-fluoro-N-methyl-benzamide base) benzamide; N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-fluoro-3-(4-fluoro-N-methyl-benzamide base) benzamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical)-2-fluorophenyl)-2-chloro niacinamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical)-2-fluorophenyl)-6-chloro niacinamide; N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-(3-cyano group benzoylamino)-2-fluorobenzamide; N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-fluoro-3-(2-fluorobenzoyl amido) benzamide; N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-fluoro-3-(3-fluorobenzoyl amido) benzamide; N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-fluoro-3-(4-fluorobenzoyl amido) benzamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical)-2-fluorophenyl)-N-methylnicotinamide; 2-chloro-N-(2-fluoro-3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methylnicotinamide;

2-fluoro-3-(4-fluorobenzoyl amido)-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 3-(2; 6-difluorobenzamide base)-2-fluoro-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 6-chloro-N-(2-fluoro-3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methylnicotinamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-6-chloro niacinamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-2-fluorobenzamide; N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-(3-fluorobenzoyl amido) benzamide; N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-(4-fluorobenzoyl amido) benzamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-2; the 6-difluorobenzamide; N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-(2; 6-difluorobenzamide base)-the 2-fluorobenzamide; 3-fluoro-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) benzamide; 3-(4-fluorobenzoyl amido)-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 2-fluoro-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) benzamide; 2,6-two fluoro-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) benzamide; 6-chloro-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) niacinamide; 6-chloro-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methylnicotinamide; 3-cyano group-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide; 2-fluoro-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide; 3-fluoro-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide; 4-fluoro-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-2-fluoro-N-methyl-benzamide;

N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-3-fluoro-N-methyl-benzamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-4-fluoro-N-methyl-benzamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-2; 6-two fluoro-N-methyl-benzamides; 2; 4-two chloro-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) benzamide; 3-(2; 4-dichlorobenzene formamido-)-2-fluoro-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 2; 6-two fluoro-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide; 3-(2-chloro-4-fluorobenzoyl amido)-2-fluoro-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide; 3-benzoylamino-N-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 2-chloro-N-(3-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) niacinamide; 6-chloro-N-(3-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) niacinamide; 3-cyano group-N-(3-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) benzamide; 3-(4-cyano group benzoylamino)-N-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 2-fluoro-N-(3-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) benzamide; 3-fluoro-N-(3-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) benzamide; 3-(4-fluorobenzoyl amido)-N-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 2,6-two fluoro-N-(3-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) benzamide; N-(3-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide; 2-chloro-N-(3-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methylnicotinamide; 3-cyano group-N-(3-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide; 4-cyano group-N-(3-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide;

3-fluoro-N-(3-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide; 4-fluoro-N-(3-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical)-2-fluorophenyl)-N-methyl Isonicotinamide; 1-oxidation 3-((3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical)-2-fluorophenyl) (methyl) formamyl) pyridine; 1-oxidation 4-((3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical)-2-fluorophenyl) (methyl) formamyl) pyridine; 2-chloro-4-fluoro-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) benzamide; N-(3-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-2-chloro niacinamide; N-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl)-3-(3-cyano group benzoylamino) benzamide; N-(3-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-2-fluorobenzamide; N-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl)-3-(3-fluorobenzoyl amido) benzamide; N-(3-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-6-chloro niacinamide; N-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl)-3-(4-cyano group benzoylamino) benzamide; N-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl)-3-(4-fluorobenzoyl amido) benzamide; N-(3-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-2, the 6-difluorobenzamide; N-(3-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-2-chloro-N-methylnicotinamide; N-(3-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-3-cyano group-N-methyl-benzamide; N-(3-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-2-fluoro-N-methyl-benzamide; N-(3-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-3-fluoro-N-methyl-benzamide; N-(3-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-6-chloro-N-methylnicotinamide; N-(3-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-4-cyano group-N-methyl-benzamide;

N-(3-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-4-fluoro-N-methyl-benzamide; N-(3-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-2; 6-two fluoro-N-methyl-benzamides; 6-chloro-N-(2-fluoro-3-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) niacinamide; 3-(3-cyano group benzoylamino)-2-fluoro-N-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 3-(4-cyano group benzoylamino)-2-fluoro-N-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 2-fluoro-3-(2-fluorobenzoyl amido)-N-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 2-fluoro-3-(3-fluorobenzoyl amido)-N-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 2-fluoro-3-(4-fluorobenzoyl amido)-N-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 3-(2; 6-difluorobenzamide base)-2-fluoro-N-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; N-(3-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical)-2-fluorophenyl)-6-chloro niacinamide; N-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl)-3-(3-cyano group benzoylamino)-2-fluorobenzamide; N-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl)-3-(4-cyano group benzoylamino)-2-fluorobenzamide; N-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl)-2-fluoro-3-(2-fluorobenzoyl amido) benzamide; N-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl)-2-fluoro-3-(3-fluorobenzoyl amido) benzamide; N-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl)-2-fluoro-3-(4-fluorobenzoyl amido) benzamide; N-(2-bromo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl)-3-(2,6-difluorobenzamide base)-2-fluorobenzamide; 2-chloro-N-(2-fluoro-3-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methylnicotinamide; 6-chloro-N-(2-fluoro-3-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methylnicotinamide; 3-(3-cyano group-N-methyl-benzamide base)-2-fluoro-N-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 2-fluoro-N-(2-fluoro-3-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide;

2-fluoro-3-(3-fluoro-N-methyl-benzamide base)-N-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 2-fluoro-3-(4-fluoro-N-methyl-benzamide base)-N-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 2-chloro-4,5-two fluoro-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) benzamide; 2-chloro-4-fluoro-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-2-chloro-4-fluorobenzamide; 2-chloro-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) benzamide; 3-(2-chlorinated benzene formamido-)-2-fluoro-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide; 2-chloro-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methyl-benzamide; N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-2-chlorinated benzene methane amide; 2-chloro-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-4-nitrobenzamide; N-(2-fluoro-3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl)-N-methylnicotinamide; 1-oxidation 3-((2-fluoro-3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) (methyl) formamyl) pyridine; 4-bromo-2-chloro-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) benzamide; 2-bromo-4-chloro-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) benzamide; 2-bromo-4-fluoro-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) benzamide; 2-fluoro-3-(3-fluoro-N-methyl-benzamide base)-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-N-methyl-benzamide; N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-fluoro-N-methyl-3-(N-methyl-benzamide base) benzamide; or N-(2-chloro-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-fluoro-3-(N-methyl-benzamide base) benzamide.

＜12〉as above-mentioned＜2〉described amide derivatives; in the above-mentioned general formula (7); among the X at least one is the chlorine atom; bromine atoms; the iodine atom; the C1-C6 alkyl; the C1-C6 haloalkyl; the C3-C9 cycloalkyl; the C3-C9 halogenated cycloalkyl; the C2-C6 alkenyl; the C2-C6 halogenated alkenyl; the C2-C6 alkynyl; C2-C6 halo alkynyl; the C1-C6 alkoxyl group; the C1-C6 halogenated alkoxy; the C2-C6 alkenyl oxy; the C2-C6 halogenated alkenyl oxy; C2-C6 alkynyloxy base; C2-C6 halo alkynyloxy base; the C3-C9 cycloalkyloxy; C3-C9 halo cycloalkyloxy; C1-C6 alkyl sulfenyl; C1-C6 haloalkyl sulfenyl; the C1-C6 alkyl sulphinyl; C1-C6 haloalkyl sulfinyl; the C1-C6 alkyl sulphonyl; the C1-C6 halogenated alkyl sulfonyl; C1-C6 alkyl sulphonyl oxygen base; C1-C6 halogenated alkyl sulfonyl oxygen base; the C2-C7 alkyl-carbonyl; the C2-C7 halogenated alkyl carbonyl; the C3-C7 alkenyl carbonyl; C3-C7 halogenated alkenyl carbonyl; C3-C7 alkynyl carbonyl; C3-C7 halo alkynyl carbonyl; the C4-C10 naphthene base carbonyl; C4-C10 halogenated cycloalkyl carbonyl; C2-C7 alkyl-carbonyl oxygen base; C2-C7 halogenated alkyl carbonyl oxygen base; aryl carbonyl oxygen base; the C2-C7 alkoxy carbonyl; the C2-C7 halo alkoxy carbonyl; C3-C7 alkenyl oxy carbonyl; C3-C7 halogenated alkenyl oxy carbonyl; C3-C7 alkynyloxy base carbonyl; C3-C7 halo alkynyloxy base carbonyl; C4-C10 cycloalkyl oxy carbonyl; C4-C10 halogenated cycloalkyl oxygen base carbonyl; the C2-C7 alkyl-carbonyl-amino; C2-C7 halogenated alkyl carbonyl amino; the C2-C7 alkoxycarbonyl amino; C2-C7 halo alkoxy carbonyl amino; the C2-C7 alkoxy-carbonyl oxy; C2-C7 halo alkoxy carbonyl oxygen base; aryl-amino-carbonyl; amino; formamyl; cyano group; hydroxyl; Pentafluorosulfanyl; the C1-C6 alkylamino; C1-C6 haloalkyl amino; the C2-C6 alkenyl amino; C2-C6 halogenated alkenyl amino; C2-C6 alkynyl amino; C2-C6 halo alkynyl amino; the C3-C9 cycloalkyl amino; C3-C9 halogenated cycloalkyl amino; the C2-C7 alkyl amino-carbonyl; C2-C7 haloalkyl aminocarboxyl; C3-C7 alkenyl amino carbonyl; C3-C7 halogenated alkenyl aminocarboxyl; C3-C7 alkynyl aminocarboxyl; C3-C7 halo alkynyl aminocarboxyl; C4-C10 cycloalkyl amino carbonyl; C4-C10 halogenated cycloalkyl aminocarboxyl; phenyl; or heterocyclic radical; when having a plurality of X; each X is same to each other or different to each other, Y ₁Expression halogen atom, C1-C6 halogenated alkoxy or C1-C3 haloalkyl, Y ₅Be C1-C6 halogenated alkoxy or C1-C3 haloalkyl.

＜13〉as above-mentioned＜12〉described amide derivatives, in the above-mentioned general formula (7), Y ₃Be the C2-C4 perfluoroalkyl.

＜14〉as above-mentioned＜13〉described amide derivatives, in the above-mentioned general formula (7), Y ₁Be halogen atom or C1-C3 haloalkyl, Y ₅Be the C1-C3 haloalkyl.

＜15〉as above-mentioned＜14〉described amide derivatives, in the above-mentioned general formula (7), Y ₂And Y ₄Be hydrogen atom.

＜16〉as above-mentioned＜15〉described amide derivatives, in the above-mentioned general formula (7), 4 X are hydrogen atom, halogen atom or cyano group respectively independently.

＜17〉as above-mentioned＜1〉described amide derivatives, represent with following general formula (9).

{ in the general formula (9), n is 4, X, Y ₁～Y ₅, Q ₂, G ₁～G ₃, R ₁, and R ₂With X, the Y in the general formula (1) ₁～Y ₅, Q ₂, G ₁～G ₃, R ₁, and R ₂The difference synonym.}

＜18〉as above-mentioned＜17〉described amide derivatives, in the above-mentioned general formula (9), Y ₁Be halogen atom, C1-C6 halogenated alkoxy or C1-C3 haloalkyl, Y ₅Be C1-C6 halogenated alkoxy or C1-C3 haloalkyl.

＜19〉as above-mentioned＜18〉described amide derivatives, in the above-mentioned general formula (9), Y ₃Be the C2-C4 perfluoroalkyl.

＜20〉as above-mentioned＜19〉described amide derivatives, in the above-mentioned general formula (9), Y ₁And Y ₅Be halogen atom or C1-C3 haloalkyl, Y ₁And Y ₅In the either party be the C1-C3 haloalkyl.

＜21〉as above-mentioned＜20〉described amide derivatives, in the above-mentioned general formula (9), Y ₂And Y ₄Be hydrogen atom.

＜22〉as above-mentioned＜21〉described amide derivatives, in the above-mentioned general formula (9), 4 X are hydrogen atom, halogen atom or cyano group respectively independently.

＜23〉as above-mentioned＜1〉described amide derivatives, in the above-mentioned general formula (1), K is necessary non-metallic atom group when 2 carbon atoms with A and A bonding form cyclic linker group, and described cyclic linker group is from pyridine, N-pyridine oxide, pyrimidine, pyrazine, pyridazine, triazine, pyrroles, pyrazoles, imidazoles, oxazole, isoxazole, thiazole, isothiazole, furans, thiophene, oxadiazole, thiadiazoles or triazole.

＜24〉as above-mentioned＜23〉described amide derivatives, in the above-mentioned general formula (1), K necessary non-metallic atom group when forming the cyclic linker group from pyridine at 2 carbon atoms with A and A bonding, T is-C (=G ₁)-Q ₁The time, Y ₁And Y ₅Be halogen atom or C1-C3 haloalkyl independently respectively.

＜25〉as above-mentioned＜23〉described amide derivatives, in the above-mentioned general formula (1), K is necessary non-metallic atom group when 2 carbon atoms with A and A bonding form cyclic linker group, described cyclic linker group is from pyrroles, pyrazoles, imidazoles, oxazole, isoxazole, thiazole, isothiazole, furans, thiophene, oxadiazole, thiadiazoles or triazole, and T is-C (=G ₁)-Q ₁The time, R ₁The expression Sauerstoffatom; halogen atom; hydroxyl; nitro; nitroso-group; trimethyl silyl; t-butyldimethylsilyl; cyano group; amino; can have substituent C1-C6 alkyl; can have substituent C1-C6 haloalkyl; the C2-C7 alkyl-carbonyl; the C2-C7 halogenated alkyl carbonyl; can have substituent C2-C6 alkenyl; can have substituent C2-C6 halogenated alkenyl; can have substituent C2-C6 alkynyl; can have substituent C2-C6 halo alkynyl; the C2-C7 alkoxy carbonyl; the C2-C7 halo alkoxy carbonyl; C3-C7 alkenyl oxy carbonyl; C3-C7 halogenated alkenyl oxy carbonyl; C3-C7 alkynyloxy base carbonyl; C3-C7 halo alkynyloxy base carbonyl; phenyloxycarbonyl; the C2-C7 alkyl amino-carbonyl; C2-C7 haloalkyl aminocarboxyl; C2-C7 alkyl-carbonyl oxygen base; C2-C7 halogenated alkyl carbonyl oxygen base; benzoyl; the C1-C6 alkoxyl group; the C1-C6 halogenated alkoxy; C1-C6 alkyl sulfenyl; C1-C6 haloalkyl sulfenyl; the C1-C6 alkyl sulphinyl; C1-C6 haloalkyl sulfinyl; the C1-C6 alkyl sulphonyl; the C1-C6 halogenated alkyl sulfonyl; benzenesulfonyl; the benzyl alkylsulfonyl; benzyl; or-C (=O) C (=O) R ₇(in the formula, R ₇Expression C1-C6 alkyl, C1-C6 haloalkyl, C1-C6 alkoxyl group or C1-C6 halogenated alkoxy.)。

＜26〉as above-mentioned＜23〉described amide derivatives, in the above-mentioned general formula (1), K is necessary non-metallic atom group when 2 carbon atoms with A and A bonding form cyclic linker group, described cyclic linker group is from pyrroles, pyrazoles, imidazoles, oxazole, isoxazole, thiazole, isothiazole, furans, thiophene, oxadiazole, thiadiazoles or triazole, and T is-C (=G ₁)-Q ₁The time, R ₂The expression Sauerstoffatom; halogen atom; hydroxyl; nitro; nitroso-group; trimethyl silyl; t-butyldimethylsilyl; cyano group; amino; can have substituent C1-C6 alkyl; can have substituent C1-C6 haloalkyl; the C2-C7 alkyl-carbonyl; the C2-C7 halogenated alkyl carbonyl; can have substituent C2-C6 alkenyl; can have substituent C2-C6 halogenated alkenyl; can have substituent C2-C6 alkynyl; can have substituent C2-C6 halo alkynyl; the C2-C7 alkoxy carbonyl; the C2-C7 halo alkoxy carbonyl; C3-C7 alkenyl oxy carbonyl; C3-C7 halogenated alkenyl oxy carbonyl; C3-C7 alkynyloxy base carbonyl; C3-C7 halo alkynyloxy base carbonyl; phenyloxycarbonyl; the C2-C7 alkyl amino-carbonyl; C2-C7 haloalkyl aminocarboxyl; C2-C7 alkyl-carbonyl oxygen base; C2-C7 halogenated alkyl carbonyl oxygen base; benzoyl; the C1-C6 alkoxyl group; the C1-C6 halogenated alkoxy; C1-C6 alkyl sulfenyl; C1-C6 haloalkyl sulfenyl; the C1-C6 alkyl sulphinyl; C1-C6 haloalkyl sulfinyl; the C1-C6 alkyl sulphonyl; the C1-C6 halogenated alkyl sulfonyl; benzenesulfonyl; the benzyl alkylsulfonyl; benzyl; or-C (=O) C (=O) R ₇(in the formula, R ₇Expression C1-C6 alkyl, C1-C6 haloalkyl, C1-C6 alkoxyl group or C1-C6 halogenated alkoxy.)。

＜27〉as above-mentioned＜23 〉～＜26 in each described amide derivatives, in the above-mentioned general formula (1), Y ₃Be the C2-C4 perfluoroalkyl.

＜28〉as above-mentioned＜27〉described amide derivatives, in the above-mentioned general formula (1), Y ₁And Y ₅Be halogen atom or C1-C3 haloalkyl independently respectively, Y ₁And Y ₅In the either party be the C1-C3 haloalkyl.

＜29〉as above-mentioned＜28〉described amide derivatives, in the above-mentioned general formula (1), Y ₂And Y ₄Be hydrogen atom.

＜30〉as above-mentioned＜29〉described amide derivatives, in the above-mentioned general formula (1), K is necessary non-metallic atom group when 2 carbon atoms with A and A bonding form cyclic linker group, and described cyclic linker group is from pyridine, N-pyridine oxide, pyrroles, thiazole, furans or thiophene.

＜31〉as above-mentioned＜29〉described amide derivatives, in the above-mentioned general formula (1), K is necessary non-metallic atom group when 2 carbon atoms with A and A bonding form cyclic linker group, and described cyclic linker group is from pyridine, N-pyridine oxide or thiazole.

＜32〉as above-mentioned＜16〉described amide derivatives, in the above-mentioned general formula (7), G ₁And G ₃Be Sauerstoffatom.

＜33〉as＜22〉described amide derivatives, in the above-mentioned general formula (9), G ₁, G ₂And G ₃Be Sauerstoffatom.

＜34〉as＜31〉described amide derivatives, in the above-mentioned general formula (1), G ₁, G ₂And G ₃Be Sauerstoffatom.

＜35〉a kind of noxious organism control agent contains above-mentioned＜1 〉～＜34 in each described amide derivatives at least a kind as effective constituent.

＜36〉a kind of agricultural chemicals contains above-mentioned＜1 〉～＜34 in each described amide derivatives at least a kind as effective constituent.

＜37〉a kind of sterilant contains above-mentioned＜1 〉～＜34 in each described amide derivatives at least a kind as effective constituent.

＜38〉the method for control of a kind of harmful organism is suitable for above-mentioned＜35 〉～＜37 in each described medicine.

＜39〉compound of following general formula (56) expression.

(in the formula, Y ₅Expression C1-C3 haloalkyl, Y ₂, Y ₃, and Y ₄Respectively the expression with above-mentioned＜1 in Y ₂, Y ₃, and Y ₄Identical implication.)

＜40〉compound of following general formula (57) expression.

(in the formula, Y ₅Expression C1-C3 haloalkyl, Y ₁, Y ₂, Y ₃, and Y ₄With above-mentioned＜1〉in Y ₁, Y ₂, Y ₃, and Y ₄Represent identical implication respectively.)

＜41〉as above-mentioned＜40〉described compound, in the above-mentioned general formula (57), Y ₁Be halogen atom.

＜42〉above-mentioned＜41〉preparation method of compound of described following general formula (57a) expression, it is characterized in that, make above-mentioned＜39〉compound and the halogenating agent of described general formula (56) expression react.

(in the formula, Y ₅Expression C1-C3 haloalkyl, Y ₂, Y ₃, and Y ₄With above-mentioned＜1〉described Y ₂, Y ₃, and Y ₄Represent identical implication respectively, Y ₁The expression halogen atom.)

＜43〉compound of following general formula (60a) expression.

(in the formula, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.Wherein, K with 2 carbon atoms of A and A bonding form phenyl ring, when X is hydrogen atom, Y ₅Be the C1-C3 haloalkyl.In addition, K with 2 carbon atoms of A and A bonding form phenyl ring, when X is cyano group, Y ₅Be C1-C6 halogenated alkoxy or C1-C3 haloalkyl.)

＜44〉above-mentioned＜43〉preparation method of compound of described following general formula (60a) expression, it is characterized in that the compound that makes following general formula (59) expression reacts with the compound of following general formula (57b) expression.

(in the formula, LG represents that halogen atom, hydroxyl etc. have the functional group of the ability of leaving away, A, K, X, n, and G ₃With above-mentioned＜1〉in A, K, X, n, and G ₃Represent identical implication respectively.)

(in the formula, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

(in the formula, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.Wherein, K with 2 carbon atoms of A and A bonding form phenyl ring, when X is hydrogen atom, Y ₅Be the C1-C3 haloalkyl.In addition, K with 2 carbon atoms of A and A bonding form phenyl ring, when X is cyano group, Y ₅Be C1-C6 halogenated alkoxy or C1-C3 haloalkyl.)

＜45〉compound of following general formula (61a) expression.

(in the formula, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.Wherein, K with 2 carbon atoms of A and A bonding form phenyl ring, when X is hydrogen atom, Y ₅Be the C1-C3 haloalkyl.In addition, K with 2 carbon atoms of A and A bonding form phenyl ring, when X is cyano group, Y ₅Be C1-C6 halogenated alkoxy or C1-C3 haloalkyl.)

＜46〉above-mentioned＜45〉preparation method of compound of described following general formula (61a) expression, it is characterized in that, make above-mentioned＜43〉compound of described general formula (60a) expression reacts in the presence of reductive agent.

(in the formula, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.Wherein, K with 2 carbon atoms of A and A bonding form phenyl ring, when X is hydrogen atom, Y ₅Be the C1-C3 haloalkyl.In addition, K with 2 carbon atoms of A and A bonding form phenyl ring, when X is cyano group, Y ₅Be C1-C6 halogenated alkoxy or C1-C3 haloalkyl.)

＜47〉compound of following general formula (69) expression.

(in the formula, T, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in T, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜48〉above-mentioned＜47〉preparation method of compound of described following general formula (69) expression, it is characterized in that the compound that makes following general formula (61b) expression reacts with the compound of following general formula (62) expression.

(in the formula, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

T-LG general formula (62)

(in the formula, LG represents that halogen atom, hydroxyl etc. have the functional group of the ability of leaving away, T and above-mentioned＜1〉in T represent identical implication.)

(in the formula, T, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in T, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜49〉compound of following general formula (51a) expression.

(in the formula, T, R ₁, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in T, R ₁, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜50〉preparation method of the compound of following general formula (51b) expression is characterized in that, makes above-mentioned＜47〉compound of described following general formula (69) expression and the compound reaction of following general formula (64) expression.

(in the formula, T, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in T, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

R ₁-LG general formula (64)

(in the formula, LG represents that halogen atom, hydroxyl etc. have the functional group of the ability of leaving away, R ₁The expression trimethyl silyl; t-butyldimethylsilyl; cyano group; can have substituent C1-C6 alkyl; can have substituent C1-C6 haloalkyl; the C2-C7 alkyl-carbonyl; the C2-C7 halogenated alkyl carbonyl; can have substituent C2-C6 alkenyl; can have substituent C2-C6 halogenated alkenyl; can have substituent C2-C6 alkynyl; can have substituent C2-C6 halo alkynyl; the C2-C7 alkoxy carbonyl; the C2-C7 halo alkoxy carbonyl; C3-C7 alkenyl oxy carbonyl; C3-C7 halogenated alkenyl oxy carbonyl; C3-C7 alkynyloxy base carbonyl; C3-C7 halo alkynyloxy base carbonyl; phenyloxycarbonyl; the C2-C7 alkyl amino-carbonyl; C2-C7 haloalkyl aminocarboxyl; C2-C7 alkyl-carbonyl oxygen base; C2-C7 halogenated alkyl carbonyl oxygen base; benzoyl; the C1-C6 alkyl sulphinyl; C1-C6 haloalkyl sulfinyl; the C1-C6 alkyl sulphonyl; the C1-C6 halogenated alkyl sulfonyl; benzenesulfonyl; the benzyl alkylsulfonyl; benzyl; or-C (=O) C (=O) R ₇(in the formula, R ₇Expression C1-C6 alkyl, C1-C6 haloalkyl, C1-C6 alkoxyl group or C1-C6 halogenated alkoxy.)。)

(in the formula, R ₁With the R in the above-mentioned general formula (64) ₁Represent identical implication, T, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in T, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜51〉compound of following general formula (57c) expression.

(in the formula, Y ₅Expression C1-C6 halogenated alkoxy or C1-C3 haloalkyl, R ₂The expression Sauerstoffatom; halogen atom; hydroxyl; nitro; nitroso-group; trimethyl silyl; t-butyldimethylsilyl; cyano group; amino; can have substituent C1-C6 alkyl; can have substituent C1-C6 haloalkyl; the C2-C7 alkyl-carbonyl; the C2-C7 halogenated alkyl carbonyl; can have substituent C2-C6 alkenyl; can have substituent C2-C6 halogenated alkenyl; can have substituent C2-C6 alkynyl; can have substituent C2-C6 halo alkynyl; the C2-C7 alkoxy carbonyl; the C2-C7 halo alkoxy carbonyl; C3-C7 alkenyl oxy carbonyl; C3-C7 halogenated alkenyl oxy carbonyl; C3-C7 alkynyloxy base carbonyl; C3-C7 halo alkynyloxy base carbonyl; phenyloxycarbonyl; the C2-C7 alkyl amino-carbonyl; C2-C7 haloalkyl aminocarboxyl; C2-C7 alkyl-carbonyl oxygen base; C2-C7 halogenated alkyl carbonyl oxygen base; benzoyl; the C1-C6 alkoxyl group; the C1-C6 halogenated alkoxy; C1-C6 alkyl sulfenyl; C1-C6 haloalkyl sulfenyl; the C1-C6 alkyl sulphinyl; C1-C6 haloalkyl sulfinyl; the C1-C6 alkyl sulphonyl; the C1-C6 halogenated alkyl sulfonyl; benzenesulfonyl; the benzyl alkylsulfonyl; benzyl; or-C (=O) C (=O) R ₇(in the formula, R ₇Expression C1-C6 alkyl, C1-C6 haloalkyl, C1-C6 alkoxyl group or C1-C6 halogenated alkoxy.), Y ₁, Y ₂, Y ₃, and Y ₄With above-mentioned＜1〉in Y ₁, Y ₂, Y ₃, and Y ₄Represent identical implication respectively.)

＜52〉preparation method of the compound of following general formula (57m) expression is characterized in that, makes the compound of following general formula (57k) expression and the compound reaction of following general formula (66) expression.

(in the formula, Y ₅Expression C1-C6 halogenated alkoxy or C1-C3 haloalkyl, Y ₁, Y ₂, Y ₃, and Y ₄With above-mentioned＜1〉in Y ₁, Y ₂, Y ₃, and Y ₄Represent identical implication respectively.)

R ₂-LG general formula (66)

(in the formula, LG represents that halogen atom, hydroxyl etc. have the functional group of the ability of leaving away, R ₂The expression trimethyl silyl; t-butyldimethylsilyl; cyano group; can have substituent C1-C6 alkyl; can have substituent C1-C6 haloalkyl; the C2-C7 alkyl-carbonyl; the C2-C7 halogenated alkyl carbonyl; can have substituent C2-C6 alkenyl; can have substituent C2-C6 halogenated alkenyl; can have substituent C2-C6 alkynyl; can have substituent C2-C6 halo alkynyl; the C2-C7 alkoxy carbonyl; the C2-C7 halo alkoxy carbonyl; C3-C7 alkenyl oxy carbonyl; C3-C7 halogenated alkenyl oxy carbonyl; C3-C7 alkynyloxy base carbonyl; C3-C7 halo alkynyloxy base carbonyl; phenyloxycarbonyl; the C2-C7 alkyl amino-carbonyl; C2-C7 haloalkyl aminocarboxyl; C2-C7 alkyl-carbonyl oxygen base; C2-C7 halogenated alkyl carbonyl oxygen base; benzoyl; the C1-C6 alkyl sulphinyl; C1-C6 haloalkyl sulfinyl; the C1-C6 alkyl sulphonyl; the C1-C6 halogenated alkyl sulfonyl; benzenesulfonyl; the benzyl alkylsulfonyl; benzyl; or-C (=O) C (=O) R ₇(in the formula, R ₇Expression C1-C6 alkyl, C1-C6 haloalkyl, C1-C6 alkoxyl group or C1-C6 halogenated alkoxy.)。)

(in the formula, Y ₅Expression C1-C6 halogenated alkoxy or C1-C3 haloalkyl, R ₂With the R in the above-mentioned general formula (66) ₂Represent identical implication, Y ₁, Y ₂, Y ₃, and Y ₄With above-mentioned＜1〉in Y ₁, Y ₂, Y ₃, and Y ₄Represent identical implication respectively.)

＜53〉preparation method of the compound of following general formula (57n) expression is characterized in that, makes above-mentioned＜52〉compound and the aldehydes of described following general formula (57k) expression react.

(in the formula, Y ₅Expression C1-C6 halogenated alkoxy or C1-C3 haloalkyl, Y ₁, Y ₂, Y ₃, and Y ₄With above-mentioned＜1〉in Y ₁, Y ₂, Y ₃, and Y ₄Represent identical implication respectively.)

(in the formula, Y ₅Expression C1-C6 halogenated alkoxy or C1-C3 haloalkyl, R ₂Expression can have substituent C1-C6 alkyl, can have substituent C1-C6 haloalkyl, benzyl, Y ₁, Y ₂, Y ₃, and Y ₄With above-mentioned＜1〉in Y ₁, Y ₂, Y ₃, and Y ₄Represent identical implication respectively.)

＜54〉compound of following general formula (60) expression.

(in the formula, R ₂With above-mentioned＜51〉in R ₂Represent identical implication, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜55〉following general formula＜60e〉preparation method of compound of expression, it is characterized in that, make compound and above-mentioned＜52 of following general formula (60f) expression〉compound of described following general formula (66) expression reacts.

(in the formula, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

R ₂-LG general formula (66)

(in the formula, LG represents that halogen atom, hydroxyl etc. have the functional group of the ability of leaving away, R ₂The expression trimethyl silyl; t-butyldimethylsilyl; cyano group; can have substituent C1-C6 alkyl; can have substituent C1-C6 haloalkyl; the C2-C7 alkyl-carbonyl; the C2-C7 halogenated alkyl carbonyl; can have substituent C2-C6 alkenyl; can have substituent C2-C6 halogenated alkenyl; can have substituent C2-C6 alkynyl; can have substituent C2-C6 halo alkynyl; the C2-C7 alkoxy carbonyl; the C2-C7 halo alkoxy carbonyl; C3-C7 alkenyl oxy carbonyl; C3-C7 halogenated alkenyl oxy carbonyl; C3-C7 alkynyloxy base carbonyl; C3-C7 halo alkynyloxy base carbonyl; phenyloxycarbonyl; the C2-C7 alkyl amino-carbonyl; C2-C7 haloalkyl aminocarboxyl; C2-C7 alkyl-carbonyl oxygen base; C2-C7 halogenated alkyl carbonyl oxygen base; benzoyl; the C1-C6 alkyl sulphinyl; C1-C6 haloalkyl sulfinyl; the C1-C6 alkyl sulphonyl; the C1-C6 halogenated alkyl sulfonyl; benzenesulfonyl; the benzyl alkylsulfonyl; benzyl; or-C (=O) C (=O) R ₇(in the formula, R ₇Expression C1-C6 alkyl, C1-C6 haloalkyl, C1-C6 alkoxyl group or C1-C6 halogenated alkoxy.)。)

(in the formula, R ₂With the R in the above-mentioned general formula (66) ₂Represent identical implication, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜56〉above-mentioned＜54〉preparation method of compound of described following general formula (60) expression, it is characterized in that, make compound and above-mentioned＜44 of following general formula (57d) expression〉compound of described following general formula (59) expression reacts.

(in the formula, R ₂With above-mentioned＜51〉in R ₂Represent identical implication, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

(in the formula, LG represents that halogen atom, hydroxyl etc. have the functional group of the ability of leaving away, A, K, X, n, and G ₃With above-mentioned＜1〉in A, K, X, n, and G ₃Represent identical implication respectively.)

(in the formula, R ₂With above-mentioned＜51〉in R ₂Represent identical implication, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜57〉compound of following general formula (61) expression.

(in the formula, R ₂With above-mentioned＜51〉in R ₂Represent identical implication, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜58〉above-mentioned＜57〉preparation method of compound of described following general formula (61) expression, it is characterized in that, make above-mentioned＜54〉compound of described general formula (60) expression reacts in the presence of reductive agent.

(in the formula, R ₂With above-mentioned＜51〉in R ₂Represent identical implication, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜59〉compound of following general formula (63) expression.

(in the formula, T, R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in T, R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜60〉above-mentioned＜59〉preparation method of compound of described following general formula (63) expression, it is characterized in that, make compound and above-mentioned＜48 of following general formula (61e) expression〉described following general formula (62) reacts.

(in the formula, R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

T-LG general formula (62)

(in the formula, LG represents that halogen atom, hydroxyl etc. have the functional group of the ability of leaving away, T and above-mentioned＜1〉in T represent identical implication.)

(in the formula, T, R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in T, R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜61〉preparation method of the compound of following general formula (1b) expression is characterized in that, makes above-mentioned＜59〉compound and above-mentioned＜50 of described following general formula (63) expression〉described following general formula (64) reacts.

(in the formula, T, R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in T, R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

R ₁-LG general formula (64)

(in the formula, LG represents that halogen atom, hydroxyl etc. have the functional group of the ability of leaving away, R ₁The expression trimethyl silyl; t-butyldimethylsilyl; cyano group; can have substituent C1-C6 alkyl; can have substituent C1-C6 haloalkyl; the C2-C7 alkyl-carbonyl; the C2-C7 halogenated alkyl carbonyl; can have substituent C2-C6 alkenyl; can have substituent C2-C6 halogenated alkenyl; can have substituent C2-C6 alkynyl; can have substituent C2-C6 halo alkynyl; the C2-C7 alkoxy carbonyl; the C2-C7 halo alkoxy carbonyl; C3-C7 alkenyl oxy carbonyl; C3-C7 halogenated alkenyl oxy carbonyl; C3-C7 alkynyloxy base carbonyl; C3-C7 halo alkynyloxy base carbonyl; phenyloxycarbonyl; the C2-C7 alkyl amino-carbonyl; C2-C7 haloalkyl aminocarboxyl; C2-C7 alkyl-carbonyl oxygen base; C2-C7 halogenated alkyl carbonyl oxygen base; benzoyl; the C1-C6 alkyl sulphinyl; C1-C6 haloalkyl sulfinyl; the C1-C6 alkyl sulphonyl; the C1-C6 halogenated alkyl sulfonyl; benzenesulfonyl; the benzyl alkylsulfonyl; benzyl; or-C (=O) C (=O) R ₇(in the formula, R ₇Expression C1-C6 alkyl, C1-C6 haloalkyl, C1-C6 alkoxyl group or C1-C6 halogenated alkoxy.)。)

(in the formula, R ₁With the R in the general formula (64) ₁Represent identical implication, R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜62〉compound of following general formula (65a) expression.

(in the formula, R ₁, R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in R ₁, R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.Wherein, K with 2 carbon atoms of A and A bonding form phenyl ring, X is hydrogen atom, R ₂During for hydrogen atom, Y ₅Be the C1-C3 haloalkyl.In addition, K with 2 carbon atoms of A and A bonding form phenyl ring, X is cyano group, R ₁And R ₂During for hydrogen atom, Y ₅Be C1-C6 halogenated alkoxy or C1-C3 haloalkyl.)

＜63〉preparation method of the compound of following general formula (65c) expression is characterized in that, makes above-mentioned＜60〉compound and the aldehydes of described following general formula (61e) expression react.

(in the formula, R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

(in the formula, R ₁Expression can have substituent C1-C6 alkyl, can have substituent C1-C6 haloalkyl or benzyl, R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.Wherein, K with 2 carbon atoms of A and A bonding form phenyl ring, X is hydrogen atom, R ₂During for hydrogen atom, Y ₅Be the C1-C3 haloalkyl.)

＜64〉above-mentioned＜1〉preparation method of compound of described following general formula (1) expression, it is characterized in that, make compound and above-mentioned＜48 of following general formula (65b) expression〉described following general formula (62) reacts.

(in the formula, R ₁, R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in R ₁, R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

T-LG general formula (62)

(in the formula, LG represents that halogen atom, hydroxyl etc. have the functional group of the ability of leaving away, T and above-mentioned＜1〉in T represent identical implication.)

＜65〉compound of following general formula (68) expression.

(in the formula, Xa represents chlorine atom, bromine atoms or iodine atom, R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜23〉in R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜66〉above-mentioned＜65〉preparation method of compound of described following general formula (68) expression, it is characterized in that, the compound of following general formula (57j) expression and following general formula (67) are reacted.

(in the formula, R ₂, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜1〉in R ₂, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

(in the formula, LG represents that halogen atom, hydroxyl etc. have the functional group of the ability of leaving away, and Xa represents chlorine atom, bromine atoms or iodine atom, A, K, X, n, and G ₃With above-mentioned＜23〉in A, K, X, n, and G ₃Represent identical implication respectively.)

(in the formula, Xa represents chlorine atom, bromine atoms or iodine atom, R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜23〉in R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜67〉preparation method of the compound of following general formula (65d) expression is characterized in that, makes above-mentioned＜65〉compound and the amination agent of described following general formula (68) expression react.

(in the formula, Xa represents chlorine atom, bromine atoms or iodine atom, R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜23〉in R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

(in the formula, R ₁, R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜23〉in R ₁, R ₂, A, K, X, n, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜68〉compound of following general formula (70) expression.

(in the formula, Xb represents chlorine atom, bromine atoms, iodine atom, R ₂, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, Y ₅With above-mentioned＜1〉the identical implication of expression.)

＜69〉compound of following general formula (72) expression.

(in the formula, R ₂, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, Y ₅With above-mentioned＜1〉in R ₂, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, Y ₅Represent identical implication respectively.)

＜70〉above-mentioned＜69〉preparation method of compound of described following general formula (72) expression, it is characterized in that, make above-mentioned＜68〉compound and the fluorizating agent of described general formula (70) expression react.

(in the formula, R ₂, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, Y ₅With above-mentioned＜1〉in R ₂, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, Y ₅Represent identical implication respectively.)

＜71〉compound of following general formula (73) expression.

(in the formula, Xc represents halogen atom, R ₂, G ₃, Y ₁, Y ₂, Y ₃, Y ₄And Y ₅With above-mentioned＜1〉in R ₂, G ₃, Y ₁, Y ₂, Y ₃, Y ₄And Y ₅Represent identical implication respectively.)

＜72〉compound of following general formula (75) expression.

(in the formula, Y ₅Expression C1-C6 halogenated alkoxy or C1-C3 haloalkyl, R ₂, G ₃, Y ₁, Y ₂, Y ₃, and Y ₄With above-mentioned＜1〉in R ₂, G ₃, Y ₁, Y ₂, Y ₃, and Y ₄Represent identical implication respectively.)

＜73〉above-mentioned＜72〉preparation method of compound of described following general formula (75) expression, it is characterized in that, make above-mentioned＜71〉Y in the described general formula (73) ₅Compound and cyano group agent reaction for C1-C6 halogenated alkoxy or C1-C3 haloalkyl.

(in the formula, Y ₅Expression C1-C6 halogenated alkoxy or C1-C3 haloalkyl, R ₂, G ₃, Y ₁, Y ₂, Y ₃, and Y ₄With above-mentioned＜1〉in R ₂, G ₃, Y ₁, Y ₂, Y ₃, and Y ₄Represent identical implication respectively.)

＜74〉compound of following general formula (56a) expression.

(in the formula, Y ₅Expression C1-C3 haloalkyl, Y ₂, Y ₃, and Y ₄With above-mentioned＜3〉in Y ₂, Y ₃, and Y ₄Represent identical implication respectively.)

＜75〉compound of following general formula (57e) expression.

(in the formula, Y ₅Expression C1-C3 haloalkyl, Y ₁, Y ₂, Y ₃, and Y ₄With above-mentioned＜3〉in Y ₁, Y ₂, Y ₃, and Y ₄Represent identical implication respectively.)

＜76〉above-mentioned＜75〉the middle Y of described general formula (57e) ₁Compound for halogen atom.

＜77〉above-mentioned＜76〉preparation method of compound of described following general formula (57f) expression, it is characterized in that, make above-mentioned＜74〉compound and the halogenating agent of described general formula (56a) expression react.

(in the formula, Y ₅Expression C1-C3 haloalkyl, Y ₂, Y ₃, and Y ₄With above-mentioned＜3〉in Y ₂, Y ₃, and Y ₄Represent identical implication respectively, Y ₁The expression halogen atom.)

＜78〉compound of following general formula (60b) expression.

(in the formula, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.Wherein, X ₁, X ₂, X ₃, and X ₄When being hydrogen atom, Y ₅Be the C1-C3 haloalkyl, in addition, X ₂Be cyano group, X ₁, X ₃, and X ₄During for hydrogen atom, Y ₅Be C1-C3 halogenated alkoxy or C1-C3 haloalkyl.)

＜79〉above-mentioned＜78〉preparation method of compound of described following general formula (60b) expression, it is characterized in that the compound that makes following general formula (59a) expression reacts with the compound of following general formula (57g) expression.

(in the formula, LG represents that halogen atom, hydroxyl etc. have the functional group of the ability of leaving away, X ₁, X ₂, X ₃, and X ₄With above-mentioned＜3〉in X ₁, X ₂, X ₃, and X ₄Represent identical implication respectively.)

(in the formula, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

(in the formula, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.Wherein, X ₁, X ₂, X ₃, and X ₄When being hydrogen atom, Y ₅Be the C1-C3 haloalkyl, in addition, X ₂Be cyano group, X ₁, X ₃, and X ₄During for hydrogen atom, Y ₅Be C1-C3 halogenated alkoxy or C1-C3 haloalkyl.)

＜80〉compound of following general formula (61f) expression.

(in the formula, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.Wherein, X ₁, X ₂, X ₃, and X ₄When being hydrogen atom, Y ₅Be the C1-C3 haloalkyl, in addition, X ₂Be cyano group, X ₁, X ₃, and X ₄During for hydrogen atom, Y ₅Be C1-C3 halogenated alkoxy or C1-C3 haloalkyl.)

＜81〉above-mentioned＜80〉preparation method of compound of described following general formula (61f) expression, it is characterized in that, make above-mentioned＜78〉compound of described general formula (60b) expression reacts in the presence of reductive agent.

(in the formula, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.Wherein, X ₁, X ₂, X ₃, and X ₄When being hydrogen atom, Y ₅Be the C1-C3 haloalkyl, in addition, X ₂Be cyano group, X ₁, X ₃, and X ₄During for hydrogen atom, Y ₅Be C1-C3 halogenated alkoxy or C1-C3 haloalkyl.)

＜82〉compound of following general formula (69a) expression.

(in the formula, Q ₁, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in Q ₁, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜83〉above-mentioned＜82〉preparation method of compound of described following general formula (69a) expression, it is characterized in that, the compound of following general formula (61c) expression and following general formula (62a) are reacted.

(in the formula, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

(in the formula, LG represents that halogen atom, hydroxyl etc. have the functional group of the ability of leaving away, Q ₁With above-mentioned＜3〉in Q ₁Represent identical implication.)

(in the formula, Q ₁, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in Q ₁, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜84〉compound of following general formula (53a) expression.

(in the formula, Q ₁, R ₁, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in Q ₁, R ₁, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜85〉preparation method of the compound of following general formula (53b) expression is characterized in that, makes above-mentioned＜82〉compound and the following general formula (64a) of described following general formula (69a) expression react.

(in the formula, Q ₁, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in Q ₁, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

R ₁-LG general formula (64a)

(in the formula, LG represents that halogen atom, hydroxyl etc. have the functional group of the ability of leaving away, R ₁Expression C1-C3 alkyl.)

(in the formula, R ₁With the R in the general formula (64a) ₁Represent identical implication, Q ₁, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in Q ₁, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜86〉compound of following general formula (57h) expression.

(in the formula, Y ₅Expression C1-C3 halogenated alkoxy or C1-C3 haloalkyl, R ₂Expression C1-C3 alkyl, Y ₁, Y ₂, Y ₃, and Y ₄With above-mentioned＜3〉in Y ₁, Y ₂, Y ₃, and Y ₄Represent identical implication respectively.)

＜87〉above-mentioned＜86〉preparation method of compound of described following general formula (57h) expression, it is characterized in that, the compound of following general formula (571) expression and following general formula (66a) are reacted.

(in the formula, Y ₅Expression C1-C3 halogenated alkoxy or C1-C3 haloalkyl, Y ₁, Y ₂, Y ₃, and Y ₄With above-mentioned＜3〉in Y ₁, Y ₂, Y ₃, and Y ₄Represent identical implication respectively.)

R ₂-LG general formula (66a)

(in the formula, LG represents that halogen atom, hydroxyl etc. have the functional group of the ability of leaving away, R ₂Expression C1-C3 alkyl.)

(in the formula, Y ₅Expression C1-C3 halogenated alkoxy or C1-C3 haloalkyl, R ₂Expression C1-C3 alkyl, Y ₁, Y ₂, Y ₃, and Y ₄With above-mentioned＜3〉in Y ₁, Y ₂, Y ₃, and Y ₄Represent identical implication respectively.)

＜88〉above-mentioned＜86〉preparation method of compound of described following general formula (57h) expression, it is characterized in that, make above-mentioned＜87〉compound and the aldehydes of described following general formula (571) expression react.

(in the formula, Y ₅Expression C1-C3 halogenated alkoxy or C1-C3 haloalkyl, Y ₁, Y ₂, Y ₃, and Y ₄With above-mentioned＜3〉in Y ₁, Y ₂, Y ₃, and Y ₄Represent identical implication respectively.)

(in the formula, Y ₅Expression C1-C3 halogenated alkoxy or C1-C3 haloalkyl, R ₂Expression C1-C3 alkyl, Y ₁, Y ₂, Y ₃, and Y ₄With above-mentioned＜3〉in Y ₁, Y ₂, Y ₃, and Y ₄Represent identical implication respectively.)

＜89〉compound of following general formula (60c) expression.

(in the formula, R ₂Expression C1-C3 alkyl, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜90〉above-mentioned＜89〉preparation method of compound of described following general formula (60c) expression, it is characterized in that, make compound and above-mentioned＜87 of following general formula (60d) expression〉described following general formula (66a) reacts.

(in the formula, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

R ₂-LG general formula (66a)

(in the formula, LG represents that halogen atom, hydroxyl etc. have the functional group of the ability of leaving away, R ₂Expression C1-C3 alkyl.)

(in the formula, R ₂Expression C1-C3 alkyl, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜91〉above-mentioned＜89〉preparation method of compound of described following general formula (60c) expression, it is characterized in that, make compound and above-mentioned＜79 of following general formula (57i) expression〉compound of described following general formula (59a) expression reacts.

(in the formula, R ₂Expression C1-C3 alkyl, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

(in the formula, LG represents that halogen atom, hydroxyl etc. have the functional group of the ability of leaving away, X ₁, X ₂, X ₃, and X ₄With above-mentioned＜3〉in X ₁, X ₂, X ₃, and X ₄Represent identical implication respectively.)

(in the formula, R ₂Expression C1-C3 alkyl, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜92〉compound of following general formula (61g) expression.

(in the formula, R ₂Expression C1-C3 alkyl, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜93〉above-mentioned＜92〉preparation method of compound of described following general formula (61g) expression, it is characterized in that, make above-mentioned＜89〉compound of described general formula (60c) expression reacts in the presence of reductive agent.

(in the formula, R ₂Expression C1-C3 alkyl, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜94〉compound of following general formula (63c) expression.

(in the formula, Q ₁, R ₂, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in Q ₁, R ₂, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜95〉above-mentioned＜94〉preparation method of compound of described following general formula (63c) expression, it is characterized in that, make compound and above-mentioned＜83 of following general formula (61d) expression〉described following general formula (62a) reacts.

(in the formula, R ₂, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in R ₂, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

(in the formula, LG represents that halogen atom, hydroxyl etc. have the functional group of the ability of leaving away, Q ₁With above-mentioned＜3〉in Q ₁Represent identical implication.)

(in the formula, Q ₁, R ₂, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in Q ₁, R ₂, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜96〉preparation method of the compound of following general formula (3a) expression is characterized in that, makes above-mentioned＜94〉compound and above-mentioned＜85 of described following general formula (63c) expression〉described following general formula (64a) reacts.

(in the formula, Q ₁, R ₂, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in Q ₁, R ₂, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

R ₁-LG general formula (64a)

(in the formula, LG represents that halogen atom, hydroxyl etc. have the functional group of the ability of leaving away, R ₁Expression C1-C3 alkyl.)

(in the formula, R ₁With the R in the general formula (64a) ₁Represent identical implication, Q ₁, R ₂, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in Q ₁, R ₂, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜97〉compound of following general formula (65e) expression.

(in the formula, R ₁, R ₂, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in R ₁, R ₂, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.Wherein, X ₁, X ₂, X ₃, X ₄Be hydrogen atom, R ₂During for hydrogen atom, Y ₅Be the C1-C3 haloalkyl, in addition, X ₂Be cyano group, X ₁, X ₃, and X ₄Be hydrogen atom, R ₁And R ₂During for hydrogen atom, Y ₅Be C1-C3 halogenated alkoxy or C1-C3 haloalkyl.)

＜98〉preparation method of the compound of following general formula (65f) expression is characterized in that, makes the compound and the aldehydes reaction of following general formula (61d) expression.

(in the formula, R ₂, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in R ₂, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

(in the formula, R ₁Expression C1-C3 alkyl, R ₂, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in R ₂, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.Wherein, X ₁, X ₂, X ₃, X ₄Be hydrogen atom, R ₂During for hydrogen atom, Y ₅Be the C1-C3 haloalkyl.)

＜99〉above-mentioned＜3〉preparation method of compound of described following general formula (3) expression, it is characterized in that, make compound and above-mentioned＜83 of following general formula (65g) expression〉described following general formula (62a) reacts.

(in the formula, R ₁, R ₂, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in R ₁, R ₂, X ₁, X ₂, X ₃, X ₄, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

(in the formula, LG represents that halogen atom, hydroxyl etc. have the functional group of the ability of leaving away, Q ₁With above-mentioned＜3〉in Q ₁Represent identical implication.)

＜100〉compound of following general formula (70a) expression.

(in the formula, Xb represents chlorine atom, bromine atoms, iodine atom, R ₂, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in R ₂, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜101〉compound of following general formula (72a) expression.

(in the formula, R ₂, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in R ₂, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

＜102〉above-mentioned＜101〉preparation method of compound of described following general formula (72a) expression, it is characterized in that, make above-mentioned＜100〉compound and the fluorizating agent of described general formula (70a) expression react.

(in the formula, R ₂, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅With above-mentioned＜3〉in R ₂, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Represent identical implication respectively.)

According to the present invention, can be provided at and operable in the agricultural gardening field of wider range insect is shown the acid amides biology of insecticidal effect and contains this amide derivatives as the noxious organism control agent of effective constituent and the method for control of harmful organism.

Embodiment

Amide compound of the present invention is shown in following general formula (1).

In the general formula (1), A represents carbon atom, Sauerstoffatom, nitrogen-atoms, oxidized nitrogen-atoms or sulphur atom.Necessary non-metallic atom group when K is illustrated in 2 carbon atoms with A and A bonding and forms cyclic linker group, described cyclic linker group is from benzene, pyridine, N-pyridine oxide, pyrimidine, pyrazine, pyridazine, triazine, pyrroles, pyrazoles, imidazoles, oxazole, isoxazole, thiazole, isothiazole, furans, thiophene, oxadiazole, thiadiazoles or triazole.

X represents hydrogen atom; halogen atom; the C1-C6 alkyl; the C1-C6 haloalkyl; the C3-C9 cycloalkyl; the C3-C9 halogenated cycloalkyl; the C2-C6 alkenyl; the C2-C6 halogenated alkenyl; the C2-C6 alkynyl; C2-C6 halo alkynyl; the C1-C6 alkoxyl group; the C1-C6 halogenated alkoxy; C1-C6 alkyl sulfenyl; C1-C6 haloalkyl sulfenyl; the C1-C6 alkyl sulphinyl; C1-C6 haloalkyl sulfinyl; the C1-C6 alkyl sulphonyl; the C1-C6 halogenated alkyl sulfonyl; C1-C6 alkyl sulphonyl oxygen base; C1-C6 halogenated alkyl sulfonyl oxygen base; the C2-C7 alkyl-carbonyl; the C2-C7 halogenated alkyl carbonyl; C2-C7 alkyl-carbonyl oxygen base; C2-C7 halogenated alkyl carbonyl oxygen base; aryl carbonyl oxygen base; the C2-C7 alkoxy carbonyl; the C2-C7 halo alkoxy carbonyl; the C2-C7 alkyl-carbonyl-amino; C2-C7 halogenated alkyl carbonyl amino; the C2-C7 alkoxycarbonyl amino; C2-C7 halo alkoxy carbonyl amino; the C2-C7 alkoxy-carbonyl oxy; C2-C7 halo alkoxy carbonyl oxygen base; aryl-amino-carbonyl; amino; formamyl; cyano group; hydroxyl; Pentafluorosulfanyl; the C1-C6 alkylamino; C1-C6 haloalkyl amino; the C2-C6 alkenyl amino; C2-C6 halogenated alkenyl amino; C2-C6 alkynyl amino; C2-C6 halo alkynyl amino; the C3-C9 cycloalkyl amino; C3-C9 halogenated cycloalkyl amino; the C2-C7 alkyl amino-carbonyl; C2-C7 haloalkyl aminocarboxyl; C3-C7 alkenyl amino carbonyl; C3-C7 halogenated alkenyl aminocarboxyl; C3-C7 alkynyl aminocarboxyl; C3-C7 halo alkynyl aminocarboxyl; C4-C10 cycloalkyl amino carbonyl; C4-C10 halogenated cycloalkyl aminocarboxyl; phenyl; or heterocyclic radical; when having a plurality of X, each X can be same to each other or different to each other.

N represents 0～4 integer.T represents-C (=G ₁)-Q ₁, or-C (=G ₁)-G ₂Q ₂G ₁And G ₂Represent Sauerstoffatom or sulphur atom, Q respectively independently ₁And Q ₂Represent hydrogen atom, C1-C6 alkyl, C1-C6 haloalkyl, C2-C6 alkenyl, C2-C6 halogenated alkenyl, C2-C6 alkynyl, C2-C6 halo alkynyl, C3-C9 cycloalkyl, C3-C9 halogenated cycloalkyl, benzyl, can have substituent phenyl, naphthyl, maybe can have substituent heterocyclic radical.

Y ₁And Y ₅Represent halogen atom, C1-C6 halogenated alkoxy or C1-C3 haloalkyl respectively independently, Y ₂And Y ₄Represent hydrogen atom, halogen atom or C1-C4 alkyl respectively independently, Y ₃Expression C2-C5 haloalkyl.

Need to prove Q ₁And Q ₂In; the substituting group that can have substituent phenyl and can have a substituent heterocyclic radical represents to be selected from the substituting group more than 1 in the following radicals; described group is: halogen atom; the C1-C6 alkyl; the C1-C6 haloalkyl; the C3-C9 cycloalkyl; the C3-C9 halogenated cycloalkyl; the C2-C6 alkenyl; the C2-C6 halogenated alkenyl; the C2-C6 alkynyl; C2-C6 halo alkynyl; the C1-C6 alkoxyl group; the C1-C6 halogenated alkoxy; C1-C6 alkyl sulfenyl; C1-C6 haloalkyl sulfenyl; the C1-C6 alkyl sulphinyl; C1-C6 haloalkyl sulfinyl; the C1-C6 alkyl sulphonyl; the C1-C6 halogenated alkyl sulfonyl; the C2-C7 alkyl-carbonyl; the C2-C7 halogenated alkyl carbonyl; C2-C7 alkyl-carbonyl oxygen base; C2-C7 halogenated alkyl carbonyl oxygen base; C1-C6 alkyl sulphonyl oxygen base; C1-C6 halogenated alkyl sulfonyl oxygen base; the C2-C7 alkoxy carbonyl; the C2-C7 halo alkoxy carbonyl; the C2-C7 alkyl-carbonyl-amino; C2-C7 halogenated alkyl carbonyl amino; the C2-C7 alkoxycarbonyl amino; C2-C7 halo alkoxy carbonyl amino; the C1-C6 alkylamino; C1-C6 haloalkyl amino; the C2-C6 alkenyl amino; C2-C6 halogenated alkenyl amino; C2-C6 alkynyl amino; C2-C6 halo alkynyl amino; the C3-C9 cycloalkyl amino; C3-C9 halogenated cycloalkyl amino; the C2-C7 alkyl amino-carbonyl; C2-C7 haloalkyl aminocarboxyl; C3-C7 alkenyl amino carbonyl; C3-C7 halogenated alkenyl aminocarboxyl; C3-C7 alkynyl aminocarboxyl; C3-C7 halo alkynyl aminocarboxyl; C4-C10 cycloalkyl amino carbonyl; C4-C10 halogenated cycloalkyl aminocarboxyl; amino; formamyl; cyano group; nitro; hydroxyl; Pentafluorosulfanyl; can have substituent phenyl; and can have substituent heterocyclic radical; when having 2 above substituting groups, each substituting group can be the same or different.

And then, X, Q ₁, and Q ₂In heterocyclic radical represent pyridyl, N-pyridine oxide base, pyrimidyl, pyrazinyl, pyridazinyl, furyl, thienyl, oxazolyl, isoxazolyl, oxadiazole base, thiazolyl, isothiazolyl, thiadiazolyl group, pyrryl, imidazolyl, triazolyl, pyrazolyl or tetrazyl.

G ₃Expression Sauerstoffatom or sulphur atom.

R ₁And R ₂Represent hydrogen atom respectively independently; Sauerstoffatom; halogen atom; hydroxyl; nitro; nitroso-group; trimethyl silyl; t-butyldimethylsilyl; cyano group; amino; can have substituent C1-C6 alkyl; can have substituent C1-C6 haloalkyl; the C2-C7 alkyl-carbonyl; the C2-C7 halogenated alkyl carbonyl; can have substituent C2-C6 alkenyl; can have substituent C2-C6 halogenated alkenyl; can have substituent C2-C6 alkynyl; can have substituent C2-C6 halo alkynyl; the C2-C7 alkoxy carbonyl; the C2-C7 halo alkoxy carbonyl; C3-C7 alkenyl oxy carbonyl; C3-C7 halogenated alkenyl oxy carbonyl; C3-C7 alkynyloxy base carbonyl; C3-C7 halo alkynyloxy base carbonyl; phenyloxycarbonyl; the C2-C7 alkyl amino-carbonyl; C2-C7 haloalkyl aminocarboxyl; C2-C7 alkyl-carbonyl oxygen base; C2-C7 halogenated alkyl carbonyl oxygen base; benzoyl; the C1-C6 alkoxyl group; the C1-C6 halogenated alkoxy; C1-C6 alkyl sulfenyl; C1-C6 haloalkyl sulfenyl; the C1-C6 alkyl sulphinyl; C1-C6 haloalkyl sulfinyl; the C1-C6 alkyl sulphonyl; the C1-C6 halogenated alkyl sulfonyl; benzenesulfonyl; the benzyl alkylsulfonyl; benzyl; or-C (=O) C (=O) R ₇(in the formula, R ₇Expression C1-C6 alkyl, C1-C6 haloalkyl, C1-C6 alkoxyl group or C1-C6 halogenated alkoxy.)。

But the amide derivatives that does not comprise above-mentioned general formula (1) expression is any one the situation in following (A)～(I).

(A) in the above-mentioned general formula (1), K necessary non-metallic atom group when forming the cyclic linker group from pyridine at 2 carbon atoms, Y with A and A bonding ₁Be halogen atom, Y ₅Be the C1-C6 halogenated alkoxy, T is-C (=G ₁)-Q ₁

(B) in the above-mentioned general formula (1), K is necessary non-metallic atom group when 2 carbon atoms with A and A bonding form cyclic linker group, described cyclic linker group is from pyrroles, pyrazoles, imidazoles, oxazole, isoxazole, thiazole, isothiazole, furans, thiophene, oxadiazole, thiadiazoles or triazole, Y ₁And Y ₅Be halogen atom independently respectively, T is-C (=G ₁)-G ₂Q ₂

(C) in the above-mentioned general formula (1), K is necessary non-metallic atom group when 2 carbon atoms with A and A bonding form cyclic linker group, described cyclic linker group is from pyrroles, pyrazoles, imidazoles, oxazole, isoxazole, thiazole, isothiazole, furans, thiophene, oxadiazole, thiadiazoles or triazole, and T is-C (=G ₁)-Q ₁, Y ₁Be halogen atom, Y ₅Be halogen atom or halogenated alkoxy.

(D) amide compound of following general formula (2) expression.

In the general formula (2), Y ₂～Y ₄, Q ₁, G ₁, G ₃, R ₁, and R ₂With the Y in the general formula (1) ₂～Y ₄, Q ₁, G ₁, G ₃, R ₁, and R ₂Implication respectively identical, Y ₁Be halogen atom, Y ₅Be the C1-C2 halogenated alkoxy.

(E) in the above-mentioned general formula (2), Y ₁And Y ₅Be halogen atom, X is hydrogen atom, Y ₃Be the C2-C3 haloalkyl.

(F) be the amide compound of following general formula (3) expression.

In the general formula (3), Y ₁And Y ₅Be halogen atom independently respectively, X ₁And X ₃Be hydrogen atom or fluorine atom independently respectively, Q ₁With the Q in the general formula (1) ₁Implication identical, R ₁Be hydrogen atom or methyl, Y ₃Be the C3-C4 perfluoroalkyl.

(G) amide compound of following general formula (4) expression.

In the general formula (4), X ₁Be fluorine atom, X ₂, X ₃, and X ₄Be hydrogen atom, Y ₁And Y ₅Differ from one another, be bromine atoms or trifluoromethoxy, Y ₂And Y ₄Be hydrogen atom, Y ₃Be seven fluorine sec.-propyls, Q ₁Be phenyl or 2-chloropyridine-3-base, R ₁And R ₂Differ from one another, be hydrogen atom or methyl.

Perhaps, X ₁Be fluorine atom, X ₂, X ₃, and X ₄Be hydrogen atom, Y ₁And Y ₅Be bromine atoms, Y ₂And Y ₄Be hydrogen atom, Y ₃Be pentafluoroethyl group, Q ₁Be 2-fluorophenyl, R ₁And R ₂Be hydrogen atom or methyl independently respectively.

(H) amide compound of following general formula (5) expression.

In the general formula (5), Y ₁And Y ₅Be halogen atom independently respectively, X ₁Be hydrogen atom or fluorine atom, Q ₂Be 2,2,2-three chloroethyls and 3,3,3-three fluoro-n-propyl group, Y ₃Be the C2-C4 haloalkyl.

(I) amide compound of following general formula (6) expression.

In the general formula (6), Y ₁And Y ₅Be halogen atom independently respectively, Q ₂With the Q in the general formula (1) ₂Implication is identical, R ₁Be hydrogen atom or methyl, Y ₃Be the C3-C4 haloalkyl.

Considering that from the active viewpoint of Pesticidal the amide derivatives among the present invention is preferably the compound of following general formula (7) expression, more preferably is the compound of following general formula (8) expression.

In the general formula (7), X, n are 4, Y ₁～Y ₅, Q ₁, G ₁, G ₃, R ₁, and R ₂With X, the Y in the general formula (1) ₁～Y ₅, Q ₁, G ₁, G ₃, R ₁, and R ₂Implication respectively identical.

In the general formula (8), Q ₁Expression can have substituent phenyl maybe can have substituent pyridyl.X ₁, X ₂, X ₃, and X ₄Represent hydrogen atom or fluorine atom respectively independently.R ₁And R ₂Represent hydrogen atom or C1-C3 alkyl respectively independently.

Y ₁And Y ₅Represent halogen atom, C1-C3 halogenated alkoxy or C1-C3 haloalkyl respectively independently, Y ₂And Y ₄Represent hydrogen atom, halogen atom or C1-C4 alkyl, Y respectively independently ₃Expression C3-C4 haloalkyl.

Wherein, Y ₁And Y ₅When being halogen atom simultaneously, X ₁And X ₂In at least one side be fluorine atom.In addition, Y ₁Or Y ₅During for the C1-C3 halogenated alkoxy, X ₂Be fluorine atom.

The definition of the term that uses in the general formula of the present invention general formulas such as (1) has following illustrated implication respectively.

" halogen atom " expression fluorine atom, chlorine atom, bromine atoms or iodine atom.

The implication of the mark of " Ca-Cb (a, b represent the integer more than 1) " is: for example, " C1-C3 " expression carbonatoms is 1～3, and " C2-C6 " expression carbonatoms is 2～6, and " C1-C4 " expression carbonatoms is 1～4.

" n-" just representing, " i-" expression is different, and " s-" represents secondary, and " t-" represents uncle.

The alkyl that a straight chain shape such as " C1-C3 alkyl " among the present invention expression methyl, ethyl, n-propyl group, i-propyl group or a catenate carbonatoms are 1～3.

" C1-C3 haloalkyl " represents for example trifluoromethyl, pentafluoroethyl group, seven fluoro-n-propyl group, seven fluoro-i-propyl group, 2,2-two fluoro ethyls, 2, the 2-Dichloroethyl, 2,2, the 2-trifluoroethyl, the 2-fluoro ethyl, the 2-chloroethyl, the 2-bromotrifluoromethane, 2-iodine ethyl, 2,2,2-three chloroethyls, 2,2, the 2-three bromomethyl, 1,3-two fluoro-2-propyl group, 1,3-two chloro-2-propyl group, 1-chloro-3-fluoro-2-propyl group, 1,1,1-three fluoro-2-propyl group, 2,3,3,3-three fluoro-n-propyl group, 1,1,1,3,3,3-hexafluoro-2-propyl group, 1,1,1,3,3,3-hexafluoro-2-chloro-2-propyl group, 1,1,1,3,3,3-hexafluoro-2-bromo-2-propyl group, 1,1,2,3,3,3-hexafluoro-2-chloro-n-propyl group, 1,1,2,3,3,3-hexafluoro-2-bromo-n-propyl group, 1,1,2,3,3,3-hexafluoro-1-bromo-2-propyl group, 2,2,3,3,3-five fluoro-n-propyl group, 3-fluoro-n-propyl group, 3-chloro-n-propyl group, the alkyl that a straight chain shape that 3-bromo-n-propyl group etc. are replaced by halogen atom that can be identical or different more than 1 or a catenate carbonatoms are 1～3.

" C1-C4 alkyl " represents the alkyl of 1～4 of straight chain shape such as for example methyl, ethyl, n-propyl group, i-propyl group, n-butyl, s-butyl, t-butyl or a catenate carbonatoms.

" C1-C3 halogenated alkoxy " represents for example trifluoromethoxy, five fluorine oxyethyl groups, seven fluoro-n-propyl group oxygen bases, seven fluoro-i-propyl group oxygen bases, 2, the 2-difluoroethoxy, 2,2-two chloroethoxies, 2,2, the 2-trifluoro ethoxy, 2-fluorine oxyethyl group, the 2-chloroethoxy, the 2-bromine oxethyl, 2-iodine oxyethyl group, 2,2,2-three chloroethoxies, 2,2,2-three bromine oxethyls, 1,3-two fluoro-2-propyl group oxygen bases, 1,3-two chloro-2-propyl group oxygen bases, 1-chloro-3-fluoro-2-propyl group oxygen base, 1,1,1-three fluoro-2-propyl group oxygen bases, 2,3,3,3-three fluoro-n-propyl group oxygen bases, 1,1,1,3,3,3-hexafluoro-2-propyl group oxygen base, 1,1,1,3,3,3-hexafluoro-2-chloro-2-propyl group oxygen base, 1,1,1,3,3,3-hexafluoro-2-bromo-2-propyl group oxygen base, 1,1,2,3,3,3-hexafluoro-2-chloro-n-propyl group oxygen base, 1,1,2,3,3,3-hexafluoro-2-bromo-n-propyl group oxygen base, 1,1,2,3,3,3-hexafluoro-1-bromo-2-propyl group oxygen base, 2,2,3,3,3-five fluoro-n-propyl group oxygen bases, 3-fluoro-n-propyl group oxygen base, 3-chloro-n-propyl group oxygen base, the alkoxyl group that a straight chain shape that 3-bromo-n-propyl group oxygen base etc. are replaced by halogen atom that can be identical or different more than 1 or a catenate carbonatoms are 1～3.

" C3-C4 perfluoroalkyl " expression perfluor-n-propyl group, perfluor-i-propyl group, perfluor-n-butyl, perfluor-i-butyl, perfluor-s-butyl, perfluor-t-butyl etc. are the alkyl of 3～4 of the straight chain shape that replaced by fluorine atom of hydrogen atoms or catenate carbonatomss all.

" C1 haloalkyl " expression trifluoromethyl, 1, the methyl that 1-two fluoro-1-brooethyls etc. are replaced by halogen atom that can be identical or different more than 1.

" C1-C6 alkyl " represents the alkyl of 1～6 of straight chain shape such as for example methyl, ethyl, n-propyl group, i-propyl group, n-butyl, s-butyl, t-butyl, n-amyl group, 2-amyl group, neo-pentyl, 4-methyl-2-amyl group, n-hexyl, 3-methyl-n-amyl group or a catenate carbonatoms.

" C1-C6 haloalkyl " represents for example trifluoromethyl, pentafluoroethyl group, seven fluoro-n-propyl group, seven fluoro-i-propyl group, 2,2-two fluoro ethyls, 2, the 2-Dichloroethyl, 2,2, the 2-trifluoroethyl, the 2-fluoro ethyl, the 2-chloroethyl, the 2-bromotrifluoromethane, 2-iodine ethyl, 2,2,2-three chloroethyls, 2,2, the 2-three bromomethyl, 1,3-two fluoro-2-propyl group, 1,3-two chloro-2-propyl group, 1-chloro-3-fluoro-2-propyl group, 1,1,1-three fluoro-2-propyl group, 2,3,3,3-three fluoro-n-propyl group, 4,4,4-three fluoro-n-butyl, 1,1,1,3,3,3-hexafluoro-2-propyl group, 1,1,1,3,3,3-hexafluoro-2-chloro-2-propyl group, 1,1,1,3,3,3-hexafluoro-2-bromo-2-propyl group, 1,1,2,3,3,3-hexafluoro-2-chloro-n-propyl group, 1,1,2,3,3,3-hexafluoro-2-bromo-n-propyl group, 1,1,2,3,3,3-hexafluoro-1-bromo-2-propyl group, 2,2,3,3,3-five fluoro-n-propyl group, 3-fluoro-n-propyl group, 3-chloro-n-propyl group, 3-bromo-n-propyl group, 3,3,4,4,4-five fluoro-2-butyl, nine fluoro-n-butyl, nine fluoro-2-butyl, 5,5,5-three fluoro-n-amyl groups, 4,4,5,5,5-five fluoro-2-amyl groups, 3-chloro-n-amyl group, the alkyl that a straight chain shape that 4-bromo-2-amyl group etc. are replaced by halogen atom that can be identical or different more than 1 or a catenate carbonatoms are 1～6.

" C3-C9 cycloalkyl " represents that for example cyclopropyl, cyclobutyl, cyclopentyl, 2-methylcyclopentyl, 3-methylcyclopentyl, cyclohexyl, 2-methylcyclohexyl, 3-methylcyclohexyl, 4-methylcyclohexyl etc. have the cycloalkyl of 3～9 of the carbonatomss of ring texture.

The cycloalkyl that the carbonatoms with ring texture that " C3-C9 halogenated cycloalkyl " expression for example 2,2,3,3-ptfe ring butyl, 2-chlorine cyclohexyl, 4-chlorine cyclohexyl etc. are replaced by halogen atom that can be identical or different more than 1 is 3～9.

" C2-C6 alkenyl " represents to have in the carbochains such as vinyl, allyl group, crotyl, 3-butenyl for example the alkenyl of 2～6 of the carbonatomss of two keys.

" C2-C6 halogenated alkenyl " expression for example 3,3-two fluoro-2-propenyl, 3,3-two chloro-2-propenyl, 3,3-two bromo-2-propenyl, 2,3-two bromo-2-propenyl, 4, have the straight chain shape of two keys in the carbochain that 4-two fluoro-3-butenyls, 3,4,4-three bromo-3-butenyls etc. are replaced by halogen atom that can be identical or different more than 1 or prop up the alkenyl of 2～6 of catenate carbonatomss.

" C2-C6 alkynyl " represents to have in for example propargyl, ethyl acetylene-3-base, the ethyl acetylene-3-methyl-carbochains such as 3-base the alkynyl of 2～6 of triple-linked carbonatomss.

" C2-C6 halo alkynyl " represents for example fluorine ethynyl, chloroethene alkynyl, bromoacetylene base, 3,3,3-three fluoro-1-proyls, 3,3,3-three chloro-1-proyls, 3,3,3-three bromo-1-proyls, 4,4,4-three fluoro-ethyl acetylene bases, 4,4,4-three chloro-ethyl acetylene bases, 4,4, have the alkynyl of 2～6 of a triple-linked straight chain shape or catenate carbonatomss in the carbochain that 4-three bromo-ethyl acetylene bases etc. are replaced by halogen atom that can be identical or different more than 1.

" C1-C6 alkoxyl group " represents the alkoxyl group of 1～6 of straight chain shape such as methoxyl group for example, oxyethyl group, n-propyl group oxygen base, i-propyl group oxygen base, ring propoxy-, n-butoxy, s-butoxy, i-butoxy, t-butoxy, n-amyl group oxygen base, i-amyl group oxygen base, n-hexyl oxygen base, cyclohexyl oxygen base or a chain or cyclic carbonatoms.

" C1-C6 halogenated alkoxy " represents for example trifluoromethoxy, five fluorine oxyethyl groups, the 2-chloroethoxy, 2,2, the 2-trifluoro ethoxy, seven fluoro-n-propoxy-, seven fluoro-i-propoxy-, 1,1,1,3,3,3-hexafluoro-2-propoxy-, 3-fluoro-n-propoxy-, 1-chlorine ring propoxy-, 2-bromine ring propoxy-, 3,3,4,4,4-five fluoro-2-butoxy, nine fluoro-n-butoxy, nine fluoro-2-butoxy, 5,5,5-three fluoro-n-amyl group oxygen bases, 4,4,5,5,5-five fluoro-2-amyl group oxygen bases, 3-chloro-n-amyl group oxygen base, 4-bromo-2-amyl group oxygen base, 4-chlorobutyl oxygen base, the alkoxyl group that a straight chain shape that 2-iodo-n-propyl group oxygen base etc. are replaced by halogen atom that can be identical or different more than 1 or a chain or cyclic carbonatoms are 1～6.

" C1-C6 alkyl sulfenyl " represents the alkyl sulfenyl of 1～6 of straight chain shape such as methylthio group for example, ethylmercapto group, n-rosickyite base, i-rosickyite base, ring rosickyite base, n-butylthio, s-butylthio, i-butylthio, t-butylthio, n-penta sulfenyl, i-penta sulfenyl, the own sulfenyl of n-, hexamethylene sulfenyl or a chain or cyclic carbonatoms.

" C1-C6 haloalkyl sulfenyl " represents for example trifluoromethylthio, five fluorine ethylmercapto groups, 2-chloroethene sulfenyl, 2,2,2-trifluoro ethylmercapto group, seven fluoro-n-rosickyite bases, seven fluoro-i-rosickyite bases, 1,1,1,3,3,3-hexafluoro-2-rosickyite base, 3-fluoro-n-rosickyite base, 1-chlorine ring rosickyite base, 2-bromine ring rosickyite base, 3,3,4,4,4-five fluoro-2-butylthios, nine fluoro-n-butylthios, nine fluoro-2-butylthios, 5,5,5-three fluoro-n-penta sulfenyl, 4,4,5,5,5-five fluoro-2-penta sulfenyl, 3-chloro-n-penta sulfenyl, 4-bromo-2-penta sulfenyl, 4-neoprene sulfenyl, the alkyl sulfenyl that a straight chain shape that 2-iodo-n-rosickyite base etc. are replaced by halogen atom that can be identical or different more than 1 or a chain or cyclic carbonatoms are 1～6.

" C1-C6 alkyl sulphinyl " represents the alkyl sulphinyl of 1～6 of straight chain shape such as for example methylsulfinyl, ethyl sulfinyl, n-propyl group sulfinyl, i-propyl group sulfinyl, cyclopropyl sulfinyl, n-butyl sulfinyl, s-butyl sulfinyl, i-butyl sulfinyl, t-butyl sulfinyl, n-amyl group sulfinyl, i-amyl group sulfinyl, n-hexyl sulfinyl, cyclohexyl sulfinyl or a chain or cyclic carbonatoms.

" C1-C6 haloalkyl sulfinyl " represents for example trifluoromethyl sulphinyl base; the pentafluoroethyl group sulfinyl; 2-chloroethyl sulfinyl; 2; 2; 2-trifluoroethyl sulfinyl; seven fluoro-n-propyl group sulfinyls; seven fluoro-i-propyl group sulfinyls; 1; 1; 1; 3; 3; 3-hexafluoro-2-propyl group sulfinyl; 3-fluoro-n-propyl group sulfinyl; 1-chlorine cyclopropyl sulfinyl; 2-bromine cyclopropyl sulfinyl; 3; 3; 4,4,4-five fluoro-2-butyl sulfinyls; nine fluoro-n-butyl sulfinyls; nine fluoro-2-butyl sulfinyls; 5; 5; 5-three fluoro-n-amyl group sulfinyls; 4,4,5; 5,5-five fluoro-2-amyl group sulfinyls; 3-chloro-n-amyl group sulfinyl; 4-bromo-2-amyl group sulfinyl; 4-chlorobutyl sulfinyl; the alkyl sulphinyl that a straight chain shape that 2-iodo-n-propyl group sulfinyl etc. are replaced by halogen atom that can be identical or different more than 1 or a chain or cyclic carbonatoms are 1～6.

" C1-C6 alkyl sulphonyl " represents the alkyl sulphonyl of 1～6 of straight chain shape such as for example methyl sulphonyl, ethylsulfonyl, n-sulfonyl propyl base, i-sulfonyl propyl base, cyclopropyl alkylsulfonyl, n-butyl alkylsulfonyl, s-butyl alkylsulfonyl, i-butyl alkylsulfonyl, t-butyl alkylsulfonyl, n-amyl group alkylsulfonyl, i-amyl group alkylsulfonyl, n-hexyl alkylsulfonyl, cyclohexyl alkylsulfonyl or a chain or cyclic carbonatoms.

" C1-C6 halogenated alkyl sulfonyl " represents for example trifluoromethyl sulfonyl; the pentafluoroethyl group alkylsulfonyl; 2-chloroethyl alkylsulfonyl; 2; 2; 2-trifluoroethyl alkylsulfonyl; seven fluoro-n-sulfonyl propyl bases; seven fluoro-i-sulfonyl propyl bases; 1; 1; 1; 3; 3; 3-hexafluoro-2-sulfonyl propyl base; 3-fluoro-n-sulfonyl propyl base; 1-chlorine cyclopropyl alkylsulfonyl; 2-bromine cyclopropyl alkylsulfonyl; 3; 3; 4,4,4-five fluoro-2-butyl alkylsulfonyls; nine fluoro-n-butyl alkylsulfonyls; nine fluoro-2-butyl alkylsulfonyls; 5; 5; 5-three fluoro-n-amyl group alkylsulfonyls; 4,4,5; 5,5-five fluoro-2-amyl group alkylsulfonyls; 3-chloro-n-amyl group alkylsulfonyl; 4-bromo-2-amyl group alkylsulfonyl; 4-chlorobutyl alkylsulfonyl; the alkyl sulphonyl that a straight chain shape that 2-iodo-n-sulfonyl propyl base etc. are replaced by halogen atom that can be identical or different more than 1 or a chain or cyclic carbonatoms are 1～6.

" C1-C6 alkyl sulphonyl oxygen base " represents the alkyl sulphonyl oxygen base of 1～6 of straight chain shape such as methylsulfonyl oxygen base for example, ethylsulfonyl oxygen base, the n-third alkylsulfonyl oxygen base, the i-third alkylsulfonyl oxygen base, the ring third alkylsulfonyl oxygen base, n-fourth alkylsulfonyl oxygen base, s-fourth alkylsulfonyl oxygen base, i-fourth alkylsulfonyl oxygen base, t-fourth alkylsulfonyl oxygen base, n-penta alkylsulfonyl oxygen base, i-penta alkylsulfonyl oxygen base, the own alkylsulfonyl oxygen of n-base, hexamethylene alkylsulfonyl oxygen base or a chain or cyclic carbonatoms.

" C1-C6 halogenated alkyl sulfonyl oxygen base " represents for example trifyl oxygen base; five fluorine, the third alkylsulfonyl oxygen base; the 2-chlorine third alkylsulfonyl oxygen base; 2; 2; 2-trifluoropropyl alkylsulfonyl oxygen base; seven fluoro-n-, the third alkylsulfonyl oxygen base; seven fluoro-i-, the third alkylsulfonyl oxygen base; 1; 1; 1; 3; 3; 3-hexafluoro-2-third alkylsulfonyl oxygen base; the 3-fluoro-n-third alkylsulfonyl oxygen base; the 1-chlorine ring third alkylsulfonyl oxygen base; the 2-bromine ring third alkylsulfonyl oxygen base; 3; 3; 4,4,4-five fluoro-2-fourth alkylsulfonyl oxygen bases; nine fluoro-n-fourth alkylsulfonyl oxygen bases; nine fluoro-2-fourth alkylsulfonyl oxygen bases; 5; 5; 5-three fluoro-n-penta alkylsulfonyl oxygen base; 4,4,5; 5,5-five fluoro-2-penta alkylsulfonyl oxygen base; 3-chloro-n-penta alkylsulfonyl oxygen base; 4-bromo-2-penta alkylsulfonyl oxygen base; 4-neoprene alkylsulfonyl oxygen base; the alkyl sulphonyl oxygen base that a straight chain shape that the 2-iodo-n-third alkylsulfonyl oxygen base etc. are replaced by halogen atom that can be identical or different more than 1 or a chain or cyclic carbonatoms are 1～6.

" C2-C7 alkyl-carbonyl " represents the alkyl-carbonyl of 2～7 of straight chain shape such as for example ethanoyl, propionyl, i-propyl group carbonyl, cyclopropyl carbonyl, n-butyl carbonyl, s-butyl carbonyl, t-butyl carbonyl, n-amyl group carbonyl, 2-amyl group carbonyl, neo-pentyl carbonyl, cyclopentylcarbonyl or a chain or cyclic carbonatomss.

" C2-C7 halogenated alkyl carbonyl " represents for example trifluoroacetyl group; five fluorine propionyls; 2-chlorine propionyl; 2; 2; 2-trifluoropropyl acyl group; seven fluoro-n-propyl group carbonyls; seven fluoro-i-propyl group carbonyls; 1; 1; 1; 3,3,3-hexafluoro-2-propyl group carbonyl; 3-fluoro-n-propyl group carbonyl; 1-chlorine cyclopropyl carbonyl; 2-bromine cyclopropyl carbonyl; 3; 3; 4,4,4-five fluoro-2-butyl carbonyls; nine fluoro-n-butyl carbonyls; nine fluoro-2-butyl carbonyls; 5; 5; 5-three fluoro-n-amyl group carbonyls; 4,4,5; 5,5-five fluoro-2-amyl group carbonyls; 3-chloro-n-amyl group carbonyl; 4-bromo-2-amyl group carbonyl; 4-chlorobutyl carbonyl; the alkyl-carbonyl that a straight chain shape that 2-iodo-n-propyl group carbonyl etc. are replaced by halogen atom that can be identical or different more than 1 or a chain or cyclic carbonatoms are 2～7.

" C2-C7 alkyl-carbonyl oxygen base " represents the alkyl-carbonyl oxygen base of 2～7 of straight chain shape such as for example acetoxyl group, propionyloxy, i-propyl group ketonic oxygen base, cyclopropyl carbonyl oxygen base, n-butyl ketonic oxygen base, s-butyl ketonic oxygen base, t-butyl ketonic oxygen base, n-amyl group ketonic oxygen base, 2-amyl group ketonic oxygen base, neo-pentyl ketonic oxygen base, cyclopentylcarbonyl oxygen base or a chain or cyclic carbonatomss.

" C2-C7 halogenated alkyl carbonyl oxygen base " represents for example trifluoroacetyl oxygen base, five fluorine propionyloxies, 2-chlorine propionyloxy, 2,2,2-trifluoropropyl acyloxy, seven fluoro-n-propyl group ketonic oxygen bases, seven fluoro-i-propyl group ketonic oxygen bases, 1,1,1,3,3,3-hexafluoro-2-propyl group ketonic oxygen base, 3-fluoro-n-propyl group ketonic oxygen base, 1-chlorine cyclopropyl carbonyl oxygen base, 2-bromine cyclopropyl carbonyl oxygen base, 3,3,4,4,4-five fluoro-2-butyl ketonic oxygen bases, nine fluoro-n-butyl ketonic oxygen bases, nine fluoro-2-butyl ketonic oxygen bases, 5,5,5-three fluoro-n-amyl group ketonic oxygen bases, 4,4,5,5,5-five fluoro-2-amyl group ketonic oxygen bases, 3-chloro-n-amyl group ketonic oxygen base, 4-bromo-2-amyl group ketonic oxygen base, 4-chlorobutyl ketonic oxygen base, the alkyl-carbonyl oxygen base that a straight chain shape that 2-iodo-n-propyl group ketonic oxygen base etc. are replaced by halogen atom that can be identical or different more than 1 or a chain or cyclic carbonatoms are 2～7.

" C2-C7 alkoxy carbonyl " represents the alkoxy carbonyl of 2～7 of straight chain shape such as for example methoxycarbonyl, ethoxy carbonyl, isopropoxy carbonyl, ring propoxycarbonyl, n-butoxy carbonyl, s-butoxy carbonyl, t-butoxy carbonyl, n-amyl group oxygen base carbonyl, 2-amyl group oxygen base carbonyl, neo-pentyl oxygen base carbonyl, cyclopentyloxy carbonyl or a chain or cyclic carbonatomss.

" C2-C7 halo alkoxy carbonyl " represents for example trifluoromethoxy carbonyl, five fluorine ethoxy carbonyls, 2-chloroethoxy carbonyl, 2,2,2-trifluoro ethoxy carbonyl, seven fluoro-n-propoxycarbonyl, seven fluoro-i-propoxycarbonyl, 1,1,1,3,3,3-hexafluoro-2-propoxycarbonyl, 3-fluoro-n-propoxycarbonyl, 1-chlorine ring propoxycarbonyl, 2-bromine ring propoxycarbonyl, 3,3,4,4,4-five fluoro-2-butoxy carbonyls, nine fluoro-n-butoxy carbonyls, nine fluoro-2-butoxy carbonyls, 5,5,5-three fluoro-n-amyl group oxygen base carbonyls, 4,4,5,5,5-five fluoro-2-amyl group oxygen base carbonyls, 3-chloro-n-amyl group oxygen base carbonyl, 4-bromo-2-amyl group oxygen base carbonyl, 4-chlorobutyl oxygen base carbonyl, the alkoxy carbonyl that a straight chain shape that 2-iodo-n-propyl group oxygen base carbonyl etc. are replaced by halogen atom that can be identical or different more than 1 or a chain or cyclic carbonatoms are 2～7.

" C2-C7 alkyl-carbonyl-amino " represents the alkyl-carbonyl-amino of 2～7 of straight chain shape such as for example acetylamino, propionyl amino, n-propyl group carbonylamino, i-propyl group carbonylamino, cyclopropyl carbonyl amino, n-butyl carbonylamino, s-butyl carbonylamino, i-butyl carbonylamino, t-butyl carbonylamino, n-amyl group carbonylamino, i-amyl group carbonylamino, n-hexyl carbonylamino, cyclohexyl-carbonyl amino or a chain or cyclic carbonatomss.

" C2-C7 halogenated alkyl carbonyl amino " represents for example trifluoroacetyl group amino; five fluorine propionyl amino; 2-chlorine propionyl amino; 2; 2; 2-trifluoropropyl acyl amino; seven fluoro-n-propyl group carbonylaminos; seven fluoro-i-propyl group carbonylaminos; 1; 1; 1; 3; 3; 3-hexafluoro-2-propyl group carbonylamino; 3-fluoro-n-propyl group carbonylamino; 1-chlorine cyclopropyl carbonyl amino; 2-bromine cyclopropyl carbonyl amino; 3; 3; 4,4,4-five fluoro-2-butyl carbonylaminos; nine fluoro-n-butyl carbonylaminos; nine fluoro-2-butyl carbonylaminos; 5; 5; 5-three fluoro-n-amyl group carbonylaminos; 4,4,5; 5,5-five fluoro-2-amyl group carbonylaminos; 3-chloro-n-amyl group carbonylamino; 4-bromo-2-amyl group carbonylamino; 4-chlorobutyl carbonylamino; the alkyl-carbonyl-amino that a straight chain shape that 2-iodo-n-propyl group carbonylamino etc. are replaced by halogen atom that can be identical or different more than 1 or a chain or cyclic carbonatoms are 2～7.

" C2-C7 alkoxycarbonyl amino " represents for example methoxycarbonyl amino, ethoxy carbonyl amino, n-propyl group oxygen base carbonylamino, i-propyl group oxygen base carbonylamino, ring propoxycarbonyl amino, n-butoxy carbonyl amino, s-butoxy carbonyl amino, i-butoxy carbonyl amino, t-butoxy carbonyl amino, n-amyl group oxygen base carbonylamino, i-amyl group oxygen base carbonylamino, n-hexyl oxygen base carbonylamino, the alkoxycarbonyl amino that a straight chain shape such as cyclohexyl oxygen base carbonylamino or a chain or cyclic carbonatoms are 2～7.

" C2-C7 halo alkoxy carbonyl amino " represents for example trifluoromethyl oxygen base carbonylamino, five fluorine ethoxy carbonyl amino, 2-chloroethoxy carbonylamino, 2,2, the 2-trifluoro-ethoxy carbonyl-amino, seven fluoro-n-propyl group oxygen base carbonylaminos, seven fluoro-i-propyl group oxygen base carbonylaminos, 1,1,1,3,3,3-hexafluoro-2-propyl group oxygen base carbonylamino, 3-fluoro-n-propyl group oxygen base carbonylamino, 1-chlorine cyclopropyl oxygen base carbonylamino, 2-bromine cyclopropyl oxygen base carbonylamino, 3,3,4,4,4-five fluoro-2-butyl oxygen base carbonylaminos, nine fluoro-n-butyl oxygen base carbonylaminos, nine fluoro-2-butyl oxygen base carbonylaminos, 5,5,5-three fluoro-n-amyl group oxygen base carbonylaminos, 4,4,5,5,5-five fluoro-2-amyl group oxygen base carbonylaminos, 3-chloro-n-amyl group oxygen base carbonylamino, 4-bromo-2-amyl group oxygen base carbonylamino, 4-chlorobutyl oxygen base carbonylamino, the alkoxycarbonyl amino that a straight chain shape that 2-iodo-n-propyl group oxygen base carbonylamino etc. are replaced by halogen atom that can be identical or different more than 1 or a chain or cyclic carbonatoms are 2～7.

" C2-C7 alkoxy-carbonyl oxy " represents for example methoxycarbonyl oxygen base, ethoxy carbonyl oxygen base, n-propyl group oxygen base ketonic oxygen base, i-propyl group oxygen base ketonic oxygen base, ring propoxycarbonyl oxygen base, n-butoxy carbonyl oxygen base, s-butoxy carbonyl oxygen base, i-butoxy carbonyl oxygen base, t-butoxy carbonyl oxygen base, n-amyl group oxygen base ketonic oxygen base, i-amyl group oxygen base ketonic oxygen base, n-hexyl oxygen base ketonic oxygen base, the alkoxy-carbonyl oxy that a straight chain shape such as cyclohexyl oxygen base ketonic oxygen base or a chain or cyclic carbonatoms are 2～7.

" C2-C7 halo alkoxy carbonyl oxygen base " represents for example trifluoromethyl oxygen base ketonic oxygen base, five fluorine ethoxy carbonyl oxygen bases, 2-chloroethoxy ketonic oxygen base, 2,2,2-trifluoro ethoxy ketonic oxygen base, seven fluoro-n-propyl group oxygen base ketonic oxygen bases, seven fluoro-i-propyl group oxygen base ketonic oxygen bases, 1,1,1,3,3,3-hexafluoro-2-propyl group oxygen base ketonic oxygen base, 3-fluoro-n-propyl group oxygen base ketonic oxygen base, 1-chlorine cyclopropyl oxygen base ketonic oxygen base, 2-bromine cyclopropyl oxygen base ketonic oxygen base, 3,3,4,4,4-five fluoro-2-butyl oxygen base ketonic oxygen bases, nine fluoro-n-butyl oxygen base ketonic oxygen bases, nine fluoro-2-butyl oxygen base ketonic oxygen bases, 5,5,5-three fluoro-n-amyl group oxygen base ketonic oxygen bases, 4,4,5,5,5-five fluoro-2-amyl group oxygen base ketonic oxygen bases, 3-chloro-n-amyl group oxygen base ketonic oxygen base, 4-bromo-2-amyl group oxygen base ketonic oxygen base, 4-chlorobutyl oxygen base ketonic oxygen base, the alkoxy-carbonyl oxy that a straight chain shape that 2-iodo-n-propyl group oxygen base ketonic oxygen base etc. are replaced by halogen atom that can be identical or different more than 1 or a chain or cyclic carbonatoms are 2～7.

" C1-C6 alkylamino " represents the alkylamino of 1～6 of straight chain shape such as for example methylamino, dimethylamino, ethylamino, diethylamino, n-propyl group amino, i-propyl group amino, cyclopropyl amino, n-butyl amino, s-butyl amino, i-butyl amino, t-butyl amino, n-amyl group amino, i-amyl group amino, n-hexyl amino, cyclohexyl amino or a chain or cyclic carbonatoms.

" C1-C6 haloalkyl amino " represents for example trifluoromethyl amino, two (trifluoromethyl) amino, pentafluoroethyl group amino, two (pentafluoroethyl group) amino, the 2-chloroethyl amino, 2,2,2-trifluoroethyl amino, seven fluoro-n-propyl group amino, seven fluoro-i-propyl group amino, 1,1,1,3,3,3-hexafluoro-2-propyl group amino, 3-fluoro-n-propyl group amino, 1-chlorine cyclopropyl amino, 2-bromine cyclopropyl amino, 3,3,4,4,4-five fluoro-2-butyl amino, nine fluoro-n-butyl amino, nine fluoro-2-butyl amino, 5,5,5-three fluoro-n-amyl group amino, 4,4,5,5,5-five fluoro-2-amyl group amino, 3-chloro-n-amyl group amino, 4-bromo-2-amyl group amino, 4-chlorobutyl amino, the alkylamino that a straight chain shape that 2-iodo-n-propyl group amino etc. are replaced by halogen atom that can be identical or different more than 1 or a chain or cyclic carbonatoms are 1～6.

" C2-C6 alkenyl oxy " represents to have in the carbochains such as vinyl oxygen base, allyl group oxygen base, crotyl oxygen base, 3-butenyl oxygen base for example the alkenyl oxy of 2～6 of the carbonatomss of two keys.

" C2-C6 halogenated alkenyl oxy " expression for example 3,3-two fluoro-2-propenyl oxygen bases, 3,3-two chloro-2-propenyl oxygen bases, 3,3-two bromo-2-propenyl oxygen bases, 2,3-two bromo-2-propenyl oxygen bases, 4, have the straight chain shape of two keys in the carbochain that 4-two fluoro-3-butenyl oxygen bases, 3,4,4-three bromo-3-butenyl oxygen bases etc. are replaced by halogen atom that can be identical or different more than 1 or prop up the alkenyl oxy of 2～6 of catenate carbonatomss.

" C2-C6 alkynyloxy base " represents to have in propargyloxy for example, ethyl acetylene-3-base oxygen base, the ethyl acetylene-3-methyl-carbochains such as 3-base oxygen base the alkynyloxy base of 2～6 of triple-linked carbonatomss.

" C2-C6 halo alkynyloxy base " represents for example fluorine ethynyl oxygen base, chloroethene alkynyloxy base, bromoacetylene base oxygen base, 3,3,3-three fluoro-1-proyl oxygen bases, 3,3,3-three chloro-1-proyl oxygen bases, 3,3,3-three bromo-1-proyl oxygen bases, 4,4,4-three fluoro-ethyl acetylene base oxygen bases, 4,4,4-three chloro-ethyl acetylene base oxygen bases, 4,4, have the alkynyloxy base of 2～6 of a triple-linked straight chain shape or catenate carbonatomss in the carbochain that 4-three bromo-ethyl acetylene base oxygen bases etc. are replaced by halogen atom that can be identical or different more than 1.

" C3-C9 cycloalkyloxy " represents that for example cyclopropyl oxygen base, cyclobutyl oxygen base, cyclopentyloxy, 2-methylcyclopentyl oxygen base, 3-methylcyclopentyl oxygen base, cyclohexyl oxygen base, 2-methylcyclohexyl oxygen base, 3-methylcyclohexyl oxygen base, 4-methylcyclohexyl oxygen base etc. have the cycloalkyl oxy of 3～9 of the carbonatomss of ring texture.

" C3-C9 halo cycloalkyloxy " expression for example 2,2,3, the cycloalkyl oxy that the carbonatoms with ring texture that 3-ptfe ring butyl oxygen base, 2-chlorine cyclohexyl oxygen base, 4-chlorine cyclohexyl oxygen base etc. are replaced by halogen atom that can be identical or different more than 1 is 3～9.

" C3-C7 alkenyl carbonyl " represents to have in the carbochains such as vinyl carbonyl, allyl group carbonyl, crotyl carbonyl, 3-butenyl carbonyl for example the alkenyl carbonyl of 3～7 of the carbonatomss of two keys.

" C3-C7 halogenated alkenyl carbonyl " expression for example 3,3-two fluoro-2-propenyl carbonyls, 3,3-two chloro-2-propenyl carbonyls, 3,3-two bromo-2-propenyl carbonyls, 2,3-two bromo-2-propenyl carbonyls, 4, have the straight chain shape of two keys in the carbochain that 4-two fluoro-3-butenyl carbonyls, 3,4,4-three bromo-3-butenyl carbonyls etc. are replaced by halogen atom that can be identical or different more than 1 or prop up the alkenyl carbonyl of 3～7 of catenate carbonatomss.

The alkynyl carbonyl that has 3～7 of triple-linked carbonatomss in " C3-C7 alkynyl carbonyl " expression propargyl carbonyl, ethyl acetylene-3-base carbonyl, the ethyl acetylene-3-methyl-carbochains such as 3-base carbonyl.

" C3-C7 halo alkynyl carbonyl " represents for example fluorine ethynyl carbonyl, chloroethene alkynyl carbonyl, bromoacetylene base carbonyl, 3,3,3-three fluoro-1-proyl carbonyls, 3,3,3-three chloro-1-proyl carbonyls, 3,3,3-three bromo-1-proyl carbonyls, 4,4,4-three fluoro-ethyl acetylene base carbonyls, 4,4,4-three chloro-ethyl acetylene base carbonyls, 4,4, have the alkynyl carbonyl of 3～7 of a triple-linked straight chain shape or catenate carbonatomss in the carbochain that 4-three bromo-ethyl acetylene base carbonyls etc. are replaced by halogen atom that can be identical or different more than 1.

" C4-C10 naphthene base carbonyl " represents that for example cyclopropyl carbonyl, cyclobutyl carbonyl, cyclopentylcarbonyl, 2-methylcyclopentyl carbonyl, 3-methylcyclopentyl carbonyl, cyclohexyl-carbonyl, 2-methylcyclohexyl carbonyl, 3-methylcyclohexyl carbonyl, 4-methylcyclohexyl carbonyl etc. have the naphthene base carbonyl of 4～10 of the carbonatomss of ring texture.

" C4-C10 halogenated cycloalkyl carbonyl " expression for example 2,2,3, the naphthene base carbonyl that the carbonatoms with ring texture that 3-tetrafluoro cyclobutyl carbonyl, 2-chlorine cyclohexyl-carbonyl, 4-chlorine cyclohexyl-carbonyl etc. are replaced by halogen atom that can be identical or different more than 1 is 4～10.

The alkenyl oxy carbonyl that has 3～7 of the carbonatomss of two keys in the carbochains such as " C3-C7 alkenyl oxy carbonyl " expression vinyl oxygen base carbonyl, allyl group oxygen base carbonyl, crotyl oxygen base carbonyl, 3-butenyl oxygen base carbonyl.

" C3-C7 halogenated alkenyl oxy carbonyl " expression for example 3,3-two fluoro-2-propenyl oxygen base carbonyls, 3,3-two chloro-2-propenyl oxygen base carbonyls, 3,3-two bromo-2-propenyl oxygen base carbonyls, 2,3-two bromo-2-propenyl oxygen base carbonyls, 4,4-two fluoro-3-butenyl oxygen base carbonyls, 3,4, have the straight chain shape of two keys in the carbochain that 4-three bromo-3-butenyl oxygen base carbonyls etc. are replaced by halogen atom that can be identical or different more than 1 or prop up the alkenyl oxy carbonyl of 3～7 of catenate carbonatomss.

" C3-C7 alkynyloxy base carbonyl " expression for example has the alkynyloxy base carbonyl of 3～7 of triple-linked carbonatomss in propargyloxy carbonyl, ethyl acetylene-3-base oxygen base carbonyl, the ethyl acetylene-3-methyl-carbochains such as 3-base oxygen base carbonyl.

" C3-C7 halo alkynyloxy base carbonyl " represents for example fluorine ethynyl oxygen base carbonyl, chloroethene alkynyloxy base carbonyl, bromoacetylene base oxygen base carbonyl, 3,3,3-three fluoro-1-proyl oxygen base carbonyls, 3,3,3-three chloro-1-proyl oxygen base carbonyls, 3,3,3-three bromo-1-proyl oxygen base carbonyls, 4,4,4-three fluoro-ethyl acetylene base oxygen base carbonyls, 4,4,4-three chloro-ethyl acetylene base oxygen base carbonyls, 4,4, have the alkynyloxy base carbonyl of 3～7 of a triple-linked straight chain shape or catenate carbonatomss in the carbochain that 4-three bromo-ethyl acetylene base oxygen base carbonyls etc. are replaced by halogen atom that can be identical or different more than 1.

" C4-C10 cycloalkyl oxy carbonyl " represents that for example cyclopropyl oxygen base carbonyl, cyclobutyl oxygen base carbonyl, cyclopentyloxy carbonyl, 2-methylcyclopentyl oxygen base carbonyl, 3-methylcyclopentyl oxygen base carbonyl, cyclohexyl oxygen base carbonyl, 2-methylcyclohexyl oxygen base carbonyl, 3-methylcyclohexyl oxygen base carbonyl, 4-methylcyclohexyl oxygen base carbonyl etc. have the cycloalkyl oxy carbonyl of 4～10 of the carbonatomss of ring texture.

" C4-C10 halogenated cycloalkyl oxygen base carbonyl " expression for example 2,2,3, the cycloalkyl oxy carbonyl that the carbonatoms with ring texture that 3-ptfe ring butyl oxygen base carbonyl, 2-chlorine cyclohexyl oxygen base carbonyl, 4-chlorine cyclohexyl oxygen base carbonyl etc. are replaced by halogen atom that can be identical or different more than 1 is 4～10.

" C2-C6 alkenyl amino " represents to have in the carbochains such as vinyl amino, allyl amino, crotyl amino, 3-butenyl amino for example the alkenyl amino of 2～6 of the carbonatomss of two keys.

" C2-C6 halogenated alkenyl amino " expression 3,3-two fluoro-2-propenyl amino, 3,3-two chloro-2-propenyl amino, 3,3-two bromo-2-propenyl amino, 2,3-two bromo-2-propenyl amino, 4, have the straight chain shape of two keys in the carbochain that 4-two fluoro-3-butenyl amino, 3,4,4-three bromo-3-butenyl amino etc. are replaced by halogen atom that can be identical or different more than 1 or prop up the alkenyl amino of 2～6 of catenate carbonatomss.

" C2-C6 alkynyl amino " represents propargyl amino for example, ethyl acetylene-3-base is amino, have the alkynyl amino of 2～6 of triple-linked carbonatomss in ethyl acetylene-3-methyl-carbochains such as 3-base amino.

" C2-C6 halo alkynyl amino " represents for example fluorine ethynyl amino, chloroethene alkynyl amino, bromoacetylene base amino, 3,3,3-three fluoro-1-proyl amino, 3,3,3-three chloro-1-proyl amino, 3,3,3-three bromo-1-proyl amino, 4,4,4-three fluoro-ethyl acetylene base amino, 4,4,4-three chloro-ethyl acetylene base amino, 4,4, have the alkynyl amino of 2～6 of a triple-linked straight chain shape or catenate carbonatomss in the carbochain that 4-three bromo-ethyl acetylene base amino etc. are replaced by halogen atom that can be identical or different more than 1.

" C3-C9 cycloalkyl amino " represents that for example cyclopropyl amino, cyclobutyl amino, cyclopentyl amino, 2-methylcyclopentyl amino, 3-methylcyclopentyl amino, cyclohexyl amino, 2-methylcyclohexyl amino, 3-methylcyclohexyl amino, 4-methylcyclohexyl amino etc. have the cycloalkyl amino of 3～9 of the carbonatomss of ring texture.

" C3-C9 halogenated cycloalkyl amino " expression for example 2,2,3, the cycloalkyl amino that the carbonatoms with ring texture that 3-ptfe ring butyl amino, 2-chlorine cyclohexyl amino, 4-chlorine cyclohexyl amino etc. are replaced by halogen atom that can be identical or different more than 1 is 3～9.

" C2-C7 alkyl amino-carbonyl " represents the alkyl amino-carbonyl of 2～7 of straight chain shape such as for example methylamino carbonyl, ethylamino carbonyl, n-propyl group aminocarboxyl, i-propyl group aminocarboxyl, n-butyl aminocarboxyl, s-butyl aminocarboxyl, t-butyl aminocarboxyl, n-amyl group aminocarboxyl, 2-amyl group aminocarboxyl, neo-pentyl aminocarboxyl, 4-methyl-2-amyl group aminocarboxyl, n-hexyl aminocarboxyl, 3-methyl-n-amyl group aminocarboxyl or catenate carbonatomss.

" C2-C7 haloalkyl aminocarboxyl " represents for example trifluoromethyl aminocarboxyl, the pentafluoroethyl group aminocarboxyl, seven fluoro-n-propyl group aminocarboxyls, seven fluoro-i-propyl group aminocarboxyls, 2,2-difluoro ethylamino carbonyl, 2,2-Dichloroethyl aminocarboxyl, 2,2,2-trifluoroethyl aminocarboxyl, 2-fluoro ethyl aminocarboxyl, 2-chloroethyl amino carbonyl, 2-bromotrifluoromethane aminocarboxyl, 2-iodine ethylamino carbonyl, 2,2,2-three chloroethyl amino carbonyls, 2,2,2-three bromomethyl aminocarboxyl, 1,3-two fluoro-2-propyl group aminocarboxyls, 1,3-two chloro-2-propyl group aminocarboxyls, 1-chloro-3-fluoro-2-propyl group aminocarboxyl, 1,1,1-three fluoro-2-propyl group aminocarboxyls, 2,3,3,3-three fluoro-n-propyl group aminocarboxyls, 4,4,4-three fluoro-n-butyl aminocarboxyls, 1,1,1,3,3,3-hexafluoro-2-propyl group aminocarboxyl, 1,1,1,3,3,3-hexafluoro-2-chloro-2-propyl group aminocarboxyl, 1,1,1,3,3,3-hexafluoro-2-bromo-2-propyl group aminocarboxyl, 1,1,2,3,3,3-hexafluoro-2-chloro-n-propyl group aminocarboxyl, 1,1,2,3,3,3-hexafluoro-2-bromo-n-propyl group aminocarboxyl, 1,1,2,3,3,3-hexafluoro-1-bromo-2-propyl group aminocarboxyl, 2,2,3,3,3-five fluoro-n-propyl group aminocarboxyls, 3-fluoro-n-propyl group aminocarboxyl, 3-chloro-n-propyl group aminocarboxyl, 3-bromo-n-propyl group aminocarboxyl, 3,3,4,4,4-five fluoro-2-butyl aminocarboxyls, nine fluoro-n-butyl aminocarboxyls, nine fluoro-2-butyl aminocarboxyls, 5,5,5-three fluoro-n-amyl group aminocarboxyls, 4,4,5,5,5-five fluoro-2-amyl group aminocarboxyls, 3-chloro-n-amyl group aminocarboxyl, the alkyl amino-carbonyl that a straight chain shape that 4-bromo-2-amyl group aminocarboxyl etc. are replaced by halogen atom that can be identical or different more than 1 or a catenate carbonatoms are 2～7.

" C3-C7 alkenyl amino carbonyl " represents to have in the carbochains such as vinyl aminocarboxyl, allyl amino carbonyl, crotyl aminocarboxyl, 3-butenyl aminocarboxyl for example the alkenyl amino carbonyl of 3～7 of the carbonatomss of two keys.

" C3-C7 halogenated alkenyl aminocarboxyl " expression for example 3,3-two fluoro-2-propenyl aminocarboxyls, 3,3-two chloro-2-propenyl aminocarboxyls, 3,3-two bromo-2-propenyl aminocarboxyls, 2,3-two bromo-2-propenyl aminocarboxyls, 4,4-two fluoro-3-butenyl aminocarboxyls, 3,4, have the straight chain shape of two keys in the carbochain that 4-three bromo-3-butenyl aminocarboxyls etc. are replaced by halogen atom that can be identical or different more than 1 or prop up the alkenyl amino carbonyl of 3～7 of catenate carbonatomss.

" C3-C7 alkynyl aminocarboxyl " represents to have in propargyl aminocarboxyl for example, ethyl acetylene-3-base aminocarboxyl, the ethyl acetylene-3-methyl-carbochains such as 3-base aminocarboxyl the alkynyl aminocarboxyl of 3～7 of triple-linked carbonatomss.

" C3-C7 halo alkynyl aminocarboxyl " represents for example fluorine ethynyl aminocarboxyl, chloroethene alkynyl aminocarboxyl, bromoacetylene base aminocarboxyl, 3,3,3-three fluoro-1-proyl aminocarboxyls, 3,3,3-three chloro-1-proyl aminocarboxyls, 3,3,3-three bromo-1-proyl aminocarboxyls, 4,4,4-three fluoro-ethyl acetylene base aminocarboxyls, 4,4,4-three chloro-ethyl acetylene base aminocarboxyls, 4,4, have the alkynyl aminocarboxyl of 3～7 of a triple-linked straight chain shape or catenate carbonatomss in the carbochain that 4-three bromo-ethyl acetylene base aminocarboxyls etc. are replaced by halogen atom that can be identical or different more than 1.

" C4-C10 cycloalkyl amino carbonyl " represents that for example cyclopropyl aminocarboxyl, cyclobutyl aminocarboxyl, cyclopentyl aminocarboxyl, 2-methylcyclopentyl aminocarboxyl, 3-methylcyclopentyl aminocarboxyl, cyclohexyl aminocarboxyl, 2-methylcyclohexyl aminocarboxyl, 3-methylcyclohexyl aminocarboxyl, 4-methylcyclohexyl aminocarboxyl etc. have the cycloalkyl amino carbonyl of 4～10 of the carbonatomss of ring texture.

" C4-C10 halogenated cycloalkyl aminocarboxyl " expression for example 2,3, the cycloalkyl amino carbonyl that the carbonatoms with ring texture that 3-ptfe ring butyl aminocarboxyl, 2-chlorine cyclohexyl aminocarboxyl, 4-chlorine cyclohexyl aminocarboxyl etc. are replaced by halogen atom that can be identical or different more than 1 is 4～10.

" aryl " represents for example monocycle or Ppolynuclear aromatic alkyl such as phenyl or naphthyl.

" aryl carbonyl oxygen base " represents for example aryl carbonyl oxygen base such as phenylcarbonyl group oxygen base, naphthyl carbonyl oxygen base.

" aryl-amino-carbonyl " represents for example aryl-amino-carbonyl such as phenylcarbonyl group amino, naphthyl carbonyl amino.

R ₁And R ₂In the straight chain shape that do not have to replace of " can have substituent C1-C6 alkyl " expression, a chain or the alkyl of 1～6 of cyclic carbonatoms, or by nitro, can have substituent phenyl and can have the straight chain shape, a chain of at least a kind of replacement in the substituent unsaturated heterocycle base or the alkyl of 1～6 of cyclic carbonatoms.Need to prove that substituting group is 2 when above, above-mentioned substituting group can be the same or different.

R ₁And R ₂In the straight chain shape that only replaced of " can have substituent C1-C6 haloalkyl " expression, a chain by 1 above halogen atom or the alkyl of 1～6 of cyclic carbonatoms, or except that 1 above halogen atom, also by nitro, can have substituent phenyl and can have the straight chain shape, chain of at least a kind of replacement in the substituent unsaturated heterocycle base or the alkyl of 1～6 of cyclic carbonatoms.

R ₁And R ₂In the straight chain shape that do not have to replace of " can have substituent C2-C6 alkenyl " expression, a chain or the alkenyl of 2～6 of cyclic carbonatomss, or by nitro, can have substituent phenyl and can have the straight chain shape, a chain of at least a kind of replacement in the substituent unsaturated heterocycle base or the alkenyl of 2～6 of cyclic carbonatomss.Need to prove that substituting group is 2 when above, above-mentioned substituting group can be the same or different.

R ₁And R ₂In the straight chain shape that only replaced of " can have substituent C2-C6 halogenated alkenyl " expression, a chain by 1 above halogen atom or the alkenyl of 2～6 of cyclic carbonatomss, or except that 1 above halogen atom, also by nitro, can have substituent phenyl and can have the straight chain shape, chain of at least a kind of replacement in the substituent unsaturated heterocycle base or the alkenyl of 2～6 of cyclic carbonatomss.

R ₁And R ₂In the straight chain shape that do not have to replace of " can have substituent C2-C6 alkynyl " expression, a chain or the alkynyl of 2～6 of cyclic carbonatomss, or by nitro, can have substituent phenyl and can have the straight chain shape, a chain of at least a kind of replacement in the substituent unsaturated heterocycle base or the alkynyl of 2～6 of cyclic carbonatomss.Need to prove that substituting group is 2 when above, above-mentioned substituting group can be the same or different.

R ₁And R ₂In the straight chain shape that only replaced of " can have substituent C2-C6 halo alkynyl " expression, a chain by 1 above halogen atom or the alkynyl of 2～6 of cyclic carbonatomss, or except that 1 above halogen atom, also by nitro, can have substituent phenyl and can have the straight chain shape, chain of at least a kind of replacement in the substituent unsaturated heterocycle base or the alkynyl of 2～6 of cyclic carbonatomss.

Need to prove that above-mentioned each substituting group further can have substituting group among the present invention under possible situation, as described below as its substituent example.

Described substituting group is the substituting group more than 1 that is selected from the following radicals; described group is: halogen atom; the C1-C6 alkyl; the C1-C6 haloalkyl; the C3-C9 cycloalkyl; the C3-C9 halogenated cycloalkyl; the C2-C6 alkenyl; the C2-C6 halogenated alkenyl; the C2-C6 alkynyl; C2-C6 halo alkynyl; the C1-C6 alkoxyl group; the C1-C6 halogenated alkoxy; C1-C6 alkyl sulfenyl; C1-C6 haloalkyl sulfenyl; the C1-C6 alkyl sulphinyl; C1-C6 haloalkyl sulfinyl; the C1-C6 alkyl sulphonyl; the C1-C6 halogenated alkyl sulfonyl; the C2-C7 alkyl-carbonyl; the C2-C7 halogenated alkyl carbonyl; C2-C7 alkyl-carbonyl oxygen base; C2-C7 halogenated alkyl carbonyl oxygen base; C1-C6 alkyl sulphonyl oxygen base; C1-C6 halogenated alkyl sulfonyl oxygen base; the C2-C7 alkoxy carbonyl; the C2-C7 halo alkoxy carbonyl; the C2-C7 alkyl-carbonyl-amino; C2-C7 halogenated alkyl carbonyl amino; the C2-C7 alkoxycarbonyl amino; C2-C7 halo alkoxy carbonyl amino; the C2-C7 alkyl amino-carbonyl; C2-C7 haloalkyl aminocarboxyl; the C1-C6 alkylamino; C1-C6 haloalkyl amino; the C2-C6 alkenyl amino; C2-C6 halogenated alkenyl amino; C2-C6 alkynyl amino; C2-C6 halo alkynyl amino; the C3-C9 cycloalkyl amino; C3-C9 halogenated cycloalkyl amino; C3-C7 alkenyl amino carbonyl; C3-C7 halogenated alkenyl aminocarboxyl; C3-C7 alkynyl aminocarboxyl; C3-C7 halo alkynyl aminocarboxyl; C4-C10 cycloalkyl amino carbonyl; C4-C10 halogenated cycloalkyl aminocarboxyl; amino; formamyl; sulfamyl; cyano group; nitro; hydroxyl; carboxyl; Pentafluorosulfanyl; can have substituent phenyl; can have substituent heterocyclic radical; can have substituent benzyl; can have substituent phenylcarbonyl group; and can have substituent phenyl amino; when having 2 above substituting groups, each substituting group can be the same or different.

General formula of the present invention (1), general formula (7), and the compound of general formula expressions such as (8) in its structural formula, contain one or more unsymmetrical carbons or asymmetric center sometimes, sometimes there is the optical isomer more than 2 kinds, each optical isomer and also all be included in the present invention with the mixture that arbitrary proportion contains them.In addition, general formula of the present invention (1), general formula (7), and the compound of general formula (8) expression of etc.ing in its structural formula, exist the geometrical isomer more than 2 kinds from carbon-to-carbon double bond, each geometrical isomer to reach the mixture that contains them with arbitrary proportion sometimes also all to be included in the present invention.

The preferred substituents of the substituting group in the amide derivatives of general formula of the present invention (1) expression etc. or the combination of atom are as described below.

Be preferably-C (=G as T ₁)-Q ₁As G ₁Be preferably Sauerstoffatom; As Q ₁Be preferably and have substituent phenyl, maybe can have substituent pyridyl; As Q ₁More preferably phenyl or pyridyl, described phenyl or pyridyl have be selected from halogen atom, C1 haloalkyl, nitro, and cyano group in the substituting group more than 1, when having 2 above substituting groups, each substituting group can be the same or different.

As G ₃Be preferably Sauerstoffatom.

As R ₁Be preferably hydrogen atom or C1-C3 alkyl.

As R ₂Be preferably hydrogen atom.

Be preferably carbon atom as A, be preferably the non-metallic atom group that forms phenyl ring with 2 carbon atoms of A and A bonding as K.

Be preferably hydrogen atom, halogen atom or cyano group as X, more preferably hydrogen atom, fluorine atom or cyano group.

N as X during for substituting group except that hydrogen atom is preferably 0,1 or 2.

As Y ₁Be preferably halogen atom or C1-C3 haloalkyl.

As Y ₅Be preferably the C1-C3 haloalkyl.

As Y ₂And Y ₄Be preferably hydrogen atom, halogen atom or C1-C4 alkyl, more preferably hydrogen atom.

As Y ₃Be preferably the C2-C5 haloalkyl, more preferably the C2-C4 perfluoroalkyl.

In addition, the combination of the preferred substituents of the substituting group in the amide derivatives of general formula (8) expression etc. or atom is as described below.

As Q ₁Be preferably phenyl or pyridyl, described phenyl or pyridyl have be selected from halogen atom, C1 haloalkyl, nitro, and cyano group in the substituting group more than 1, when having 2 above substituting groups, each substituting group can be the same or different.

As R ₁Be preferably hydrogen atom or C1-C3 alkyl.

As R ₂Be preferably hydrogen atom.

As X ₁, and X ₂Be preferably hydrogen atom or fluorine atom, as X ₃, X ₄Be preferably hydrogen atom.

As Y ₁, and Y ₅Be preferably halogen atom or C1-C3 haloalkyl.As Y ₂, and Y ₄Be preferably hydrogen atom.As Y ₃Be preferably the C3-C4 perfluoroalkyl.

Below provide the representative preparation method of compound of the present invention, but the preparation method of amide derivatives of the present invention is not limited to preparation method shown below.

In the general formula shown in the following preparation method, A, K, X, n, R ₁, R ₂, T, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅A, K, X, n, R in expression and the above-mentioned general formula (1) ₁, R ₂, T, G ₃, Y ₁, Y ₂, Y ₃, Y ₄, and Y ₅Identical respectively implication.LG represents that halogen atom, hydroxyl etc. have the functional group of the ability of leaving away, and Hal represents chlorine atom or bromine atoms, Xa, Xb, and Xc represent chlorine atom, bromine atoms or iodine atom.

＜preparation method 1 〉

1-(i): general formula (21)+general formula (22) → general formula (23)

General formula (21)+general formula (22) → general formula (28)

The nitryl aromatic family carboxylic acid derivative with leavings group of general formula (21) expression and the aromatic amine derivative of general formula (22) expression are reacted in appropriate solvent or under the non-solvent, can prepare the nitryl aromatic family carboxylic acid amide derivative of general formula (23) or general formula (28) expression thus.Also can use suitable alkali in this step.

As solvent, do not get final product so long as significantly do not suppress the solvent that this reaction carries out.For example can enumerate halogenated hydrocarbon, ether, dioxane, tetrahydrofuran (THF)s, 1 such as water, benzene,toluene,xylene etc. are aromatic hydrocarbon based, methylene dichloride, chloroform, tetracol phenixin, nitriles, 1 such as amidess such as ketones such as alcohols such as ester class, methyl alcohol, ethanol, acetone, methyl iso-butyl ketone (MIBK), pimelinketone, dimethyl formamide, N,N-DIMETHYLACETAMIDE, acetonitrile such as chains such as 2-glycol dimethyl ether or ring-type ethers, ethyl acetate, butylacetate, 3-dimethyl-inert solvents such as 2-imidazolone.Above-mentioned solvent can use separately or be mixed with two or more.

In addition, as alkali, can enumerate lithium amide classes such as alkali metal alcoholate class, lithium diisopropylamines such as hydrogenated alkali metal salt, sodium methylate, sodium ethylates such as phosphoric acid salts such as carbonates such as alkali hydroxide metal species, sodium bicarbonate, salt of wormwood, dipotassium hydrogen phosphate, tertiary sodium phosphate, sodium hydrides such as organic bases, sodium hydroxide, potassium hydroxide such as triethylamine, three-n-butylamine, pyridine, 4-dimethylaminopyridine etc.

Above-mentioned alkali can be suitably selection in the scope of 0.01～5 times of molar equivalent at the compound with respect to general formula (21) expression.

Temperature of reaction can suitably be selected to the scope of the reflux temperature of solvent for use at-20 ℃.Reaction times can suitably be selected in several minutes to 96 hours scope in addition.

In the compound of general formula (21) expression, aromatic series etheride derivative can easily adopt and use the ordinary method of halogenating agent to be prepared by aromatic carboxylic acid.As halogenating agent, can enumerate for example halogenating agents such as thionyl chloride, thionyl bromide, phosphorus oxychloride, oxalyl chloride, phosphorus trichloride.

On the other hand, can not use halogenating agent ground by the compound general formula (23) of nitryl aromatic family carboxylic acid derivative and general formula (22) expression or the compound of general formula (28) expression.As this method, can enumerate for example method of the middle record of Chem.Ber.788 page or leaf (1970).Particularly, additives such as suitable use I-hydroxybenzotriazole be can enumerate, and N, the method for N '-condensing agents such as dicyclohexylcarbodiimide used.As other condensing agents that use this moment, can enumerate 1-ethyl-3-(3-dimethylaminopropyl) carbodiimide, 1,1 '-carbonyl is two-the 1H-imidazoles etc.

In addition, as the additive method of the compound for preparing the expression of general formula (23) or general formula (28), also can enumerate the mixed anhydride method of using the chloro-formic ester class.For example can enumerate the method for record in the J.Am.Chem.Soc.5012 page or leaf (1967), can prepare the compound of general formula (23) or general formula (28) expression.Isobutyl chlorocarbonate, isopropyl chlorocarbonate etc. can be enumerated as the chloro-formic ester class that use this moment, outside the dechlorination formate ester, diethyl ethanoyl chlorine, pivaloyl chlorine etc. can also be enumerated.

Use the method for condensing agent and solvent, temperature of reaction, the reaction times that mixed anhydride method all is not limited to above-mentioned document record.As solvent, the inert solvent that suitably uses not remarkable inhibited reaction to carry out gets final product.Temperature of reaction, reaction times are also as long as suitably select according to the carrying out of reaction in addition.

1-is (ii): general formula (23) → general formula (24)

General formula (28) → general formula (29)

The aromatic carboxylic acid amide derivatives with nitro of general formula (23) or general formula (28) expression can pass through reduction reaction, is derivatized to the amino aromatic carboxylic acid amide derivatives that has of general formula (24) or general formula (29) expression.Can enumerate the method for using hydrogenation reaction and the method for using metallic compound (for example, tin protochloride (anhydride), iron powder, zinc powder etc.) as reduction reaction.

The former method can be in appropriate solvent in the presence of catalyzer, and normal pressure descends or add to depress under nitrogen atmosphere to react.As catalyzer, can enumerate nickel catalyzators such as palladium catalyst, Raney nickel, cobalt catalyst, ruthenium catalyst, rhodium catalyst, platinum catalysts etc. such as palladium-carbon, as solvent, can enumerate chain or ester classes such as ring-type ethers, ethyl acetate such as alcohols such as water, methyl alcohol, ethanol, benzene, toluene etc. are aromatic hydrocarbon based, ether, dioxane, tetrahydrofuran (THF).Pressure is suitably selected to get final product at-20 ℃ to the scope of the reflux temperature of solvent for use in 0.1～10MPa, temperature of reaction.Reaction times can suitably be selected to get final product in several minutes to 96 hours scope in addition.The compound that can prepare general formula (24) or general formula (29) thus efficiently.

As the latter's method, can enumerate according to the condition of putting down in writing among " Organic Syntheses " Coll.Vol.IIIP.453, use the method for tin protochloride (anhydride) as metallic compound.

1-is (iii): general formula (24)+general formula (26) → general formula (25)

Aromatic amine derivative by making general formula (24) expression and the carboxylic acid derivative of general formula (26) expression or the carbonic acid ester derivative with leavings group react in appropriate solvent, can prepare aromatic carboxylic acid acid amides or carbamate derivatives that general formula (25) is represented.Suitable alkali or solvent can be used in this step,, the material of enumerating among the 1-(i) can be used as this alkali or solvent.Temperature of reaction, reaction times etc. are also as shown in 1-(i).

In the general formula (26), carboxylic acid chloride (carboxylic acid chloride) derivative can easily be prepared by carboxylic acid derivative by the ordinary method of using halogenating agent.As halogenating agent, as shown in 1-(i).

Do not use halogenating agent in addition but, can be prepared according to the method for enumerating among the 1-(i) by the method for the compound of compound general formula (25) expression of carboxylic acid derivative (26) and general formula (24) expression.

1-is (iv): general formula (25)+general formula (27) → general formula (1)

The compound with leavings group such as halogen of amide compound that can be by making general formula (25) expression and general formula (27) expression reacts the The compounds of this invention that preparation general formula (1) is represented in solvent or under the non-solvent.Suitable alkali or solvent can be used in this step,, the material of enumerating among the 1-(i) can be used as its alkali or solvent.Temperature of reaction, reaction times etc. are also as shown in 1-(i).

1-(v): general formula (28)+general formula (30) → general formula (23)

Amide compound that can be by making general formula (28) expression, in solvent or under the non-solvent, react the compound of preparation general formula (23) expression with the compound with leavings group such as halogen of general formula (30) expression.Suitable alkali or solvent can be used in this step,, the material of in 1-(i), enumerating can be used as this alkali or solvent.Temperature of reaction, reaction times etc. are also as shown in 1-(i).

1-(vi): general formula (29) → general formula (31)

(method A)

The compound of general formula (29) expression is reacted with aldehydes or ketone in solvent, and add catalyzer, under nitrogen atmosphere, react, prepare the compound of general formula (31) expression thus.

As solvent, do not get final product so long as significantly do not suppress the solvent that this reaction carries out, can enumerate for example hexane, hexanaphthene, aliphatic hydrocarbons such as methylcyclohexane, benzene, dimethylbenzene, toluene etc. are aromatic hydrocarbon based, methylene dichloride, chloroform, tetracol phenixin, 1, halogenated hydrocarbons such as 2-ethylene dichloride, ether, dioxane, tetrahydrofuran (THF), 1, ethers such as 2-glycol dimethyl ether, dimethyl formamide, amidess such as N,N-DIMETHYLACETAMIDE, acetonitrile, nitriles such as propionitrile, acetone, methyl iso-butyl ketone (MIBK), pimelinketone, ketones such as methyl ethyl ketone, ethyl acetate, ester classes such as butylacetate, 1,3-dimethyl-2-imidazolone, tetramethylene sulfone, dimethyl sulfoxide (DMSO), methyl alcohol, alcohols such as ethanol, the water equal solvent, above-mentioned solvent can use separately or be mixed with two or more.

As catalyzer, can enumerate nickel catalyzator classes such as palladium catalyst class, Raney nickels such as palladium-carbon, palladium hydroxide-carbon, cobalt catalyst class, platinum catalyst class, ruthenium catalyst class, rhodium catalyst class etc.

As aldehydes, can enumerate for example aldehydes such as formaldehyde, acetaldehyde, propionic aldehyde, trifluoro acetaldehyde, difluoro acetaldehyde, fluorine acetaldehyde, monochloroacetaldehyde, dichloro acetaldehyde, trichoro-aldehyde, bromoacetaldehyde.

As ketone, can enumerate for example ketones such as acetone, perfluoro acetone, methyl ethyl ketone.

Reaction pressure can be distinguished suitably selection in the scope of 1 air pressure to 100 air pressure.Temperature of reaction can suitably be selected to the scope of the reflux temperature of solvent for use at-20 ℃.Reaction times can suitably be selected in several minutes to 96 hours scope in addition.

(method B)

The compound of general formula (29) expression is reacted with aldehydes or ketone in solvent, handle, can prepare the compound of general formula (31) expression by reductive agent.

As solvent, do not get final product so long as significantly do not suppress the solvent that this reaction carries out, can enumerate for example hexane, hexanaphthene, aliphatic hydrocarbons such as methylcyclohexane, benzene, dimethylbenzene, toluene etc. are aromatic hydrocarbon based, methylene dichloride, chloroform, tetracol phenixin, 1, halogenated hydrocarbons such as 2-ethylene dichloride, ether, dioxane, tetrahydrofuran (THF), 1, ethers such as 2-glycol dimethyl ether, dimethyl formamide, amidess such as N,N-DIMETHYLACETAMIDE, acetonitrile, nitriles such as propionitrile, acetone, methyl iso-butyl ketone (MIBK), pimelinketone, ketones such as methyl ethyl ketone, ethyl acetate, ester classes such as butylacetate, 1,3-dimethyl-2-imidazolone, tetramethylene sulfone, dimethyl sulfoxide (DMSO), methyl alcohol, alcohols such as ethanol, the water equal solvent, above-mentioned solvent can use separately or be mixed with two or more.

As reductive agent, can enumerate for example sodium borohydride, sodium cyanoborohydride, sodium triacetoxy borohydride hydroborate classes such as (sodium triacetateborohydride) etc.

As aldehydes, can enumerate for example aldehydes such as formaldehyde, acetaldehyde, propionic aldehyde, trifluoro acetaldehyde, difluoro acetaldehyde, fluorine acetaldehyde, monochloroacetaldehyde, dichloro acetaldehyde, trichoro-aldehyde, bromoacetaldehyde.

As ketone, can enumerate for example ketones such as acetone, perfluoro acetone, methyl ethyl ketone.

Temperature of reaction can suitably be selected to the scope of the reflux temperature of solvent for use at-20 ℃.Reaction times can suitably be selected in several minutes to 96 hours scope in addition.

(method C)

The compound that makes general formula (29) expression in solvent, or in the non-solvent with the aldehydes reaction, can prepare the compound of general formula (31) thus.

As solvent, do not get final product so long as significantly do not suppress the solvent that this reaction carries out, can enumerate for example hexane, hexanaphthene, aliphatic hydrocarbons such as methylcyclohexane, benzene, dimethylbenzene, toluene etc. are aromatic hydrocarbon based, methylene dichloride, chloroform, tetracol phenixin, 1, halogenated hydrocarbons such as 2-ethylene dichloride, ether, dioxane, tetrahydrofuran (THF), 1, ethers such as 2-glycol dimethyl ether, dimethyl formamide, amidess such as N,N-DIMETHYLACETAMIDE, acetonitrile, nitriles such as propionitrile, acetone, methyl iso-butyl ketone (MIBK), pimelinketone, ketones such as methyl ethyl ketone, ethyl acetate, ester classes such as butylacetate, 1,3-dimethyl-2-imidazolone, tetramethylene sulfone, dimethyl sulfoxide (DMSO), methyl alcohol, alcohols such as ethanol, sulfuric acid, inorganic acids such as hydrochloric acid, formic acid, organic acids such as acetate, the water equal solvent, above-mentioned solvent can use separately or be mixed with two or more.

As aldehydes, can enumerate for example formaldehyde, acetaldehyde, propionic aldehyde etc.

Temperature of reaction can suitably be selected to the scope of the reflux temperature of solvent for use at-20 ℃, and the reaction times can be distinguished suitably selection in several minutes to 96 hours scope.

1-(vii): general formula (31)+general formula (26) → general formula (32)

The aromatic amine derivative of general formula (31) expression and the carboxylic acid derivative that general formula (26) is represented or the carbonic acid ester derivative with leavings group are reacted in appropriate solvent, can prepare the aromatic carboxylic acid acid amides or the carbamate derivatives of general formula (32) expression thus.Suitable alkali or solvent can be used in this step,, the material of in 1-(i), enumerating can be used as this alkali or solvent.Temperature of reaction, reaction times etc. are also as shown in 1-(i).

In the general formula (26), the carboxylic acid chloride derivative can easily be prepared by carboxylic acid derivative by the ordinary method of using halogenating agent.As halogenating agent, can use the material of enumerating among the 1-(i).

Do not use halogenating agent in addition but, can be prepared according to the method for enumerating among the 1-(i) by the method for the compound of compound general formula (32) expression of carboxylic acid derivative (26) and general formula (31) expression.

1-(viii): general formula (32)+general formula (30) → general formula (1)

Make general formula (32) expression amide compound, react in solvent or in the non-solvent with the compound with leavings group such as halogen of general formula (30) expression, can prepare the The compounds of this invention of general formula (1) expression thus.Suitable alkali or solvent can be used in this step,, the material of in 1-(i), enumerating can be used as this alkali or solvent.Temperature of reaction, reaction times etc. are also as shown in 1-(i).

＜preparation method 2 〉

2-(i): general formula (33)+general formula (22) → general formula (34)

Compound that makes general formula (33) expression and the conditioned response of the compound of general formula (22) expression according to record among the 1-(i) can prepare the compound that general formula (34) is represented thus.

2-is (ii): general formula (34) → general formula (36)

For example, according to the condition of record in the J.Org.Chem.280 page or leaf (1958), ammoxidation is carried out in amination agent such as use ammonia, can prepare the compound of general formula (36) expression.Conditions such as reaction solvent are not limited to the condition of document record, and the inert solvent that suitably uses not remarkable inhibited reaction to carry out gets final product.Temperature of reaction, reaction times are also as long as suitably select according to the carrying out of reaction in addition.Need to prove,, except that ammonia, also can enumerate methylamine, ethamine etc. as the amination agent.

2-is (iii): general formula (36)+general formula (26) → general formula (1)

Compound that makes general formula (36) expression and the conditioned response of the compound of general formula (26) expression according to record among the 1-(i) can prepare the compound that general formula (1) is represented thus.

＜preparation method 3 〉

3-(i): general formula (29)+general formula (26) → general formula (35)

The aromatic amine derivative of general formula (29) expression and the carboxylic acid derivative that general formula (26) is represented or the carbonic acid ester derivative with leavings group are reacted in appropriate solvent, can prepare the aromatic carboxylic acid acid amides or the carbamate derivatives of general formula (35) expression thus.Suitable alkali or solvent can be used in this step,, the material of in 1-(i), enumerating can be used as this alkali or solvent.Temperature of reaction, reaction times etc. are also as shown in 1-(i).

In the general formula (26), the carboxylic acid chloride derivative can easily be prepared by carboxylic acid derivative by the ordinary method of using halogenating agent.As halogenating agent, can use the material of enumerating among the 1-(i).

Do not use halogenating agent in addition but, can be prepared according to the method for enumerating among the 1-(i) by the method for the compound of compound general formula (35) expression of carboxylic acid derivative (26) and general formula (29) expression.

3-is (ii): general formula (35)+general formula (27) → general formula (1a)

The compound with leavings group such as halogen of the amide compound that makes general formula (35) expression and general formula (27) expression reacts in solvent or in the non-solvent, can prepare the The compounds of this invention that general formula (1a) is represented thus.Suitable alkali or solvent can be used in this step,, the material of in 1-(i), enumerating can be used as this alkali or solvent.Temperature of reaction, reaction times etc. are also as shown in 1-(i).

＜preparation method 4 〉

4-(i): general formula (24) → general formula (36)

As starting raw material, (vi) the conditioned response of Ji Zai (method A), (method B) or (method C) can prepare the compound that general formula (36) is represented thus according to 1-with the compound of general formula (24) expression.

4-(i '): general formula (24)+general formula (27) → general formula (36)

The aromatic amine derivative of general formula (24) expression and the carboxylic acid derivative that general formula (27) is represented or the carbonic acid ester derivative with leavings group are reacted in appropriate solvent, can prepare the aromatic carboxylic acid acid amides of general formula (36) expression thus.Suitable alkali or solvent can be used in this step,, the material of in 1-(i), enumerating can be used as this alkali or solvent.Temperature of reaction, reaction times etc. are also as shown in 1-(i).

In the general formula (27), the carboxylic acid chloride derivative can easily be prepared by carboxylic acid derivative by the ordinary method of using halogenating agent.As halogenating agent, can use the material of enumerating among the 1-(i).

Do not use halogenating agent in addition but, can be prepared according to the method for enumerating among the 1-(i) by the method for the compound of compound general formula (36) expression of carboxylic acid derivative (27) and general formula (24) expression.

4-is (ii): general formula (36)+general formula (26) → general formula (1)

As starting raw material,, can prepare the compound of general formula (1) expression thus with the compound of the compound of general formula (36) expression and general formula (26) expression according to the conditioned response of record among the 1-(i).

＜preparation method 5 〉

5-(i): general formula (37)+general formula (22) → general formula (38)

Compound that makes general formula (37) expression and the conditioned response of the compound of general formula (22) expression according to record among the 1-(i) can prepare the compound that general formula (38) is represented thus.

5-is (ii): general formula (38) → general formula (39)

The nitryl aromatic family carboxylic acid amide derivative that makes general formula (38) expression in appropriate solvent or in the non-solvent with suitable fluorizating agent reaction, can prepare the compound of general formula (39) expression thus.

As solvent, do not get final product so long as significantly do not suppress the solvent that this reaction carries out, can enumerate for example hexane, hexanaphthene, aliphatic hydrocarbons such as methylcyclohexane, benzene, toluene, dimethylbenzene etc. are aromatic hydrocarbon based, methylene dichloride, chloroform, tetracol phenixin, 1, halogenated hydrocarbons such as 2-ethylene dichloride, ether, dioxane, tetrahydrofuran (THF), 1, chain or ring-type ethers such as 2-glycol dimethyl ether, ethyl acetate, ester classes such as butylacetate, acetone, methyl iso-butyl ketone (MIBK), pimelinketone, ketones such as methyl ethyl ketone, acetonitrile, nitriles such as propionitrile, 1,3-dimethyl-2-imidazolone, tetramethylene sulfone, dimethyl sulfoxide (DMSO), N, dinethylformamide, N-Methyl pyrrolidone, N, non-proton property polar solvents such as N-N,N-DIMETHYLACETAMIDE, above-mentioned solvent can use separately or be mixed with two or more.

Can enumerate 1 as fluorizating agent, 1,2,2-tetrafluoro ethyl diethylamide, 2-chloro-1,1,2-trifluoroethyl diethylamide, trifluoro phenylbenzene phosphorane, difluoro triphenyl phosphorane, the fluorofomates class, sulfur tetrafluoride, Potassium monofluoride, potassium bifluoride, cesium fluoride, rubidium fluoride, Sodium Fluoride, lithium fluoride, antimonic fluoride (III), antimonic fluoride (V), zinc fluoride, cobaltous fluoride, plumbous fluoride, cupric fluoride, Mercury difluoride (II), silver fluoride, silver fluoborate, thallium fluoride (I), molybdenum fluoride (Vl), fluoridize arsenic (III), bromine fluoride, selenium tetrafluoride, three (dimethylamino) sulfonium halide atom hydrochlorate, sodium hexafluorisilicate, fluoridize quaternary ammonium salt, (2-chloroethyl) diethylamide, three fluoridize diethylamino sulphur, three fluoridize morpholino sulphur, silicon tetrafluoride, hydrogen fluoride, hydrofluoric acid, the hydrogen fluoride pyridine coordination compound, hydrogen fluoride triethylamine coordination compound, the hydrogen fluoride salt, two (2-methoxy ethyl) amino sulfur trifluoride, 2,2-two fluoro-1,3-dimethyl-2-imidazolone, iodine pentafluoride, three (diethylamino) Phosphonium-2,2,3,3,4,4-hexafluoro-tetramethylene inner salt (tris (diethylamino) phosphonium 2,2,3,3,4,4-hexafluorocyclobutanilide), triethyl ammonium trans-1,1,2,2,3,4-Hexafluorocyclobutane inner salt, R 1216 etc.Above-mentioned fluorizating agent can use separately or mix more than 2 kinds and use.

Above-mentioned fluorizating agent uses in the scope of 1 to 10 times of molar equivalent or suitably selects to use as solvent with respect to the nitryl aromatic family carboxylic acid amide derivative of general formula (38) expression.

Also can use additive, as additive, can enumerate for example metal oxide-type such as inorganic salts such as phase-transfer catalyst class, Calcium Fluoride (Fluorspan), calcium chloride, red precipitate, ion exchange resin etc. such as crown ether-like, tetraphenyl phosphonium salt such as hexaoxacyclooctadecane-6-6, above-mentioned additive not only can add in the reaction system, and can be used as the pretreating reagent use of fluorizating agent.

Temperature of reaction is suitably selected to get final product to the scope of the reflux temperature of solvent for use at-80 ℃.Reaction times is suitably selected to get final product in several minutes to 96 hours scope in addition.

＜preparation method 6 〉

6-(i): general formula (40)+general formula (22) → general formula (41)

Compound that makes general formula (40) expression and the conditioned response of the compound of general formula (22) expression according to record among the 1-(i) can prepare the compound that general formula (41) is represented thus.

6-is (ii): general formula (41) → general formula (42)

The halogen aromatic carboxylic acid amide derivatives of general formula (41) expression is reacted with suitable cyano group agent in appropriate solvent or in the non-solvent, can prepare the compound of general formula (42) expression thus.

As solvent, do not get final product so long as significantly do not suppress the solvent that this reaction carries out.Can enumerate for example hexane, hexanaphthene, aliphatic hydrocarbons such as methylcyclohexane, benzene, toluene, dimethylbenzene etc. are aromatic hydrocarbon based, methylene dichloride, chloroform, tetracol phenixin, 1, halogenated hydrocarbons such as 2-ethylene dichloride, ether, dioxane, tetrahydrofuran (THF), 1, chain or ring-type ethers such as 2-glycol dimethyl ether, ethyl acetate, ester classes such as butylacetate, acetone, methyl iso-butyl ketone (MIBK), pimelinketone, ketones such as methyl ethyl ketone, acetonitrile, nitriles such as propionitrile, 1,3-dimethyl-2-imidazolone, tetramethylene sulfone, dimethyl sulfoxide (DMSO), N, dinethylformamide, N-Methyl pyrrolidone, N, non-proton property polar solvents such as N-N,N-DIMETHYLACETAMIDE, above-mentioned solvent can use separately or be mixed with two or more.

As the cyano group agent, can enumerate metal cyanides classes such as prussiate salt, cupric cyanide, silver cyanide, lithium cyanides such as sodium cyanide, potassium cyanide, sodium cyanoborohydride, prussic acid, cyaniding Tetrylammonium etc.

Above-mentioned cyano group agent can suitably be selected to use in the scope of 1 to 1O times of molar equivalent with respect to the halogen aromatic carboxylic acid amide derivatives of general formula (41) expression.

Additive can be used,, for example inorganic salts such as phase-transfer catalyst class, sodium iodide such as crown ether-like, tetraphenyl phosphonium salt such as hexaoxacyclooctadecane-6-6 can be enumerated as additive.

Temperature of reaction can suitably be selected to the scope of the reflux temperature of solvent for use at-20 ℃.Reaction times can suitably be selected in several minutes to 96 hours scope in addition.

＜preparation method 7 〉

7-(i): general formula (43) → general formula (44)

According to the known condition of record in Synthesis463 page or leaf (1993) or the Synthesis829 page or leaf (1984) etc., make the compound and the lawesson reagent reaction of general formula (43) expression, can prepare the compound of general formula (44) expression thus.Condition such as solvent, temperature of reaction is not limited to the condition of document record.

2-is (ii): general formula (44)+general formula (26) → general formula (45)

Compound that makes general formula (44) expression and the conditioned response of the compound of general formula (26) expression according to record among the 1-(i) can prepare the compound that general formula (45) is represented thus.

＜preparation method 8 〉

8: general formula (46) → general formula (47)+general formula (48)

According to the condition of record among the 7-(i), can prepare the compound of general formula (47) and general formula (48) expression by the compound of general formula (46) expression.Condition such as solvent, temperature of reaction is not limited to the condition of document record.Above-mentioned 2 kinds of compounds can be by known separation and purification technology such as silica gel column chromatography separation and purification easily.

＜preparation method 9 〉

9-(i): general formula (49)+general formula (26) → general formula (50)

Have amino carboxylic-acid as starting raw material with what general formula (49) was represented, according to the condition of record among the 1-(i), the compound of representing with general formula (26) reacts, and can prepare the carboxylic-acid with acyl amino of general formula (50) expression thus.

9-is (ii): general formula (50) → general formula (51)

By known ordinary method, promptly, make the compound and reactions such as thionyl chloride, oxalyl chloride, carbonyl chloride, phosphorus oxychloride, phosphorus pentachloride, phosphorus trichloride, thionyl bromide, phosphorus tribromide, diethylaminosulfurtrifluoride of general formula (50) expression, can prepare the compound that general formula (51) is represented.

9-is (iii): general formula (51)+general formula (22) → general formula (1)

Compound that makes general formula (51) expression and the conditioned response of the compound of general formula (22) expression according to record among the 1-(i) can prepare the compound that general formula (1) is represented thus.

9-is (iv): general formula (50)+general formula (22) → general formula (1)

According to the condition of using the use condensing agent of record among the 1-(i) or according to the condition of using mixed anhydride method, make the compound of general formula (50) expression and the compound reaction of general formula (22) expression, can prepare the compound of general formula (1) expression thus.

Among whole preparation methods shown in above-mentioned, target substance can finish the back in reaction to be separated from reaction system according to ordinary method, as required, can carry out operations such as recrystallization, column chromatography, distillation and make with extra care.In addition, can target substance not separated from reaction system yet but it directly is supplied to next reactions steps.

Below, the 1st table provides the example of representative compounds of the amide derivatives of general formula (1) as the effective constituent of noxious organism control agent of the present invention, general formula (7) or general formula (8) expression to the 51st table, but the present invention is not limited thereto.

Need to prove that " n-" expression just in the table; " i-" expression is different; " s-" represents secondary; " t-" represents uncle; " Me " represents methyl; " Et " represents ethyl; " n-Pr " represents n-propyl; " i-Pr " represents sec.-propyl; " n-Bu " represents normal-butyl; " i-Bu " represents isobutyl-; " s-Bu " represents sec-butyl; " t-Bu " represents the tertiary butyl; " CF3 " represents trifluoromethyl; " C2F5 " represents pentafluoroethyl group; " n-C3F7 " represents seven fluorine n-propyls; " i-C3F7 " represents seven fluorine sec.-propyls; " OCF3 " represents trifluoromethoxy; " OC2F5 " represents five fluorine oxyethyl groups; " H " represents hydrogen atom; " F " represents fluorine atom; " Cl " expression chlorine atom; " Br " represents bromine atoms; " I " expression iodine atom; " O " represents Sauerstoffatom; " C (O) " represents carbonyl; " CN " represents cyano group; " Py " represents pyridyl; " Ph " represents phenyl; " S (O) 2 " represents alkylsulfonyl.

[table 1]

The 1st table (1)

[table 2]

The 1st table (2)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

1-478

The 3-bromophenyl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-479

The 4-bromophenyl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-480

The 2-iodophenyl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-481

The 3-iodophenyl

H

H

H

CN

H

H

Cl

H

Pentafluoroethyl group

H

CF3

1-482

The 4-iodophenyl

H

H

H

CN

H

H

Cl

H

Pentafluoroethyl group

H

CF3

1-483

(2-trifluoromethyl) phenyl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-484

(3-trifluoromethyl) phenyl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-485

(4-trifluoromethyl) phenyl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-486

The 2-nitrophenyl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-487

The 3-nitrophenyl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-488

The 4-nitrophenyl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-489

The 2-cyano-phenyl

H

H

H

CN

H

H

Cl

H

Pentafluoroethyl group

H

C2F5

1-490

The 3-cyano-phenyl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-491

The 4-cyano-phenyl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-492

2, the 6-difluorophenyl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-493

3, the 4-dichlorophenyl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-494

The 2,4 dichloro benzene base

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

C2F5

1-495

2-chloro-4-fluorophenyl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-496

2-chloro-4, the 5-difluorophenyl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-497

4-bromo-2-chloro-phenyl-

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-498

2-bromo-4-chloro-phenyl-

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

n-C3F7

1-499

2-bromo-4-fluorophenyl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-500

2-chloro-4-nitrophenyl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-501

3,5-dicyano phenyl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-502

4-cyano group-2-fluorophenyl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-503

2-chloro-4-cyano-phenyl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-504

Pyridin-3-yl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-505

2-fluorine pyridin-3-yl

H

H

H

CN

H

H

Cl

H

Pentafluoroethyl group

H

CF3

1-506

2-chloropyridine-3-base

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-507

2-bromopyridine-3-base

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-508

2-iodine pyridine-3-base

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-509

2-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-510

2-nitropyridine-3-base

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-511

2-cyanopyridine-3-base

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-512

6-fluorine pyridin-3-yl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-513

6-chloropyridine-3-base

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-514

6-bromopyridine-3-base

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-515

6-iodine pyridine-3-base

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-516

6-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-517

6-nitropyridine-3-base

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-518

6-cyanopyridine-3-base

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-519

5-fluorine pyridin-3-yl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

C2F5

[table 3]

The 1st table (3)

[table 4]

The 1st table (4)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

1-608

4-iodine pyridine-3-base

H

H

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

1-609

4-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

n-C3F7

1-610

4-nitropyridine-3-base

H

H

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

i-C3F7

1-611

4-cyanopyridine-3-base

H

H

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

1-612

2,6-dichloropyridine-3-base

H

H

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

1-613

N-pyridine oxide-3-base

H

H

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

1-614

Pyridin-4-yl

H

H

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

1-615

2-chloropyridine-4-base

H

H

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

1-616

3-bromopyridine-4-base

H

H

H

CN

H

H

C?l

H

Nine fluoro-2-butyl

H

CF3

1-617

3,5-dichloropyridine-4-base

H

H

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

1-618

3-(trifluoromethyl) pyridin-4-yl

H

H

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

1-619

2,6-dicyanopyridine-4-base

H

H

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

1-620

N-pyridine oxide-4-base

H

H

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

1-621

Pyridine-2-base

H

H

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

1-622

3-chloropyridine-2-base

H

H

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

1-623

4-bromopyridine-2-base

H

H

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

1-624

5-iodine pyridine-2-base

H

H

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

1-625

6-chloropyridine-2-base

H

H

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

1-626

4-cyanopyridine-2-base

H

H

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

C2F5

1-627

Phenyl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-628

The 2-fluorophenyl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-629

The 3-fluorophenyl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-630

The 4-fluorophenyl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-631

The 2-chloro-phenyl-

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-632

The 3-chloro-phenyl-

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-633

The 4-chloro-phenyl-

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-634

The 2-bromophenyl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-635

The 3-bromophenyl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-636

The 4-bromophenyl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-637

The 2-iodophenyl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-638

The 3-iodophenyl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-639

The 4-iodophenyl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-640

(2-trifluoromethyl) phenyl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-641

(3-trifluoromethyl) phenyl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-642

(4-trifluoromethyl) phenyl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-643

The 2-nitrophenyl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-644

The 3-nitrophenyl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-645

The 4-nitrophenyl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-646

The 2-cyano-phenyl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-647

The 3-cyano-phenyl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-648

The 4-cyano-phenyl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-649

2, the 6-difluorophenyl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

[table 5]

The 1st table (5)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

1-672

6-iodine pyridine-3-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-673

6-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-674

6-nitropyridine-3-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-675

6-cyanopyridine-3-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-676

5-fluorine pyridin-3-yl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-677

5-chloropyridine-3-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-678

5-bromopyridine-3-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-679

5-iodine pyridine-3-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-680

5-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-681

5-nitropyridine-3-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-682

5-cyanopyridine-3-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-683

4-fluorine pyridin-3-yl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-684

4-chloropyridine-3-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-685

4-bromopyridine-3-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-686

4-iodine pyridine-3-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-687

4-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-688

4-nitropyridine-3-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-689

4-cyanopyridine-3-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-690

2,6-dichloropyridine-3-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-691

N-pyridine oxide-3-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-692

Pyridin-4-yl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-693

2-chloropyridine-4-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-694

3-bromopyridine-4-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-695

3,5-dichloropyridine-4-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-696

3-(trifluoromethyl) pyridin-4-yl

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-697

2,6-dicyanopyridine-4-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-698

N-pyridine oxide-4-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-699

Pyridine-2-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-700

3-chloropyridine-2-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-701

4-bromopyridine-2-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-702

5-iodine pyridine-2-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-703

6-chloropyridine-2-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-704

4-cyanopyridine-2-base

H

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-705

Phenyl

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-706

The 2-fluorophenyl

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-707

The 3-fluorophenyl

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-708

The 4-fluorophenyl

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-709

The 2-chloro-phenyl-

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-710

The 3-chloro-phenyl-

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-711

The 4-chloro-phenyl-

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-712

The 2-bromophenyl

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-713

The 3-bromophenyl

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

[table 6]

The 1st table (6)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

1-736

3,5-dicyano phenyl

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-737

4-cyano group-2-fluorophenyl

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-738

2-chloro-4-cyano-phenyl

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-739

Pyridin-3-yl

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-740

2-fluorine pyridin-3-yl

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-741

2-chloropyridine-3-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-742

2-bromopyridine-3-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-743

2-iodine pyridine-3-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-744

2-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-745

2-nitropyridine-3-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-746

2-cyanopyridine-3-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-747

6-fluorine pyridin-3-yl

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-748

6-chloropyridine-3-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-749

6-bromopyridine-3-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-750

6-iodine pyridine-3-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-751

6-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-752

6-nitropyridine-3-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-753

6-cyanopyridine-3-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-754

5-fluorine pyridin-3-yl

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-755

5-chloropyridine-3-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-756

5-bromopyridine-3-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-757

5-iodine pyridine-3-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-758

5-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-759

5-nitropyridine-3-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-760

5-cyanopyridine-3-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-761

4-fluorine pyridin-3-yl

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-762

4-chloropyridine-3-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-763

4-bromopyridine-3-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-764

4-iodine pyridine-3-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-765

4-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-766

4-nitropyridine-3-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-767

4-cyanopyridine-3-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-768

2,6-dichloropyridine-3-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-769

N-pyridine oxide-3-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-770

Pyridin-4-yl

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-771

2-chloropyridine-4-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-772

3-bromopyridine-4-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-773

3,5-dichloropyridine-4-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-774

3-(trifluoromethyl) pyridin-4-yl

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-775

2,6-dicyanopyridine-4-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-776

N-pyridine oxide-4-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-777

Pyridine-2-base

H

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

[table 7]

The 1st table (7)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

1-800

The 3-nitrophenyl

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-801

The 4-nitrophenyl

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-802

The 2-cyano-phenyl

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-803

The 3-cyano-phenyl

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-804

The 4-cyano-phenyl

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-805

2, the 6-difluorophenyl

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-806

3, the 4-dichlorophenyl

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-807

The 2,4 dichloro benzene base

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-808

2-chloro-4-fluorophenyl

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-809

2-chloro-4, the 5-difluorophenyl

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-810

4-bromo-2-chloro-phenyl-

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-811

2-bromo-4-chloro-phenyl-

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-812

2-bromo-4-fluorophenyl

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-813

2-chloro-4-nitrophenyl

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-814

3,5-dicyano phenyl

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-815

4-cyano group-2-fluorophenyl

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-816

2-chloro-4-cyano-phenyl

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-817

Pyridin-3-yl

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-818

2-fluorine pyridin-3-yl

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-819

2-chloropyridine-3-base

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-820

2-bromopyridine-3-base

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-821

2-iodine pyridine-3-base

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-822

2-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-823

2-nitropyridine-3-base

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-824

2-cyanopyridine-3-base

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-825

6-fluorine pyridin-3-yl

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-826

6-chloropyridine-3-base

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-827

6-bromopyridine-3-base

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-828

6-iodine pyridine-3-base

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-829

6-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-830

6-nitropyridine-3-base

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-831

6-cyanopyridine-3-base

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-832

5-fluorine pyridin-3-yl

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-833

5-chloropyridine-3-base

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-834

5-bromopyridine-3-base

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-835

5-iodine pyridine-3-base

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-836

5-(trifluoromethyl) pyridin-3-yl

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-837

5-nitropyridine-3-base

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-838

5-cyanopyridine-3-base

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-839

4-fluorine pyridin-3-yl

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-840

4-chloropyridine-3-base

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-841

4-bromopyridine-3-base

H

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

[table 8]

The 1st table (8)

[table 9]

The 1st table (9)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

1-927

2-chloropyridine-4-base

H

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

1-928

3-bromopyridine-4-base

H

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

1-929

3,5-dichloropyridine-4-base

H

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

1-930

3-(trifluoromethyl) pyridin-4-yl

H

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

1-931

2,6-dicyanopyridine-4-base

H

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

1-932

N-pyridine oxide-4-base

H

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

1-933

Pyridine-2-base

H

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

1-934

3-chloropyridine-2-base

H

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

1-935

4-bromopyridine-2-base

H

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

1-936

5-iodine pyridine-2-base

H

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

1-937

6-chloropyridine-2-base

H

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

1-938

4-cyanopyridine-2-base

H

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

1-939

Phenyl

H

H

H

CN

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

1-954

The 3-cyano-phenyl

H

H

H

CN

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

1-955

The 4-cyano-phenyl

H

H

H

CN

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

1-970

2-chloropyridine-3-base

H

H

H

CN

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

1-995

Phenyl

H

H

H

CN

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

1-1010

The 3-cyano-phenyl

H

H

H

CN

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

1-1011

The 4-cyano-phenyl

H

H

H

CN

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

1-1026

2-chloropyridine-3-base

H

H

H

CN

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

1-1051

Phenyl

H

H

H

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

1-1066

The 3-cyano-phenyl

H

H

H

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

1-1067

The 4-cyano-phenyl

H

H

H

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

1-1082

2-chloropyridine-3-base

H

H

H

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

1-1107

Phenyl

H

H

H

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

1-1122

The 3-cyano-phenyl

H

H

H

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

1-1123

The 4-cyano-phenyl

H

H

H

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

1-1138

2-chloropyridine-3-base

H

H

H

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

1-1163

Phenyl

H

H

H

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

1-1175

The 4-iodophenyl

H

H

H

CN

H

H

CF3

H

Pentafluoroethyl group

H

CF3

1-1177

(3-trifluoromethyl) phenyl

H

H

H

CN

H

H

C2F5

H

Seven fluorine sec.-propyls

H

CF3

1-1183

The 3-cyano-phenyl

H

H

H

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

1-1184

The 4-cyano-phenyl

H

H

H

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

1-1190

4-bromo-2-chloro-phenyl-

H

H

H

CN

H

H

n-C3F7

H

Seven fluorine sec.-propyls

H

CF3

1-1195

4-cyano group-2-fluorophenyl

H

H

H

CN

H

H

i-C3F7

H

Seven fluorine sec.-propyls

H

CF3

1-1199

2-chloropyridine-3-base

H

H

H

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

1-1200

2-bromopyridine-3-base

H

H

H

CN

H

H

C2F5

H

Seven fluorine sec.-propyls

H

C2F5

1-1211

6-cyanopyridine-3-base

H

H

H

CN

H

H

C2F5

H

Seven fluorine sec.-propyls

H

n-C3F7

1-1215

4-cyanopyridine-3-base

H

H

H

CN

H

H

C2F5

H

Seven fluorine sec.-propyls

H

i-C3F7

1-1231

Phenyl

H

H

H

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

1-1243

The 4-iodophenyl

H

H

H

CN

H

H

C2F5

H

Nine fluoro-2-butyl

H

CF3

1-1251

The 3-cyano-phenyl

H

H

H

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

[table 10]

The 1st table (10)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

1-1554

The 4-cyano-phenyl

H

H

F

CN

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

1-1569

2-chloropyridine-3-base

H

H

F

CN

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

1-1611

Phenyl

H

H

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

1-1631

The 3-cyano-phenyl

H

H

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

1-1632

The 4-cyano-phenyl

H

H

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

1-1647

2-chloropyridine-3-base

H

H

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

1-1689

Phenyl

H

H

F

CN

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

1-1709

The 3-cyano-phenyl

H

H

F

CN

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

1-1710

The 4-cyano-phenyl

H

H

F

CN

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

1-1725

2-chloropyridine-3-base

H

H

F

CN

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

1-1767

Phenyl

H

H

F

CN

H

H

F

H

Seven fluorine sec.-propyls

H

CF3

1-1768

Phenyl

H

H

F

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-1788

The 3-cyano-phenyl

H

H

F

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-1789

The 4-cyano-phenyl

H

H

F

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-1804

2-chloropyridine-3-base

H

H

F

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-1846

Phenyl

H

H

F

CN

H

H

F

H

Nine fluoro-2-butyl

H

CF3

1-1847

Phenyl

H

H

F

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

1-1867

The 3-cyano-phenyl

H

H

F

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

1-1868

The 4-cyano-phenyl

H

H

F

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

1-1883

2-chloropyridine-3-base

H

H

F

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

1-1925

Phenyl

H

H

F

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-1945

The 3-cyano-phenyl

H

H

F

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-1946

The 4-cyano-phenyl

H

H

F

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-1961

2-chloropyridine-3-base

H

H

F

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-1968

6-chloropyridine-3-base

H

H

F

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-2003

Phenyl

H

H

F

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-2023

The 3-cyano-phenyl

H

H

F

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-2024

The 4-cyano-phenyl

H

H

F

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-2039

2-chloropyridine-3-base

H

H

F

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-2081

Phenyl

H

H

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-2101

The 3-cyano-phenyl

H

H

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-2102

The 4-cyano-phenyl

H

H

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-2117

2-chloropyridine-3-base

H

H

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-2159

Phenyl

H

H

F

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

1-2179

The 3-cyano-phenyl

H

H

F

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

1-2180

The 4-cyano-phenyl

H

H

F

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

1-2195

2-chloropyridine-3-base

H

H

F

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

1-2237

Phenyl

H

H

F

CN

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

1-2252

The 3-cyano-phenyl

H

H

F

CN

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

1-2253

The 4-cyano-phenyl

H

H

F

CN

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

1-2268

2-chloropyridine-3-base

H

H

F

CN

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

1-2293

Phenyl

H

H

F

CN

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

[table 11]

The 1st table (11)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

1-2618

The 4-cyano-phenyl

H

H

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

1-2633

2-chloropyridine-3-base

H

H

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

1-2675

Phenyl

H

H

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

1-2695

The 3-cyano-phenyl

H

H

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

1-2696

The 4-cyano-phenyl

H

H

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

1-2711

2-chloropyridine-3-base

H

H

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

1-2753

Phenyl

H

H

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

1-2773

The 3-cyano-phenyl

H

H

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

1-2774

The 4-cyano-phenyl

H

H

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

1-2789

2-chloropyridine-3-base

H

H

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

1-2831

Phenyl

H

H

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

OCF3

1-2851

The 3-cyano-phenyl

H

H

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

OCF3

1-2852

The 4-cyano-phenyl

H

H

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

OCF3

1-2867

2-chloropyridine-3-base

H

H

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

OCF3

1-2909

Phenyl

H

H

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

OCF3

1-2929

The 3-cyano-phenyl

H

H

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

OCF3

1-2930

The 4-cyano-phenyl

H

H

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

OCF3

1-2945

2-chloropyridine-3-base

H

H

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

OCF3

1-2987

Phenyl

H

H

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

OCF3

1-3007

The 3-cyano-phenyl

H

H

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

OCF3

1-3008

The 4-cyano-phenyl

H

H

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

OCF3

1-3023

2-chloropyridine-3-base

H

H

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

OCF3

1-3065

Phenyl

H

H

F

CN

F

H

F

H

Seven fluorine sec.-propyls

H

CF3

1-3066

Phenyl

H

H

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-3086

The 3-cyano-phenyl

H

H

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-3087

The 4-cyano-phenyl

H

H

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-3102

2-chloropyridine-3-base

H

H

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

1-3144

Phenyl

H

H

F

CN

F

H

F

H

Nine fluoro-2-butyl

H

CF3

1-3145

Phenyl

H

H

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

CF3

1-3165

The 3-cyano-phenyl

H

H

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

CF3

1-3166

The 4-cyano-phenyl

H

H

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

CF3

1-3181

2-chloropyridine-3-base

H

H

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

CF3

1-3223

Phenyl

H

H

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-3243

The 3-cyano-phenyl

H

H

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-3244

The 4-cyano-phenyl

H

H

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-3259

2-chloropyridine-3-base

H

H

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

CF3

1-3301

Phenyl

H

H

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-3321

The 3-cyano-phenyl

H

H

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-3322

The 4-cyano-phenyl

H

H

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-3337

2-chloropyridine-3-base

H

H

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

1-3379

Phenyl

H

H

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

1-3399

The 3-cyano-phenyl

H

H

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

[table 12]

The 1st table (12)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

1-3759

Phenyl

H

H

F

CN

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

1-3779

The 3-cyano-phenyl

H

H

F

CN

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

1-3780

The 4-cyano-phenyl

H

H

F

CN

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

1-3795

2-chloropyridine-3-base

H

H

F

CN

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

1-3827

Phenyl

H

H

F

CN

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

1-3847

The 3-cyano-phenyl

H

H

F

CN

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

1-3848

The 4-cyano-phenyl

H

H

F

CN

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

1-3863

2-chloropyridine-3-base

H

H

F

CN

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

[table 13]

The 2nd table (1)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

2-1

Phenyl

Me

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

2-21

The 3-cyano-phenyl

Me

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

2-22

The 4-cyano-phenyl

Me

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

2-37

2-chloropyridine-3-base

Me

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

2-79

Phenyl

Me

H

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

2-99

The 3-cyano-phenyl

Me

H

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

2-100

The 4-cyano-phenyl

Me

H

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

2-115

2-chloropyridine-3-base

Me

H

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

2-157

Phenyl

Me

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

2-177

The 3-cyano-phenyl

Me

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

2-178

The 4-cyano-phenyl

Me

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

2-193

2-chloropyridine-3-base

Me

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

2-235

Phenyl

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

2-255

The 3-cyano-phenyl

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

2-256

The 4-cyano-phenyl

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

2-271

2-chloropyridine-3-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

2-313

Phenyl

Me

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

2-333

The 3-cyano-phenyl

Me

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

2-334

The 4-cyano-phenyl

Me

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

2-349

2-chloropyridine-3-base

Me

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

2-391

Phenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

2-411

The 3-cyano-phenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

2-412

The 4-cyano-phenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

2-427

2-chloropyridine-3-base

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

2-469

Phenyl

Me

H

H

CN

H

H

F

H

Seven fluorine sec.-propyls

H

CF3

2-470

Phenyl

Me

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

2-481

The 3-iodophenyl

Me

H

H

CN

H

H

Cl

H

Pentafluoroethyl group

H

CF3

2-482

The 4-iodophenyl

Me

H

H

CN

H

H

Cl

H

Pentafluoroethyl group

H

CF3

2-484

(3-trifluoromethyl) phenyl

Et

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

2-489

The 2-cyano-phenyl

Me

H

H

CN

H

H

Cl

H

Pentafluoroethyl group

H

C2F5

2-490

The 3-cyano-phenyl

Me

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

2-491

The 4-cyano-phenyl

Me

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

2-494

The 2,4 dichloro benzene base

Me

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

C2F5

2-495

2-chloro-4-fluorophenyl

n-Pr

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

2-498

2-bromo-4-chloro-phenyl-

Me

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

n-C3F7

[table 14]

The 2nd table (2)

[table 15]

The 2nd table (3)

[table 16]

The 2nd table (4)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

2-739

Pyridin-3-yl

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-740

2-fluorine pyridin-3-yl

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-741

2-chloropyridine-3-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-742

2-bromopyridine-3-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-743

2-iodine pyridine-3-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-744

2-(trifluoromethyl) pyridin-3-yl

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-745

2-nitropyridine-3-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-746

2-cyanopyridine-3-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-747

6-fluorine pyridin-3-yl

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-748

6-chloropyridine-3-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-749

6-bromopyridine-3-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-750

6-iodine pyridine-3-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-751

6-(trifluoromethyl) pyridin-3-yl

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-752

6-nitropyridine-3-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-753

6-cyanopyridine-3-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-754

5-fluorine pyridin-3-yl

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-755

5-chloropyridine-3-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-756

5-bromopyridine-3-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-757

5-iodine pyridine-3-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-758

5-(trifluoromethyl) pyridin-3-yl

CN

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-759

5-nitropyridine-3-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-760

5-cyanopyridine-3-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-761

4-fluorine pyridin-3-yl

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-762

4-chloropyridine-3-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-763

4-bromopyridine-3-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-764

4-iodine pyridine-3-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-765

4-(trifluoromethyl) pyridin-3-yl

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-766

4-nitropyridine-3-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-767

4-cyanopyridine-3-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-768

2,6-dichloropyridine-3-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-769

N-pyridine oxide-3-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-770

Pyridin-4-yl

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-771

2-chloropyridine-4-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-772

3-bromopyridine-4-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-773

3,5-dichloropyridine-4-base

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

[table 17]

The 2nd table (5)

[table 18]

The 2nd table (6)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

2-867

The 4-chloro-phenyl-

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-868

The 2-bromophenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-869

The 3-bromophenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-870

The 4-bromophenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-871

The 2-iodophenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-872

The 3-iodophenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-873

The 4-iodophenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-874

(2-trifluoromethyl) phenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-875

(3-trifluoromethyl) phenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-876

(4-trifluoromethyl) phenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-877

The 2-nitrophenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-878

The 3-nitrophenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-879

The 4-nitrophenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-880

The 2-cyano-phenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-881

The 3-cyano-phenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-882

The 4-cyano-phenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-883

2, the 6-difluorophenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-884

3, the 4-dichlorophenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-885

The 2,4 dichloro benzene base

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-886

2-chloro-4-fluorophenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-887

2-chloro-4, the 5-difluorophenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-888

4-bromo-2-chloro-phenyl-

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-889

2-bromo-4-chloro-phenyl-

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-890

2-bromo-4-fluorophenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-891

2-chloro-4-nitrophenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-892

3,5-dicyano phenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-893

4-cyano group-2-fluorophenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-894

2-chloro-4-cyano-phenyl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-895

Pyridin-3-yl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-896

2-fluorine pyridin-3-yl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-897

2-chloropyridine-3-base

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-898

2-bromopyridine-3-base

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-899

2-iodine pyridine-3-base

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-900

2-(trifluoromethyl) pyridin-3-yl

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-901

2-nitropyridine-3-base

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

[table 19]

The 2nd table (7)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

2-931

2,6-dicyanopyridine-4-base

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-932

N-pyridine oxide-4-base

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-933

Pyridine-2-base

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-934

3-chloropyridine-2-base

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-935

4-bromopyridine-2-base

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-936

5-iodine pyridine-2-base

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-937

6-chloropyridine-2-base

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-938

4-cyanopyridine-2-base

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-939

Phenyl

Me

H

H

CN

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

2-970

2-chloropyridine-3-base

Me

H

H

CN

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

2-995

Phenyl

Me

H

H

CN

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

2-1026

2-chloropyridine-3-base

Me

H

H

CN

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

2-1051

Phenyl

Me

H

H

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

2-1082

2-chloropyridine-3-base

Me

H

H

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

2-1107

Phenyl

Me

H

H

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

2-1138

2-chloropyridine-3-base

Me

H

H

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

2-1163

Phenyl

Me

H

H

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

2-1183

The 3-cyano-phenyl

Me

H

H

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

2-1184

The 4-cyano-phenyl

Me

H

H

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

2-1199

2-chloropyridine-3-base

Me

H

H

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

2-1231

Phenyl

Me

H

H

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

2-1251

The 3-cyano-phenyl

Me

H

H

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

2-1252

The 4-cyano-phenyl

Me

H

H

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

2-1267

2-chloropyridine-3-base

Me

H

H

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

2-1299

Phenyl

Me

H

F

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

2-1319

The 3-cyano-phenyl

Me

H

F

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

2-1320

The 4-cyano-phenyl

Me

H

F

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

2-1335

2-chloropyridine-3-base

Me

H

F

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

2-1377

Phenyl

Me

H

F

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

2-1397

The 3-cyano-phenyl

Me

H

F

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

2-1398

The 4-cyano-phenyl

Me

H

F

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

2-1413

2-chloropyridine-3-base

Me

H

F

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

2-1455

Phenyl

Me

H

F

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

2-1475

The 3-cyano-phenyl

Me

H

F

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

2-1476

The 4-cyano-phenyl

Me

H

F

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

2-1491

2-chloropyridine-3-base

Me

H

F

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

2-1533

Phenyl

Me

H

F

CN

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

2-1553

The 3-cyano-phenyl

Me

H

F

CN

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

2-1554

The 4-cyano-phenyl

Me

H

F

CN

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

2-1569

2-chloropyridine-3-base

Me

H

F

CN

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

2-1611

Phenyl

Me

H

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

2-1631

The 3-cyano-phenyl

Me

H

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

[table 20]

The 2nd table (8)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

2-2024

The 4-cyano-phenyl

Me

H

F

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-2039

2-chloropyridine-3-base

Me

H

F

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-2081

Phenyl

Me

H

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

2-2101

The 3-cyano-phenyl

Me

H

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

2-2102

The 4-cyano-phenyl

Me

H

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

2-2117

2-chloropyridine-3-base

Me

H

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

2-2159

Phenyl

Me

H

F

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-2179

The 3-cyano-phenyl

Me

H

F

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-2180

The 4-cyano-phenyl

Me

H

F

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-2195

2-chloropyridine-3-base

Me

H

F

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

2-2237

Phenyl

Me

H

F

CN

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

2-2268

2-chloropyridine-3-base

Me

H

F

CN

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

2-2293

Phenyl

Me

H

F

CN

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

2-2324

2-chloropyridine-3-base

Me

H

F

CN

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

2-2349

Phenyl

Me

H

F

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

2-2380

2-chloropyridine-3-base

Me

H

F

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

2-2405

Phenyl

Me

H

F

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

2-2436

2-chloropyridine-3-base

Me

H

F

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

2-2461

Phenyl

Me

H

F

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

2-2481

The 3-cyano-phenyl

Me

H

F

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

2-2482

The 4-cyano-phenyl

Me

H

F

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

2-2497

2-chloropyridine-3-base

Me

H

F

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

2-2529

Phenyl

Me

H

F

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

2-2549

The 3-cyano-phenyl

Me

H

F

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

2-2550

The 4-cyano-phenyl

Me

H

F

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

2-2565

2-chloropyridine-3-base

Me

H

F

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

2-2597

Phenyl

Me

H

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

2-2617

The 3-cyano-phenyl

Me

H

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

2-2618

The 4-cyano-phenyl

Me

H

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

2-2633

2-chloropyridine-3-base

Me

H

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

2-2675

Phenyl

Me

H

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

2-2695

The 3-cyano-phenyl

Me

H

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

2-2696

The 4-cyano-phenyl

Me

H

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

2-2711

2-chloropyridine-3-base

Me

H

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

2-2753

Phenyl

Me

H

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

2-2773

The 3-cyano-phenyl

Me

H

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

2-2774

The 4-cyano-phenyl

Me

H

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

2-2789

2-chloropyridine-3-base

Me

H

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

2-2831

Phenyl

Me

H

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

OCF3

2-2851

The 3-cyano-phenyl

Me

H

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

OCF3

2-2852

The 4-cyano-phenyl

Me

H

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

OCF3

2-2867

2-chloropyridine-3-base

Me

H

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

OCF3

[table 21]

The 2nd table (9)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

2-3321

The 3-cyano-phenyl

Me

H

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-3322

The 4-cyano-phenyl

Me

H

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-3337

2-chloropyridine-3-base

Me

H

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

2-3379

Phenyl

Me

H

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

2-3399

The 3-cyano-phenyl

Me

H

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

2-3400

The 4-cyano-phenyl

Me

H

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

2-3415

2-chloropyridine-3-base

Me

H

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

2-3457

Phenyl

Me

H

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

CF3

2-3477

The 3-cyano-phenyl

Me

H

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

CF3

2-3478

The 4-cyano-phenyl

Me

H

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

CF3

2-3493

2-chloropyridine-3-base

Me

H

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

CF3

2-3494

2-bromopyridine-3-base

Me

H

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

CF3

2-3535

Phenyl

Me

H

F

CN

F

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

2-3566

2-chloropyridine-3-base

Me

H

F

CN

F

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

2-3591

Phenyl

Me

H

F

CN

F

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

2-3622

2-chloropyridine-3-base

Me

H

F

CN

F

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

2-3647

Phenyl

Me

H

F

CN

F

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

2-3678

2-chloropyridine-3-base

Me

H

F

CN

F

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

2-3703

Phenyl

Me

H

F

CN

F

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

2-3734

2-chloropyridine-3-base

Me

H

F

CN

F

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

2-3759

Phenyl

Me

H

F

CN

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

2-3779

The 3-cyano-phenyl

Me

H

F

CN

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

2-3780

The 4-cyano-phenyl

Me

H

F

CN

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

2-3795

2-chloropyridine-3-base

Me

H

F

CN

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

2-3827

Phenyl

Me

H

F

CN

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

2-3847

The 3-cyano-phenyl

Me

H

F

CN

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

2-3848

The 4-cyano-phenyl

Me

H

F

CN

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

2-3863

2-chloropyridine-3-base

Me

H

F

CN

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

[table 22]

The 3rd table (1)

[table 23]

The 3rd table (2)

[table 24]

The 3rd table (3)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

3-1925

Phenyl

H

Me

F

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

3-1945

The 3-cyano-phenyl

H

Me

F

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

3-1946

The 4-cyano-phenyl

H

Me

F

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

3-1961

2-chloropyridine-3-base

H

Me

F

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

3-2003

Phenyl

H

Me

F

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

3-2023

The 3-cyano-phenyl

H

Me

F

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

3-2024

The 4-cyano-phenyl

H

Me

F

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

3-2039

2-chloropyridine-3-base

H

Me

F

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

3-2081

Phenyl

H

Me

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

3-2101

The 3-cyano-phenyl

H

Me

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

3-2102

The 4-cyano-phenyl

H

Me

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

3-2117

2-chloropyridine-3-base

H

Me

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

3-2159

Phenyl

H

Me

F

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

3-2179

The 3-cyano-phenyl

H

Me

F

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

3-2180

The 4-cyano-phenyl

H

Me

F

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

3-2195

2-chloropyridine-3-base

H

Me

F

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

3-2237

Phenyl

H

Me

F

CN

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

3-2268

2-chloropyridine-3-base

H

Me

F

CN

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

3-2293

Phenyl

H

Me

F

CN

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

3-2324

2-chloropyridine-3-base

H

Me

F

CN

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

3-2349

Phenyl

H

Me

F

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

3-2380

2-chloropyridine-3-base

H

Me

F

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

3-2405

Phenyl

H

Me

F

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

3-2436

2-chloropyridine-3-base

H

Me

F

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

3-2461

Phenyl

H

Me

F

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

3-2481

The 3-cyano-phenyl

H

Me

F

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

3-2482

The 4-cyano-phenyl

H

Me

F

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

3-2497

2-chloropyridine-3-base

H

Me

F

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

3-2529

Phenyl

H

Me

F

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

3-2549

The 3-cyano-phenyl

H

Me

F

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

3-2550

The 4-cyano-phenyl

H

Me

F

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

3-2565

2-chloropyridine-3-base

H

Me

F

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

3-2597

Phenyl

H

Me

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

3-2617

The 3-cyano-phenyl

H

Me

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

3-2618

The 4-cyano-phenyl

H

Me

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

3-2633

2-chloropyridine-3-base

H

Me

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

3-2675

Phenyl

H

Me

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

3-2695

The 3-cyano-phenyl

H

Me

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

3-2696

The 4-cyano-phenyl

H

Me

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

3-2711

2-chloropyridine-3-base

H

Me

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

3-2753

Phenyl

H

Me

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

[table 25]

The 3rd table (4)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

3-3102

2-chloropyridine-3-base

H

Me

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

3-3144

Phenyl

H

Me

F

CN

F

H

F

H

Nine fluoro-2-butyl

H

CF3

3-3145

Phenyl

H

Me

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

CF3

3-3165

The 3-cyano-phenyl

H

Me

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

CF3

3-3166

The 4-cyano-phenyl

H

Me

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

CF3

3-3181

2-chloropyridine-3-base

H

Me

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

CF3

3-3223

Phenyl

H

Me

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

CF3

3-3243

The 3-cyano-phenyl

H

Me

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

CF3

3-3244

The 4-cyano-phenyl

H

Me

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

CF3

3-3259

2-chloropyridine-3-base

H

Me

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

CF3

3-3301

Phenyl

H

Me

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

3-3321

The 3-cyano-phenyl

H

Me

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

3-3322

The 4-cyano-phenyl

H

Me

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

3-3337

2-chloropyridine-3-base

H

Me

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

3-3379

Phenyl

H

Me

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

3-3399

The 3-cyano-phenyl

H

Me

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

3-3400

The 4-cyano-phenyl

H

Me

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

3-3415

2-chloropyridine-3-base

H

Me

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

3-3457

Phenyl

H

Me

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

CF3

3-3477

The 3-cyano-phenyl

H

Me

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

CF3

3-3478

The 4-cyano-phenyl

H

Me

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

CF3

3-3493

2-chloropyridine-3-base

H

Me

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

CF3

3-3535

Phenyl

H

Me

F

CN

F

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

3-3566

2-chloropyridine-3-base

H

Me

F

CN

F

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

3-3591

Phenyl

H

Me

F

CN

F

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

3-3622

2-chloropyridine-3-base

H

Me

F

CN

F

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

3-3647

Phenyl

H

Me

F

CN

F

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

3-3678

2-chloropyridine-3-base

H

Me

F

CN

F

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

3-3703

Phenyl

H

Me

F

CN

F

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

3-3734

2-chloropyridine-3-base

H

Me

F

CN

F

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

3-3759

Phenyl

H

Me

F

CN

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

3-3779

The 3-cyano-phenyl

H

Me

F

CN

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

3-3780

The 4-cyano-phenyl

H

Me

F

CN

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

3-3795

2-chloropyridine-3-base

H

Me

F

CN

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

[table 26]

The 4th table (1)

[table 27]

The 4th table (2)

[table 28]

The 4th table (3)

[table 29]

The 4th table (4)

[table 30]

The 4th table

(5)

[table 31]

The 4th table (6)

[table 32]

The 4th table (7)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

4-3745

Phenyl

Me

Me

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

4-3765

The 3-cyano-phenyl

Me

Me

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

4-3766

The 4-cyano-phenyl

Me

Me

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

4-3781

2-chloropyridine-3-base

Me

Me

F

CN

F

H

C?l

H

Seven fluorine sec.-propyls

H

OCF3

4-3823

Phenyl

Me

Me

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

4-3843

The 3-cyano-phenyl

Me

Me

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

4-3844

The 4-cyano-phenyl

Me

Me

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

4-3859

2-chloropyridine-3-base

Me

Me

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

4-3901

Phenyl

Me

Me

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

4-3921

The 3-cyano-phenyl

Me

Me

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

4-3922

The 4-cyano-phenyl

Me

Me

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

4-3937

2-chloropyridine-3-base

Me

Me

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

4-3979

Phenyl

Me

Me

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

OCF3

4-3999

The 3-cyano-phenyl

Me

Me

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

OCF3

4-4000

The 4-cyano-phenyl

Me

Me

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

OCF3

4-4015

2-chloropyridine-3-base

Me

Me

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

OCF3

4-4057

Phenyl

Me

Me

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

OCF3

4-4077

The 3-cyano-phenyl

Me

Me

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

OCF3

4-4078

The 4-cyano-phenyl

Me

Me

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

OCF3

4-4093

2-chloropyridine-3-base

Me

Me

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

OCF3

4-4135

Phenyl

Me

Me

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

OCF3

4-4155

The 3-cyano-phenyl

Me

Me

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

OCF3

4-4156

The 4-cyano-phenyl

Me

Me

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

OCF3

4-4171

2-chloropyridine-3-base

Me

Me

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

OCF3

4-4409

Phenyl

Me

Me

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

4-4410

Phenyl

Et

Me

F

CN

F

H

F

H

Seven fluorine sec.-propyls

H

CF3

4-4416

The 3-cyano-phenyl

Me

Me

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

4-4417

The 4-cyano-phenyl

Me

Me

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

4-4432

2-chloropyridine-3-base

Me

Me

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

4-4474

Phenyl

Me

Me

F

CN

F

H

F

H

Nine fluoro-2-butyl

H

CF3

4-4475

Phenyl

Me

Me

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

CF3

4-4495

The 3-cyano-phenyl

Me

Me

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

CF3

4-4496

The 4-cyano-phenyl

Me

Me

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

CF3

4-4511

2-chloropyridine-3-base

Me

Me

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

CF3

4-4553

Phenyl

Me

Me

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

CF3

4-4573

The 3-cyano-phenyl

Me

Me

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

CF3

4-4574

The 4-cyano-phenyl

Me

Me

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

CF3

4-4589

2-chloropyridine-3-base

Me

Me

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

CF3

4-4631

Phenyl

Me

Me

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

4-4651

The 3-cyano-phenyl

Me

Me

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

4-4652

The 4-cyano-phenyl

Me

Me

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

[table 33]

The 5th table (1)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

5-9

The 3-bromophenyl

H

E?t

H

CN

H

H

Cl

F

Seven fluorine sec.-propyls

F

OCF3

5-39

2-iodine pyridine-3-base

H

H

H

CN

H

H

Cl

Me

Nine fluoro-2-butyl

Me

OCF3

5-144

Phenyl

H

H

H

CN

H

H

Cl

F

Seven fluorine sec.-propyls

H

CF3

5-145

The 2-fluorophenyl

Me

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

F

CF3

5-146

The 3-fluorophenyl

H

Me

H

CN

H

H

Cl

Cl

Seven fluorine sec.-propyls

H

CF3

5-147

The 4-fluorophenyl

Me

Me

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

Cl

CF3

5-148

The 2-chloro-phenyl-

H

H

H

CN

H

H

F

Br

Seven fluorine sec.-propyls

H

CF3

5-149

The 3-chloro-phenyl-

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

Br

CF3

5-150

The 4-chloro-phenyl-

Et

H

H

CN

H

H

Cl

I

Seven fluorine sec.-propyls

H

C2F5

5-151

The 2-bromophenyl

H

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

I

CF3

5-152

The 3-bromophenyl

H

Et

H

CN

H

H

Cl

F

Seven fluorine sec.-propyls

F

CF3

5-153

The 4-bromophenyl

H

H

H

CN

H

H

Cl

F

Seven fluorine sec.-propyls

Cl

CF3

5-154

The 2-iodophenyl

H

H

H

CN

H

H

Cl

F

Seven fluorine sec.-propyls

Br

CF3

5-155

The 3-iodophenyl

Et

Et

H

CN

H

H

Cl

F

Pentafluoroethyl group

I

C2F5

5-156

The 4-iodophenyl

H

H

H

CN

H

H

Cl

Cl

Pentafluoroethyl group

F

CF3

5-157

(2-trifluoromethyl) phenyl

H

H

H

CN

H

H

Cl

Cl

Seven fluorine sec.-propyls

Cl

CF3

5-158

(3-trifluoromethyl) phenyl

n-Pr

H

H

CN

H

H

Cl

Cl

Seven fluorine sec.-propyls

Br

CF3

5-159

(4-trifluoromethyl) phenyl

H

H

H

CN

H

H

Cl

Cl

Seven fluorine sec.-propyls

I

n-C3F7

5-160

The 2-nitrophenyl

H

n-Pr

H

CN

H

H

Cl

Br

Seven fluorine sec.-propyls

F

CF3

5-161

The 3-nitrophenyl

H

H

H

CN

H

H

Cl

Br

Seven fluorine sec.-propyls

Cl

CF3

5-162

The 4-nitrophenyl

H

H

H

CN

H

H

Cl

Br

Seven fluorine sec.-propyls

Br

CF3

5-163

The 2-cyano-phenyl

n-Pr

n-Pr

H

CN

H

H

Cl

Br

Pentafluoroethyl group

I

CF3

5-164

The 3-cyano-phenyl

H

H

H

CN

H

H

F

I

Nine fluoro-2-butyl

F

CF3

5-165

The 4-cyano-phenyl

H

H

H

CN

H

H

Cl

I

Nine fluoro-2-butyl

Cl

CF3

5-166

2, the 6-difluorophenyl

H

H

H

CN

H

H

Cl

I

Nine fluoro-2-butyl

Br

CF3

5-167

3, the 4-dichlorophenyl

H

H

H

CN

H

H

Cl

I

Nine fluoro-2-butyl

I

CF3

[table 34]

The 5th table (2)

[table 35]

The 5th table (3)

[table 36]

The 5th table (4)

[table 37]

The 6th table (1)

[table 38]

The 6th table (2)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

6-349

The 4-fluorophenyl

H

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-366

The 3-cyano-phenyl

H

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-367

The 4-cyano-phenyl

H

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-368

2, the 6-difluorophenyl

H

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-382

2-chloropyridine-3-base

H

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-389

6-chloropyridine-3-base

H

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-424

Phenyl

H

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-425

The 2-fluorophenyl

H

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-426

The 3-fluorophenyl

H

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-427

The 4-fluorophenyl

H

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-428

The 2-chloro-phenyl-

H

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-444

The 3-cyano-phenyl

H

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-445

The 4-cyano-phenyl

H

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-446

2, the 6-difluorophenyl

H

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-448

The 2,4 dichloro benzene base

H

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-449

2-chloro-4-fluorophenyl

H

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-450

2-chloro-4, the 5-difluorophenyl

H

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-451

4-bromo-2-chloro-phenyl-

H

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-452

2-bromo-4-chloro-phenyl-

H

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-453

2-bromo-4-fluorophenyl

H

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-454

2-chloro-4-nitrophenyl

H

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-460

2-chloropyridine-3-base

H

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-461

2-bromopyridine-3-base

H

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-467

6-chloropyridine-3 base

H

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-502

Phenyl

H

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-503

The 2-fluorophenyl

H

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-504

The 3-fluorophenyl

H

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-505

The 4-fluorophenyl

H

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-522

The 3-cyano-phenyl

H

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-523

The 4-cyano-phenyl

H

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-524

2, the 6-difluorophenyl

H

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-538

2-chloropyridine-3-base

H

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-545

6-chloropyridine-3-base

H

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-580

Phenyl

H

H

H

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

6-595

The 3-cyano-phenyl

H

H

H

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

6-596

The 4-cyano-phenyl

H

H

H

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

6-611

2-chloropyridine-3-base

H

H

H

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

6-636

Phenyl

H

H

H

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

6-651

The 3-cyano-phenyl

H

H

H

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

6-652

The 4-cyano-phenyl

H

H

H

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

6-667

2-chloropyridine-3-base

H

H

H

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

[table 39]

The 6th table (3)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

6-946

The 4-cyano-phenyl

H

H

F

H

H

H

F

H

Nine fluoro-2-butyl

H

F

6-947

2-chloropyridine-3-base

H

H

F

H

H

H

F

H

Nine fluoro-2-butyl

H

F

6-948

Phenyl

H

H

F

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

6-952

The 2-chloro-phenyl-

H

H

F

H

H

H

F

H

Seven fluorine sec.-propyls

H

Cl

6-956

The 3-bromophenyl

H

H

F

H

H

H

F

H

Seven fluorine sec.-propyls

H

Br

6-961

(2-trifluoromethyl) phenyl

H

H

F

H

H

H

F

H

Seven fluorine sec.-propyls

H

I

6-964

The 2-nitrophenyl

H

H

F

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Br

6-968

The 3-cyano-phenyl

H

H

F

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

6-969

The 4-cyano-phenyl

H

H

F

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

6-970

2, the 6-difluorophenyl

H

H

F

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

H

6-982

Pyridin-3-yl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

I

6-984

2-chloropyridine-3-base

H

H

F

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

6-1026

Phenyl

H

H

F

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

6-1046

The 3-cyano-phenyl

H

H

F

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

6-1047

The 4-cyano-phenyl

H

H

F

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

6-1062

2-chloropyridine-3-base

H

H

F

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

6-1104

Phenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

6-1105

The 2-fluorophenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

6-1106

The 3-fluorophenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

6-1107

The 4-fluorophenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

6-1124

The 3-cyano-phenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

6-1125

The 4-cyano-phenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

6-1126

2, the 6-difluorophenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

6-1140

2-chloropyridine-3-base

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

6-1147

6-chloropyridine-3-base

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

6-1182

Phenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

6-1183

The 2-fluorophenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

6-1184

The 3-fluorophenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

6-1185

The 4-fluorophenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

6-1202

The 3-cyano-phenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

6-1203

The 4-cyano-phenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

6-1204

2, the 6-difluorophenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

6-1218

2-chloropyridine-3-base

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

6-1225

6-chloropyridine-3-base

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

6-1260

Phenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

6-1261

The 2-fluorophenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

6-1262

The 3-fluorophenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

6-1263

The 4-fluorophenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

6-1280

The 3-cyano-phenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

6-1281

The 4-cyano-phenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

6-1282

2, the 6-difluorophenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

[table 40]

The 6th table (4)

[table 41]

The 6th table (5)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

6-1582

The 3-bromophenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1583

The 4-bromophenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1584

The 2-iodophenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1585

The 3-iodophenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1586

The 4-iodophenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1587

(2-trifluoromethyl) phenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1588

(3-trifluoromethyl) phenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1589

(4-trifluoromethyl) phenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1590

The 2-nitrophenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1591

The 3-nitrophenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1592

The 4-nitrophenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1593

The 2-cyano-phenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1594

The 3-cyano-phenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1595

The 4-cyano-phenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1596

2, the 6-difluorophenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1597

3, the 4-dichlorophenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1598

The 2,4 dichloro benzene base

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1599

2-chloro-4-fluorophenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1600

2-chloro-4, the 5-difluorophenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1601

4-bromo-2-chloro-phenyl-

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1602

2-bromo-4-chloro-phenyl-

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1603

2-bromo-4-fluorophenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1604

2-chloro-4-nitrophenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1605

3,5-dicyano phenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1606

4-cyano group-2-fluorophenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1607

2-chloro-4-cyano-phenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1608

Pyridin-3-yl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1609

2-fluorine pyridin-3-yl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1610

2-chloropyridine-3-base

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1611

2-bromopyridine-3-base

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1612

2-iodine pyridine-3-base

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1613

2-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1614

2-nitropyridine-3-base

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1615

2-cyanopyridine-3-base

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1616

6-fluorine pyridin-3-yl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1617

6-chloropyridine-3-base

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1618

6-bromopyridine-3-base

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1619

6-iodine pyridine-3-base

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1620

6-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1621

6-nitropyridine-3-base

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1622

6-cyanopyridine-3-base

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

[table 42]

The 6th table (6)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

6-1647

3-chloropyridine-2-base

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1648

4-bromopyridine-2-base

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1649

5-iodine pyridine-2-base

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1650

6-chloropyridine-2-base

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1651

4-cyanopyridine-2-base

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-1652

Phenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1653

The 2-fluorophenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1654

The 3-fluorophenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1655

The 4-fluorophenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1656

The 2-chloro-phenyl-

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1657

The 3-chloro-phenyl-

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1658

The 4-chloro-phenyl-

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1659

The 2-bromophenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1660

The 3-bromophenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1661

The 4-bromophenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1662

The 2-iodophenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1663

The 3-iodophenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1664

The 4-iodophenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1665

(2-trifluoromethyl) phenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1666

(3-trifluoromethyl) phenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1667

(4-trifluoromethyl) phenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1668

The 2-nitrophenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1669

The 3-nitrophenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1670

The 4-nitrophenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1671

The 2-cyano-phenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1672

The 3-cyano-phenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1673

The 4-cyano-phenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1674

2, the 6-difluorophenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1675

3, the 4-dichlorophenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1676

The 2,4 dichloro benzene base

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1677

2-chloro-4-fluorophenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1678

2-chloro-4, the 5-difluorophenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1679

4-bromo-2-chloro-phenyl-

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1680

2-bromo-4-chloro-phenyl-

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1681

2-bromo-4-fluorophenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1682

2-chloro-4-nitrophenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1683

3,5-dicyano phenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1684

4-cyano group-2-fluorophenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1685

2-chloro-4-cyano-phenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1686

Pyridin-3-yl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1687

2-fluorine pyridin-3-yl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

[table 43]

The 6th table (7)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

6-1710

4-bromopyridine-3-base

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1711

4-iodine pyridine-3-base

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1712

4-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1713

4-nitropyridine-3-base

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1714

4-cyanopyridine-3-base

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1715

2,6-dichloropyridine-3-base

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1716

N-pyridine oxide-3-base

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1717

Pyridin-4-yl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1718

2-chloropyridine-4-base

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1719

3-bromopyridine-4-base

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1720

3,5-dichloropyridine-4-base

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1721

3-(trifluoromethyl) pyridin-4-yl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1722

2,6-dicyanopyridine-4-base

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1723

N-pyridine oxide-4-base

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1724

Pyridine-2-base

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1725

3-chloropyridine-2-base

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1726

4-bromopyridine-2-base

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1727

5-iodine pyridine-2-base

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1728

6-chloropyridine-2-base

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1729

4-cyanopyridine-2-base

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-1730

Phenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1731

The 2-fluorophenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1732

The 3-fluorophenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1733

The 4-fluorophenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1734

The 2-chloro-phenyl-

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1735

The 3-chloro-phenyl-

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1736

The 4-chloro-phenyl-

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1737

The 2-bromophenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1738

The 3-bromophenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1739

The 4-bromophenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1740

The 2-iodophenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1741

The 3-iodophenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1742

The 4-iodophenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1743

(2-trifluoromethyl) phenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1744

(3-trifluoromethyl) phenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1745

(4-trifluoromethyl) phenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1746

The 2-nitrophenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1747

The 3-nitrophenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1748

The 4-nitrophenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1749

The 2-cyano-phenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1750

The 3-cyano-phenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1751

The 4-cyano-phenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

[table 44]

The 6th table (8)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

6-1775

6-iodine pyridine-3-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1776

6-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1777

6-nitropyridine-3-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1778

6-cyanopyridine-3-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1779

5-fluorine pyridin-3-yl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1780

5-chloropyridine-3-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1781

5-bromopyridine-3-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1782

5-iodine pyridine-3-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1783

5-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1784

5-nitropyridine-3-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1785

5-cyanopyridine-3-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1786

4-fluorine pyridin-3-yl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1787

4-chloropyridine-3-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1788

4-bromopyridine-3-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1789

4-iodine pyridine-3-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1790

4-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1791

4-nitropyridine-3-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1792

4-cyanopyridine-3-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1793

2,6-dichloropyridine-3-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1794

N-pyridine oxide-3-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1795

Pyridin-4-yl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1796

2-chloropyridine-4-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1797

3-bromopyridine-4-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1798

3,5-dichloropyridine-4-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1799

3-(trifluoromethyl) pyridin-4-yl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1800

2,6-dicyanopyridine-4-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1801

N-pyridine oxide-4-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1802

Pyridine-2-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1803

3-chloropyridine-2-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1804

4-bromopyridine-2-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1805

5-iodine pyridine-2-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1806

6-chloropyridine-2-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1807

4-cyanopyridine-2-base

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-1808

Phenyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1809

The 2-fluorophenyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1810

The 3-fluorophenyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1811

The 4-fluorophenyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1812

The 2-chloro-phenyl-

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1813

The 3-chloro-phenyl-

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1814

The 4-chloro-phenyl-

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1815

The 2-bromophenyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

[table 45]

The 6th table (9)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

6-1839

3,5-dicyano phenyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1840

4-cyano group-2-fluorophenyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1841

2-chloro-4-cyano-phenyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1842

Pyridin-3-yl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1843

2-fluorine pyridin-3-yl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1844

2-chloropyridine-3-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1845

2-bromopyridine-3-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1846

2-iodine pyridine-3-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1847

2-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1848

2-nitropyridine-3-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1849

2-cyanopyridine-3-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1850

6-fluorine pyridin-3-yl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1851

6-chloropyridine-3-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1852

6-bromopyridine-3-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1853

6-iodine pyridine-3-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1854

6-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1855

6-nitropyridine-3-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1856

6-cyanopyridine-3-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1857

5-fluorine pyridin-3-yl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1858

5-chloropyridine-3-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1859

5-bromopyridine-3-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1860

5-iodine pyridine-3-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1861

5-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1862

5-nitropyridine-3-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1863

5-cyanopyridine-3-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1864

4-fluorine pyridin-3-yl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1865

4-chloropyridine-3-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1866

4-bromopyridine-3-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1867

4-iodine pyridine-3-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1868

4-(trifluoromethyl) pyridin-3-yl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1869

4-nitropyridine-3-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1870

4-cyanopyridine-3-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1871

2,6-dichloropyridine-3-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1872

N-pyridine oxide-3-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1873

Pyridin-4-yl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1874

2-chloropyridine-4-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1875

3-bromopyridine-4-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1876

3,5-dichloropyridine-4-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1877

3-(trifluoromethyl) pyridin-4-yl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1878

2,6-dicyanopyridine-4-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-1879

N-pyridine oxide-4-base

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

[table 46]

The 6th table (10)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

6-2130

The 3-cyano-phenyl

H

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

6-2131

The 4-cyano-phenyl

H

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

6-2146

2-chloropyridine-3-base

H

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

6-2178

Phenyl

H

H

F

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

6-2198

The 3-cyano-phenyl

H

H

F

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

6-2199

The 4-cyano-phenyl

H

H

F

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

6-2214

2-chloropyridine-3-base

H

H

F

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

6-2246

Phenyl

H

H

H

F

H

H

F

H

Seven fluorine sec.-propyls

H

F

6-2247

The 3-cyano-phenyl

H

H

H

F

H

H

F

H

Seven fluorine sec.-propyls

H

F

6-2248

The 4-cyano-phenyl

H

H

H

F

H

H

F

H

Seven fluorine sec.-propyls

H

F

6-2249

2-chloropyridine-3-base

H

H

H

F

H

H

F

H

Seven fluorine sec.-propyls

H

F

6-2250

Phenyl

H

H

H

F

H

H

F

H

Nine fluoro-2-butyl

H

F

6-2251

The 3-cyano-phenyl

H

H

H

F

H

H

F

H

Nine fluoro-2-butyl

H

F

6-2252

The 4-cyano-phenyl

H

H

H

F

H

H

F

H

Nine fluoro-2-butyl

H

F

6-2253

2-chloropyridine-3-base

H

H

H

F

H

H

F

H

Nine fluoro-2-butyl

H

F

6-2254

Phenyl

H

H

H

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

6-2274

The 3-cyano-phenyl

H

H

H

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

6-2275

The 4-cyano-phenyl

H

H

H

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

6-2290

2-chloropyridine-3-base

H

H

H

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

6-2332

Phenyl

H

H

H

F

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

6-2352

The 3-cyano-phenyl

H

H

H

F

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

6-2353

The 4-cyano-phenyl

H

H

H

F

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

6-2368

2-chloropyridine-3-base

H

H

H

F

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

6-2410

Phenyl

H

H

H

F

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

6-2430

The 3-cyano-phenyl

H

H

H

F

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

6-2431

The 4-cyano-phenyl

H

H

H

F

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

6-2446

2-chloropyridine-3-base

H

H

H

F

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

6-2488

Phenyl

H

H

H

F

H

H

Br

H

Nine fluoro-2-butyl

H

Br

6-2508

The 3-cyano-phenyl

H

H

H

F

H

H

Br

H

Nine fluoro-2-butyl

H

Br

6-2509

The 4-cyano-phenyl

H

H

H

F

H

H

Br

H

Nine fluoro-2-butyl

H

Br

6-2524

2-chloropyridine-3-base

H

H

H

F

H

H

Br

H

Nine fluoro-2-butyl

H

Br

6-2566

Phenyl

H

H

H

F

H

H

I

H

Seven fluorine sec.-propyls

H

I

6-2586

The 3-cyano-phenyl

H

H

H

F

H

H

I

H

Seven fluorine sec.-propyls

H

I

6-2587

The 4-cyano-phenyl

H

H

H

F

H

H

I

H

Seven fluorine sec.-propyls

H

I

6-2602

2-chloropyridine-3-base

H

H

H

F

H

H

I

H

Seven fluorine sec.-propyls

H

I

6-2644

Phenyl

H

H

H

F

H

H

I

H

Nine fluoro-2-butyl

H

I

6-2664

The 3-cyano-phenyl

H

H

H

F

H

H

I

H

Nine fluoro-2-butyl

H

I

6-2665

The 4-cyano-phenyl

H

H

H

F

H

H

I

H

Nine fluoro-2-butyl

H

I

6-2680

2-chloropyridine-3-base

H

H

H

F

H

H

I

H

Nine fluoro-2-butyl

H

I

6-2722

Phenyl

H

H

H

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

6-2742

The 3-cyano-phenyl

H

H

H

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

[table 47]

The 6th table (11)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

6-3191

Phenyl

H

H

H

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

6-3211

The 3-cyano-phenyl

H

H

H

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

6-3212

The 4-cyano-phenyl

H

H

H

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

6-3227

2-chloropyridine-3-base

H

H

H

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

6-3269

Phenyl

H

H

H

F

H

H

F

H

Nine fluoro-2-butyl

H

CF3

6-3270

Phenyl

H

H

H

F

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

6-3290

The 3-cyano-phenyl

H

H

H

F

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

6-3291

The 4-cyano-phenyl

H

H

H

F

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

6-3306

2-chloropyridine-3-base

H

H

H

F

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

6-3348

Phenyl

H

H

H

F

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-3368

The 3-cyano-phenyl

H

H

H

F

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-3369

The 4-cyano-phenyl

H

H

H

F

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-3384

2-chloropyridine-3-base

H

H

H

F

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

6-3426

Phenyl

H

H

H

F

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-3446

The 3-cyano-phenyl

H

H

H

F

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-3447

The 4-cyano-phenyl

H

H

H

F

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-3462

2-chloropyridine-3-base

H

H

H

F

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-3504

Phenyl

H

H

H

F

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-3524

The 3-cyano-phenyl

H

H

H

F

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-3525

The 4-cyano-phenyl

H

H

H

F

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-3540

2-chloropyridine-3-base

H

H

H

F

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-3582

Phenyl

H

H

H

F

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-3602

The 3-cyano-phenyl

H

H

H

F

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-3603

The 4-cyano-phenyl

H

H

H

F

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-3618

2-chloropyridine-3-base

H

H

H

F

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-3660

Phenyl

H

H

H

F

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

6-3675

The 3-cyano-phenyl

H

H

H

F

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

6-3676

The 4-cyano-phenyl

H

H

H

F

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

6-3691

2-chloropyridine-3-base

H

H

H

F

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

6-3716

Phenyl

H

H

H

F

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

6-3731

The 3-cyano-phenyl

H

H

H

F

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

6-3732

The 4-cyano-phenyl

H

H

H

F

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

6-3747

2-chloropyridine-3-base

H

H

H

F

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

6-3772

Phenyl

H

H

H

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

6-3787

The 3-cyano-phenyl

H

H

H

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

6-3788

The 4-cyano-phenyl

H

H

H

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

6-3803

2-chloropyridine-3-base

H

H

H

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

6-3828

Phenyl

H

H

H

F

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

6-3843

The 3-cyano-phenyl

H

H

H

F

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

6-3844

The 4-cyano-phenyl

H

H

H

F

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

6-3859

2-chloropyridine-3-base

H

H

H

F

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

[table 48]

The 6th table (12)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

6-4142

2-chloropyridine-3-base

H

H

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

6-4184

Phenyl

H

H

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

6-4204

The 3-cyano-phenyl

H

H

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

6-4205

The 4-cyano-phenyl

H

H

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

6-4220

2-chloropyridine-3-base

H

H

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

6-4262

Phenyl

H

H

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

Br

6-4282

The 3-cyano-phenyl

H

H

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

Br

6-4283

The 4-cyano-phenyl

H

H

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

Br

6-4298

2-chloropyridine-3-base

H

H

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

Br

6-4340

Phenyl

H

H

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

I

6-4360

The 3-cyano-phenyl

H

H

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

I

6-4361

The 4-cyano-phenyl

H

H

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

I

6-4376

2-chloropyridine-3-base

H

H

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

I

6-4418

Phenyl

H

H

F

F

H

H

I

H

Nine fluoro-2-butyl

H

I

6-4438

The 3-cyano-phenyl

H

H

F

F

H

H

I

H

Nine fluoro-2-butyl

H

I

6-4439

The 4-cyano-phenyl

H

H

F

F

H

H

I

H

Nine fluoro-2-butyl

H

I

6-4454

2-chloropyridine-3-base

H

H

F

F

H

H

I

H

Nine fluoro-2-butyl

H

I

6-4496

Phenyl

H

H

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

6-4516

The 3-cyano-phenyl

H

H

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

6-4517

The 4-cyano-phenyl

H

H

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

6-4532

2-chloropyridine-3-base

H

H

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

6-4574

Phenyl

H

H

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

6-4594

The 3-cyano-phenyl

H

H

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

6-4595

The 4-cyano-phenyl

H

H

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

6-4610

2-chloropyridine-3-base

H

H

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

6-4652

Phenyl

H

H

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

6-4672

The 3-cyano-phenyl

H

H

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

6-4673

The 4-cyano-phenyl

H

H

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

6-4688

2-chloropyridine-3-base

H

H

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

6-4730

Phenyl

H

H

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

6-4750

The 3-cyano-phenyl

H

H

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

6-4751

The 4-cyano-phenyl

H

H

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

6-4766

2-chloropyridine-3-base

H

H

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

6-4808

Phenyl

H

H

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

6-4828

The 3-cyano-phenyl

H

H

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

6-4829

The 4-cyano-phenyl

H

H

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

6-4844

2-chloropyridine-3-base

H

H

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

6-4886

Phenyl

H

H

F

F

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

6-4906

The 3-cyano-phenyl

H

H

F

F

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

6-4907

The 4-cyano-phenyl

H

H

F

F

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

6-4922

2-chloropyridine-3-base

H

H

F

F

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

[table 49]

The 6th table (13)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

6-5376

The 3-cyano-phenyl

H

H

F

F

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-5377

The 4-cyano-phenyl

H

H

F

F

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-5392

2-chloropyridine-3-base

H

H

F

F

H

H

I

H

Nine fluoro-2-butyl

H

CF3

6-5434

Phenyl

H

H

F

F

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

6-5449

The 3-cyano-phenyl

H

H

F

F

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

6-5450

The 4-cyano-phenyl

H

H

F

F

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

6-5465

2-chloropyridine-3-base

H

H

F

F

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

6-5490

Phenyl

H

H

F

F

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

6-5505

The 3-cyano-phenyl

H

H

F

F

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

6-5506

The 4-cyano-phenyl

H

H

F

F

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

6-5521

2-chloropyridine-3-base

H

H

F

F

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

6-5546

Phenyl

H

H

F

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

6-5561

The 3-cyano-phenyl

H

H

F

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

6-5562

The 4-cyano-phenyl

H

H

F

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

6-5577

2-chloropyridine-3-base

H

H

F

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

6-5602

Phenyl

H

H

F

F

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

6-5617

The 3-cyano-phenyl

H

H

F

F

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

6-5633

2-chloropyridine-3-base

H

H

F

F

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

6-5658

Phenyl

H

H

F

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

6-5678

The 3-cyano-phenyl

H

H

F

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

6-5694

2-chloropyridine-3-base

H

H

F

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

6-5726

Phenyl

H

H

F

F

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

6-5746

The 3-cyano-phenyl

H

H

F

F

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

6-5747

The 4-cyano-phenyl

H

H

F

F

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

6-5762

2-chloropyridine-3-base

H

H

F

F

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

6-5794

Phenyl

H

H

F

F

F

H

Cl

H

Pentafluoroethyl group

H

Cl

6-5795

Phenyl

H

H

F

F

F

H

Br

H

Seven fluorine sec.-propyls

H

Br

6-5796

Phenyl

H

H

F

F

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

6-5797

Phenyl

H

H

F

F

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-5798

Phenyl

H

H

F

F

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

6-5799

Phenyl

H

H

F

F

F

H

I

H

Nine fluoro-2-butyl

H

I

6-5800

Phenyl

H

H

F

F

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

6-5801

Phenyl

H

H

F

F

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-5802

Phenyl

H

H

F

F

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

6-5803

Phenyl

H

H

H

H

F

H

Cl

H

Pentafluoroethyl group

H

Cl

6-5804

Phenyl

H

H

H

H

F

H

Br

H

Seven fluorine sec.-propyls

H

Br

6-5805

Phenyl

H

H

H

H

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

6-5806

Phenyl

H

H

H

H

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-5807

Phenyl

H

H

H

H

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

6-5808

Phenyl

H

H

H

H

F

H

I

H

Nine fluoro-2-butyl

H

I

6-5809

Phenyl

H

H

H

H

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

[table 50]

The 6th table (14)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

6-5833

Phenyl

H

H

F

H

H

F

I

H

Seven fluorine sec.-propyls

H

CF3

6-5834

Phenyl

H

H

F

H

H

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

6-5835

Phenyl

H

H

F

H

H

F

I

H

Nine fluoro-2-butyl

H

I

6-5836

Phenyl

H

H

F

H

H

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

6-5837

Phenyl

H

H

F

H

H

F

Br

H

Nine fluoro-2-butyl

H

CF3

6-5838

Phenyl

H

H

F

H

H

F

CF3

H

Nine fluoro-2-butyl

H

CF3

6-5839

Phenyl

H

H

H

F

F

H

Cl

H

Pentafluoroethyl group

H

Cl

6-5840

Phenyl

H

H

H

F

F

H

Br

H

Seven fluorine sec.-propyls

H

Br

6-5841

Phenyl

H

H

H

F

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

6-5842

Phenyl

H

H

H

F

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-5843

Phenyl

H

H

H

F

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

6-5844

Phenyl

H

H

H

F

F

H

I

H

Nine fluoro-2-butyl

H

I

6-5845

Phenyl

H

H

H

F

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

6-5846

Phenyl

H

H

H

F

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

6-5847

Phenyl

H

H

H

F

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

6-5848

Phenyl

H

H

H

F

H

F

Cl

H

Pentafluoroethyl group

H

Cl

6-5849

Phenyl

H

H

H

F

H

F

Br

H

Seven fluorine sec.-propyls

H

Br

6-5850

Phenyl

H

H

H

F

H

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

6-5851

Phenyl

H

H

H

F

H

F

I

H

Seven fluorine sec.-propyls

H

CF3

6-5852

Phenyl

H

H

H

F

H

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

6-5853

Phenyl

H

H

H

F

H

F

I

H

Nine fluoro-2-butyl

H

I

6-5854

Phenyl

H

H

H

F

H

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

6-5855

Phenyl

H

H

H

F

H

F

Br

H

Nine fluoro-2-butyl

H

CF3

6-5856

Phenyl

H

H

H

F

H

F

CF3

H

Nine fluoro-2-butyl

H

CF3

6-5857

Phenyl

H

H

H

H

F

F

Cl

H

Pentafluoroethyl group

H

Cl

6-5858

Phenyl

H

H

H

H

F

F

Br

H

Seven fluorine sec.-propyls

H

Br

6-5859

Phenyl

H

H

H

H

F

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

6-5860

Phenyl

H

H

H

H

F

F

I

H

Seven fluorine sec.-propyls

H

CF3

6-5861

Phenyl

H

H

H

H

F

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

6-5862

Phenyl

H

H

H

H

F

F

I

H

Nine fluoro-2-butyl

H

I

6-5863

Phenyl

H

H

H

H

F

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

6-5864

Phenyl

H

H

H

H

F

F

Br

H

Nine fluoro-2-butyl

H

CF3

6-5865

Phenyl

H

H

H

H

F

F

CF3

H

Nine fluoro-2-butyl

H

CF3

6-5866

Phenyl

H

H

F

F

H

F

Cl

H

Pentafluoroethyl group

H

Cl

6-5867

Phenyl

H

H

F

F

H

F

Br

H

Seven fluorine sec.-propyls

H

Br

6-5868

Phenyl

H

H

F

F

H

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

6-5869

Phenyl

H

H

F

F

H

F

I

H

Seven fluorine sec.-propyls

H

CF3

6-5870

Phenyl

H

H

F

F

H

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

6-5871

Phenyl

H

H

F

F

H

F

I

H

Nine fluoro-2-butyl

H

I

6-5872

Phenyl

H

H

F

F

H

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

6-5873

Phenyl

H

H

F

F

H

F

Br

H

Nine fluoro-2-butyl

H

CF3

[table 51]

The 6th table (15)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

6-5897

Phenyl

H

H

F

F

F

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

6-5898

Phenyl

H

H

F

F

F

F

I

H

Nine fluoro-2-butyl

H

I

6-5899

Phenyl

H

H

F

F

F

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

6-5900

Phenyl

H

H

F

F

F

F

Br

H

Nine fluoro-2-butyl

H

CF3

6-5901

Phenyl

H

H

F

F

F

F

CF3

H

Nine fluoro-2-butyl

H

CF3

6-5902

Phenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Cl

6-5903

The 3-fluorophenyl

H

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

I

6-5904

The 4-fluorophenyl

H

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

I

6-5905

The 3-fluorophenyl

H

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

6-5906

The 4-fluorophenyl

H

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

6-5907

Phenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

6-5908

2-chloropyridine-3-base

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

6-5909

The 4-cyano-phenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

6-5910

Phenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

C2F5

6-5911

The 4-cyano-phenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

C2F5

6-5912

2-chloro-4-(methyl sulphonyl) phenyl

H

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

6-5913

Phenyl

H

H

H

H

H

H

Br

H

Pentafluoroethyl group

H

CF3

6-5914

2-chloropyridine-3-base

H

H

H

H

H

H

Br

H

Pentafluoroethyl group

H

CF3

[table 52]

The 7th table (1)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

7-1

Phenyl

Me

H

H

H

H

H

F

H

Nine fluoro-2-butyl

H

F

7-2

The 3-cyano-phenyl

Me

H

H

H

H

H

F

H

Nine fluoro-2-butyl

H

F

7-3

The 4-cyano-phenyl

Me

H

H

H

H

H

F

H

Nine fluoro-2-butyl

H

F

7-4

2-chloropyridine-3-base

Me

H

H

H

H

H

F

H

Nine fluoro-2-butyl

H

F

7-5

Phenyl

Me

H

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

7-12

The 3-cyano-phenyl

Me

H

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

7-13

The 4-cyano-phenyl

Me

H

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

7-24

2-chloropyridine-3-base

Me

H

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

7-38

Phenyl

Me

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

7-39

The 2-fluorophenyl

Me

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

7-45

The 3-cyano-phenyl

Me

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

7-46

The 4-cyano-phenyl

Me

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

7-47

2, the 6-difluorophenyl

Me

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

7-57

2-chloropyridine-3-base

Me

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

7-60

6-chloropyridine-3-base

Me

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

7-71

Phenyl

Me

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

I

7-72

The 2-fluorophenyl

Me

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

I

7-78

The 3-cyano-phenyl

Me

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

I

7-79

The 4-cyano-phenyl

Me

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

I

7-80

2, the 6-difluorophenyl

Me

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

I

7-90

2-chloropyridine-3-base

Me

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

I

7-93

6-chloropyridine-3-base

Me

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

I

7-104

Phenyl

Me

H

H

H

H

H

F

H

Nine fluoro-2-butyl

H

Cl

7-105

Phenyl

Me

H

H

H

H

H

F

H

Nine fluoro-2-butyl

H

Br

7-106

Phenyl

Me

H

H

H

H

H

F

H

Nine fluoro-2-butyl

H

I

7-107

Phenyl

Me

H

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Br

7-108

Phenyl

Me

H

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

I

7-109

Phenyl

Me

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

I

7-110

Phenyl

Me

H

H

H

H

H

F

H

Seven fluorine sec.-propyls

H

CF3

7-111

Phenyl

Me

H

H

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

7-131

The 3-cyano-phenyl

Me

H

H

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

7-132

The 4-cyano-phenyl

Me

H

H

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

[table 53]

The 7th table (2)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

7-346

Phenyl

Me

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-347

The 2-fluorophenyl

Me

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-348

The 3-fluorophenyl

Me

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-349

The 4-fluorophenyl

Me

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-366

The 3-cyano-phenyl

Me

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-367

The 4-cyano-phenyl

Me

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-368

2, the 6-difluorophenyl

Me

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-382

2-chloropyridine-3-base

Me

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-389

6-chloropyridine-3-base

Me

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-424

Phenyl

Me

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

7-425

The 2-fluorophenyl

Me

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

7-426

The 3-fluorophenyl

Me

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

7-427

The 4-fluorophenyl

Me

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

7-428

The 2-chloro-phenyl-

Me

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

7-444

The 3-cyano-phenyl

Me

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

7-445

The 4-cyano-phenyl

Me

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

7-446

2, the 6-difluorophenyl

Me

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

7-449

2-chloro-4-fluorophenyl

Me

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

7-460

2-chloropyridine-3-base

Me

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

7-467

6-chloropyridine-3-base

Me

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

7-502

Phenyl

Me

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-504

The 3-fluorophenyl

Me

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-505

The 4-fluorophenyl

Me

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-522

The 3-cyano-phenyl

Me

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-523

The 4-cyano-phenyl

Me

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-538

2-chloropyridine-3-base

Me

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-580

Phenyl

Me

H

H

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

7-611

2-chloropyridine-3-base

Me

H

H

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

7-636

Phenyl

Me

H

H

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

7-667

2-chloropyridine-3-base

Me

H

H

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

7-692

Phenyl

Me

H

H

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

7-723

2-chloropyridine-3-base

Me

H

H

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

7-748

Phenyl

Me

H

H

H

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

7-779

2-chloropyridine-3-base

Me

H

H

H

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

7-804

Phenyl

Me

H

H

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

7-824

The 3-cyano-phenyl

Me

H

H

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

7-825

The 4-cyano-phenyl

Me

H

H

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

7-840

2-chloropyridine-3-base

Me

H

H

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

7-841

2-bromopyridine-3-base

Me

H

H

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

7-872

Phenyl

Me

H

H

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

7-892

The 3-cyano-phenyl

Me

H

H

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

[table 54]

The 7th table (3)

[table 55]

The 7th table (4)

[table 56]

The 7th table (5)

[table 57]

The 7th table (6)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

7-1694

6-fluorine pyridin-3-yl

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1695

6-chloropyridine-3-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1696

6-bromopyridine-3-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1697

6-iodine pyridine-3-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1698

6-(trifluoromethyl) pyridin-3-yl

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1699

6-nitropyridine-3-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1700

6-cyanopyridine-3-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1701

5-fluorine pyridin-3-yl

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1702

5-chloropyridine-3-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1703

5-bromopyridine-3-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1704

5-iodine pyridine-3-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1705

5-(trifluoromethyl) pyridin-3-yl

CN

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1706

5-nitropyridine-3-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1707

5-cyanopyridine-3-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1708

4-fluorine pyridin-3-yl

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1709

4-chloropyridine-3-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1710

4-bromopyridine-3-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1711

4-iodine pyridine-3-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1712

4-(trifluoromethyl) pyridin-3-yl

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1713

4-nitropyridine-3-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1714

4-cyanopyridine-3-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1715

2,6-dichloropyridine-3-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1716

N-pyridine oxide-3-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1717

Pyridin-4-yl

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1718

2-chloropyridine-4-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1719

3-bromopyridine-4-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1720

3,5-dichloropyridine-4-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1721

3-(trifluoromethyl) pyridin-4-yl

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1722

2,6-dicyanopyridine-4-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1723

N-pyridine oxide-4-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1724

Pyridine-2-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1725

3-chloropyridine-2-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1726

4-bromopyridine-2-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1727

5-iodine pyridine-2-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1728

6-chloropyridine-2-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1729

4-cyanopyridine-2-base

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-1730

Phenyl

Me

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

7-1731

The 2-fluorophenyl

Me

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

7-1732

The 3-fluorophenyl

Me

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

7-1733

The 4-fluorophenyl

Me

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

7-1734

The 2-chloro-phenyl-

Me

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

[table 58]

The 7th table (7)

[table 59]

The 7th table (8)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

7-1822

(3-trifluoromethyl) phenyl

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1823

(4-trifluoromethyl) phenyl

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1824

The 2-nitrophenyl

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1825

The 3-nitrophenyl

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1826

The 4-nitrophenyl

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1827

The 2-cyano-phenyl

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1828

The 3-cyano-phenyl

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1829

The 4-cyano-phenyl

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1830

2, the 6-difluorophenyl

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1831

3, the 4-dichlorophenyl

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1832

The 2,4 dichloro benzene base

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1833

2-chloro-4-fluorophenyl

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1834

2-chloro-4, the 5-difluorophenyl

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1835

4-bromo-2-chloro-phenyl-

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1836

2-bromo-4-chloro-phenyl-

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1837

2-bromo-4-fluorophenyl

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1838

2-chloro-4-nitrophenyl

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1839

3,5-dicyano phenyl

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1840

4-cyano group-2-fluorophenyl

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1841

2-chloro-4-cyano-phenyl

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1842

Pyridin-3-yl

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1843

2-fluorine pyridin-3-yl

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1844

2-chloropyridine-3-base

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1845

2-bromopyridine-3-base

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1846

2-iodine pyridine-3-base

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1847

2-(trifluoromethyl) pyridin-3-yl

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1848

2-nitropyridine-3-base

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1849

2-cyanopyridine-3-base

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1850

6-fluorine pyridin-3-yl

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1851

6-chloropyridine-3-base

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1852

6-bromopyridine-3-base

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1853

6-iodine pyridine-3-base

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1854

6-(trifluoromethyl) pyridin-3-yl

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1855

6-nitropyridine-3-base

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1856

6-cyanopyridine-3-base

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1857

5-fluorine pyridin-3-yl

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1858

5-chloropyridine-3-base

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1859

5-bromopyridine-3-base

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-1860

5-iodine pyridine-3-base

Me

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

[table 60]

The 7th table (9)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

7-1886

Phenyl

Me

H

F

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

7-1901

The 3-cyano-phenyl

Me

H

F

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

7-1902

The 4-cyano-phenyl

Me

H

F

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

7-1917

2-chloropyridine-3-base

Me

H

F

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

7-1942

Phenyl

Me

H

F

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

7-1957

The 3-cyano-phenyl

Me

H

F

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

7-1958

The 4-cyano-phenyl

Me

H

F

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

7-1973

2-chloropyridine-3-base

Me

H

F

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

7-1998

Phenyl

Me

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

7-2013

The 3-cyano-phenyl

Me

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

7-2014

The 4-cyano-phenyl

Me

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

7-2029

2-chloropyridine-3-base

Me

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

7-2054

Phenyl

Me

H

F

H

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

7-2069

The 3-cyano-phenyl

Me

H

F

H

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

7-2070

The 4-cyano-phenyl

Me

H

F

H

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

7-2085

2-chloropyridine-3-base

Me

H

F

H

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

7-2110

Phenyl

Me

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

7-2130

The 3-cyano-phenyl

Me

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

7-2131

The 4-cyano-phenyl

Me

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

7-2146

2-chloropyridine-3-base

Me

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

7-2178

Phenyl

Me

H

F

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

7-2198

The 3-cyano-phenyl

Me

H

F

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

7-2199

The 4-cyano-phenyl

Me

H

F

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

7-2214

2-chloropyridine-3-base

Me

H

F

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

7-2246

Phenyl

Me

H

H

F

H

H

F

H

Seven fluorine sec.-propyls

H

F

7-2247

The 3-cyano-phenyl

Me

H

H

F

H

H

F

H

Seven fluorine sec.-propyls

H

F

7-2248

The 4-cyano-phenyl

Me

H

H

F

H

H

F

H

Seven fluorine sec.-propyls

H

F

7-2249

2-chloropyridine-3-base

Me

H

H

F

H

H

F

H

Seven fluorine sec.-propyls

H

F

7-2250

Phenyl

Me

H

H

F

H

H

F

H

Nine fluoro-2-butyl

H

F

7-2251

The 3-cyano-phenyl

Me

H

H

F

H

H

F

H

Nine fluoro-2-butyl

H

F

7-2252

The 4-cyano-phenyl

Me

H

H

F

H

H

F

H

Nine fluoro-2-butyl

H

F

7-2253

2-chloropyridine-3-base

Me

H

H

F

H

H

F

H

Nine fluoro-2-butyl

H

F

7-2254

Phenyl

Me

H

H

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

7-2274

The 3-cyano-phenyl

Me

H

H

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

7-2275

The 4-cyano-phenyl

Me

H

H

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

7-2290

2-chloropyridine-3-base

Me

H

H

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

7-2332

Phenyl

Me

H

H

F

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

7-2352

The 3-cyano-phenyl

Me

H

H

F

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

7-2353

The 4-cyano-phenyl

Me

H

H

F

H

H

Cl

H

Nine fluoro-2-butyl

H

CH

[table 61]

The 7th table (10)

[table 62]

The 7th table (11)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

7-4027

2-chloropyridine-3-base

Me

H

F

F

H

H

F

H

Nine fluoro-2-butyl

H

F

7-4028

Phenyl

Me

H

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

7-4048

The 3-cyano-phenyl

Me

H

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

7-4049

The 4-cyano-phenyl

Me

H

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

7-4064

2-chloropyridine-3-base

Me

H

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

7-4106

Phenyl

Me

H

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

7-4126

The 3-cyano-phenyl

Me

H

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

7-4127

The 4-cyano-phenyl

Me

H

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

7-4142

2-chloropyridine-3-base

Me

H

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

7-4184

Phenyl

Me

H

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

7-4204

The 3-cyano-phenyl

Me

H

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

7-4205

The 4-cyano-phenyl

Me

H

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

7-4220

2-chloropyridine-3-base

Me

H

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

7-4262

Phenyl

Me

H

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

Br

7-4282

The 3-cyano-phenyl

Me

H

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

Br

7-4283

The 4-cyano-phenyl

Me

H

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

Br

7-4298

2-chloropyridine-3-base

Me

H

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

Br

7-4340

Phenyl

Me

H

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

I

7-4360

The 3-cyano-phenyl

Me

H

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

I

7-4361

The 4-cyano-phenyl

Me

H

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

I

7-4376

2-chloropyridine-3-base

Me

H

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

I

7-4418

Phenyl

Me

H

F

F

H

H

I

H

Nine fluoro-2-butyl

H

I

7-4438

The 3-cyano-phenyl

Me

H

F

F

H

H

I

H

Nine fluoro-2-butyl

H

I

7-4439

The 4-cyano-phenyl

Me

H

F

F

H

H

I

H

Nine fluoro-2-butyl

H

I

7-4454

2-chloropyridine-3-base

Me

H

F

F

H

H

I

H

Nine fluoro-2-butyl

H

I

7-4496

Phenyl

Me

H

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

7-4516

The 3-cyano-phenyl

Me

H

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

7-4517

The 4-cyano-phenyl

Me

H

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

7-4532

2-chloropyridine-3-base

Me

H

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

7-4574

Phenyl

Me

H

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

7-4594

The 3-cyano-phenyl

Me

H

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

7-4595

The 4-cyano-phenyl

Me

H

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

7-4610

2-chloropyridine-3-base

Me

H

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

7-4652

Phenyl

Me

H

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

7-4672

The 3-cyano-phenyl

Me

H

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

7-4673

The 4-cyano-phenyl

Me

H

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

7-4688

2-chloropyridine-3-base

Me

H

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

7-4730

Phenyl

Me

H

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

7-4750

The 3-cyano-phenyl

Me

H

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

7-4751

The 4-cyano-phenyl

Me

H

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

7-4766

2-chloropyridine-3-base

Me

H

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

[table 63]

The 7th table (12)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

7-5220

The 3-cyano-phenyl

Me

H

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-5221

The 4-cyano-phenyl

Me

H

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-5236

2-chloropyridine-3-base

Me

H

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-5278

Phenyl

Me

H

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

7-5298

The 3-cyano-phenyl

Me

H

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

7-5299

The 4-cyano-phenyl

Me

H

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

7-5314

2-chloropyridine-3-base

Me

H

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

7-5356

Phenyl

Me

H

F

F

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-5376

The 3-cyano-phenyl

Me

H

F

F

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-5377

The 4-cyano-phenyl

Me

H

F

F

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-5392

2-chloropyridine-3-base

Me

H

F

F

H

H

I

H

Nine fluoro-2-butyl

H

CF3

7-5434

Phenyl

Me

H

F

F

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

7-5465

2-chloropyridine-3-base

Me

H

F

F

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

7-5490

Phenyl

Me

H

F

F

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

7-5521

2-chloropyridine-3-base

Me

H

F

F

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

7-5546

Phenyl

Me

H

F

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

7-5577

2-chloropyridine-3-base

Me

H

F

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

7-5602

Phenyl

Me

H

F

F

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

7-5633

2-chloropyridine-3-base

Me

H

F

F

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

7-5658

Phenyl

Me

H

F

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

7-5678

The 3-cyano-phenyl

Me

H

F

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

7-5679

The 4-cyano-phenyl

Me

H

F

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

7-5694

2-chloropyridine-3-base

Me

H

F

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

7-5726

Phenyl

Me

H

F

F

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

7-5746

The 3-cyano-phenyl

Me

H

F

F

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

7-5747

The 4-cyano-phenyl

Me

H

F

F

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

7-5762

2-chloropyridine-3-base

Me

H

F

F

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

7-5794

Phenyl

Me

H

F

F

F

H

Cl

H

Pentafluoroethyl group

H

Cl

7-5795

Phenyl

Me

H

F

F

F

H

Br

H

Seven fluorine sec.-propyls

H

Br

7-5796

Phenyl

Me

H

F

F

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

7-5797

Phenyl

Me

H

F

F

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

7-5798

Phenyl

Me

H

F

F

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

7-5799

Phenyl

Me

H

F

F

F

H

I

H

Nine fluoro-2-butyl

H

I

7-5800

Phenyl

Me

H

F

F

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

7-5801

Phenyl

Me

H

F

F

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-5802

Phenyl

Me

H

F

F

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

7-5803

Phenyl

Me

H

H

H

F

H

Cl

H

Pentafluoroethyl group

H

Cl

7-5804

Phenyl

Me

H

H

H

F

H

Br

H

Seven fluorine sec.-propyls

H

Br

7-5805

Phenyl

Me

H

H

H

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

7-5806

Phenyl

Me

H

H

H

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

7-5807

Phenyl

Me

H

H

H

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

[table 64]

The 7th table (13)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

7-5831

Phenyl

Me

H

F

H

H

F

Br

H

Seven fluorine sec.-propyls

H

Br

7-5832

Phenyl

Me

H

F

H

H

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

7-5833

Phenyl

Me

H

F

H

H

F

I

H

Seven fluorine sec.-propyls

H

CF3

7-5834

Phenyl

Me

H

F

H

H

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

7-5835

Phenyl

Me

H

F

H

H

F

I

H

Nine fluoro-2-butyl

H

I

7-5836

Phenyl

Me

H

F

H

H

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

7-5837

Phenyl

Me

H

F

H

H

F

Br

H

Nine fluoro-2-butyl

H

CF3

7-5838

Phenyl

Me

H

F

H

H

F

CF3

H

Nine fluoro-2-butyl

H

CF3

7-5839

Phenyl

Me

H

H

F

F

H

Cl

H

Pentafluoroethyl group

H

Cl

7-5840

Phenyl

Me

H

H

F

F

H

Br

H

Seven fluorine sec.-propyls

H

Br

7-5841

Phenyl

Me

H

H

F

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

7-5842

Phenyl

Me

H

H

F

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

7-5843

Phenyl

Me

H

H

F

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

7-5844

Phenyl

Me

H

H

F

F

H

I

H

Nine fluoro-2-butyl

H

I

7-5845

Phenyl

Me

H

H

F

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

7-5846

Phenyl

Me

H

H

F

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

7-5847

Phenyl

Me

H

H

F

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

7-5848

Phenyl

Me

H

H

F

H

F

Cl

H

Pentafluoroethyl group

H

Cl

7-5849

Phenyl

Me

H

H

F

H

F

Br

H

Seven fluorine sec.-propyls

H

Br

7-5850

Phenyl

Me

H

H

F

H

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

7-5851

Phenyl

Me

H

H

F

H

F

I

H

Seven fluorine sec.-propyls

H

CF3

7-5852

Phenyl

Me

H

H

F

H

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

7-5853

Phenyl

Me

H

H

F

H

F

I

H

Nine fluoro-2-butyl

H

I

7-5854

Phenyl

Me

H

H

F

H

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

7-5855

Phenyl

Me

H

H

F

H

F

Br

H

Nine fluoro-2-butyl

H

CF3

7-5856

Phenyl

Me

H

H

F

H

F

CF3

H

Nine fluoro-2-butyl

H

CF3

7-5857

Phenyl

Me

H

H

H

F

F

Cl

H

Pentafluoroethyl group

H

Cl

7-5858

Phenyl

Me

H

H

H

F

F

Br

H

Seven fluorine sec.-propyls

H

Br

7-5859

Phenyl

Me

H

H

H

F

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

7-5860

Phenyl

Me

H

H

H

F

F

I

H

Seven fluorine sec.-propyls

H

CF3

7-5861

Phenyl

Me

H

H

H

F

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

7-5862

Phenyl

Me

H

H

H

F

F

I

H

Nine fluoro-2-butyl

H

I

7-5863

Phenyl

Me

H

H

H

F

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

7-5864

Phenyl

Me

H

H

H

F

F

Br

H

Nine fluoro-2-butyl

H

CF3

[table 65]

The 7th table (14)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

7-5894

Phenyl

Me

H

F

F

F

F

Br

H

Seven fluorine sec.-propyls

H

Br

7-5895

Phenyl

Me

H

F

F

F

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

7-5896

Phenyl

Me

H

F

F

F

F

I

H

Seven fluorine sec.-propyls

H

CF3

7-5897

Phenyl

Me

H

F

F

F

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

7-5898

Phenyl

Me

H

F

F

F

F

I

H

Nine fluoro-2-butyl

H

I

7-5899

Phenyl

Me

H

F

F

F

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

7-5900

Phenyl

Me

H

F

F

F

F

Br

H

Nine fluoro-2-butyl

H

CF3

7-5901

Phenyl

Me

H

F

F

F

F

CF3

H

Nine fluoro-2-butyl

H

CF3

7-5902

Phenyl

Me

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

Br

7-5903

2-chloropyridine-3-base

Me

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

Br

7-5904

The 3-fluorophenyl

Me

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

I

7-5905

The 4-fluorophenyl

Me

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

I

7-5906

The 3-fluorophenyl

Me

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

7-5907

The 4-fluorophenyl

Me

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

7-5908

4-(methyl sulphonyl) phenyl

Me

H

H

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

7-5909

Pyrimidine-5-base

Me

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

7-5910

3-cyano group-5-(methoxycarbonyl) phenyl

Me

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

7-5911

Phenyl

Me

H

H

H

H

H

Br

H

Pentafluoroethyl group

H

CF3

7-5912

2-chloropyridine-3-base

Me

H

H

H

H

H

Br

H

Pentafluoroethyl group

H

CF3

[table 66]

The 8th table (1)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

8-1

Phenyl

H

Me

H

H

H

H

F

H

Nine fluoro-2-butyl

H

F

8-2

The 3-cyano-phenyl

H

Me

H

H

H

H

F

H

Nine fluoro-2-butyl

H

F

8-3

The 4-cyano-phenyl

H

Me

H

H

H

H

F

H

Nine fluoro-2-butyl

H

F

8-4

2-chloropyridine-3-base

H

Me

H

H

H

H

F

H

Nine fluoro-2-butyl

H

F

8-5

Phenyl

H

Me

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

8-12

The 3-cyano-phenyl

H

Me

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

8-13

The 4-cyano-phenyl

H

Me

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

8-24

2-chloropyridine-3-base

H

Me

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

8-38

Phenyl

H

Me

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

8-45

The 3-cyano-phenyl

H

Me

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

8-46

The 4-cyano-phenyl

H

Me

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

8-57

2-chloropyridine-3-base

H

Me

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

8-71

Phenyl

H

Me

H

H

H

H

I

H

Nine fluoro-2-butyl

H

I

8-78

The 3-cyano-phenyl

H

Me

H

H

H

H

I

H

Nine fluoro-2-butyl

H

I

8-79

The 4-cyano-phenyl

H

Me

H

H

H

H

I

H

Nine fluoro-2-butyl

H

I

8-90

2-chloropyridine-3-base

H

Me

H

H

H

H

I

H

Nine fluoro-2-butyl

H

I

8-104

Phenyl

H

Me

H

H

H

H

F

H

Nine fluoro-2-butyl

H

Cl

8-105

Phenyl

H

Me

H

H

H

H

F

H

Nine fluoro-2-butyl

H

Br

8-106

Phenyl

H

Me

H

H

H

H

F

H

Nine fluoro-2-butyl

H

I

8-107

Phenyl

H

Me

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Br

8-108

Phenyl

H

Me

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

I

8-109

Phenyl

H

Me

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

I

8-110

Phenyl

H

Me

H

H

H

H

F

H

Seven fluorine sec.-propyls

H

CF3

8-111

Phenyl

H

Me

H

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

8-131

The 3-cyano-phenyl

H

Me

H

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

8-132

The 4-cyano-phenyl

H

Me

H

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

8-147

2-chloropyridine-3-base

H

Me

H

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

8-189

Phenyl

H

Me

H

H

H

H

F

H

Nine fluoro-2-butyl

H

CF3

8-190

Phenyl

H

Me

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

8-210

The 3-cyano-phenyl

H

Me

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

8-211

The 4-cyano-phenyl

H

Me

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

8-226

2-chloropyridine-3-base

H

Me

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

[table 67]

The 8th table (2)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

8-748

Phenyl

H

Me

H

H

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

8-779

2-chloropyridine-3-base

H

Me

H

H

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

8-804

Phenyl

H

Me

H

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

8-824

The 3-cyano-phenyl

H

Me

H

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

8-825

The 4-cyano-phenyl

H

Me

H

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

8-840

2-chloropyridine-3-base

H

Me

H

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

8-841

2-bromopyridine-3-base

H

Me

H

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

8-872

Phenyl

H

Me

H

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

8-892

The 3-cyano-phenyl

H

Me

H

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

8-893

The 4-cyano-phenyl

H

Me

H

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

8-908

2-chloropyridine-3-base

H

Me

H

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

8-940

Phenyl

H

Me

F

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

8-941

The 3-cyano-phenyl

H

Me

F

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

8-942

The 4-cyano-phenyl

H

Me

F

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

8-943

2-chloropyridine-3-base

H

Me

F

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

8-944

Phenyl

H

Me

F

H

H

H

F

H

Nine fluoro-2-butyl

H

F

8-945

The 3-cyano-phenyl

H

Me

F

H

H

H

F

H

Nine fluoro-2-butyl

H

F

8-946

The 4-cyano-phenyl

H

Me

F

H

H

H

F

H

Nine fluoro-2-butyl

H

F

8-947

2-chloropyridine-3-base

H

Me

F

H

H

H

F

H

Nine fluoro-2-butyl

H

F

8-948

Phenyl

H

Me

F

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

8-952

The 2-chloro-phenyl-

H

Me

F

H

H

H

F

H

Seven fluorine sec.-propyls

H

Cl

8-956

The 3-bromophenyl

H

Me

F

H

H

H

F

H

Seven fluorine sec.-propyls

H

Br

8-961

(2-trifluoromethyl) phenyl

H

i-Pr

F

H

H

H

F

H

Seven fluorine sec.-propyls

H

I

8-964

The 2-nitrophenyl

H

Me

F

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Br

8-968

The 3-cyano-phenyl

H

Me

F

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

8-969

The 4-cyano-phenyl

H

Me

F

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

8-970

2, the 6-difluorophenyl

H

Me

F

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

I

8-982

Pyridin-3-yl

H

Me

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

I

8-984

2-chloropyridine-3-base

H

Me

F

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

8-1026

Phenyl

H

Me

F

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

8-1046

The 3-cyano-phenyl

H

Me

F

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

8-1047

The 4-cyano-phenyl

H

Me

F

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

8-1062

2-chloropyridine-3-base

H

Me

F

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

8-1104

Phenyl

H

Me

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

8-1124

The 3-cyano-phenyl

H

Me

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

8-1125

The 4-cyano-phenyl

H

Me

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

8-1140

2-chloropyridine-3-base

H

Me

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

8-1182

Phenyl

H

Me

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

8-1202

The 3-cyano-phenyl

H

Me

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

8-1203

The 4-cyano-phenyl

H

Me

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

8-1218

2-chloropyridine-3-base

H

Me

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

[table 68]

The 8th table (3)

[table 69]

The 8th table (4)

8-3112

Phenyl

H

Me

H

F

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

8-3132

The 3-cyano-phenyl

H

Me

H

F

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

8-3133

The 4-cyano-phenyl

H

Me

H

F

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

8-3148

2-chloropyridine-3-base

H

Me

H

F

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

8-3190

Phenyl

H

Me

H

F

H

H

F

H

Seven fluorine sec.-propyls

H

CF3

8-3191

Phenyl

H

Me

H

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

8-3211

The 3-cyano-phenyl

H

Me

H

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

8-3212

The 4-cyano-phenyl

H

Me

H

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

8-3227

2-chloropyridine-3-base

H

Me

H

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

8-3269

Phenyl

H

Me

H

F

H

H

F

H

Nine fluoro-2-butyl

H

CF3

8-3270

Phenyl

H

Me

H

F

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

8-3290

The 3-cyano-phenyl

H

Me

H

F

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

8-3291

The 4-cyano-phenyl

H

Me

H

F

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

8-3306

2-chloropyridine-3-base

H

Me

H

F

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

8-3348

Phenyl

H

Me

H

F

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

8-3368

The 3-cyano-phenyl

H

Me

H

F

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

8-3369

The 4-cyano-phenyl

H

Me

H

F

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

8-3384

2-chloropyridine-3-base

H

Me

H

F

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

8-3426

Phenyl

H

Me

H

F

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

8-3446

The 3-cyano-phenyl

H

Me

H

F

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

8-3447

The 4-cyano-phenyl

H

Me

H

F

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

[table 70]

The 8th table (5)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

8-3462

2-chloropyridine-3-base

H

Me

H

F

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

8-3504

Phenyl

H

Me

H

F

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

8-3524

The 3-cyano-phenyl

H

Me

H

F

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

8-3525

The 4-cyano-phenyl

H

Me

H

F

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

8-3540

2-chloropyridine-3-base

H

Me

H

F

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

8-3582

Phenyl

H

Me

H

F

H

H

I

H

Nine fluoro-2-butyl

H

CF3

8-3602

The 3-cyano-phenyl

H

Me

H

F

H

H

I

H

Nine fluoro-2-butyl

H

CF3

8-3603

The 4-cyano-phenyl

H

Me

H

F

H

H

I

H

Nine fluoro-2-butyl

H

CF3

8-3618

2-chloropyridine-3-base

H

Me

H

F

H

H

I

H

Nine fluoro-2-butyl

H

CF3

8-3660

Phenyl

H

Me

H

F

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

8-3691

2-chloropyridine-3-base

H

Me

H

F

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

8-3716

Phenyl

H

Me

H

F

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

8-3747

2-chloropyridine-3-base

H

Me

H

F

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

8-3772

Phenyl

H

Me

H

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

8-3803

2-chloropyridine-3-base

H

Me

H

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

8-3828

Phenyl

H

Me

H

F

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

8-3859

2-chloropyridine-3-base

H

Me

H

F

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

8-3884

Phenyl

H

Me

H

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

8-3904

The 3-cyano-phenyl

H

Me

H

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

8-3905

The 4-cyano-phenyl

H

Me

H

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

8-3920

2-chloropyridine-3-base

H

Me

H

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

8-3952

Phenyl

H

Me

H

F

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

8-3972

The 3-cyano-phenyl

H

Me

H

F

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

8-3973

The 4-cyano-phenyl

H

Me

H

F

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

8-3988

2-chloropyridine-3-base

H

Me

H

F

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

8-4020

Phenyl

H

Me

F

F

H

H

F

H

Seven fluorine sec.-propyls

H

F

8-4021

The 3-cyano-phenyl

H

Me

F

F

H

H

F

H

Seven fluorine sec.-propyls

H

F

8-4022

The 4-cyano-phenyl

H

Me

F

F

H

H

F

H

Seven fluorine sec.-propyls

H

F

8-4023

2-chloropyridine-3-base

H

Me

F

F

H

H

F

H

Seven fluorine sec.-propyls

H

F

8-4024

Phenyl

H

Me

F

F

H

H

F

H

Nine fluoro-2-butyl

H

F

8-4025

The 3-cyano-phenyl

H

Me

F

F

H

H

F

H

Nine fluoro-2-butyl

H

F

8-4026

The 4-cyano-phenyl

H

Me

F

F

H

H

F

H

Nine fluoro-2-butyl

H

F

8-4027

2-chloropyridine-3-base

H

Me

F

F

H

H

F

H

Nine fluoro-2-butyl

H

F

8-4028

Phenyl

H

Me

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

8-4048

The 3-cyano-phenyl

H

Me

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

8-4049

The 4-cyano-phenyl

H

Me

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

8-4064

2-chloropyridine-3-base

H

Me

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

8-4106

Phenyl

H

Me

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

8-4126

The 3-cyano-phenyl

H

Me

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

8-4127

The 4-cyano-phenyl

H

Me

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

8-4142

2-chloropyridine-3-base

H

Me

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

8-4184

Phenyl

H

Me

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

[table 71]

The 8th table (6)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

8-4610

2-chloropyridine-3-base

H

Me

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

8-4652

Phenyl

H

Me

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

8-4672

The 3-cyano-phenyl

H

Me

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

8-4673

The 4-cyano-phenyl

H

Me

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

8-4688

2-chloropyridine-3-base

H

Me

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

8-4730

Phenyl

H

Me

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

8-4750

The 3-cyano-phenyl

H

Me

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

8-4751

The 4-cyano-phenyl

H

Me

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

8-4808

Phenyl

H

Me

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

8-4828

The 3-cyano-phenyl

H

Me

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

8-4829

The 4-cyano-phenyl

H

Me

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

8-4844

2-chloropyridine-3-base

H

Me

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

8-4886

Phenyl

H

Me

F

F

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

8-4906

The 3-cyano-phenyl

H

Me

F

F

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

8-4907

The 4-cyano-phenyl

H

Me

F

F

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

8-4922

2-chloropyridine-3-base

H

Me

F

F

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

8-4964

Phenyl

H

Me

F

F

H

H

F

H

Seven fluorine sec.-propyls

H

CF3

8-4965

Phenyl

H

Me

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

8-4985

The 3-cyano-phenyl

H

Me

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

8-4986

The 4-cyano-phenyl

H

Me

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

8-5001

2-chloropyridine-3-base

H

Me

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

8-5043

Phenyl

H

Me

F

F

H

H

F

H

Nine fluoro-2-butyl

H

CF3

8-5044

Phenyl

H

Me

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

8-5064

The 3-cyano-phenyl

H

Me

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

8-5065

The 4-cyano-phenyl

H

Me

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

8-5080

2-chloropyridine-3-base

H

Me

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

8-5122

Phenyl

H

Me

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

8-5142

The 3-cyano-phenyl

H

Me

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

8-5143

The 4-cyano-phenyl

H

Me

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

8-5158

2-chloropyridine-3-base

H

Me

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

8-5200

Phenyl

H

Me

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

8-5220

The 3-cyano-phenyl

H

Me

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

8-5221

The 4-cyano-phenyl

H

Me

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

8-5236

2-chloropyridine-3-base

H

Me

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

8-5278

Phenyl

H

Me

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

8-5298

The 3-cyano-phenyl

H

Me

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

8-5299

The 4-cyano-phenyl

H

Me

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

8-5314

2-chloropyridine-3-base

H

Me

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

8-5356

Phenyl

H

Me

F

F

H

H

I

H

Nine fluoro-2-butyl

H

CF3

8-5376

The 3-cyano-phenyl

H

Me

F

F

H

H

I

H

Nine fluoro-2-butyl

H

CF3

8-5377

The 4-cyano-phenyl

H

Me

F

F

H

H

I

H

Nine fluoro-2-butyl

H

CF3

8-5392

2-chloropyridine-3-base

H

Me

F

F

H

H

I

H

Nine fluoro-2-butyl

H

CF3

[table 72]

The 8th table (7)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

8-5801

Phenyl

H

Me

F

F

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

8-5802

Phenyl

H

Me

F

F

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

8-5803

Phenyl

H

Me

H

H

F

H

Cl

H

Pentafluoroethyl group

H

Cl

8-5804

Phenyl

H

Me

H

H

F

H

Br

H

Seven fluorine sec.-propyls

H

Br

8-5805

Phenyl

H

Me

H

H

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

8-5806

Phenyl

H

Me

H

H

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

8-5807

Phenyl

H

Me

H

H

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

8-5808

Phenyl

H

Me

H

H

F

H

I

H

Nine fluoro-2-butyl

H

I

8-5809

Phenyl

H

Me

H

H

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

8-5810

Phenyl

H

Me

H

H

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

8-5811

Phenyl

H

Me

H

H

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

8-5812

Phenyl

H

Me

H

H

H

F

Cl

H

Pentafluoroethyl group

H

Cl

8-5813

Phenyl

H

Me

H

H

H

F

Br

H

Seven fluorine sec.-propyls

H

Br

8-5814

Phenyl

H

Me

H

H

H

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

8-5815

Phenyl

H

Me

H

H

H

F

I

H

Seven fluorine sec.-propyls

H

CF3

8-5816

Phenyl

H

Me

H

H

H

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

8-5817

Phenyl

H

Me

H

H

H

F

I

H

Nine fluoro-2-butyl

H

I

8-5818

Phenyl

H

Me

H

H

H

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

8-5819

Phenyl

H

Me

H

H

H

F

Br

H

Nine fluoro-2-butyl

H

CF3

8-5820

Phenyl

H

Me

H

H

H

F

CF3

H

Nine fluoro-2-butyl

H

CF3

8-5821

Phenyl

H

Me

F

H

F

H

Cl

H

Pentafluoroethyl group

H

Cl

8-5822

Phenyl

H

Me

F

H

F

H

Br

H

Seven fluorine sec.-propyls

H

Br

8-5823

Phenyl

H

Me

F

H

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

8-5824

Phenyl

H

Me

F

H

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

8-5825

Phenyl

H

Me

F

H

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

8-5826

Phenyl

H

Me

F

H

F

H

I

H

Nine fluoro-2-butyl

H

I

8-5827

Phenyl

H

Me

F

H

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

8-5828

Phenyl

H

Me

F

H

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

8-5829

Phenyl

H

Me

F

H

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

8-5830

Phenyl

H

Me

F

H

H

F

Cl

H

Pentafluoroethyl group

H

Cl

8-5831

Phenyl

H

Me

F

H

H

F

Br

H

Seven fluorine sec.-propyls

H

Br

8-5832

Phenyl

H

Me

F

H

H

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

8-5833

Phenyl

H

Me

F

H

H

F

I

H

Seven fluorine sec.-propyls

H

CF3

8-5834

Phenyl

H

Me

F

H

H

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

8-5835

Phenyl

H

Me

F

H

H

F

I

H

Nine fluoro-2-butyl

H

I

8-5836

Phenyl

H

Me

F

H

H

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

8-5837

Phenyl

H

Me

F

H

H

F

Br

H

Nine fluoro-2-butyl

H

CF3

8-5838

Phenyl

H

Me

F

H

H

F

CF3

H

Nine fluoro-2-butyl

H

CF3

8-5839

Phenyl

H

Me

H

F

F

H

Cl

H

Pentafluoroethyl group

H

Cl

8-5840

Phenyl

H

Me

H

F

F

H

Br

H

Seven fluorine sec.-propyls

H

Br

8-5841

Phenyl

H

Me

H

F

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

8-5842

Phenyl

H

Me

H

F

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

[table 73]

The 8th table (8)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

8-5865

Phenyl

H

Me

H

H

F

F

CF3

H

Nine fluoro-2-butyl

H

CF3

8-5866

Phenyl

H

Me

F

F

H

F

Cl

H

Pentafluoroethyl group

H

Cl

8-5867

Phenyl

H

Me

F

F

H

F

Br

H

Seven fluorine sec.-propyls

H

Br

8-5868

Phenyl

H

Me

F

F

H

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

8-5869

Phenyl

H

Me

F

F

H

F

I

H

Seven fluorine sec.-propyls

H

CF3

8-5870

Phenyl

H

Me

F

F

H

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

8-5871

Phenyl

H

Me

F

F

H

F

I

H

Nine fluoro-2-butyl

H

I

8-5872

Phenyl

H

Me

F

F

H

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

8-5873

Phenyl

H

Me

F

F

H

F

Br

H

Nine fluoro-2-butyl

H

CF3

8-5874

Phenyl

H

Me

F

F

H

F

CF3

H

Nine fluoro-2-butyl

H

CF3

8-5875

Phenyl

H

Me

F

H

F

F

Cl

H

Pentafluoroethyl group

H

Cl

8-5876

Phenyl

H

Me

F

H

F

F

Br

H

Seven fluorine sec.-propyls

H

Br

8-5877

Phenyl

H

Me

F

H

F

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

8-5878

Phenyl

H

Me

F

H

F

F

I

H

Seven fluorine sec.-propyls

H

CF3

8-5879

Phenyl

H

Me

F

H

F

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

8-5880

Phenyl

H

Me

F

H

F

F

I

H

Nine fluoro-2-butyl

H

I

8-5881

Phenyl

H

Me

F

H

F

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

8-5882

Phenyl

H

Me

F

H

F

F

Br

H

Nine fluoro-2-butyl

H

CF3

8-5883

Phenyl

H

Me

F

H

F

F

CF3

H

Nine fluoro-2-butyl

H

CF3

8-5884

Phenyl

H

Me

H

F

F

F

Cl

H

Pentafluoroethyl group

H

Cl

8-5885

Phenyl

H

Me

H

F

F

F

Br

H

Seven fluorine sec.-propyls

H

Br

8-5886

Phenyl

H

Me

H

F

F

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

8-5887

Phenyl

H

Me

H

F

F

F

I

H

Seven fluorine sec.-propyls

H

CF3

8-5888

Phenyl

H

Me

H

F

F

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

8-5889

Phenyl

H

Me

H

F

F

F

I

H

Nine fluoro-2-butyl

H

I

8-5890

Phenyl

H

Me

H

F

F

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

8-5891

Phenyl

H

Me

H

F

F

F

Br

H

Nine fluoro-2-butyl

H

CF3

8-5892

Phenyl

H

Me

H

F

F

F

CF3

H

Nine fluoro-2-butyl

H

CF3

8-5893

Phenyl

H

Me

F

F

F

F

Cl

H

Pentafluoroethyl group

H

Cl

8-5894

Phenyl

H

Me

F

F

F

F

Br

H

Seven fluorine sec.-propyls

H

Br

8-5895

Phenyl

H

Me

F

F

F

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

8-5896

Phenyl

H

Me

F

F

F

F

I

H

Seven fluorine sec.-propyls

H

CF3

8-5897

Phenyl

H

Me

F

F

F

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

8-5898

Phenyl

H

Me

F

F

F

F

I

H

Nine fluoro-2-butyl

H

I

8-5899

Phenyl

H

Me

F

F

F

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

8-5900

Phenyl

H

Me

F

F

F

F

Br

H

Nine fluoro-2-butyl

H

CF3

8-5901

Phenyl

H

Me

F

F

F

F

CF3

H

Nine fluoro-2-butyl

H

CF3

[table 74]

The 9th table (1)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

9-1

Phenyl

Me

Me

H

H

H

H

F

H

Nine fluoro-2-butyl

H

F

9-2

The 3-cyano-phenyl

Me

Me

H

H

H

H

F

H

Nine fluoro-2-butyl

H

F

9-3

The 4-cyano-phenyl

Me

Me

H

H

H

H

F

H

Nine fluoro-2-butyl

H

F

9-4

2-chloropyridine-3-base

Me

Me

H

H

H

H

F

H

Nine fluoro-2-butyl

H

F

9-5

Phenyl

Me

Me

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

9-12

The 3-cyano-phenyl

Me

Me

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

9-13

The 4-cyano-phenyl

Me

Me

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

9-24

2-chloropyridine-3-base

Me

Me

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

9-38

Phenyl

Me

Me

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

9-45

The 3-cyano-phenyl

Me

Me

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

9-46

The 4-cyano-phenyl

Me

Me

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

9-57

2-chloropyridine-3-base

Me

Me

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

9-71

Phenyl

Me

Me

H

H

H

H

I

H

Nine fluoro-2-butyl

H

I

9-78

The 3-cyano-phenyl

Me

Me

H

H

H

H

I

H

Nine fluoro-2-butyl

H

I

9-79

The 4-cyano-phenyl

Me

Me

H

H

H

H

I

H

Nine fluoro-2-butyl

H

I

9-90

2-chloropyridine-3-base

Me

Me

H

H

H

H

I

H

Nine fluoro-2-butyl

H

I

9-109

Phenyl

Me

Me

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Br

9-112

Phenyl

Me

Me

H

H

H

H

F

H

Seven fluorine sec.-propyls

H

CF3

9-113

Phenyl

Me

Me

H

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

9-133

The 3-cyano-phenyl

Me

Me

H

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

9-134

The 4-cyano-phenyl

Me

Me

H

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

9-149

2-chloropyridine-3-base

Me

Me

H

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

9-191

Phenyl

Me

Me

H

H

H

H

F

H

Nine fluoro-2-butyl

H

CF3

9-192

Phenyl

Me

Me

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

9-212

The 3-cyano-phenyl

Me

Me

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

9-213

The 4-cyano-phenyl

Me

Me

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

9-228

2-chloropyridine-3-base

Me

Me

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

9-270

Phenyl

Me

Me

H

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

9-290

The 3-cyano-phenyl

Me

Me

H

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

9-291

The 4-cyano-phenyl

Me

Me

H

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

9-306

2-chloropyridine-3-base

Me

Me

H

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

9-348

Phenyl

Me

Me

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

9-368

The 3-cyano-phenyl

Me

Me

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

9-369

The 4-cyano-phenyl

Me

Me

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

[table 75]

The 9th table (2)

[table 76]

The 9th table (3)

[table 77]

The 9th table (4)

[table 78]

The 9th table (5)

[table 79]

The 9th table (6)

[table 80]

The 9th table (7)

[table 81]

The 9th table (8)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

9-4601

2-chloropyridine-3-base

Me

Me

H

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

9-4643

Phenyl

Me

Me

H

F

H

H

F

H

Nine fluoro-2-butyl

H

CF3

9-4644

Phenyl

Me

Me

H

F

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

9-4664

The 3-cyano-phenyl

Me

Me

H

F

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

9-4665

The 4-cyano-phenyl

Me

Me

H

F

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

9-4680

2-chloropyridine-3-base

Me

Me

H

F

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

9-4722

Phenyl

Me

Me

H

F

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

9-4742

The 3-cyano-phenyl

Me

Me

H

F

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

9-4743

The 4-cyano-phenyl

Me

Me

H

F

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

9-4758

2-chloropyridine-3-base

Me

Me

H

F

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

9-4800

Phenyl

Me

Me

H

F

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

9-4820

The 3-cyano-phenyl

Me

Me

H

F

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

9-4821

The 4-cyano-phenyl

Me

Me

H

F

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

9-4836

2-chloropyridine-3-base

Me

Me

H

F

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

9-4878

Phenyl

Me

Me

H

F

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

9-4898

The 3-cyano-phenyl

Me

Me

H

F

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

9-4899

The 4-cyano-phenyl

Me

Me

H

F

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

9-4914

2-chloropyridine-3-base

Me

Me

H

F

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

9-4956

Phenyl

Me

Me

H

F

H

H

I

H

Nine fluoro-2-butyl

H

CF3

9-4976

The 3-cyano-phenyl

Me

Me

H

F

H

H

I

H

Nine fluoro-2-butyl

H

CF3

9-4977

The 4-cyano-phenyl

Me

Me

H

F

H

H

I

H

Nine fluoro-2-butyl

H

CF3

9-4992

2-chloropyridine-3-base

Me

Me

H

F

H

H

I

H

Nine fluoro-2-butyl

H

CF3

9-5230

Phenyl

Me

Me

H

F

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

9-5261

2-chloropyridine-3-base

Me

Me

H

F

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

9-5286

Phenyl

Me

Me

H

F

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

9-5317

2-chloropyridine-3-base

Me

Me

H

F

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

9-5342

Phenyl

Me

Me

H

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

9-5373

2-chloropyridine-3-base

Me

Me

H

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

9-5398

Phenyl

Me

Me

H

F

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

9-5429

2-chloropyridine-3-base

Me

Me

H

F

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

9-5454

Phenyl

Me

Me

H

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

9-5474

The 3-cyano-phenyl

Me

Me

H

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

9-5475

The 4-cyano-phenyl

Me

Me

H

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

9-5490

2-chloropyridine-3-base

Me

Me

H

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

9-5522

Phenyl

Me

Me

H

F

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

9-5542

The 3-cyano-phenyl

Me

Me

H

F

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

9-5543

The 4-cyano-phenyl

Me

Me

H

F

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

9-5558

2-chloropyridine-3-base

Me

Me

H

F

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

9-5786

Phenyl

Me

Me

F

F

H

H

F

H

Seven fluorine sec.-propyls

H

F

9-5787

The 3-cyano-phenyl

Me

Me

F

F

H

H

F

H

Seven fluorine sec.-propyls

H

F

9-5788

The 4-cyano-phenyl

Me

Me

F

F

H

H

F

H

Seven fluorine sec.-propyls

H

F

[table 82]

The 9th table (9)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

9-6127

The 4-cyano-phenyl

Me

Me

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

I

9-6142

2-chloropyridine-3-base

Me

Me

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

I

9-6184

Phenyl

Me

Me

F

F

H

H

I

H

Nine fluoro-2-butyl

H

I

9-6204

The 3-cyano-phenyl

Me

Me

F

F

H

H

I

H

Nine fluoro-2-butyl

H

I

9-6205

The 4-cyano-phenyl

Me

Me

F

F

H

H

I

H

Nine fluoro-2-butyl

H

I

9-6220

2-chloropyridine-3-base

Me

Me

F

F

H

H

I

H

Nine fluoro-2-butyl

H

I

9-6458

Phenyl

Me

Me

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

9-6478

The 3-cyano-phenyl

Me

Me

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

9-6479

The 4-cyano-phenyl

Me

Me

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

9-6494

2-chloropyridine-3-base

Me

Me

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

9-6536

Phenyl

Me

Me

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

9-6556

The 3-cyano-phenyl

Me

Me

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

9-6557

The 4-cyano-phenyl

Me

Me

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

9-6572

2-chloropyridine-3-base

Me

Me

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

9-6614

Phenyl

Me

Me

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

9-6634

The 3-cyano-phenyl

Me

Me

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

9-6635

The 4-cyano-phenyl

Me

Me

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

9-6650

2-chloropyridine-3-base

Me

Me

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

9-6692

Phenyl

Me

Me

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

9-6712

The 3-cyano-phenyl

Me

Me

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

9-6713

The 4-cyano-phenyl

Me

Me

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

9-6728

2-chloropyridine-3-base

Me

Me

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

9-6770

Phenyl

Me

Me

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

9-6790

The 3-cyano-phenyl

Me

Me

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

9-6791

The 4-cyano-phenyl

Me

Me

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

9-6806

2-chloropyridine-3-base

Me

Me

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

9-6848

Phenyl

Me

Me

F

F

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

9-6868

The 3-cyano-phenyl

Me

Me

F

F

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

9-6869

The 4-cyano-phenyl

Me

Me

F

F

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

9-6884

2-chloropyridine-3-base

Me

Me

F

F

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

9-7122

Phenyl

Me

Me

F

F

H

H

F

H

Seven fluorine sec.-propyls

H

CF3

9-7123

Phenyl

Me

Me

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

9-7143

The 3-cyano-phenyl

Me

Me

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

9-7144

The 4-cyano-phenyl

Me

Me

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

9-7159

2-chloropyridine-3-base

Me

Me

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

9-7201

Phenyl

Me

Me

F

F

H

H

F

H

Nine fluoro-2-butyl

H

CF3

9-7202

Phenyl

Me

Me

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

9-7222

The 3-cyano-phenyl

Me

Me

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

9-7223

The 4-cyano-phenyl

Me

Me

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

9-7238

2-chloropyridine-3-base

Me

Me

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

9-7280

Phenyl

Me

Me

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

[table 83]

The 9th table (10)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

9-8012

Phenyl

Me

Me

F

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

9-8032

The 3-cyano-phenyl

Me

Me

F

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

9-8033

The 4-cyano-phenyl

Me

Me

F

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

9-8048

2-chloropyridine-3-base

Me

Me

F

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

9-8080

Phenyl

Me

Me

F

F

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

9-8100

The 3-cyano-phenyl

Me

Me

F

F

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

9-8101

The 4-cyano-phenyl

Me

Me

F

F

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

9-8116

2-chloropyridine-3-base

Me

Me

F

F

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

9-8344

Phenyl

Me

Me

F

F

F

H

Cl

H

Pentafluoroethyl group

H

Cl

9-8345

Phenyl

Me

Me

F

F

F

H

Br

H

Seven fluorine sec.-propyls

H

Br

9-8346

Phenyl

Me

Me

F

F

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

9-8347

Phenyl

Me

Me

F

F

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

9-8348

Phenyl

Me

Me

F

F

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

9-8349

Phenyl

Me

Me

F

F

F

H

I

H

Nine fluoro-2-butyl

H

I

9-8350

Phenyl

Me

Me

F

F

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

9-8351

Phenyl

Me

Me

F

F

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

9-8352

Phenyl

Me

Me

F

F

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

9-8353

Phenyl

Me

Me

H

H

F

H

Cl

H

Pentafluoroethyl group

H

Cl

9-8354

Phenyl

Me

Me

H

H

F

H

Br

H

Seven fluorine sec.-propyls

H

Br

9-8355

Phenyl

Me

Me

H

H

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

9-8356

Phenyl

Me

Me

H

H

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

9-8357

Phenyl

Me

Me

H

H

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

9-8358

Phenyl

Me

Me

H

H

F

H

I

H

Nine fluoro-2-butyl

H

I

9-8359

Phenyl

Me

Me

H

H

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

9-8360

Phenyl

Me

Me

H

H

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

9-8361

Phenyl

Me

Me

H

H

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

9-8362

Phenyl

Me

Me

H

H

H

F

Cl

H

Pentafluoroethyl group

H

Cl

9-8363

Phenyl

Me

Me

H

H

H

F

Br

H

Seven fluorine sec.-propyls

H

Br

9-8364

Phenyl

Me

Me

H

H

H

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

9-8365

Phenyl

Me

Me

H

H

H

F

I

H

Seven fluorine sec.-propyls

H

CF3

9-8366

Phenyl

Me

Me

H

H

H

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

9-8367

Phenyl

Me

Me

H

H

H

F

I

H

Nine fluoro-2-butyl

H

I

9-8368

Phenyl

Me

Me

H

H

H

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

9-8369

Phenyl

Me

Me

H

H

H

F

Br

H

Nine fluoro-2-butyl

H

CF3

9-8370

Phenyl

Me

Me

H

H

H

F

CF3

H

Nine fluoro-2-butyl

H

CF3

9-8371

Phenyl

Me

Me

F

H

F

H

Cl

H

Pentafluoroethyl group

H

Cl

9-8372

Phenyl

Me

Me

F

H

F

H

Br

H

Seven fluorine sec.-propyls

H

Br

9-8373

Phenyl

Me

Me

F

H

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

9-8374

Phenyl

Me

Me

F

H

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

9-8375

Phenyl

Me

Me

F

H

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

9-8376

Phenyl

Me

Me

F

H

F

H

I

H

Nine fluoro-2-butyl

H

I

[table 84]

The 9th table (11)

The compound sequence number

Q 1

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

9-8400

Phenyl

Me

Me

H

F

H

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

9-8401

Phenyl

Me

Me

H

F

H

F

I

H

Seven fluorine sec.-propyls

H

CF3

9-8402

Phenyl

Me

Me

H

F

H

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

9-8403

Phenyl

Me

Me

H

F

H

F

I

H

Nine fluoro-2-butyl

H

I

9-8404

Phenyl

Me

Me

H

F

H

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

9-8405

Phenyl

Me

Me

H

F

H

F

Br

H

Nine fluoro-2-butyl

H

CF3

9-8406

Phenyl

Me

Me

H

F

H

F

CF3

H

Nine fluoro-2-butyl

H

CF3

9-8407

Phenyl

Me

Me

H

H

F

F

Cl

H

Pentafluoroethyl group

H

Cl

9-8408

Phenyl

Me

Me

H

H

F

F

Br

H

Seven fluorine sec.-propyls

H

Br

9-8409

Phenyl

Me

Me

H

H

F

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

9-8410

Phenyl

Me

Me

H

H

F

F

I

H

Seven fluorine sec.-propyls

H

CF3

9-8411

Phenyl

Me

Me

H

H

F

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

9-8412

Phenyl

Me

Me

H

H

F

F

I

H

Nine fluoro-2-butyl

H

I

9-8413

Phenyl

Me

Me

H

H

F

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

9-8414

Phenyl

Me

Me

H

H

F

F

Br

H

Nine fluoro-2-butyl

H

CF3

9-8415

Phenyl

Me

Me

H

H

F

F

CF3

H

Nine fluoro-2-butyl

H

CF3

9-8416

Phenyl

Me

Me

F

F

H

F

Cl

H

Pentafluoroethyl group

H

Cl

9-8417

Phenyl

Me

Me

F

F

H

F

Br

H

Seven fluorine sec.-propyls

H

Br

9-8418

Phenyl

Me

Me

F

F

H

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

9-8419

Phenyl

Me

Me

F

F

H

F

I

H

Seven fluorine sec.-propyls

H

CF3

9-8420

Phenyl

Me

Me

F

F

H

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

9-8421

Phenyl

Me

Me

F

F

H

F

I

H

Nine fluoro-2-butyl

H

I

9-8422

Phenyl

Me

Me

F

F

H

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

9-8423

Phenyl

Me

Me

F

F

H

F

Br

H

Nine fluoro-2-butyl

H

CF3

9-8424

Phenyl

Me

Me

F

F

H

F

CF3

H

Nine fluoro-2-butyl

H

CF3

9-8425

Phenyl

Me

Me

F

H

F

F

Cl

H

Pentafluoroethyl group

H

Cl

9-8426

Phenyl

Me

Me

F

H

F

F

Br

H

Seven fluorine sec.-propyls

H

Br

9-8427

Phenyl

Me

Me

F

H

F

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

9-8428

Phenyl

Me

Me

F

H

F

F

I

H

Seven fluorine sec.-propyls

H

CF3

9-8429

Phenyl

Me

Me

F

H

F

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

9-8430

Phenyl

Me

Me

F

H

F

F

I

H

Nine fluoro-2-butyl

H

I

9-8431

Phenyl

Me

Me

F

H

F

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

9-8432

Phenyl

Me

Me

F

H

F

F

Br

H

Nine fluoro-2-butyl

H

CF3

9-8433

Phenyl

Me

Me

F

H

F

F

CF3

H

Nine fluoro-2-butyl

H

CF3

9-8434

Phenyl

Me

Me

H

F

F

F

Cl

H

Pentafluoroethyl group

H

Cl

9-8435

Phenyl

Me

Me

H

F

F

F

Br

H

Seven fluorine sec.-propyls

H

Br

9-8436

Phenyl

Me

Me

H

F

F

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

9-8437

Phenyl

Me

Me

H

F

F

F

I

H

Seven fluorine sec.-propyls

H

CF3

9-8438

Phenyl

Me

Me

H

F

F

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

9-8439

Phenyl

Me

Me

H

F

F

F

I

H

Nine fluoro-2-butyl

H

I

9-8440

Phenyl

Me

Me

H

F

F

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

[table 85]

The 10th table (1)

[table 86]

The 10th table (2)

[table 87]

The 10th table (3)

[table 88]

The 10th table (4)

[table 89]

The 10th table (5)

[table 90]

The 11st table (1)

[table 91]

The 11st table (2)

The compound sequence number

Q 2

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

11-612

3,3,3-three fluoro-n-propyl group

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

11-613

The n-butyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

11-614

4,4,4-three fluoro-n-butyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

11-615

The i-butyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

11-616

The s-butyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

11-617

Vinyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

11-618

Benzyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

11-619

Phenyl

H

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

11-620

Methyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-621

Ethyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-622

The 2-fluoro ethyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-623

The 2-chloroethyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-624

The 2-bromotrifluoromethane

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-625

2-iodine ethyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-626

The 2-cyano ethyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-627

2,2-two fluoro ethyls

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-628

2, the 2-Dichloroethyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-629

2,2, the 2-trifluoroethyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-630

2,2,2-three chloroethyls

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-631

2,2, the 2-three bromomethyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-632

The n-propyl group

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OC2F5

11-633

3-fluoro-n-propyl group

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-634

3-chloro-n-propyl group

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-635

3-bromo-n-propyl group

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-636

The i-propyl group

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-637

1,2-two fluoro-2-propyl group

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-638

1,3-two fluoro-2-propyl group

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-639

1,3-two chloro-2-propyl group

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-640

1-chloro-3-fluoro-2-propyl group

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-641

3,3,3-three fluoro-n-propyl group

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-642

The n-butyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-643

4,4,4-three fluoro-n-butyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-644

The i-butyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-645

The s-butyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-646

Vinyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-647

Benzyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-648

Phenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

11-649

Methyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

11-650

Ethyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

11-651

The 2-fluoro ethyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

11-652

The 2-chloroethyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

[table 92]

The 11st table (3)

The compound sequence number

Q 2

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

11-676

Benzyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

11-677

Phenyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

11-678

Methyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-679

Ethyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-680

The 2-fluoro ethyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-681

The 2-chloroethyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-682

The 2-bromotrifluoromethane

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-683

2-iodine ethyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-684

The 2-cyano ethyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-685

2,2-two fluoro ethyls

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-686

2, the 2-Dichloroethyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-687

2,2, the 2-trifluoroethyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-688

2,2,2-three chloroethyls

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-689

2,2, the 2-three bromomethyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-690

The n-propyl group

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-691

3-fluoro-n-propyl group

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-692

3-chloro-n-propyl group

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-693

3-bromo-n-propyl group

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-694

The i-propyl group

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-695

1,2-two fluoro-2-propyl group

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-696

1,3-two fluoro-2-propyl group

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-697

1,3-two chloro-2-propyl group

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-698

1-chloro-3-fluoro-2-propyl group

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-699

3,3,3-three fluoro-n-propyl group

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-700

The n-butyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-701

4,4,4-three fluoro-n-butyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-702

The i-butyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-703

The s-butyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-704

Vinyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-705

Benzyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OC2F5

11-706

Phenyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

11-707

2,2,2-three chloroethyls

H

H

F

H

H

H

F

H

Seven fluorine sec.-propyls

H

CF3

11-708

2,2,2-three chloroethyls

H

H

F

H

H

H

F

H

Nine fluoro-2-butyl

H

CF3

11-709

Methyl

H

H

F

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

11-710

Ethyl

H

H

F

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

11-711

The 2-fluoro ethyl

H

H

F

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

11-712

The 2-chloroethyl

H

H

F

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

11-713

The 2-bromotrifluoromethane

H

H

F

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

11-714

2-iodine ethyl

H

H

F

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

11-715

The 2-cyano ethyl

H

H

F

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

C2F5

11-716

2,2-two fluoro ethyls

H

H

F

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

[table 93]

The 11st table (4)

[table 94]

The 11st table (5)

The compound sequence number

Q 2

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

11-804

2, the 2-Dichloroethyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

11-805

2,2, the 2-trifluoroethyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

11-806

2,2,2-three chloroethyls

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

11-807

2,2, the 2-three bromomethyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

11-808

The n-propyl group

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

11-809

3-fluoro-n-propyl group

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

11-810

3-chloro-n-propyl group

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

11-811

3-bromo-n-propyl group

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

11-812

The i-propyl group

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

11-813

1,2-two fluoro-2-propyl group

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

11-814

1,3-two fluoro-2-propyl group

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

11-815

1,3-two chloro-2-propyl group

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

11-816

1-chloro-3-fluoro-2-propyl group

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

11-817

3,3,3-three fluoro-n-propyl group

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

11-818

The n-butyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

11-819

4,4,4-three fluoro-n-butyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

11-820

The i-butyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

11-821

The s-butyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

11-822

Vinyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

11-823

Benzyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

11-824

Phenyl

H

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

i-C3F7

11-825

Methyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

11-826

Ethyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

11-827

The 2-fluoro ethyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

11-828

The 2-chloroethyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

11-829

The 2-bromotrifluoromethane

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

11-830

2-iodine ethyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

11-831

The 2-cyano ethyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

11-832

2,2-two fluoro ethyls

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

11-833

2, the 2-Dichloroethyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

11-834

2,2, the 2-trifluoroethyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

11-835

2,2,2-three chloroethyls

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

11-836

2,2, the 2-three bromomethyl

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

11-837

The n-propyl group

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

11-838

3-fluoro-n-propyl group

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

11-839

3-chloro-n-propyl group

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

11-840

3-bromo-n-propyl group

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

C2F5

11-841

The i-propyl group

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

11-842

1,2-two fluoro-2-propyl group

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

11-843

1,3-two fluoro-2-propyl group

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

11-844

1,3-two chloro-2-propyl group

H

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

[table 95]

The 11st table (6)

The compound sequence number

Q 2

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

11-868

3-chloro-n-propyl group

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

11-869

3-bromo-n-propyl group

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

11-870

The i-propyl group

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

11-871

1,2-two fluoro-2-propyl group

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

11-872

1,3-two fluoro-2-propyl group

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

11-873

1,3-two chloro-2-propyl group

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

11-874

1-chloro-3-fluoro-2-propyl group

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

11-875

3,3,3-three fluoro-n-propyl group

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

11-876

The n-butyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

11-877

4,4,4-three fluoro-n-butyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

11-878

The i-butyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

11-879

The s-butyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

11-880

Vinyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

i-C3F7

11-881

Benzyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

11-882

Phenyl

H

H

F

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

11-893

2,2,2-three chloroethyls

H

H

F

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

11-922

2,2,2-three chloroethyls

H

H

F

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

11-951

2,2,2-three chloroethyls

H

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

11-980

2,2,2-three chloroethyls

H

H

F

H

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

11-999

Methyl

H

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

11-1000

Ethyl

H

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

11-1001

The 2-fluoro ethyl

H

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

11-1002

The 2-chloroethyl

H

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

11-1003

The 2-bromotrifluoromethane

H

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

11-1004

2-iodine ethyl

H

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

11-1005

The 2-cyano ethyl

H

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

11-1006

2,2-two fluoro ethyls

H

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

11-1007

2, the 2-Dichloroethyl

H

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

11-1008

2,2, the 2-trifluoroethyl

H

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

11-1009

2,2,2-three chloroethyls

H

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

11-1010

2,2, the 2-three bromomethyl

H

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

11-1011

The n-propyl group

H

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

11-1012

3-fluoro-n-propyl group

H

H

F

H

H

H

C2F5

H

Seven fluorine sec.-propyls

H

CF3

11-1013

3-chloro-n-propyl group

H

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

11-1014

3-bromo-n-propyl group

H

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

11-1015

The i-propyl group

H

H

F

H

H

H

i-C3F7

H

Seven fluorine sec.-propyls

H

CF3

11-1016

1,2-two fluoro-2-propyl group

H

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

11-1017

1,3-two fluoro-2-propyl group

H

H

F

H

H

H

CF3

H

Pentafluoroethyl group

H

CF3

11-1018

1,3-two chloro-2-propyl group

H

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

11-1019

1-chloro-3-fluoro-2-propyl group

H

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

11-1020

3,3,3-three fluoro-n-propyl group

H

H

F

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

[table 96]

The 11st table (7)

[table 97]

The 11st table (8)

[table 98]

The 11st table (9)

The compound sequence number

Q 2

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

11-2519

2,2,2-three chloroethyls

H

H

F

H

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

11-2520

2,2,2-three chloroethyls

H

H

F

H

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

11-2521

2,2,2-three chloroethyls

H

H

F

H

H

F

Cl

H

Pentafluoroethyl group

H

Cl

11-2522

2,2,2-three chloroethyls

H

H

F

H

H

F

Br

H

Seven fluorine sec.-propyls

H

Br

11-2523

2,2,2-three chloroethyls

H

H

F

H

H

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

11-2524

2,2,2-three chloroethyls

H

H

F

H

H

F

I

H

Seven fluorine sec.-propyls

H

CF3

11-2525

2,2,2-three chloroethyls

H

H

F

H

H

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

11-2526

2,2,2-three chloroethyls

H

H

F

H

H

F

I

H

Nine fluoro-2-butyl

H

I

11-2527

2,2,2-three chloroethyls

H

H

F

H

H

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

11-2528

2,2,2-three chloroethyls

H

H

F

H

H

F

Br

H

Nine fluoro-2-butyl

H

CF3

11-2529

2,2,2-three chloroethyls

H

H

F

H

H

F

CF3

H

Nine fluoro-2-butyl

H

CF3

11-2530

2,2,2-three chloroethyls

H

H

H

F

F

H

Cl

H

Pentafluoroethyl group

H

Cl

11-2531

2,2,2-three chloroethyls

H

H

H

F

F

H

Br

H

Seven fluorine sec.-propyls

H

Br

11-2532

2,2,2-three chloroethyls

H

H

H

F

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

11-2533

2,2,2-three chloroethyls

H

H

H

F

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

11-2534

2,2,2-three chloroethyls

H

H

H

F

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

11-2535

2,2,2-three chloroethyls

H

H

H

F

F

H

I

H

Nine fluoro-2-butyl

H

I

11-2536

2,2,2-three chloroethyls

H

H

H

F

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

11-2537

2,2,2-three chloroethyls

H

H

H

F

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

11-2538

2,2,2-three chloroethyls

H

H

H

F

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

11-2539

2,2,2-three chloroethyls

H

H

H

F

H

F

Cl

H

Pentafluoroethyl group

H

Cl

11-2540

2,2,2-three chloroethyls

H

H

H

F

H

F

Br

H

Seven fluorine sec.-propyls

H

Br

11-2541

2,2,2-three chloroethyls

H

H

H

F

H

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

11-2542

2,2,2-three chloroethyls

H

H

H

F

H

F

I

H

Seven fluorine sec.-propyls

H

CF3

11-2543

2,2,2-three chloroethyls

H

H

H

F

H

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

11-2544

2,2,2-three chloroethyls

H

H

H

F

H

F

I

H

Nine fluoro-2-butyl

H

I

11-2545

2,2,2-three chloroethyls

H

H

H

F

H

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

11-2546

2,2,2-three chloroethyls

H

H

H

F

H

F

Br

H

Nine fluoro-2-butyl

H

CF3

11-2547

2,2,2-three chloroethyls

H

H

H

F

H

F

CF3

H

Nine fluoro-2-butyl

H

CF3

11-2548

2,2,2-three chloroethyls

H

H

H

H

F

F

Cl

H

Pentafluoroethyl group

H

Cl

11-2549

2,2,2-three chloroethyls

H

H

H

H

F

F

Br

H

Seven fluorine sec.-propyls

H

Br

11-2550

2,2,2-three chloroethyls

H

H

H

H

F

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

11-2551

2,2,2-three chloroethyls

H

H

H

H

F

F

I

H

Seven fluorine sec.-propyls

H

CF3

11-2552

2,2,2-three chloroethyls

H

H

H

H

F

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

11-2553

2,2,2-three chloroethyls

H

H

H

H

F

F

I

H

Nine fluoro-2-butyl

H

I

11-2554

2,2,2-three chloroethyls

H

H

H

H

F

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

11-2555

2,2,2-three chloroethyls

H

H

H

H

F

F

Br

H

Nine fluoro-2-butyl

H

CF3

11-2556

2,2,2-three chloroethyls

H

H

H

H

F

F

CF3

H

Nine fluoro-2-butyl

H

CF3

11-2557

2,2,2-three chloroethyls

H

H

F

F

H

F

Cl

H

Pentafluoroethyl group

H

Cl

11-2558

2,2,2-three chloroethyls

H

H

F

F

H

F

Br

H

Seven fluorine sec.-propyls

H

Br

11-2559

2,2,2-three chloroethyls

H

H

F

F

H

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

[table 99]

The 11st table (10)

[table 100]

The 11st table (11)

The compound sequence number

Q 2

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

11-3483

2,2,2-three chloroethyls

H

H

F

CN

H

H

F

H

Seven fluorine sec.-propyls

H

CF3

11-3484

2,2,2-three chloroethyls

H

H

F

CN

H

H

F

H

Nine fluoro-2-butyl

H

CF3

11-3495

2,2,2-three chloroethyls

H

H

F

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

11-3524

2,2,2-three chloroethyls

H

H

F

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

11-3553

2,2,2-three chloroethyls

H

H

F

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

11-3566

4,4,4-three fluoro-n-butyl

H

H

F

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

11-3582

2,2,2-three chloroethyls

H

H

F

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

11-3595

4,4,4-three fluoro-n-butyl

H

H

F

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

11-3611

2,2,2-three chloroethyls

H

H

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

11-3624

4,4,4-three fluoro-n-butyl

H

H

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

11-3640

2,2,2-three chloroethyls

H

H

F

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

11-3653

4,4,4-three fluoro-n-butyl

H

H

F

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

11-3669

2,2,2-three chloroethyls

H

H

F

CN

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

11-3698

2,2,2-three chloroethyls

H

H

F

CN

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

11-3727

2,2,2-three chloroethyls

H

H

F

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

11-3756

2,2,2-three chloroethyls

H

H

F

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

11-3785

2,2,2-three chloroethyls

H

H

F

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

11-3814

2,2,2-three chloroethyls

H

H

F

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

11-3833

2,2,2-three chloroethyls

H

H

F

CN

F

H

F

H

Seven fluorine sec.-propyls

H

F

11-3834

2,2,2-three chloroethyls

H

H

F

CN

F

H

F

H

Nine fluoro-2-butyl

H

F

11-3845

2,2,2-three chloroethyls

H

H

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

11-3874

2,2,2-three chloroethyls

H

H

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

Cl

11-3903

2,2,2-three chloroethyls

H

H

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

Br

11-3932

2,2,2-three chloroethyls

H

H

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

Br

11-3961

2,2,2-three chloroethyls

H

H

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

I

11-3990

2,2,2-three chloroethyls

H

H

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

I

11-4009

2,2,2-three chloroethyls

H

H

F

CN

F

H

F

H

Seven fluorine sec.-propyls

H

Cl

11-4010

2,2,2-three chloroethyls

H

H

F

CN

F

H

F

H

Seven fluorine sec.-propyls

H

Br

11-4011

2,2,2-three chloroethyls

H

H

F

CN

F

H

F

H

Seven fluorine sec.-propyls

H

I

11-4012

2,2,2-three chloroethyls

H

H

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

Br

11-4013

2,2,2-three chloroethyls

H

H

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

I

11-4014

2,2,2-three chloroethyls

H

H

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

I

11-4015

2,2,2-three chloroethyls

H

H

F

CN

F

H

F

H

Nine fluoro-2-butyl

H

Cl

11-4016

2,2,2-three chloroethyls

H

H

F

CN

F

H

F

H

Nine fluoro-2-butyl

H

Br

11-4017

2,2,2-three chloroethyls

H

H

F

CN

F

H

F

H

Nine fluoro-2-butyl

H

I

11-4018

2,2,2-three chloroethyls

H

H

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

Br

11-4019

2,2,2-three chloroethyls

H

H

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

I

11-4020

2,2,2-three chloroethyls

H

H

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

I

11-4021

2,2,2-three chloroethyls

H

H

F

CN

F

H

F

H

Seven fluorine sec.-propyls

H

OCF3

11-4022

2,2,2-three chloroethyls

H

H

F

CN

F

H

F

H

Nine fluoro-2-butyl

H

OCF3

11-4033

2,2,2-three chloroethyls

H

H

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

[table 101]

The 12nd table (1)

The compound sequence number

Q 2

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

12-1

2,2,2-three chloroethyls

Me

H

H

H

H

H

F

H

Seven fluorine sec.-propyls

H

OCF3

12-2

2,2,2-three chloroethyls

Me

H

H

H

H

H

F

H

Nine fluoro-2-butyl

H

OCF3

12-13

2,2,2-three chloroethyls

Me

H

H

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

12-42

2,2,2-three chloroethyls

Me

H

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

12-71

2,2,2-three chloroethyls

Me

H

H

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

12-100

2,2,2-three chloroethyls

Me

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

12-129

2,2,2-three chloroethyls

Me

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

12-158

2,2,2-three chloroethyls

Me

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

12-177

2,2,2-three chloroethyls

Me

H

H

H

H

H

F

H

Seven fluorine sec.-propyls

H

CF3

12-178

2,2,2-three chloroethyls

Me

H

H

H

H

H

F

H

Nine fluoro-2-butyl

H

CF3

12-189

2,2,2-three chloroethyls

Me

H

H

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

12-218

2,2,2-three chloroethyls

Me

H

H

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

12-247

2,2,2-three chloroethyls

Me

H

H

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

12-276

2,2,2-three chloroethyls

Me

H

H

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

12-305

2,2,2-three chloroethyls

Me

H

H

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

12-334

2,2,2-three chloroethyls

Me

H

H

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

12-363

2,2,2-three chloroethyls

Me

H

H

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

12-392

2,2,2-three chloroethyls

Me

H

H

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

12-421

2,2,2-three chloroethyls

Me

H

H

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

12-450

2,2,2-three chloroethyls

Me

H

H

H

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

12-479

2,2,2-three chloroethyls

Me

H

H

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

12-508

2,2,2-three chloroethyls

Me

H

H

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

12-527

2,2,2-three chloroethyls

Me

H

F

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

12-528

2,2,2-three chloroethyls

Me

H

F

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

12-529

2,2,2-three chloroethyls

Me

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

12-530

2,2,2-three chloroethyls

Me

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

12-531

2,2,2-three chloroethyls

Me

H

F

H

H

H

F

H

Seven fluorine sec.-propyls

H

OCF3

12-532

2,2,2-three chloroethyls

Me

H

F

H

H

H

F

H

Nine fluoro-2-butyl

H

OCF3

12-543

2,2,2-three chloroethyls

Me

H

F

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

12-572

2,2,2-three chloroethyls

Me

H

F

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

12-601

2,2,2-three chloroethyls

Me

H

F

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

12-630

2,2,2-three chloroethyls

Me

H

F

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

12-659

2,2,2-three chloroethyls

Me

H

F

H

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

[table 102]

The 12nd table (2)

[table 103]

The 12nd table (3)

[table 104]

The 12nd table (4)

The compound sequence number

Q 2

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

12-1315

2,2,2-three chloroethyls

Me

H

H

F

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

12-1344

2,2,2-three chloroethyls

Me

H

H

F

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

12-1373

2,2,2-three chloroethyls

Me

H

H

F

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

12-1402

2,2,2-three chloroethyls

Me

H

H

F

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

12-1421

2,2,2-three chloroethyls

Me

H

H

F

H

H

F

H

Seven fluorine sec.-propyls

H

CF3

12-1422

2,2,2-three chloroethyls

Me

H

H

F

H

H

F

H

Nine fluoro-2-butyl

H

CF3

12-1433

2,2,2-three chloroethyls

Me

H

H

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

12-1462

2,2,2-three chloroethyls

Me

H

H

F

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

12-1491

2,2,2-three chloroethyls

Me

H

H

F

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

12-1520

2,2,2-three chloroethyls

Me

H

H

F

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

12-1549

2,2,2-three chloroethyls

Me

H

H

F

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

12-1578

2,2,2-three chloroethyls

Me

H

H

F

H

H

I

H

Nine fluoro-2-butyl

H

CF3

12-1607

2,2,2-three chloroethyls

Me

H

H

F

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

12-1636

2,2,2-three chloroethyls

Me

H

H

F

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

12-1665

2,2,2-three chloroethyls

Me

H

H

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

12-1694

2,2,2-three chloroethyls

Me

H

H

F

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

12-1723

2,2,2-three chloroethyls

Me

H

H

F

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

12-1752

2,2,2-three chloroethyls

Me

H

H

F

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

12-1771

2,2,2-three chloroethyls

Me

H

F

F

H

H

F

H

Seven fluorine sec.-propyls

H

F

12-1772

2,2,2-three chloroethyls

Me

H

F

F

H

H

F

H

Nine fluoro-2-butyl

H

F

12-1783

2,2,2-three chloroethyls

Me

H

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

12-1812

2,2,2-three chloroethyls

Me

H

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

12-1841

2,2,2-three chloroethyls

Me

H

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

12-1870

2,2,2-three chloroethyls

Me

H

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

Br

12-1899

2,2,2-three chloroethyls

Me

H

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

I

12-1928

2,2,2-three chloroethyls

Me

H

F

F

H

H

I

H

Nine fluoro-2-butyl

H

I

12-1956

2,2,2-three chloroethyls

Me

H

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

Br

12-1959

2,2,2-three chloroethyls

Me

H

F

F

H

H

F

H

Seven fluorine sec.-propyls

H

OCF3

12-1960

2,2,2-three chloroethyls

Me

H

F

F

H

H

F

H

Nine fluoro-2-butyl

H

OCF3

12-1971

2,2,2-three chloroethyls

Me

H

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

12-2000

2,2,2-three chloroethyls

Me

H

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

12-2029

2,2,2-three chloroethyls

Me

H

F

F

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

12-2058

2,2,2-three chloroethyls

Me

H

F

F

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

12-2087

2,2,2-three chloroethyls

Me

H

F

F

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

12-2116

2,2,2-three chloroethyls

Me

H

F

F

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

12-2135

2,2,2-three chloroethyls

Me

H

F

F

H

H

F

H

Seven fluorine sec.-propyls

H

CF3

12-2136

2,2,2-three chloroethyls

Me

H

F

F

H

H

F

H

Nine fluoro-2-butyl

H

CF3

12-2147

2,2,2-three chloroethyls

Me

H

F

F

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

12-2176

2,2,2-three chloroethyls

Me

H

F

F

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

[table 105]

The 12nd table (5)

The compound sequence number

Q 2

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

12-2500

2,2,2-three chloroethyls

Me

H

H

H

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

12-2501

2,2,2-three chloroethyls

Me

H

H

H

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

12-2502

2,2,2-three chloroethyls

Me

H

H

H

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

12-2503

2,2,2-three chloroethyls

Me

H

H

H

H

F

Cl

H

Pentafluoroethyl group

H

Cl

12-2504

2,2,2-three chloroethyls

Me

H

H

H

H

F

Br

H

Seven fluorine sec.-propyls

H

Br

12-2505

2,2,2-three chloroethyls

Me

H

H

H

H

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

12-2506

2,2,2-three chloroethyls

Me

H

H

H

H

F

I

H

Seven fluorine sec.-propyls

H

CF3

12-2507

2,2,2-three chloroethyls

Me

H

H

H

H

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

12-2508

2,2,2-three chloroethyls

Me

H

H

H

H

F

I

H

Nine fluoro-2-butyl

H

I

12-2509

2,2,2-three chloroethyls

Me

H

H

H

H

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

12-2510

2,2,2-three chloroethyls

Me

H

H

H

H

F

Br

H

Nine fluoro-2-butyl

H

CF3

12-2511

2,2,2-three chloroethyls

Me

H

H

H

H

F

CF3

H

Nine fluoro-2-butyl

H

CF3

12-2512

2,2,2-three chloroethyls

Me

H

F

H

F

H

Cl

H

Pentafluoroethyl group

H

Cl

12-2513

2,2,2-three chloroethyls

Me

H

F

H

F

H

Br

H

Seven fluorine sec.-propyls

H

Br

12-2514

2,2,2-three chloroethyls

Me

H

F

H

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

12-2515

2,2,2-three chloroethyls

Me

H

F

H

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

12-2516

2,2,2-three chloroethyls

Me

H

F

H

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

12-2517

2,2,2-three chloroethyls

Me

H

F

H

F

H

I

H

Nine fluoro-2-butyl

H

I

12-2518

2,2,2-three chloroethyls

Me

H

F

H

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

12-2519

2,2,2-three chloroethyls

Me

H

F

H

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

12-2520

2,2,2-three chloroethyls

Me

H

F

H

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

12-2521

2,2,2-three chloroethyls

Me

H

F

H

H

F

Cl

H

Pentafluoroethyl group

H

Cl

12-2522

2,2,2-three chloroethyls

Me

H

F

H

H

F

Br

H

Seven fluorine sec.-propyls

H

Br

12-2523

2,2,2-three chloroethyls

Me

H

F

H

H

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

12-2524

2,2,2-three chloroethyls

Me

H

F

H

H

F

I

H

Seven fluorine sec.-propyls

H

CF3

12-2525

2,2,2-three chloroethyls

Me

H

F

H

H

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

12-2526

2,2,2-three chloroethyls

Me

H

F

H

H

F

I

H

Nine fluoro-2-butyl

H

I

12-2527

2,2,2-three chloroethyls

Me

H

F

H

H

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

12-2528

2,2,2-three chloroethyls

Me

H

F

H

H

F

Br

H

Nine fluoro-2-butyl

H

CF3

12-2529

2,2,2-three chloroethyls

Me

H

F

H

H

F

CF3

H

Nine fluoro-2-butyl

H

CF3

12-2530

2,2,2-three chloroethyls

Me

H

H

F

F

H

Cl

H

Pentafluoroethyl group

H

Cl

12-2531

2,2,2-three chloroethyls

Me

H

H

F

F

H

Br

H

Seven fluorine sec.-propyls

H

Br

12-2532

2,2,2-three chloroethyls

Me

H

H

F

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

12-2533

2,2,2-three chloroethyls

Me

H

H

F

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

12-2534

2,2,2-three chloroethyls

Me

H

H

F

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

12-2535

2,2,2-three chloroethyls

Me

H

H

F

F

H

I

H

Nine fluoro-2-butyl

H

I

12-2536

2,2,2-three chloroethyls

Me

H

H

F

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

12-2537

2,2,2-three chloroethyls

Me

H

H

F

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

12-2538

2,2,2-three chloroethyls

Me

H

H

F

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

[table 106]

The 12nd table (6)

The compound sequence number

Q 2

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

12-2564

2,2,2-three chloroethyls

Me

H

F

F

H

F

Br

H

Nine fluoro-2-butyl

H

CF3

12-2565

2,2,2-three chloroethyls

Me

H

F

F

H

F

CF3

H

Nine fluoro-2-butyl

H

CF3

12-2566

2,2,2-three chloroethyls

Me

H

F

H

F

F

Cl

H

Pentafluoroethyl group

H

Cl

12-2567

2,2,2-three chloroethyls

Me

H

F

H

F

F

Br

H

Seven fluorine sec.-propyls

H

Br

12-2568

2,2,2-three chloroethyls

Me

H

F

H

F

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

12-2569

2,2,2-three chloroethyls

Me

H

F

H

F

F

I

H

Seven fluorine sec.-propyls

H

CF3

12-2570

2,2,2-three chloroethyls

Me

H

F

H

F

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

12-2571

2,2,2-three chloroethyls

Me

H

F

H

F

F

I

H

Nine fluoro-2-butyl

H

I

12-2572

2,2,2-three chloroethyls

Me

H

F

H

F

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

12-2573

2,2,2-three chloroethyls

Me

H

F

H

F

F

Br

H

Nine fluoro-2-butyl

H

CF3

12-2574

2,2,2-three chloroethyls

Me

H

F

H

F

F

CF3

H

Nine fluoro-2-butyl

H

CF3

12-2575

2,2,2-three chloroethyls

Me

H

H

F

F

F

Cl

H

Pentafluoroethyl group

H

Cl

12-2576

2,2,2-three chloroethyls

Me

H

H

F

F

F

Br

H

Seven fluorine sec.-propyls

H

Br

12-2577

2,2,2-three chloroethyls

Me

H

H

F

F

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

12-2578

2,2,2-three chloroethyls

Me

H

H

F

F

F

I

H

Seven fluorine sec.-propyls

H

CF3

12-2579

2,2,2-three chloroethyls

Me

H

H

F

F

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

12-2580

2,2,2-three chloroethyls

Me

H

H

F

F

F

I

H

Nine fluoro-2-butyl

H

I

12-2581

2,2,2-three chloroethyls

Me

H

H

F

F

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

12-2582

2,2,2-three chloroethyls

Me

H

H

F

F

F

Br

H

Nine fluoro-2-butyl

H

CF3

12-2583

2,2,2-three chloroethyls

Me

H

H

F

F

F

CF3

H

Nine fluoro-2-butyl

H

CF3

12-2584

2,2,2-three chloroethyls

Me

H

F

F

F

F

Cl

H

Pentafluoroethyl group

H

Cl

12-2585

2,2,2-three chloroethyls

Me

H

F

F

F

F

Br

H

Seven fluorine sec.-propyls

H

Br

12-2586

2,2,2-three chloroethyls

Me

H

F

F

F

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

12-2587

2,2,2-three chloroethyls

Me

H

F

F

F

F

I

H

Seven fluorine sec.-propyls

H

CF3

12-2588

2,2,2-three chloroethyls

Me

H

F

F

F

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

12-2589

2,2,2-three chloroethyls

Me

H

F

F

F

F

I

H

Nine fluoro-2-butyl

H

I

12-2590

2,2,2-three chloroethyls

Me

H

F

F

F

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

12-2591

2,2,2-three chloroethyls

Me

H

F

F

F

F

Br

H

Nine fluoro-2-butyl

H

CF3

12-2592

2,2,2-three chloroethyls

Me

H

F

F

F

F

CF3

H

Nine fluoro-2-butyl

H

CF3

12-2593

2,2,2-three chloroethyls

Me

H

H

CN

H

H

F

H

Seven fluorine sec.-propyls

H

OCF3

12-2594

2,2,2-three chloroethyls

Me

H

H

CN

H

H

F

H

Nine fluoro-2-butyl

H

OCF3

12-2605

2,2,2-three chloroethyls

Me

H

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

12-2634

2,2,2-three chloroethyls

Me

H

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

12-2663

2,2,2-three chloroethyls

Me

H

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

12-2692

2,2,2-three chloroethyls

Me

H

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

12-2721

2,2,2-three chloroethyls

Me

H

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

12-2750

2,2,2-three chloroethyls

Me

H

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

12-2769

2,2,2-three chloroethyls

Me

H

H

CN

H

H

F

H

Seven fluorine sec.-propyls

H

CF3

12-2770

2,2,2-three chloroethyls

Me

H

H

CN

H

H

F

H

Nine fluoro-2-butyl

H

CF3

[table 107]

The 12nd table (7)

The compound sequence number

Q 2

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

12-3377

2,2,2-three chloroethyls

Me

H

F

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

12-3406

2,2,2-three chloroethyls

Me

H

F

CN

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

12-3435

2,2,2-three chloroethyls

Me

H

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

12-3464

2,2,2-three chloroethyls

Me

H

F

CN

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

12-3483

2,2,2-three chloroethyls

Me

H

F

CN

H

H

F

H

Seven fluorine sec.-propyls

H

CF3

12-3484

2,2,2-three chloroethyls

Me

H

F

CN

H

H

F

H

Nine fluoro-2-butyl

H

CF3

12-3495

2,2,2-three chloroethyls

Me

H

F

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

12-3524

2,2,2-three chloroethyls

Me

H

F

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

12-3553

2,2,2-three chloroethyls

Me

H

F

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

12-3582

2,2,2-three chloroethyls

Me

H

F

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

12-3611

2,2,2-three chloroethyls

Me

H

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

12-3640

2,2,2-three chloroethyls

Me

H

F

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

12-3669

2,2,2-three chloroethyls

Me

H

F

CN

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

12-3698

2,2,2-three chloroethyls

Me

H

F

CN

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

12-3727

2,2,2-three chloroethyls

Me

H

F

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

12-3756

2,2,2-three chloroethyls

Me

H

F

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

12-3785

2,2,2-three chloroethyls

Me

H

F

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

12-3814

2,2,2-three chloroethyls

Me

H

F

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

12-3833

2,2,2-three chloroethyls

Me

H

F

CN

F

H

F

H

Seven fluorine sec.-propyls

H

F

12-3834

2,2,2-three chloroethyls

Me

H

F

CN

F

H

F

H

Nine fluoro-2-butyl

H

F

12-3845

2,2,2-three chloroethyls

Me

H

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

12-3874

2,2,2-three chloroethyls

Me

H

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

Cl

12-3903

2,2,2-three chloroethyls

Me

H

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

Br

12-3932

2,2,2-three chloroethyls

Me

H

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

Br

12-3961

2,2,2-three chloroethyls

Me

H

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

I

12-3990

2,2,2-three chloroethyls

Me

H

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

I

12-4018

2,2,2-three chloroethyls

Me

H

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

Br

12-4021

2,2,2-three chloroethyls

Me

H

F

CN

F

H

F

H

Seven fluorine sec.-propyls

H

OCF3

12-4022

2,2,2-three chloroethyls

Me

H

F

CN

F

H

F

H

Nine fluoro-2-butyl

H

OCF3

12-4033

2,2,2-three chloroethyls

Me

H

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

12-4062

2,2,2-three chloroethyls

Me

H

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

12-4091

2,2,2-three chloroethyls

Me

H

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

12-4120

2,2,2-three chloroethyls

Me

H

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

OCF3

12-4149

2,2,2-three chloroethyls

Me

H

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

OCF3

12-4178

2,2,2-three chloroethyls

Me

H

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

OCF3

12-4197

2,2,2-three chloroethyls

Me

H

F

CN

F

H

F

H

Seven fluorine sec.-propyls

H

CF3

12-4198

2,2,2-three chloroethyls

Me

H

F

CN

F

H

F

H

Nine fluoro-2-butyl

H

CF3

12-4209

2,2,2-three chloroethyls

Me

H

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

12-4238

2,2,2-three chloroethyls

Me

H

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

CF3

[table 108]

The 13rd table (1)

[table 109]

The 13rd table (2)

[table 110]

The 13rd table (3)

[table 111]

The 13rd table (4)

The compound sequence number

Q 2

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

13-2529

2,2,2-three chloroethyls

H

Me

F

H

H

F

CF3

H

Nine fluoro-2-butyl

H

CF3

13-2530

2,2,2-three chloroethyls

H

Me

H

F

F

H

Cl

H

Pentafluoroethyl group

H

Cl

13-2531

2,2,2-three chloroethyls

H

Me

H

F

F

H

Br

H

Seven fluorine sec.-propyls

H

Br

13-2532

2,2,2-three chloroethyls

H

Me

H

F

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

13-2533

2,2,2-three chloroethyls

H

Me

H

F

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

13-2534

2,2,2-three chloroethyls

H

Me

H

F

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

13-2535

2,2,2-three chloroethyls

H

Me

H

F

F

H

I

H

Nine fluoro-2-butyl

H

I

13-2536

2,2,2-three chloroethyls

H

Me

H

F

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

13-2537

2,2,2-three chloroethyls

H

Me

H

F

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

13-2538

2,2,2-three chloroethyls

H

Me

H

F

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

13-2539

2,2,2-three chloroethyls

H

Me

H

F

H

F

Cl

H

Pentafluoroethyl group

H

Cl

13-2540

2,2,2-three chloroethyls

H

Me

H

F

H

F

Br

H

Seven fluorine sec.-propyls

H

Br

13-2541

2,2,2-three chloroethyls

H

Me

H

F

H

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

13-2542

2,2,2-three chloroethyls

H

Me

H

F

H

F

I

H

Seven fluorine sec.-propyls

H

CF3

13-2543

2,2,2-three chloroethyls

H

Me

H

F

H

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

13-2544

2,2,2-three chloroethyls

H

Me

H

F

H

F

I

H

Nine fluoro-2-butyl

H

I

13-2545

2,2,2-three chloroethyls

H

Me

H

F

H

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

13-2546

2,2,2-three chloroethyls

H

Me

H

F

H

F

Br

H

Nine fluoro-2-butyl

H

CF3

13-2547

2,2,2-three chloroethyls

H

Me

H

F

H

F

CF3

H

Nine fluoro-2-butyl

H

CF3

13-2548

2,2,2-three chloroethyls

H

Me

H

H

F

F

Cl

H

Pentafluoroethyl group

H

Cl

13-2549

2,2,2-three chloroethyls

H

Me

H

H

F

F

Br

H

Seven fluorine sec.-propyls

H

Br

13-2550

2,2,2-three chloroethyls

H

Me

H

H

F

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

13-2551

2,2,2-three chloroethyls

H

Me

H

H

F

F

I

H

Seven fluorine sec.-propyls

H

CF3

13-2552

2,2,2-three chloroethyls

H

Me

H

H

F

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

13-2553

2,2,2-three chloroethyls

H

Me

H

H

F

F

I

H

Nine fluoro-2-butyl

H

I

13-2554

2,2,2-three chloroethyls

H

Me

H

H

F

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

13-2555

2,2,2-three chloroethyls

H

Me

H

H

F

F

Br

H

Nine fluoro-2-butyl

H

CF3

13-2556

2,2,2-three chloroethyls

H

Me

H

H

F

F

CF3

H

Nine fluoro-2-butyl

H

CF3

13-2557

2,2,2-three chloroethyls

H

Me

F

F

H

F

Cl

H

Pentafluoroethyl group

H

Cl

13-2558

2,2,2-three chloroethyls

H

Me

F

F

H

F

Br

H

Seven fluorine sec.-propyls

H

Br

13-2559

2,2,2-three chloroethyls

H

Me

F

F

H

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

13-2560

2,2,2-three chloroethyls

H

Me

F

F

H

F

I

H

Seven fluorine sec.-propyls

H

CF3

13-2561

2,2,2-three chloroethyls

H

Me

F

F

H

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

13-2562

2,2,2-three chloroethyls

H

Me

F

F

H

F

I

H

Nine fluoro-2-butyl

H

I

13-2563

2,2,2-three chloroethyls

H

Me

F

F

H

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

13-2564

2,2,2-three chloroethyls

H

Me

F

F

H

F

Br

H

Nine fluoro-2-butyl

H

CF3

13-2565

2,2,2-three chloroethyls

H

Me

F

F

H

F

CF3

H

Nine fluoro-2-butyl

H

CF3

13-2566

2,2,2-three chloroethyls

H

Me

F

H

F

F

Cl

H

Pentafluoroethyl group

H

Cl

13-2567

2,2,2-three chloroethyls

H

Me

F

H

F

F

Br

H

Seven fluorine sec.-propyls

H

Br

[table 112]

The 13rd table (5)

The compound sequence number

Q 2

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

13-2593

2,2,2-three chloroethyls

H

Me

H

CN

H

H

F

H

Seven fluorine sec.-propyls

H

OCF3

13-2594

2,2,2-three chloroethyls

H

Me

H

CN

H

H

F

H

Nine fluoro-2-butyl

H

OCF3

13-2605

2,2,2-three chloroethyls

H

Me

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

13-2634

2,2,2-three chloroethyls

H

Me

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

13-2663

2,2,2-three chloroethyls

H

Me

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

13-2692

2,2,2-three chloroethyls

H

Me

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

13-2721

2,2,2-three chloroethyls

H

Me

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

13-2750

2,2,2-three chloroethyls

H

Me

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

13-2769

2,2,2-three chloroethyls

H

Me

H

CN

H

H

F

H

Seven fluorine sec.-propyls

H

CF3

13-2770

2,2,2-three chloroethyls

H

Me

H

CN

H

H

F

H

Nine fluoro-2-butyl

H

CF3

13-2781

2,2,2-three chloroethyls

H

Me

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

13-2810

2,2,2-three chloroethyls

H

Me

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

13-2839

2,2,2-three chloroethyls

H

Me

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

13-2868

2,2,2-three chloroethyls

H

Me

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

13-2897

2,2,2-three chloroethyls

H

Me

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

13-2926

2,2,2-three chloroethyls

H

Me

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

13-2955

2,2,2-three chloroethyls

H

Me

H

CN

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

13-2984

2,2,2-three chloroethyls

H

Me

H

CN

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

13-3013

2,2,2-three chloroethyls

H

Me

H

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

13-3042

2,2,2-three chloroethyls

H

Me

H

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

13-3071

2,2,2-three chloroethyls

H

Me

H

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

13-3100

2,2,2-three chloroethyls

H

Me

H

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

13-3119

2,2,2-three chloroethyls

H

Me

F

CN

H

H

F

H

Seven fluorine sec.-propyls

H

F

13-3120

2,2,2-three chloroethyls

H

Me

F

CN

H

H

F

H

Nine fluoro-2-butyl

H

F

13-3131

2,2,2-three chloroethyls

H

Me

F

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

13-3160

2,2,2-three chloroethyls

H

Me

F

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

13-3189

2,2,2-three chloroethyls

H

Me

F

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

13-3218

2,2,2-three chloroethyls

H

Me

F

CN

H

H

Br

H

Nine fluoro-2-butyl

H

Br

13-3247

2,2,2-three chloroethyls

H

Me

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

I

13-3276

2,2,2-three chloroethyls

H

Me

F

CN

H

H

I

H

Nine fluoro-2-butyl

H

I

13-3298

2,2,2-three chloroethyls

H

Me

F

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

Br

13-3307

2,2,2-three chloroethyls

H

Me

F

CN

H

H

F

H

Seven fluorine sec.-propyls

H

OCF3

13-3308

2,2,2-three chloroethyls

H

Me

F

CN

H

H

F

H

Nine fluoro-2-butyl

H

OCF3

13-3319

2,2,2-three chloroethyls

H

Me

F

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

13-3348

2,2,2-three chloroethyls

H

Me

F

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

13-3377

2,2,2-three chloroethyls

H

Me

F

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

13-3406

2,2,2-three chloroethyls

H

Me

F

CN

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

13-3435

2,2,2-three chloroethyls

H

Me

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

13-3464

2,2,2-three chloroethyls

H

Me

F

CN

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

[table 113]

The 13rd table (6)

The compound sequence number

Q 2

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

13-4033

2,2,2-three chloroethyls

H

Me

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

13-4062

2,2,2-three chloroethyls

H

Me

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

13-4091

2,2,2-three chloroethyls

H

Me

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

13-4120

2,2,2-three chloroethyls

H

Me

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

OCF3

13-4149

2,2,2-three chloroethyls

H

Me

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

OCF3

13-4178

2,2,2-three chloroethyls

H

Me

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

OCF3

13-4197

2,2,2-three chloroethyls

H

Me

F

CN

F

H

F

H

Seven fluorine sec.-propyls

H

CF3

13-4198

2,2,2-three chloroethyls

H

Me

F

CN

F

H

F

H

Nine fluoro-2-butyl

H

CF3

13-4209

2,2,2-three chloroethyls

H

Me

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

13-4238

2,2,2-three chloroethyls

H

Me

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

CF3

13-4267

2,2,2-three chloroethyls

H

Me

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

CF3

13-4296

2,2,2-three chloroethyls

H

Me

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

13-4325

2,2,2-three chloroethyls

H

Me

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

13-4354

2,2,2-three chloroethyls

H

Me

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

CF3

13-4383

2,2,2-three chloroethyls

H

Me

F

CN

F

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

13-4412

2,2,2-three chloroethyls

H

Me

F

CN

F

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

13-4441

2,2,2-three chloroethyls

H

Me

F

CN

F

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

13-4470

2,2,2-three chloroethyls

H

Me

F

CN

F

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

13-4499

2,2,2-three chloroethyls

H

Me

F

CN

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

13-4528

2,2,2-three chloroethyls

H

Me

F

CN

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

[table 114]

The 14th table (1)

[table 115]

The 14th table (2)

[table 116]

The 14th table (3)

[table 117]

The 14th table (4)

[table 118]

The 14th table (5)

[table 119]

[table 120]

The 14th table (7)

The compound sequence number

Q 2

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

14-5230

2,2,2-three chloroethyls

Me

Me

H

H

H

F

Br

H

Nine fluoro-2-butyl

H

CF3

14-5231

2,2,2-three chloroethyls

Me

Me

H

H

H

F

CF3

H

Nine fluoro-2-butyl

H

CF3

14-5232

2,2,2-three chloroethyls

Me

Me

F

H

F

H

Cl

H

Pentafluoroethyl group

H

Cl

14-5233

2,2,2-three chloroethyls

Me

Me

F

H

F

H

Br

H

Seven fluorine sec.-propyls

H

Br

14-5234

2,2,2-three chloroethyls

Me

Me

F

H

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

14-5235

2,2,2-three chloroethyls

Me

Me

F

H

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

14-5236

2,2,2-three chloroethyls

Me

Me

F

H

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

14-5237

2,2,2-three chloroethyls

Me

Me

F

H

F

H

I

H

Nine fluoro-2-butyl

H

I

14-5238

2,2,2-three chloroethyls

Me

Me

F

H

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

14-5239

2,2,2-three chloroethyls

Me

Me

F

H

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

14-5240

2,2,2-three chloroethyls

Me

Me

F

H

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

14-5241

2,2,2-three chloroethyls

Me

Me

F

H

H

F

Cl

H

Pentafluoroethyl group

H

Cl

14-5242

2,2,2-three chloroethyls

Me

Me

F

H

H

F

Br

H

Seven fluorine sec.-propyls

H

Br

14-5243

2,2,2-three chloroethyls

Me

Me

F

H

H

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

14-5244

2,2,2-three chloroethyls

Me

Me

F

H

H

F

I

H

Seven fluorine sec.-propyls

H

CF3

14-5245

2,2,2-three chloroethyls

Me

Me

F

H

H

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

14-5246

2,2,2-three chloroethyls

Me

Me

F

H

H

F

I

H

Nine fluoro-2-butyl

H

I

14-5247

2,2,2-three chloroethyls

Me

Me

F

H

H

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

14-5248

2,2,2-three chloroethyls

Me

Me

F

H

H

F

Br

H

Nine fluoro-2-butyl

H

CF3

14-5249

2,2,2-three chloroethyls

Me

Me

F

H

H

F

CF3

H

Nine fluoro-2-butyl

H

CF3

14-5250

2,2,2-three chloroethyls

Me

Me

H

F

F

H

Cl

H

Pentafluoroethyl group

H

Cl

14-5251

2,2,2-three chloroethyls

Me

Me

H

F

F

H

Br

H

Seven fluorine sec.-propyls

H

Br

14-5252

2,2,2-three chloroethyls

Me

Me

H

F

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

14-5253

2,2,2-three chloroethyls

Me

Me

H

F

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

14-5254

2,2,2-three chloroethyls

Me

Me

H

F

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

14-5255

2,2,2-three chloroethyls

Me

Me

H

F

F

H

I

H

Nine fluoro-2-butyl

H

I

14-5256

2,2,2-three chloroethyls

Me

Me

H

F

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

14-5257

2,2,2-three chloroethyls

Me

Me

H

F

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

14-5258

2,2,2-three chloroethyls

Me

Me

H

F

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

14-5259

2,2,2-three chloroethyls

Me

Me

H

F

H

F

Cl

H

Pentafluoroethyl group

H

Cl

14-5260

2,2,2-three chloroethyls

Me

Me

H

F

H

F

Br

H

Seven fluorine sec.-propyls

H

Br

14-5261

2,2,2-three chloroethyls

Me

Me

H

F

H

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

14-5262

2,2,2-three chloroethyls

Me

Me

H

F

H

F

I

H

Seven fluorine sec.-propyls

H

CF3

14-5263

2,2,2-three chloroethyls

Me

Me

H

F

H

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

14-5264

2,2,2-three chloroethyls

Me

Me

H

F

H

F

I

H

Nine fluoro-2-butyl

H

I

14-5265

2,2,2-three chloroethyls

Me

Me

H

F

H

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

14-5266

2,2,2-three chloroethyls

Me

Me

H

F

H

F

Br

H

Nine fluoro-2-butyl

H

CF3

14-5267

2,2,2-three chloroethyls

Me

Me

H

F

H

F

CF3

H

Nine fluoro-2-butyl

H

CF3

14-5268

2,2,2-three chloroethyls

Me

Me

H

H

F

F

Cl

H

Pentafluoroethyl group

H

Cl

14-5269

2,2,2-three chloroethyls

Me

Me

H

H

F

F

Br

H

Seven fluorine sec.-propyls

H

Br

14-5270

2,2,2-three chloroethyls

Me

Me

H

H

F

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

[table 121]

The 14th table (8)

The compound sequence number

Q 2

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

14-5294

2,2,2-three chloroethyls

Me

Me

F

H

F

F

CF3

H

Nine fluoro-2-butyl

H

CF3

14-5295

2,2,2-three chloroethyls

Me

Me

H

F

F

F

Cl

H

Pentafluoroethyl group

H

Cl

14-5296

2,2,2-three chloroethyls

Me

Me

H

F

F

F

Br

H

Seven fluorine sec.-propyls

H

Br

14-5297

2,2,2-three chloroethyls

Me

Me

H

F

F

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

14-5298

2,2,2-three chloroethyls

Me

Me

H

F

F

F

I

H

Seven fluorine sec.-propyls

H

CF3

14-5299

2,2,2-three chloroethyls

Me

Me

H

F

F

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

14-5300

2,2,2-three chloroethyls

Me

Me

H

F

F

F

I

H

Nine fluoro-2-butyl

H

I

14-5301

2,2,2-three chloroethyls

Me

Me

H

F

F

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

14-5302

2,2,2-three chloroethyls

Me

Me

H

F

F

F

Br

H

Nine fluoro-2-butyl

H

CF3

14-5303

2,2,2-three chloroethyls

Me

Me

H

F

F

F

CF3

H

Nine fluoro-2-butyl

H

CF3

14-5304

2,2,2-three chloroethyls

Me

Me

F

F

F

F

Cl

H

Pentafluoroethyl group

H

Cl

14-5305

2,2,2-three chloroethyls

Me

Me

F

F

F

F

Br

H

Seven fluorine sec.-propyls

H

Br

14-5306

2,2,2-three chloroethyls

Me

Me

F

F

F

F

Br

H

Seven fluorine sec.-propyls

H

OCF3

14-5307

2,2,2-three chloroethyls

Me

Me

F

F

F

F

I

H

Seven fluorine sec.-propyls

H

CF3

14-5308

2,2,2-three chloroethyls

Me

Me

F

F

F

F

CF3

H

Seven fluorine sec.-propyls

H

CF3

14-5309

2,2,2-three chloroethyls

Me

Me

F

F

F

F

I

H

Nine fluoro-2-butyl

H

I

14-5310

2,2,2-three chloroethyls

Me

Me

F

F

F

F

Cl

H

Nine fluoro-2-butyl

H

OCF3

14-5311

2,2,2-three chloroethyls

Me

Me

F

F

F

F

Br

H

Nine fluoro-2-butyl

H

CF3

14-5312

2,2,2-three chloroethyls

Me

Me

F

F

F

F

CF3

H

Nine fluoro-2-butyl

H

CF3

14-5313

2,2,2-three chloroethyls

Me

Me

H

CN

H

H

F

H

Seven fluorine sec.-propyls

H

OCF3

14-5314

2,2,2-three chloroethyls

Me

Me

H

CN

H

H

F

H

Nine fluoro-2-butyl

H

OCF3

14-5325

2,2,2-three chloroethyls

Me

Me

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

14-5354

2,2,2-three chloroethyls

Me

Me

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

14-5383

2,2,2-three chloroethyls

Me

Me

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

14-5412

2,2,2-three chloroethyls

Me

Me

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

14-5441

2,2,2-three chloroethyls

Me

Me

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

14-5470

2,2,2-three chloroethyls

Me

Me

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

14-5685

2,2,2-three chloroethyls

Me

Me

H

CN

H

H

F

H

Seven fluorine sec.-propyls

H

CF3

14-5686

2,2,2-three chloroethyls

Me

Me

H

CN

H

H

F

H

Nine fluoro-2-butyl

H

CF3

14-5697

2,2,2-three chloroethyls

Me

Me

H

CN

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

14-5726

2,2,2-three chloroethyls

Me

Me

H

CN

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

14-5755

2,2,2-three chloroethyls

Me

Me

H

CN

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

14-5784

2,2,2-three chloroethyls

Me

Me

H

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

14-5813

2,2,2-three chloroethyls

Me

Me

H

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

14-5842

2,2,2-three chloroethyls

Me

Me

H

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

14-6067

2,2,2-three chloroethyls

Me

Me

H

CN

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

14-6096

2,2,2-three chloroethyls

Me

Me

H

CN

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

14-6125

2,2,2-three chloroethyls

Me

Me

H

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

14-6154

2,2,2-three chloroethyls

Me

Me

H

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

14-6183

2,2,2-three chloroethyls

Me

Me

H

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

14-6212

2,2,2-three chloroethyls

Me

Me

H

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

[table 122]

The 14th table (9)

The compound sequence number

Q 2

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

14-7299

2,2,2-three chloroethyls

Me

Me

F

CN

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

14-7328

2,2,2-three chloroethyls

Me

Me

F

CN

H

H

I

H

Nine fluoro-2-butyl

H

CF3

14-7553

2,2,2-three chloroethyls

Me

Me

F

CN

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

14-7582

2,2,2-three chloroethyls

Me

Me

F

CN

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

14-7611

2,2,2-three chloroethyls

Me

Me

F

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

14-7640

2,2,2-three chloroethyls

Me

Me

F

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

14-7669

2,2,2-three chloroethyls

Me

Me

F

CN

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

14-7698

2,2,2-three chloroethyls

Me

Me

F

CN

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

14-7913

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

F

H

Seven fluorine sec.-propyls

H

F

14-7914

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

F

H

Nine fluoro-2-butyl

H

F

14-7925

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

14-7954

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

Cl

14-7983

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

Br

14-8012

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

Br

14-8041

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

I

14-8070

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

I

13-4012

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

Br

14-8285

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

F

H

Seven fluorine sec.-propyls

H

OCF3

14-8286

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

F

H

Nine fluoro-2-butyl

H

OCF3

14-8297

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

14-8326

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

14-8355

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

14-8384

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

OCF3

14-8413

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

OCF3

14-8442

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

OCF3

14-8657

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

F

H

Seven fluorine sec.-propyls

H

CF3

14-8658

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

F

H

Nine fluoro-2-butyl

H

CF3

14-8669

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

14-8698

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

Cl

H

Nine fluoro-2-butyl

H

CF3

14-8727

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

Br

H

Seven fluorine sec.-propyls

H

CF3

14-8756

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

Br

H

Nine fluoro-2-butyl

H

CF3

14-8785

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

I

H

Seven fluorine sec.-propyls

H

CF3

14-8814

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

I

H

Nine fluoro-2-butyl

H

CF3

14-9039

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

14-9068

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

14-9097

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

14-9126

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

14-9155

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

14-9184

2,2,2-three chloroethyls

Me

Me

F

CN

F

H

CF3

H

Nine fluoro-2-butyl

H

CF3

[table 123]

The 15th table (1)

The compound sequence number

Q 2

R 1

R 2

X 1

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

15-9

2, the 2-Dichloroethyl

H

Et

H

H

H

H

Cl

F

Seven fluorine sec.-propyls

F

OCF3

15-39

2,2, the 2-trifluoroethyl

H

H

H

H

H

H

Cl

Me

Nine fluoro-2-butyl

Me

OCF3

15-144

Methyl

H

H

H

H

H

H

Cl

F

Seven fluorine sec.-propyls

H

CF3

15-147

The 2-chloroethyl

Me

Me

H

H

H

H

Cl

H

Seven fluorine sec.-propyls

Cl

CF3

15-148

The 2-bromotrifluoromethane

H

H

H

H

H

H

F

Br

Seven fluorine sec.-propyls

H

CF3

15-153

2,2, the 2-trifluoroethyl

H

H

H

H

H

H

Cl

F

Seven fluorine sec.-propyls

Cl

CF3

15-165

3,3,3-three fluoro-n-propyl group

H

H

H

H

H

H

Cl

I

Nine fluoro-2-butyl

Cl

CF3

15-168

The i-butyl

H

H

H

H

H

H

Cl

Me

Nine fluoro-2-butyl

H

CF3

15-169

The s-butyl

H

H

H

H

H

H

Cl

H

Nine fluoro-2-butyl

Me

CF3

15-170

Vinyl

i-Pr

H

H

H

H

H

Cl

Et

Nine fluoro-2-butyl

H

CF3

15-171

Benzyl

H

H

H

H

H

H

Cl

H

Nine fluoro-2-butyl

Et

CF3

15-182

2,2, the 2-trifluoroethyl

H

H

H

H

H

H

Cl

Me

Nine fluoro-2-butyl

Me

n-C3F7

15-183

2,2,2-three chloroethyls

H

H

H

H

H

H

Cl

Me

Nine fluoro-2-butyl

Et

i-C3F7

15-189

The i-propyl group

H

H

H

H

H

H

Cl

Et

Nine fluoro-2-butyl

Me

n-C3F7

15-190

1,2-two fluoro-2-propyl group

H

H

H

H

H

H

Cl

Et

Nine fluoro-2-butyl

Et

i-C3F7

15-196

The 2-chloroethyl

H

H

H

H

H

H

Br

n-Pr

Seven fluorine sec.-propyls

Me

CF3

15-197

The 2-bromotrifluoromethane

H

H

H

H

H

H

Br

n-Pr

Seven fluorine sec.-propyls

Et

CF3

15-203

2,2,2-three chloroethyls

H

H

H

H

H

H

Br

i-Pr

Seven fluorine sec.-propyls

Me

CF3

15-204

2,2, the 2-three bromomethyl

H

H

H

H

H

H

Br

i-Pr

Seven fluorine sec.-propyls

Et

CF3

15-210

1,2-two fluoro-2-propyl group

H

H

H

H

H

H

Br

n-Bu

Seven fluorine sec.-propyls

Me

CF3

15-211

1,3-two fluoro-2-propyl group

H

H

H

H

H

H

Br

n-Bu

Seven fluorine sec.-propyls

Et

CF3

15-217

The i-butyl

H

H

H

H

H

H

Br

i-Bu

Nine fluoro-2-butyl

Me

CF3

15-218

The s-butyl

H

H

H

H

H

H

Br

i-Bu

Nine fluoro-2-butyl

Et

CF3

15-224

The 2-fluoro ethyl

H

H

H

H

H

H

Br

s-Bu

Nine fluoro-2-butyl

Me

CF3

15-225

The 2-chloroethyl

H

H

H

H

H

H

Br

s-Bu

Nine fluoro-2-butyl

Et

CF3

15-231

2,2, the 2-trifluoroethyl

H

H

H

H

H

H

Br

F

Nine fluoro-2-butyl

Me

CF3

15-232

2,2,2-three chloroethyls

H

H

H

H

H

H

Br

F

Nine fluoro-2-butyl

Et

CF3

15-238

The i-propyl group

Et

i-Pr

H

H

H

H

Br

Cl

Nine fluoro-2-butyl

Me

CF3

15-239

1,2-two fluoro-2-propyl group

H

H

H

H

H

H

Br

Cl

Nine fluoro-2-butyl

Et

CF3

15-245

2-iodine ethyl

H

H

H

H

H

H

I

Br

Seven fluorine sec.-propyls

Me

CF3

15-246

The 2-cyano ethyl

H

H

H

H

H

H

I

Br

Seven fluorine sec.-propyls

Et

CF3

15-252

The n-propyl group

n-Pr

Me

H

H

H

H

I

I

Seven fluorine sec.-propyls

Me

CF3

15-253

3-fluoro-n-propyl group

H

H

H

H

H

H

I

I

Seven fluorine sec.-propyls

Et

CF3

[table [124]

The the 15th (2)

[table 125]

The 15th table (3)

[table 126]

The 15th table (4)

[table 127]

The 15th table (5)

[table 128]

The 15th table (6)

[table 129]

The 15th table (7)

[table 130]

[table 131]

The 15th table (9)

[table 132]

The 15th table (10)

[table 133]

Table 16 table (1)

[table 134]

The 16th table (2)

[table 135]

The 16th table (3)

[table 136]

The 16th table (4)

[table 137]

The 16th table (5)

[table 138]

The 16th table (6)

[table 139]

The 16th table (7)

[table 140]

The 16th table (8)

[table 141]

The 16th table (9)

[table 142]

The 16th table (10)

[table 143]

The 16th table (11)

[table 144]

The 16th table (12)

[table 145]

The 16th table (13)

[table 146]

The 16th table (14)

[table 147]

The 17th table (1)

The compound sequence number

Q 1

R 1

R 2

A

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

17-1

Phenyl

Me

H

N

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

17-2

The 3-cyano-phenyl

Me

H

N

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

17-3

The 4-cyano-phenyl

Me

H

N

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

17-4

2-chloropyridine-3-base

Me

H

N

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

17-5

Phenyl

Me

H

N

H

H

H

F

H

Nine fluoro-2-butyl

H

F

17-6

The 3-cyano-phenyl

Me

H

N

H

H

H

F

H

Nine fluoro-2-butyl

H

F

17-7

The 4-cyano-phenyl

Me

H

N

H

H

H

F

H

Nine fluoro-2-butyl

H

F

17-8

2-chloropyridine-3-base

Me

H

N

H

H

H

F

H

Nine fluoro-2-butyl

H

F

17-9

Phenyl

Me

H

N

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

17-29

The 3-cyano-phenyl

Me

H

N

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

17-30

The 4-cyano-phenyl

Me

H

N

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

17-45

2-chloropyridine-3-base

Me

H

N

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

17-87

Phenyl

Me

H

N

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

17-107

The 3-cyano-phenyl

Me

H

N

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

17-108

The 4-cyano-phenyl

Me

H

N

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

17-123

2-chloropyridine-3-base

Me

H

N

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

17-165

Phenyl

Me

H

N

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

17-185

The 3-cyano-phenyl

Me

H

N

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

17-186

The 4-cyano-phenyl

Me

H

N

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

17-201

2-chloropyridine-3-base

Me

H

N

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

17-243

Phenyl

Me

H

N

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

17-263

The 3-cyano-phenyl

Me

H

N

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

17-264

The 4-cyano-phenyl

Me

H

N

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

17-279

2-chloropyridine-3-base

Me

H

N

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

17-321

Phenyl

Me

H

N

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

17-341

The 3-cyano-phenyl

Me

H

N

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

17-342

The 4-cyano-phenyl

Me

H

N

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

17-357

2-chloropyridine-3-base

Me

H

N

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

17-399

Phenyl

Me

H

N

H

H

H

I

H

Nine fluoro-2-butyl

H

I

17-400

The 2-fluorophenyl

Me

H

N

H

H

H

I

H

Nine fluoro-2-butyl

H

I

17-419

The 3-cyano-phenyl

Me

H

N

H

H

H

I

H

Nine fluoro-2-butyl

H

I

17-420

The 4-cyano-phenyl

Me

H

N

H

H

H

I

H

Nine fluoro-2-butyl

H

I

[table 148]

The 17th table (2)

[table 149]

The 17th table (3)

The compound sequence number

Q 1

R 1

R 2

A

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

17-1338

The 2-fluorophenyl

Me

H

N

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

17-1357

The 3-cyano-phenyl

Me

H

N

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

17-1358

The 4-cyano-phenyl

Me

H

N

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

17-1373

2-chloropyridine-3-base

Me

H

N

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

17-1415

Phenyl

Me

H

N

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

17-1446

2-chloropyridine-3-base

Me

H

N

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

17-1471

Phenyl

Me

H

N

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

17-1502

2-chloropyridine-3-base

Me

H

N

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

17-1527

Phenyl

Me

H

N

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

17-1558

2-chloropyridine-3-base

Me

H

N

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

17-1583

Phenyl

Me

H

N

H

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

17-1614

2-chloropyridine-3-base

Me

H

N

H

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

17-1639

Phenyl

Me

H

N

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

17-1659

The 3-cyano-phenyl

Me

H

N

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

17-1660

The 4-cyano-phenyl

Me

H

N

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

17-1675

2-chloropyridine-3-base

Me

H

N

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

17-1707

Phenyl

Me

H

N

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

17-1727

The 3-cyano-phenyl

Me

H

N

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

17-1728

The 4-cyano-phenyl

Me

H

N

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

17-1743

2-chloropyridine-3-base

Me

H

N

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

17-1775

Phenyl

Me

H

N-oxygen base

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

17-1776

The 3-cyano-phenyl

Me

H

N-oxygen base

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

17-1777

The 4-cyano-phenyl

Me

H

N-oxygen base

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

17-1778

2-chloropyridine-3-base

Me

H

N-oxygen base

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

17-1779

Phenyl

Me

H

N-oxygen base

H

H

H

F

H

Nine fluoro-2-butyl

H

F

17-1780

The 3-cyano-phenyl

Me

H

N-oxygen base

H

H

H

F

H

Nine fluoro-2-butyl

H

F

17-1781

The 4-cyano-phenyl

Me

H

N-oxygen base

H

H

H

F

H

Nine fluoro-2-butyl

H

F

17-1782

2-chloropyridine-3-base

Me

H

N-oxygen base

H

H

H

F

H

Nine fluoro-2-butyl

H

F

17-1783

Phenyl

Me

H

N-oxygen base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

17-1803

The 3-cyano-phenyl

Me

H

N-oxygen base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

17-1804

The 4-cyano-phenyl

Me

H

N-oxygen base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

17-1819

2-chloropyridine-3-base

Me

H

N-oxygen base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

17-1861

Phenyl

Me

H

N-oxygen base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

17-1881

The 3-cyano-phenyl

Me

H

N-oxygen base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

17-1882

The 4-cyano-phenyl

Me

H

N-oxygen base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

17-1897

2-chloropyridine-3-base

Me

H

N-oxygen base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

17-1939

Phenyl

Me

H

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

17-1959

The 3-cyano-phenyl

Me

H

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

17-1960

The 4-cyano-phenyl

Me

H

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

17-1975

2-chloropyridine-3-base

Me

H

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

17-2017

Phenyl

Me

H

N-oxygen base

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

[table 150]

The 17th table (4)

The compound sequence number

Q 1

R 1

R 2

A

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

17-2443

2-chloropyridine-3-base

Me

H

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

17-2485

Phenyl

Me

H

N-oxygen base

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

17-2505

The 3-cyano-phenyl

Me

H

N-oxygen base

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

17-2506

The 4-cyano-phenyl

Me

H

N-oxygen base

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

17-2563

Phenyl

Me

H

N-oxygen base

H

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

17-2583

The 3-cyano-phenyl

Me

H

N-oxygen base

H

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

17-2584

The 4-cyano-phenyl

Me

H

N-oxygen base

H

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

17-2599

2-chloropyridine-3-base

Me

H

N-oxygen base

H

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

17-2641

Phenyl

Me

H

N-oxygen base

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

17-2661

The 3-cyano-phenyl

Me

H

N-oxygen base

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

17-2662

The 4-cyano-phenyl

Me

H

N-oxygen base

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

17-2677

2-chloropyridine-3-base

Me

H

N-oxygen base

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

17-2719

Phenyl

Me

H

N-oxygen base

H

H

H

F

H

Seven fluorine sec.-propyls

H

CF3

17-2720

Phenyl

Me

H

N-oxygen base

H

H

H

C?l

H

Seven fluorine sec.-propyls

H

CF3

17-2740

The 3-cyano-phenyl

Me

H

N-oxygen base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

17-2741

The 4-cyano-phenyl

Me

H

N-oxygen base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

17-2756

2-chloropyridine-3-base

Me

H

N-oxygen base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

17-2798

Phenyl

Me

H

N-oxygen base

H

H

H

F

H

Nine fluoro-2-butyl

H

CF3

17-2799

Phenyl

Me

H

N-oxygen base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

17-2819

The 3-cyano-phenyl

Me

H

N-oxygen base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

17-2820

The 4-cyano-phenyl

Me

H

N-oxygen base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

17-2835

2-chloropyridine-3-base

Me

H

N-oxygen base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

17-2877

Phenyl

Me

H

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

17-2897

The 3-cyano-phenyl

Me

H

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

17-2898

The 4-cyano-phenyl

Me

H

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

17-2913

2-chloropyridine-3-base

Me

H

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

17-2914

2-bromopyridine-3-base

Me

H

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

17-2955

Phenyl

Me

H

N-oxygen base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

17-2975

The 3-cyano-phenyl

Me

H

N-oxygen base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

17-2976

The 4-cyano-phenyl

Me

H

N-oxygen base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

17-2991

2-chloropyridine-3-base

Me

H

N-oxygen base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

17-3033

Phenyl

Me

H

N-oxygen base

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

17-3053

The 3-cyano-phenyl

Me

H

N-oxygen base

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

17-3054

The 4-cyano-phenyl

Me

H

N-oxygen base

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

17-3069

2-chloropyridine-3-base

Me

H

N-oxygen base

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

17-3111

Phenyl

Me

H

N-oxygen base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

17-3131

The 3-cyano-phenyl

Me

H

N-oxygen base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

17-3132

The 4-cyano-phenyl

Me

H

N-oxygen base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

17-3147

2-chloropyridine-3-base

Me

H

N-oxygen base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

17-3189

Phenyl

Me

H

N-oxygen base

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

17-3220

2-chloropyridine-3-base

Me

H

N-oxygen base

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

[table 151]

The 18th table (1)

The compound sequence number

Q 1

R 1

R 2

A

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

18-1

Phenyl

H

Me

N

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

18-2

The 3-cyano-phenyl

H

Me

N

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

18-3

The 4-cyano-phenyl

H

Me

N

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

18-4

2-chloropyridine-3-base

H

Me

N

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

18-5

Phenyl

H

Me

N

H

H

H

F

H

Nine fluoro-2-butyl

H

F

18-6

The 3-cyano-phenyl

H

Me

N

H

H

H

F

H

Nine fluoro-2-butyl

H

F

18-7

The 4-cyano-phenyl

H

Me

N

H

H

H

F

H

Nine fluoro-2-butyl

H

F

18-8

2-chloropyridine-3-base

H

Me

N

H

H

H

F

H

Nine fluoro-2-butyl

H

F

18-9

Phenyl

H

Me

N

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

18-29

The 3-cyano-phenyl

H

Me

N

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

18-30

The 4-cyano-phenyl

H

Me

N

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

18-45

2-chloropyridine-3-base

H

Me

N

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

18-87

Phenyl

H

Me

N

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

18-107

The 3-cyano-phenyl

H

Me

N

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

18-108

The 4-cyano-phenyl

H

Me

N

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

18-123

2-chloropyridine-3-base

H

Me

N

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

18-165

Phenyl

H

Me

N

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

18-176

The 3-iodophenyl

H

Me

N

H

H

H

Br

H

Pentafluoroethyl group

H

Br

18-177

The 4-iodophenyl

H

Me

N

H

H

H

Br

H

Pentafluoroethyl group

H

Br

18-185

The 3-cyano-phenyl

H

Me

N

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

18-186

The 4-cyano-phenyl

H

Me

N

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

18-201

2-chloropyridine-3-base

H

Me

N

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

18-243

Phenyl

H

Me

N

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

18-263

The 3-cyano-phenyl

H

Me

N

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

18-264

The 4-cyano-phenyl

H

Me

N

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

18-279

2-chloropyridine-3-base

H

Me

N

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

18-321

Phenyl

H

Me

N

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

18-341

The 3-cyano-phenyl

H

Me

N

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

18-342

The 4-cyano-phenyl

H

Me

N

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

18-357

2-chloropyridine-3-base

H

Me

N

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

18-399

Phenyl

H

Me

N

H

H

H

I

H

Nine fluoro-2-butyl

H

I

18-419

The 3-cyano-phenyl

H

Me

N

H

H

H

I

H

Nine fluoro-2-butyl

H

I

18-420

The 4-cyano-phenyl

H

Me

N

H

H

H

I

H

Nine fluoro-2-butyl

H

I

18-435

2-chloropyridine-3-base

H

Me

N

H

H

H

I

H

Nine fluoro-2-butyl

H

I

18-477

Phenyl

H

Me

N

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

[table 152]

The 18th table (2)

[table 153]

The 18th table (3)

The compound sequence number

Q 1

R 1

R 2

A

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

18-1280

The 4-cyano-phenyl

H

Me

N

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

18-1295

2-chloropyridine-3-base

H

Me

N

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

18-1308

5-fluorine pyridin-3-yl

H

C(O)Me

N

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

18-1337

Phenyl

H

Me

N

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

18-1338

The 2-fluorophenyl

H

Me

N

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

18-1357

The 3-cyano-phenyl

H

Me

N

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

18-1358

The 4-cyano-phenyl

H

Me

N

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

18-1373

2-chloropyridine-3-base

H

Me

N

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

18-1415

Phenyl

H

Me

N

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

18-1446

2-chloropyridine-3-base

H

Me

N

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

18-1471

Phenyl

H

Me

N

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

18-1502

2-chloropyridine-3-base

H

Me

N

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

18-1527

Phenyl

H

Me

N

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

18-1558

2-chloropyridine-3-base

H

Me

N

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

18-1583

Phenyl

H

Me

N

H

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

18-1614

2-chloropyridine-3-base

H

Me

N

H

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

18-1639

Phenyl

H

Me

N

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

18-1659

The 3-cyano-phenyl

H

Me

N

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

18-1660

The 4-cyano-phenyl

H

Me

N

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

18-1675

2-chloropyridine-3-base

H

Me

N

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

18-1707

Phenyl

H

Me

N

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

18-1727

The 3-cyano-phenyl

H

Me

N

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

18-1728

The 4-cyano-phenyl

H

Me

N

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

18-1743

2-chloropyridine-3-base

H

Me

N

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

18-1775

Phenyl

H

Me

N-oxygen base

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

18-1776

The 3-cyano-phenyl

H

Me

N-oxygen base

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

18-1777

The 4-cyano-phenyl

H

Me

N-oxygen base

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

18-1778

2-chloropyridine-3-base

H

Me

N-oxygen base

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

18-1779

Phenyl

H

Me

N-oxygen base

H

H

H

F

H

Nine fluoro-2-butyl

H

F

18-1780

The 3-cyano-phenyl

H

Me

N-oxygen base

H

H

H

F

H

Nine fluoro-2-butyl

H

F

18-1781

The 4-cyano-phenyl

H

Me

N-oxygen base

H

H

H

F

H

Nine fluoro-2-butyl

H

F

18-1782

2-chloropyridine-3-base

H

Me

N-oxygen base

H

H

H

F

H

Nine fluoro-2-butyl

H

F

18-1783

Phenyl

H

Me

N-oxygen base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

18-1803

The 3-cyano-phenyl

H

Me

N-oxygen base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

18-1804

The 4-cyano-phenyl

H

Me

N-oxygen base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

18-1819

2-chloropyridine-3-base

H

Me

N-oxygen base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

18-1861

Phenyl

H

Me

N-oxygen base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

18-1881

The 3-cyano-phenyl

H

Me

N-oxygen base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

18-1882

The 4-cyano-phenyl

H

Me

N-oxygen base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

18-1897

2-chloropyridine-3-base

H

Me

N-oxygen base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

18-1939

Phenyl

H

Me

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

18-1959

The 3-cyano-phenyl

H

Me

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

18-1960

The 4-cyano-phenyl

H

Me

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

18-1975

2-chloropyridine-3-base

H

Me

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

18-2017

Phenyl

H

Me

N-oxygen base

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

18-2037

The 3-cyano-phenyl

H

Me

N-oxygen base

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

18-2038

The 4-cyano-phenyl

H

Me

N-oxygen base

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

18-2053

2-chloropyridine-3-base

H

Me

N-oxygen base

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

18-2095

Phenyl

H

Me

N-oxygen base

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

18-2115

The 3-cyano-phenyl

H

Me

N-oxygen base

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

18-2116

The 4-cyano-phenyl

H

Me

N-oxygen base

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

18-2131

2-chloropyridine-3-base

H

Me

N-oxygen base

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

18-2173

Phenyl

H

Me

N-oxygen base

H

H

H

I

H

Nine fluoro-2-butyl

H

I

18-2193

The 3-cyano-phenyl

H

Me

N-oxygen base

H

H

H

I

H

Nine fluoro-2-butyl

H

I

18-2194

The 4-cyano-phenyl

H

Me

N-oxygen base

H

H

H

I

H

Nine fluoro-2-butyl

H

I

18-2209

2-chloropyridine-3-base

H

Me

N-oxygen base

H

H

H

I

H

Nine fluoro-2-butyl

H

I

18-2251

Phenyl

H

Me

N-oxygen base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

18-2271

The 3-cyano-phenyl

H

Me

N-oxygen base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

18-2272

The 4-cyano-phenyl

H

Me

N-oxygen base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

18-2287

2-chloropyridine-3-base

H

Me

N-oxygen base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

18-2291

2-nitropyridine-3-base

H

Me

N-oxygen base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OC2F5

18-2329

Phenyl

H

Me

N-oxygen base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

18-2349

The 3-cyano-phenyl

H

Me

N-oxygen base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

[table 154]

The 18th table (4)

The compound sequence number

Q 1

R 1

R 2

A

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

18-2350

The 4-cyano-phenyl

H

Me

N-oxygen base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

18-2365

2-chloropyridine-3-base

H

Me

N-oxygen base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

18-2407

Phenyl

H

Me

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

18-2427

The 3-cyano-phenyl

H

Me

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

18-2428

The 4-cyano-phenyl

H

Me

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

18-2443

2-chloropyridine-3-base

H

Me

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

18-2485

Phenyl

H

Me

N-oxygen base

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

18-2505

The 3-cyano-phenyl

H

Me

N-oxygen base

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

18-2506

The 4-cyano-phenyl

H

Me

N-oxygen base

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

18-2521

2-chloropyridine-3-base

H

Me

N-oxygen base

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

18-2563

Phenyl

H

Me

N-oxygen base

H

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

18-2583

The 3-cyano-phenyl

H

Me

N-oxygen base

H

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

18-2584

The 4-cyano-phenyl

H

Me

N-oxygen base

H

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

18-2599

2-chloropyridine-3-base

H

Me

N-oxygen base

H

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

18-2641

Phenyl

H

Me

N-oxygen base

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

18-2661

The 3-cyano-phenyl

H

Me

N-oxygen base

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

18-2662

The 4-cyano-phenyl

H

Me

N-oxygen base

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

18-2677

2-chloropyridine-3-base

H

Me

N-oxygen base

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

18-2719

Phenyl

H

Me

N-oxygen base

H

H

H

F

H

Seven fluorine sec.-propyls

H

CF3

18-2720

Phenyl

H

Me

N-oxygen base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

18-2740

The 3-cyano-phenyl

H

Me

N-oxygen base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

18-2741

The 4-cyano-phenyl

H

Me

N-oxygen base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

18-2756

2-chloropyridine-3-base

H

Me

N-oxygen base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

18-2798

Phenyl

H

Me

N-oxygen base

H

H

H

F

H

Nine fluoro-2-butyl

H

CF3

18-2799

Phenyl

H

Me

N-oxygen base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

18-2819

The 3-cyano-phenyl

H

Me

N-oxygen base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

18-2820

The 4-cyano-phenyl

H

Me

N-oxygen base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

18-2835

2-chloropyridine-3-base

H

Me

N-oxygen base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

18-2877

Phenyl

H

Me

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

18-2897

The 3-cyano-phenyl

H

Me

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

18-2898

The 4-cyano-phenyl

H

Me

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

18-2913

2-chloropyridine-3-base

H

Me

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

18-2955

Phenyl

H

Me

N-oxygen base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

18-2975

The 3-cyano-phenyl

H

Me

N-oxygen base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

18-2976

The 4-cyano-phenyl

H

Me

N-oxygen base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

18-2991

2-chloropyridine-3-base

H

Me

N-oxygen base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

18-3033

Phenyl

H

Me

N-oxygen base

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

18-3053

The 3-cyano-phenyl

H

Me

N-oxygen base

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

18-3054

The 4-cyano-phenyl

H

Me

N-oxygen base

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

18-3069

2-chloropyridine-3-base

H

Me

N-oxygen base

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

18-3111

Phenyl

H

Me

N-oxygen base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

[table 155]

Table 19 table (1)

The compound sequence number

Q 1

R 1

R 2

A

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

19-1

Phenyl

Me

Me

N

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

19-2

The 3-cyano-phenyl

Me

Me

N

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

19-3

The 4-cyano-phenyl

Me

Me

N

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

19-4

2-chloropyridine-3-base

Me

Me

N

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

19-5

Phenyl

Me

Me

N

H

H

H

F

H

Nine fluoro-2-butyl

H

F

19-6

The 3-cyano-phenyl

Me

Me

N

H

H

H

F

H

Nine fluoro-2-butyl

H

F

19-7

The 4-cyano-phenyl

Me

Me

N

H

H

H

F

H

Nine fluoro-2-butyl

H

F

19-8

2-chloropyridine-3-base

Me

Me

N

H

H

H

F

H

Nine fluoro-2-butyl

H

F

19-9

Phenyl

Me

Me

N

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

19-11

The 3-fluorophenyl

Et

Me

N

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

19-12

The 4-fluorophenyl

Me

E?t

N

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

19-29

The 3-cyano-phenyl

Me

Me

N

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

19-30

The 4-cyano-phenyl

Me

Me

N

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

19-45

2-chloropyridine-3-base

Me

Me

N

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

19-87

Phenyl

Me

Me

N

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

19-107

The 3-cyano-phenyl

Me

Me

N

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

19-108

The 4-cyano-phenyl

Me

Me

N

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

19-123

2-chloropyridine-3-base

Me

Me

N

H

H

H

Cl

H

Nine fluoro-2-butyl

H

Cl

19-165

Phenyl

Me

Me

N

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

19-185

The 3-cyano-phenyl

Me

Me

N

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

19-186

The 4-cyano-phenyl

Me

Me

N

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

19-201

2-chloropyridine-3-base

Me

Me

N

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

19-243

Phenyl

Me

Me

N

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

19-263

The 3-cyano-phenyl

Me

Me

N

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

19-264

The 4-cyano-phenyl

Me

Me

N

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

19-279

2-chloropyridine-3-base

Me

Me

N

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

19-321

Phenyl

Me

Me

N

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

19-341

The 3-cyano-phenyl

Me

Me

N

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

19-342

The 4-cyano-phenyl

Me

Me

N

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

19-357

2-chloropyridine-3-base

Me

Me

N

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

19-399

Phenyl

Me

Me

N

H

H

H

I

H

Nine fluoro-2-butyl

H

I

19-419

The 3-cyano-phenyl

Me

Me

N

H

H

H

I

H

Nine fluoro-2-butyl

H

I

19-420

The 4-cyano-phenyl

Me

Me

N

H

H

H

I

H

Nine fluoro-2-butyl

H

I

19-435

2-chloropyridine-3-base

Me

Me

N

H

H

H

I

H

Nine fluoro-2-butyl

H

I

19-673

Phenyl

Me

Me

N

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

19-693

The 3-cyano-phenyl

Me

Me

N

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

19-694

The 4-cyano-phenyl

Me

Me

N

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

19-709

2-chloropyridine-3-base

Me

Me

N

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

19-751

Phenyl

Me

Me

N

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

19-771

The 3-cyano-phenyl

Me

Me

N

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

19-772

The 4-cyano-phenyl

Me

Me

N

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

19-787

2-chloropyridine-3-base

Me

Me

N

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

19-829

Phenyl

Me

Me

N

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

19-849

The 3-cyano-phenyl

Me

Me

N

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

19-850

The 4-cyano-phenyl

Me

Me

N

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

19-865

2-chloropyridine-3-base

Me

Me

N

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

19-907

Phenyl

Me

Me

N

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

19-927

The 3-cyano-phenyl

Me

Me

N

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

19-928

The 4-cyano-phenyl

Me

Me

N

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

19-943

2-chloropyridine-3-base

Me

Me

N

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

19-985

Phenyl

Me

Me

N

H

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

19-1005

The 3-cyano-phenyl

Me

Me

N

H

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

19-1006

The 4-cyano-phenyl

Me

Me

N

H

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

19-1021

2-chloropyridine-3-base

Me

Me

N

H

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

19-1063

Phenyl

Me

Me

N

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

[table 156]

The 19th table (2)

[table 157]

The 19th table (3)

[table 158]

The 19th table (4)

[table 159]

The 19th table (5)

The compound sequence number

Q 1

R 1

R 2

A

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

19-4561

Phenyl

Me

Me

N-oxygen base

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

19-4592

2-chloropyridine-3-base

Me

Me

N-oxygen base

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

19-4617

Phenyl

Me

Me

N-oxygen base

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

19-4648

2-chloropyridine-3-base

Me

Me

N-oxygen base

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

19-4673

Phenyl

Me

Me

N-oxygen base

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

19-4704

2-chloropyridine-3-base

Me

Me

N-oxygen base

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

19-4729

Phenyl

Me

Me

N-oxygen base

H

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

19-4760

2-chloropyridine-3-base

Me

Me

N-oxygen base

H

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

19-4785

Phenyl

Me

Me

N-oxygen base

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

19-4805

The 3-cyano-phenyl

Me

Me

N-oxygen base

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

19-4806

The 4-cyano-phenyl

Me

Me

N-oxygen base

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

19-4821

2-chloropyridine-3-base

Me

Me

N-oxygen base

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

19-4853

Phenyl

Me

Me

N-oxygen base

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

19-4873

The 3-cyano-phenyl

Me

Me

N-oxygen base

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

19-4874

The 4-cyano-phenyl

Me

Me

N-oxygen base

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

19-4889

2-chloropyridine-3-base

Me

Me

N-oxygen base

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

[table 160]

The 20th table (1)

[table 161]

The 20th table (2)

[table 162]

The 20th table (3)

[table 163]

The 21st table (1)

[table 164]

The 21st table (2)

[table 165]

The 21st table (3)

[table 166]

The 21st table (4)

[table 167]

The 22nd table (1)

[table 168]

The 22nd table (2)

[table 169]

The 23rd table (1)

[table 170]

The 23rd table (2)

The compound sequence number

Q 2

R 1

R 2

A

X 2

X 3

X 4

Y 1

Y 2

Y 3

Y 4

Y 5

23-638

2,2,2-three chloroethyls

H

Me

N

H

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

23-667

2,2,2-three chloroethyls

H

Me

N

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

23-696

2,2,2-three chloroethyls

H

Me

N

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

23-715

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

F

H

Seven fluorine sec.-propyls

H

F

23-716

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

F

H

Nine fluoro-2-butyl

H

F

23-727

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

Cl

23-756

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

C?l

H

Nine fluoro-2-butyl

H

Cl

23-785

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

Br

23-814

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

Br

H

Nine fluoro-2-butyl

H

Br

23-843

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

I

H

Seven fluorine sec.-propyls

H

I

23-872

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

I

H

Nine fluoro-2-butyl

H

I

23-895

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

I

23-903

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

F

H

Seven fluorine sec.-propyls

H

OCF3

23-904

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

F

H

Nine fluoro-2-butyl

H

OCF3

23-915

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

23-944

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

23-973

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

23-1002

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

23-1031

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

23-1060

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

23-1079

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

F

H

Seven fluorine sec.-propyls

H

CF3

23-1080

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

F

H

Nine fluoro-2-butyl

H

CF3

23-1091

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

23-1120

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

23-1149

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

23-1178

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

23-1207

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

23-1236

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

23-1265

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

23-1294

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

23-1323

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

23-1352

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

23-1381

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

23-1410

2,2,2-three chloroethyls

H

Me

N-oxygen base

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

[table 171]

The 24th table (1)

[table 172]

The 24th table (2)

[table 173]

The 25th table (1)

[table 174]

The 25th table (2)

[table 175]

The 26th table (1)

The compound sequence number

Q 1

R 1

R 2

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

26-1

Phenyl

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

26-4

The 4-fluorophenyl

H

H

Cl

Cl

H

Seven fluorine sec.-propyls

H

OCF3

26-12

The 3-iodophenyl

H

H

H

Cl

H

Pentafluoroethyl group

H

OCF3

26-13

The 4-iodophenyl

H

H

H

Cl

H

Pentafluoroethyl group

H

OCF3

26-16

(4-trifluoromethyl) phenyl

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OC2F5

26-17

The 2-nitrophenyl

H

H

H

F

H

Seven fluorine sec.-propyls

H

OCF3

26-20

The 2-cyano-phenyl

H

H

H

Cl

H

Pentafluoroethyl group

H

OC2F5

26-21

The 3-cyano-phenyl

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

26-22

The 4-cyano-phenyl

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

26-28

4-bromo-2-chloro-phenyl-

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OC2F5

26-36

2-fluorine pyridin-3-yl

H

H

H

Cl

H

Pentafluoroethyl group

H

OCF3

26-37

2-chloropyridine-3-base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

26-41

2-nitropyridine-3-base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OC2F5

26-50

5-fluorine pyridin-3-yl

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OC2F5

26-55

5-nitropyridine-3-base

H

H

H

Cl

H

Pentafluoroethyl group

H

OCF3

26-59

4-bromopyridine-3-base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OC2F5

26-60

4-iodine pyridine-3-base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OC2F5

26-78

4-cyanopyridine-2-base

H

H

H

Cl

H

Pentafluoroethyl group

H

OCF3

26-79

Phenyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

26-95

The 2-nitrophenyl

H

H

H

F

H

Nine fluoro-2-butyl

H

OCF3

26-99

The 3-cyano-phenyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

26-100

The 4-cyano-phenyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

26-105

2-chloro-4, the 5-difluorophenyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OC2F5

26-115

2-chloropyridine-3-base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

26-121

6-fluorine pyridin-3-yl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OC2F5

26-130

5-bromopyridine-3-base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OC2F5

26-131

5-iodine pyridine-3-base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OC2F5

26-139

4-(trifluoromethyl) pyridin-3-yl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OC2F5

26-140

4-nitropyridine-3-base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OC2F5

26-157

Phenyl

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

26-158

The 2-fluorophenyl

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

26-177

The 3-cyano-phenyl

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

26-178

The 4-cyano-phenyl

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

26-193

2-chloropyridine-3-base

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

[table 176]

The 26th table (2)

The compound sequence number

Q 1

R 1

R 2

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

26-470

Phenyl

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

26-471

The 2-fluorophenyl

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

26-481

The 3-iodophenyl

H

H

H

Cl

H

Pentafluoroethyl group

H

CF3

26-482

The 4-iodophenyl

H

H

H

Cl

H

Pentafluoroethyl group

H

CF3

26-489

The 2-cyano-phenyl

H

H

H

Cl

H

Pentafluoroethyl group

H

C2F5

26-490

The 3-cyano-phenyl

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

26-491

The 4-cyano-phenyl

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

26-494

The 2,4 dichloro benzene base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

C2F5

26-498

2-bromo-4-chloro-phenyl-

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

n-C3F7

26-505

2-fluorine pyridin-3-yl

H

H

H

Cl

H

Pentafluoroethyl group

H

CF3

26-506

2-chloropyridine-3-base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

26-510

2-nitropyridine-3-base

H

H

Cl

Cl

H

Seven fluorine sec.-propyls

H

CF3

26-519

5-fluorine pyridin-3-yl

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

C2F5

26-521

5-bromopyridine-3-base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

n-C3F7

26-522

5-iodine pyridine-3-base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

i-C3F7

26-524

5-nitropyridine-3-base

H

H

H

Cl

H

Pentafluoroethyl group

H

CF3

26-526

4-fluorine pyridin-3-yl

H

H

H

Cl

H

Pentafluoroethyl group

H

CF3

26-528

4-bromopyridine-3-base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

n-C3F7

26-529

4-iodine pyridine-3-base

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

i-C3F7

26-548

Phenyl

H

H

H

F

H

Nine fluoro-2-butyl

H

CF3

26-549

Phenyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

26-550

The 2-fluorophenyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

26-562

(2-trifluoromethyl) phenyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

C2F5

26-569

The 3-cyano-phenyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

26-570

The 4-cyano-phenyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

26-579

2-chloro-4-nitrophenyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

i-C3F7

26-585

2-chloropyridine-3-base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

26-598

5-fluorine pyridin-3-yl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

C2F5

26-600

5-bromopyridine-3-base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

n-C3F7

26-601

5-iodine pyridine-3-base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

i-C3F7

26-605

4-fluorine pyridin-3-yl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

C2F5

26-609

4-(trifluoromethyl) pyridin-3-yl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

n-C3F7

26-610

4-nitropyridine-3-base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

i-C3F7

26-626

4-cyanopyridine-2-base

H

H

H

Cl

H

Nine fluoro-2-butyl

H

C2F5

26-627

Phenyl

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

26-628

The 2-fluorophenyl

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

26-629

The 3-fluorophenyl

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

26-630

The 4-fluorophenyl

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

26-631

The 2-chloro-phenyl-

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

26-632

The 3-chloro-phenyl-

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

26-633

The 4-chloro-phenyl-

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

[table 177]

The 26th table (3)

[table 178]

The 26th table (4)

The compound sequence number

Q 1

R 1

R 2

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

26-711

The 4-chloro-phenyl-

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-712

The 2-bromophenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-713

The 3-bromophenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-714

The 4-bromophenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-715

The 2-iodophenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-716

The 3-iodophenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-717

The 4-iodophenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-718

(2-trifluoromethyl) phenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-719

(3-trifluoromethyl) phenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-720

(4-trifluoromethyl) phenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-721

The 2-nitrophenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-722

The 3-nitrophenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-723

The 4-nitrophenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-724

The 2-cyano-phenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-725

The 3-cyano-phenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-726

The 4-cyano-phenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-727

2, the 6-difluorophenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-728

3, the 4-dichlorophenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-729

The 2,4 dichloro benzene base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-730

2-chloro-4-fluorophenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-731

2-chloro-4, the 5-difluorophenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-732

4-bromo-2-chloro-phenyl-

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-733

2-bromo-4-chloro-phenyl-

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-734

2-bromo-4-fluorophenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-735

2-chloro-4-nitrophenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-736

3,5-dicyano phenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-737

4-cyano group-2-fluorophenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-738

2-chloro-4-cyano-phenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-739

Pyridin-3-yl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-740

2-fluorine pyridin-3-yl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-741

2-chloropyridine-3-base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-742

2-bromopyridine-3-base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-743

2-iodine pyridine-3-base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-744

2-(trifluoromethyl) pyridin-3-yl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-745

2-nitropyridine-3-base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-746

2-cyanopyridine-3-base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-747

6-fluorine pyridin-3-yl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-748

6-chloropyridine-3-base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-749

6-bromopyridine-3-base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-750

6-iodine pyridine-3-base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-751

6-(trifluoromethyl) pyridin-3-yl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-752

6-nitropyridine-3-base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

[table 179]

The 26th table (5)

The compound sequence number

Q 1

R 1

R 2

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

26-768

2,6-dichloropyridine-3-base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-769

N-pyridine oxide-3-base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-770

Pyridin-4-yl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-771

2-chloropyridine-4-base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-772

3-bromopyridine-4-base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-773

3,5-dichloropyridine-4-base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-774

3-(trifluoromethyl) pyridin-4-yl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-775

2,6-dicyanopyridine-4-base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-776

N-pyridine oxide-4-base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-777

Pyridine-2-base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-778

3-chloropyridine-2-base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-779

4-bromopyridine-2-base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-780

5-iodine pyridine-2-base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-781

6-chloropyridine-2-base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-782

4-cyanopyridine-2-base

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

26-783

Phenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-784

The 2-fluorophenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-785

The 3-fluorophenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-786

The 4-fluorophenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-787

The 2-chloro-phenyl-

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-788

The 3-chloro-phenyl-

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-789

The 4-chloro-phenyl-

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-790

The 2-bromophenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-791

The 3-bromophenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-792

The 4-bromophenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-793

The 2-iodophenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-794

The 3-iodophenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-795

The 4-iodophenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-796

(2-trifluoromethyl) phenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-797

(3-trifluoromethyl) phenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-798

(4-trifluoromethyl) phenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-799

The 2-nitrophenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-800

The 3-nitrophenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-801

The 4-nitrophenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-802

The 2-cyano-phenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-803

The 3-cyano-phenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-804

The 4-cyano-phenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-805

2, the 6-difluorophenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-806

3, the 4-dichlorophenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-807

The 2,4 dichloro benzene base

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-808

2-chloro-4-fluorophenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

26-809

2-chloro-4, the 5-difluorophenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

[table 180]

The 26th table (6)

[table 181]

The 26th table (7)

The compound sequence number

Q 1

R 1

R 2

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

26-880

The 2-cyano-phenyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-881

The 3-cyano-phenyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-882

The 4-cyano-phenyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-883

2, the 6-difluorophenyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-884

3, the 4-dichlorophenyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-885

The 2,4 dichloro benzene base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-886

2-chloro-4-fluorophenyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-887

2-chloro-4, the 5-difluorophenyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-888

4-bromo-2-chloro-phenyl-

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-889

2-bromo-4-chloro-phenyl-

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-890

2-bromo-4-fluorophenyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-891

2-chloro-4-nitrophenyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-892

3,5-dicyano phenyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-893

4-cyano group-2-fluorophenyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-894

2-chloro-4-cyano-phenyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-895

Pyridin-3-yl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-896

2-fluorine pyridin-3-yl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-897

2-chloropyridine-3-base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-898

2-bromopyridine-3-base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-899

2-iodine pyridine-3-base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-900

2-(trifluoromethyl) pyridin-3-yl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-901

2-nitropyridine-3-base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-902

2-cyanopyridine-3-base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-903

6-fluorine pyridin-3-yl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-904

6-chloropyridine-3-base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-905

6-bromopyridine-3-base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-906

6-iodine pyridine-3-base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-907

6-(trifluoromethyl) pyridin-3-yl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-908

6-nitropyridine-3-base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-909

6-cyanopyridine-3-base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-910

5-fluorine pyridin-3-yl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-911

5-chloropyridine-3-base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-912

5-bromopyridine-3-base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-913

5-iodine pyridine-3-base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-914

5-(trifluoromethyl) pyridin-3-yl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-915

5-nitropyridine-3-base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-916

5-cyanopyridine-3-base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-917

4-fluorine pyridin-3-yl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-918

4-chloropyridine-3-base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-919

4-bromopyridine-3-base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-920

4-iodine pyridine-3-base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-921

4-(trifluoromethyl) pyridin-3-yl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

[table 182]

The 26th table (8)

The compound sequence number

Q 1

R 1

R 2

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

26-936

5-iodine pyridine-2-base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-937

6-chloropyridine-2-base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-938

4-cyanopyridine-2-base

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

26-939

Phenyl

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

26-946

The 2-bromophenyl

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OC2F5

26-950

The 3-iodophenyl

H

H

H

OCF3

H

Pentafluoroethyl group

H

OCF3

26-951

The 4-iodophenyl

H

H

H

OCF3

H

Pentafluoroethyl group

H

OCF3

26-954

The 3-cyano-phenyl

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

26-955

The 4-cyano-phenyl

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

26-960

2-chloro-4, the 5-difluorophenyl

H

H

H

OC2F5

H

Seven fluorine sec.-propyls

H

OC2F5

26-963

2-bromo-4-fluorophenyl

H

H

H

OC2F5

H

Seven fluorine sec.-propyls

H

OCF3

26-964

2-chloro-4-nitrophenyl

H

H

Cl

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

26-969

2-fluorine pyridin-3-yl

H

H

H

OCF3

H

Pentafluoroethyl group

H

OCF3

26-970

2-chloropyridine-3-base

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

26-979

5-cyanopyridine-3-base

H

H

H

OC2F5

H

Seven fluorine sec.-propyls

H

OC2F5

26-981

4-cyanopyridine-3-base

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OC2F5

26-994

4-cyanopyridine-2-base

H

H

H

OCF3

H

Pentafluoroethyl group

H

OCF3

26-995

Phenyl

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

26-1002

The 2-bromophenyl

H

H

H

OC2F5

H

Nine fluoro-2-butyl

H

OCF3

26-1008

(2-trifluoromethyl) phenyl

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OC2F5

26-1010

The 3-cyano-phenyl

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

26-1011

The 4-cyano-phenyl

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

26-1017

4-bromo-2-chloro-phenyl-

H

H

H

OC2F5

H

Nine fluoro-2-butyl

H

OC2F5

26-1026

2-chloropyridine-3-base

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

26-1033

6-cyanopyridine-3-base

H

H

H

OC2F5

H

Nine fluoro-2-butyl

H

OCF3

26-1035

5-cyanopyridine-3-base

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OC2F5

26-1037

4-cyanopyridine-3-base

H

H

H

OC2F5

H

Nine fluoro-2-butyl

H

OC2F5

26-1051

Phenyl

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

26-1058

The 2-bromophenyl

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

OC2F5

26-1062

The 3-iodophenyl

H

H

H

CF3

H

Pentafluoroethyl group

H

OCF3

26-1063

The 4-iodophenyl

H

H

H

CF3

H

Pentafluoroethyl group

H

OCF3

26-1064

(2-trifluoromethyl) phenyl

H

H

H

C2F5

H

Seven fluorine sec.-propyls

H

OC2F5

26-1065

The 3-nitrophenyl

H

H

H

C2F5

H

Seven fluorine sec.-propyls

H

OCF3

26-1066

The 3-cyano-phenyl

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

26-1067

The 4-cyano-phenyl

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

26-1074

2-bromo-4-chloro-phenyl-

H

H

H

n-C3F7

H

Seven fluorine sec.-propyls

H

OCF3

26-1078

4-cyano group-2-fluorophenyl

H

H

H

i-C3F7

H

Seven fluorine sec.-propyls

H

OCF3

26-1081

2-fluorine pyridin-3-yl

H

H

H

CF3

H

Pentafluoroethyl group

H

OCF3

26-1082

2-chloropyridine-3-base

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

26-1089

6-cyanopyridine-3-base

H

H

H

n-C3F7

H

Seven fluorine sec.-propyls

H

OC2F5

26-1091

5-cyanopyridine-3-base

H

H

H

i-C3F7

H

Seven fluorine sec.-propyls

H

OC2F5

26-1106

4-cyanopyridine-2-base

H

H

H

CF3

H

Pentafluoroethyl group

H

OCF3

[table 183]

The 26th table (9)

The compound sequence number

Q 1

R 1

R 2

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

26-1177

(3-trifluoromethyl) phenyl

H

H

H

C2F5

H

Seven fluorine sec.-propyls

H

CF3

26-1183

The 3-cyano-phenyl

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

26-1184

The 4-cyano-phenyl

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

26-1190

4-bromo-2-chloro-phenyl-

H

H

H

n-C3F7

H

Seven fluorine sec.-propyls

H

CF3

26-1195

4-cyano group-2-fluorophenyl

H

H

H

i-C3F7

H

Seven fluorine sec.-propyls

H

CF3

26-1198

2-fluorine pyridin-3-yl

H

H

H

CF3

H

Pentafluoroethyl group

H

CF3

26-1199

2-chloropyridine-3-base

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

26-1200

2-bromopyridine-3-base

H

H

H

C2F5

H

Seven fluorine sec.-propyls

H

C2F5

26-1203

2-nitropyridine-3-base

H

H

Cl

CF3

H

Seven fluorine sec.-propyls

H

CF3

26-1211

6-cyanopyridine-3-base

H

H

H

C2F5

H

Seven fluorine sec.-propyls

H

n-C3F7

26-1215

4-cyanopyridine-3-base

H

H

H

C2F5

H

Seven fluorine sec.-propyls

H

i-C3F7

26-1230

4-cyanopyridine-2-base

H

H

H

CF3

H

Pentafluoroethyl group

H

CF3

26-1231

Phenyl

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

26-1243

The 4-iodophenyl

H

H

H

C2F5

H

Nine fluoro-2-butyl

H

CF3

26-1251

The 3-cyano-phenyl

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

26-1252

The 4-cyano-phenyl

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

26-1258

4-bromo-2-chloro-phenyl-

H

H

H

n-C3F7

H

Nine fluoro-2-butyl

H

CF3

26-1263

4-cyano group-2-fluorophenyl

H

H

H

i-C3F7

H

Nine fluoro-2-butyl

H

CF3

26-1267

2-chloropyridine-3-base

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

26-1268

2-bromopyridine-3-base

H

H

H

C2F5

H

Nine fluoro-2-butyl

H

C2F5

26-1279

6-cyanopyridine-3-base

H

H

H

C2F5

H

Nine fluoro-2-butyl

H

n-C3F7

26-1283

4-cyanopyridine-3-base

H

H

H

C2F5

H

Nine fluoro-2-butyl

H

i-C3F7

[table 184]

The 27th table (1)

The compound sequence number

Q 1

R 1

R 2

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

27-1

Phenyl

Me

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

27-21

The 3-cyano-phenyl

Me

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

27-22

The 4-cyano-phenyl

Me

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

27-37

2-chloropyridine-3-base

Me

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

27-79

Phenyl

Me

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

27-99

The 3-cyano-phenyl

Me

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

27-100

The 4-cyano-phenyl

Me

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

27-115

2-chloropyridine-3-base

Me

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

27-157

Phenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

27-177

The 3-cyano-phenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

27-178

The 4-cyano-phenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

27-193

2-chloropyridine-3-base

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

27-235

Phenyl

Me

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

27-255

The 3-cyano-phenyl

Me

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

27-256

The 4-cyano-phenyl

Me

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

27-271

2-chloropyridine-3-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

27-313

Phenyl

Me

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

27-333

The 3-cyano-phenyl

Me

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

27-334

The 4-cyano-phenyl

Me

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

27-349

2-chloropyridine-3-base

Me

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

27-391

Phenyl

Me

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

27-411

The 3-cyano-phenyl

Me

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

27-412

The 4-cyano-phenyl

Me

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

27-427

2-chloropyridine-3-base

Me

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

27-469

Phenyl

Me

H

H

F

H

Seven fluorine sec.-propyls

H

CF3

27-470

Phenyl

Me

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

27-484

(3-trifluoromethyl) phenyl

Et

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

27-489

The 2-cyano-phenyl

Me

H

H

Cl

H

Pentafluoroethyl group

H

C2F5

27-490

The 3-cyano-phenyl

Me

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

27-491

The 4-cyano-phenyl

Me

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

27-494

The 2,4 dichloro benzene base

Me

H

H

Cl

H

Seven fluorine sec.-propyls

H

C2F5

27-495

2-chloro-4-fluorophenyl

n-Pr

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

27-498

2-bromo-4-chloro-phenyl-

Me

H

H

Cl

H

Seven fluorine sec.-propyls

H

n-C3F7

27-506

2-chloropyridine-3-base

Me

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

27-510

2-nitropyridine-3-base

Me

H

Cl

Cl

H

Seven fluorine sec.-propyls

H

CF3

[table 185]

The 27th table (2)

The compound sequence number

Q 1

R 1

R 2

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

27-605

4-fluorine pyridin-3-yl

Me

H

H

Cl

H

Nine fluoro-2-butyl

H

C2F5

27-607

4-bromopyridine-3-base

C(O)C(O)Me

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

27-609

4-(trifluoromethyl) pyridin-3-yl

Me

H

H

Cl

H

Nine fluoro-2-butyl

H

n-C3F7

27-610

4-nitropyridine-3-base

C(O)C(O)Et

H

H

Cl

H

Nine fluoro-2-butyl

H

i-C3F7

27-624

5-iodine pyridine-2-base

C(O)Me

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

27-626

4-cyanopyridine-2-base

C(O)Et

H

H

Cl

H

Nine fluoro-2-butyl

H

C2F5

27-627

Phenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-628

The 2-fluorophenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-629

The 3-fluorophenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-630

The 4-fluorophenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-631

The 2-chloro-phenyl-

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-632

The 3-chloro-phenyl-

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-633

The 4-chloro-phenyl-

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-634

The 2-bromophenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-635

The 3-bromophenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-636

The 4-bromophenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-637

The 2-iodophenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-638

The 3-iodophenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-639

The 4-iodophenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-640

(2-trifluoromethyl) phenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-641

(3-trifluoromethyl) phenyl

S(O)2Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-642

(4-trifluoromethyl) phenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-643

The 2-nitrophenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-644

The 3-nitrophenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-645

The 4-nitrophenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-646

The 2-cyano-phenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-647

The 3-cyano-phenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-648

The 4-cyano-phenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-649

2, the 6-difluorophenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-650

3, the 4-dichlorophenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-651

The 2,4 dichloro benzene base

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-652

2-chloro-4-fluorophenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-653

2-chloro-4, the 5-difluorophenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-654

4-bromo-2-chloro-phenyl-

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-655

2-bromo-4-chloro-phenyl-

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-656

2-bromo-4-fluorophenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-657

2-chloro-4-nitrophenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-658

3,5-dicyano phenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-659

4-cyano group-2-fluorophenyl

S(O)2Et

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-660

2-chloro-4-cyano-phenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-661

Pyridin-3-yl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

27-662

2-fluorine pyridin-3-yl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

[table 186]

The 27th table (3)

[table 187]

The 27th table (4)

The compound sequence number

Q 1

R 1

R 2

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

27-749

6-bromopyridine-3-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-750

6-iodine pyridine-3-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-751

6-(trifluoromethyl) pyridin-3-yl

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-752

6-nitropyridine-3-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-753

6-cyanopyridine-3-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-754

5-fluorine pyridin-3-yl

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-755

5-chloropyridine-3-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-756

5-bromopyridine-3-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-757

5-iodine pyridine-3-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-758

5-(trifluoromethyl) pyridin-3-yl

CN

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-759

5-nitropyridine-3-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-760

5-cyanopyridine-3-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-761

4-fluorine pyridin-3-yl

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-762

4-chloropyridine-3-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-763

4-bromopyridine-3-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-764

4-iodine pyridine-3-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-765

4-(trifluoromethyl) pyridin-3-yl

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-766

4-nitropyridine-3-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-767

4-cyanopyridine-3-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-768

2,6-dichloropyridine-3-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-769

N-pyridine oxide-3-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-770

Pyridin-4-yl

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-771

2-chloropyridine-4-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-772

3-bromopyridine-4-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-773

3,5-dichloropyridine-4-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-774

3-(trifluoromethyl) pyridin-4-yl

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-775

2,6-dicyanopyridine-4-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-776

N-pyridine oxide-4-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-777

Pyridine-2-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-778

3-chloropyridine-2-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-779

4-bromopyridine-2-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-780

5-iodine pyridine-2-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-781

6-chloropyridine-2-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-782

4-cyanopyridine-2-base

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

27-783

Phenyl

Me

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

27-784

The 2-fluorophenyl

Me

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

27-785

The 3-fluorophenyl

Me

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

27-786

The 4-fluorophenyl

Me

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

27-787

The 2-chloro-phenyl-

Me

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

27-788

The 3-chloro-phenyl-

Me

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

27-789

The 4-chloro-phenyl-

Me

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

[table 188]

The 27th table (5)

[table 189]

The 27th table (6)

The compound sequence number

Q 1

R 1

R 2

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

27-877

The 2-nitrophenyl

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-878

The 3-nitrophenyl

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-879

The 4-nitrophenyl

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-880

The 2-cyano-phenyl

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-881

The 3-cyano-phenyl

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-882

The 4-cyano-phenyl

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-883

2, the 6-difluorophenyl

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-884

3, the 4-dichlorophenyl

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-885

The 2,4 dichloro benzene base

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-886

2-chloro-4-fluorophenyl

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-887

2-chloro-4, the 5-difluorophenyl

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-888

4-bromo-2-chloro-phenyl-

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-889

2-bromo-4-chloro-phenyl-

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-890

2-bromo-4-fluorophenyl

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-891

2-chloro-4-nitrophenyl

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-892

3,5-dicyano phenyl

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-893

4-cyano group-2-fluorophenyl

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-894

2-chloro-4-cyano-phenyl

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-895

Pyridin-3-yl

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-896

2-fluorine pyridin-3-yl

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-897

2-chloropyridine-3-base

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-898

2-bromopyridine-3-base

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-899

2-iodine pyridine-3-base

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-900

2-(trifluoromethyl) pyridin-3-yl

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-901

2-nitropyridine-3-base

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-902

2-cyanopyridine-3-base

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-903

6-fluorine pyridin-3-yl

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-904

6-chloropyridine-3-base

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-905

6-bromopyridine-3-base

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-906

6-iodine pyridine-3-base

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-907

6-(trifluoromethyl) pyridin-3-yl

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-908

6-nitropyridine-3-base

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-909

6-cyanopyridine-3-base

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-910

5-fluorine pyridin-3-yl

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-911

5-chloropyridine-3-base

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-912

5-bromopyridine-3-base

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-913

5-iodine pyridine-3-base

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-914

5-(trifluoromethyl) pyridin-3-yl

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-915

5-nitropyridine-3-base

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-916

5-cyanopyridine-3-base

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

27-917

4-fluorine pyridin-3-yl

Me

H

H

I

H

Nine fluoro-2-butyl

H

CF3

[table 190]

The 27th table (7)

The compound sequence number

Q 1

R 1

R 2

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

27-995

Phenyl

Me

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

27-1026

2-chloropyridine-3-base

Me

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

27-1051

Phenyl

Me

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

27-1082

2-chloropyridine-3-base

Me

H

H

CF3

H

Seven fluorine sec.-propyls

H

OCF3

27-1107

Phenyl

Me

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

27-1138

2-chloropyridine-3-base

Me

H

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

27-1163

Phenyl

Me

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

27-1183

The 3-cyano-phenyl

Me

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

27-1184

The 4-cyano-phenyl

Me

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

27-1199

2-chloropyridine-3-base

Me

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

27-1231

Phenyl

Me

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

27-1251

The 3-cyano-phenyl

Me

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

27-1252

The 4-cyano-phenyl

Me

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

27-1267

2-chloropyridine-3-base

Me

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

[table 191]

The 28th table (1)

The compound sequence number

Q 1

R 1

R 2

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

28-1

Phenyl

H

Me

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

28-21

The 3-cyano-phenyl

H

Me

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

28-22

The 4-cyano-phenyl

H

Me

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

28-37

2-chloropyridine-3-base

H

Me

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

28-79

Phenyl

H

Me

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

28-99

The 3-cyano-phenyl

H

Me

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

28-100

The 4-cyano-phenyl

H

Me

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

28-115

2-chloropyridine-3-base

H

Me

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

28-157

Phenyl

H

Me

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

28-177

The 3-cyano-phenyl

H

Me

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

28-178

The 4-cyano-phenyl

H

Me

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

28-193

2-chloropyridine-3-base

H

Me

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

28-235

Phenyl

H

Me

H

Br

H

Nine fluoro-2-butyl

H

OCF3

28-255

The 3-cyano-phenyl

H

Me

H

Br

H

Nine fluoro-2-butyl

H

OCF3

28-256

The 4-cyano-phenyl

H

Me

H

Br

H

Nine fluoro-2-butyl

H

OCF3

28-271

2-chloropyridine-3-base

H

Me

H

Br

H

Nine fluoro-2-butyl

H

OCF3

28-313

Phenyl

H

Me

H

I

H

Seven fluorine sec.-propyls

H

OCF3

28-333

The 3-cyano-phenyl

H

Me

H

I

H

Seven fluorine sec.-propyls

H

OCF3

28-334

The 4-cyano-phenyl

H

Me

H

I

H

Seven fluorine sec.-propyls

H

OCF3

28-349

2-chloropyridine-3-base

H

Me

H

I

H

Seven fluorine sec.-propyls

H

OCF3

28-391

Phenyl

H

Me

H

I

H

Nine fluoro-2-butyl

H

OCF3

28-411

The 3-cyano-phenyl

H

Me

H

I

H

Nine fluoro-2-butyl

H

OCF3

28-412

The 4-cyano-phenyl

H

Me

H

I

H

Nine fluoro-2-butyl

H

OCF3

28-427

2-chloropyridine-3-base

H

Me

H

I

H

Nine fluoro-2-butyl

H

OCF3

28-469

Phenyl

H

Me

H

F

H

Seven fluorine sec.-propyls

H

CF3

28-470

Phenyl

H

Me

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

28-481

The 3-iodophenyl

H

Me

H

Cl

H

Pentafluoroethyl group

H

CF3

28-482

The 4-iodophenyl

H

Me

H

Cl

H

Pentafluoroethyl group

H

CF3

28-484

(3-trifluoromethyl) phenyl

H

Et

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

28-489

The 2-cyano-phenyl

H

Me

H

Cl

H

Pentafluoroethyl group

H

C2F5

28-490

The 3-cyano-phenyl

H

Me

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

28-491

The 4-cyano-phenyl

H

Me

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

28-494

The 2,4 dichloro benzene base

H

Me

H

Cl

H

Seven fluorine sec.-propyls

H

C2F5

28-495

2-chloro-4-fluorophenyl

H

n-Pr

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

[table 192]

The 28th table (2)

[table 193]

The 29th table (1)

[table 194]

The 29th table (2)

[table 195]

The 29th table (3)

The compound sequence number

Q 1

R 1

R 2

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

29-1530

2-chloropyridine-3-base

Me

Me

H

CF3

H

Nine fluoro-2-butyl

H

OCF3

29-1555

Phenyl

Me

Me

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

29-1575

The 3-cyano-phenyl

Me

Me

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

29-1576

The 4-cyano-phenyl

Me

Me

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

29-1591

2-chloropyridine-3-base

Me

Me

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

29-1623

Phenyl

Me

Me

H

CF3

H

Nine fluoro-2-butyl

H

CF3

29-1643

The 3-cyano-phenyl

Me

Me

H

CF3

H

Nine fluoro-2-butyl

H

CF3

29-1644

The 4-cyano-phenyl

Me

Me

H

CF3

H

Nine fluoro-2-butyl

H

CF3

29-1659

2-chloropyridine-3-base

Me

Me

H

CF3

H

Nine fluoro-2-butyl

H

CF3

[table 196]

The 30th table (1)

[table 197]

The 31st table (1)

The compound sequence number

Q 2

R 1

R 2

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

31-1

2,2,2-three chloroethyls

H

H

H

F

H

Seven fluorine sec.-propyls

H

OCF3

31-2

2,2,2-three chloroethyls

H

H

H

F

H

Nine fluoro-2-butyl

H

OCF3

31-9

The 2-chloroethyl

H

H

Cl

Cl

H

Seven fluorine sec.-propyls

H

OCF3

31-13

2,2,2-three chloroethyls

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

31-16

3-fluoro-n-propyl group

H

H

H

Cl

H

Pentafluoroethyl group

H

OCF3

31-18

3-bromo-n-propyl group

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OC2F5

31-22

1,3-two chloro-2-propyl group

H

H

H

Cl

H

Pentafluoroethyl group

H

OC2F5

31-26

4,4,4-three fluoro-n-butyl

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

31-36

The 2-bromotrifluoromethane

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OC2F5

31-42

2,2,2-three chloroethyls

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

31-55

4,4,4-three fluoro-n-butyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

31-57

The s-butyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OC2F5

31-66

2-iodine ethyl

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OC2F5

31-71

2,2,2-three chloroethyls

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

31-84

4,4,4-three fluoro-n-butyl

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

31-100

2,2,2-three chloroethyls

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

31-102

The n-propyl group

H

H

H

Br

H

Nine fluoro-2-butyl

H

OC2F5

31-113

4,4,4-three fluoro-n-butyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

31-129

2,2,2-three chloroethyls

H

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

[table 198]

The 31st table (2)

The compound sequence number

Q 2

R 1

R 2

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

31-202

4,4,4-three fluoro-n-butyl

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

31-203

The i-butyl

H

H

Cl

Cl

H

Seven fluorine sec.-propyls

H

CF3

31-204

The s-butyl

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

31-205

Vinyl

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

31-206

Benzyl

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

31-207

Phenyl

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

31-208

Methyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-209

Ethyl

H

H

H

C?l

H

Nine fluoro-2-butyl

H

i-C3F7

31-210

The 2-fluoro ethyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-211

The 2-chloroethyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-212

The 2-bromotrifluoromethane

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-213

2-iodine ethyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-214

The 2-cyano ethyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-215

2,2-two fluoro ethyls

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-216

2, the 2-Dichloroethyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-217

2,2, the 2-trifluoroethyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-218

2,2,2-three chloroethyls

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-219

2,2, the 2-three bromomethyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-220

The n-propyl group

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-221

3-fluoro-n-propyl group

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-222

3-chloro-n-propyl group

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-223

3-bromo-n-propyl group

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-224

The i-propyl group

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-225

1,2-two fluoro-2-propyl group

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-226

1,3-two fluoro-2-propyl group

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-227

1,3-two chloro-2-propyl group

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-228

1-chloro-3-fluoro-2-propyl group

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-229

3,3,3-three fluoro-n-propyl group

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-230

The n-butyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-231

4,4,4-three fluoro-n-butyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-232

The i-butyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-233

The s-butyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-234

Vinyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-235

Benzyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-236

Phenyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

31-237

Methyl

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

31-238

Ethyl

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

31-239

The 2-fluoro ethyl

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

31-240

The 2-chloroethyl

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

31-241

The 2-bromotrifluoromethane

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

31-242

2-iodine ethyl

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

31-243

The 2-cyano ethyl

H

H

H

Br

H

Seven fluorine sec.-propyls

H

C2F5

31-244

2,2-two fluoro ethyls

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

[table 199]

The 31st table (3)

The compound sequence number

Q 2

R 1

R 2

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

31-261

The i-butyl

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

31-262

The s-butyl

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

31-263

Vinyl

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

31-264

Benzyl

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

31-265

Phenyl

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

31-266

Methyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-267

Ethyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-268

The 2-fluoro ethyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-269

The 2-chloroethyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-270

The 2-bromotrifluoromethane

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-271

2-iodine ethyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-272

The 2-cyano ethyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-273

2,2-two fluoro ethyls

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-274

2, the 2-Dichloroethyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-275

2,2, the 2-trifluoroethyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-276

2,2,2-three chloroethyls

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-277

2,2, the 2-three bromomethyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-278

The n-propyl group

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-279

3-fluoro-n-propyl group

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-280

3-chloro-n-propyl group

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-281

3-bromo-n-propyl group

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-282

The i-propyl group

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-283

1,2-two fluoro-2-propyl group

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-284

1,3-two fluoro-2-propyl group

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-285

1,3-two chloro-2-propyl group

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-286

1-chloro-3-fluoro-2-propyl group

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-287

3,3,3-three fluoro-n-propyl group

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-288

The n-butyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-289

4,4,4-three fluoro-n-butyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-290

The i-butyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-291

The s-butyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-292

Vinyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-293

Benzyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

31-294

Phenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

i-C3F7

31-295

Methyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

31-296

Ethyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

31-297

The 2-fluoro ethyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

31-298

The 2-chloroethyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

31-299

The 2-bromotrifluoromethane

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

31-300

2-iodine ethyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

31-301

The 2-cyano ethyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

31-302

2,2-two fluoro ethyls

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

[table 200]

The 31st table (4)

The compound sequence number

Q 2

R 1

R 2

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

31-321

Vinyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

31-322

Benzyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

31-323

Phenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

31-324

Methyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-325

Ethyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-326

The 2-fluoro ethyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-327

The 2-chloroethyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-328

The 2-bromotrifluoromethane

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-329

2-iodine ethyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-330

The 2-cyano ethyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-331

2,2-two fluoro ethyls

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-332

2, the 2-Dichloroethyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-333

2,2, the 2-trifluoroethyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-334

2,2,2-three chloroethyls

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-335

2,2, the 2-three bromomethyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-336

The n-propyl group

H

H

H

I

H

Nine fluoro-2-butyl

H

n-C3F7

31-337

3-fluoro-n-propyl group

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-338

3-chloro-n-propyl group

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-339

3-bromo-n-propyl group

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-340

The i-propyl group

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-341

1,2-two fluoro-2-propyl group

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-342

1,3-two fluoro-2-propyl group

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-343

1,3-two chloro-2-propyl group

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-344

1-chloro-3-fluoro-2-propyl group

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-345

3,3,3-three fluoro-n-propyl group

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-346

The n-butyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-347

4,4,4-three fluoro-n-butyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-348

The i-butyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-349

The s-butyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-350

Vinyl

H

H

H

I

H

Nine fluoro-2-butyl

H

i-C3F7

31-351

Benzyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-352

Phenyl

H

H

H

I

H

Nine fluoro-2-butyl

H

CF3

31-359

The 2-cyano ethyl

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OC2F5

31-363

2,2,2-three chloroethyls

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

31-364

2,2, the 2-three bromomethyl

H

H

H

OCF3

H

Pentafluoroethyl group

H

OCF3

31-373

1-chloro-3-fluoro-2-propyl group

H

H

H

OC2F5

H

Seven fluorine sec.-propyls

H

OC2F5

31-376

4,4,4-three fluoro-n-butyl

H

H

H

OCF3

H

Seven fluorine sec.-propyls

H

OCF3

31-378

The s-butyl

H

H

H

OC2F5

H

Seven fluorine sec.-propyls

H

OCF3

31-391

2,2, the 2-trifluoroethyl

H

H

H

OC2F5

H

Nine fluoro-2-butyl

H

OCF3

31-392

2,2,2-three chloroethyls

H

H

H

OCF3

H

Nine fluoro-2-butyl

H

OCF3

31-394

The n-propyl group

H

H

Cl

OCF3

H

Nine fluoro-2-butyl

H

OC2F5

31-403

3,3,3-three fluoro-n-propyl group

H

H

H

OC2F5

H

Nine fluoro-2-butyl

H

OC2F5

[table 201]

The 31st table (5)

The compound sequence number

Q 2

R 1

R 2

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

31-479

2,2,2-three chloroethyls

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

31-482

3-fluoro-n-propyl group

H

H

H

C2F5

H

Seven fluorine sec.-propyls

H

CF3

31-485

The i-propyl group

H

H

H

i-C3F7

H

Seven fluorine sec.-propyls

H

CF3

31-487

1,3-two fluoro-2-propyl group

H

H

H

CF3

H

Pentafluoroethyl group

H

CF3

31-490

3,3,3-three fluoro-n-propyl group

H

H

H

C2F5

H

Seven fluorine sec.-propyls

H

C2F5

31-492

4,4,4-three fluoro-n-butyl

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

31-493

The i-butyl

H

H

H

C2F5

H

Seven fluorine sec.-propyls

H

n-C3F7

31-495

Vinyl

H

H

H

n-C3F7

H

Seven fluorine sec.-propyls

H

CF3

31-508

2,2,2-three chloroethyls

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

31-520

The n-butyl

H

H

H

C2F5

H

Nine fluoro-2-butyl

H

i-C3F7

31-521

4,4,4-three fluoro-n-butyl

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

31-522

The i-butyl

H

H

Cl

CF3

H

Nine fluoro-2-butyl

H

CF3

31-524

Vinyl

H

H

H

n-C3F7

H

Nine fluoro-2-butyl

H

i-C3F7

[table 202]

The 32nd table (1)

[table 203]

The 33rd table (1)

The compound sequence number

Q 2

R 1

R 2

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

33-1

2,2,2-three chloroethyls

H

Me

H

F

H

Seven fluorine sec.-propyls

H

OCF3

33-2

2,2,2-three chloroethyls

H

Me

H

F

H

Nine fluoro-2-butyl

H

OCF3

33-13

2,2,2-three chloroethyls

H

Me

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

33-42

2,2,2-three chloroethyls

H

Me

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

33-71

2,2,2-three chloroethyls

H

Me

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

33-100

2,2,2-three chloroethyls

H

Me

H

Br

H

Nine fluoro-2-butyl

H

OCF3

33-129

2,2,2-three chloroethyls

H

Me

H

I

H

Seven fluorine sec.-propyls

H

OCF3

33-158

2,2,2-three chloroethyls

H

Me

H

I

H

Nine fluoro-2-butyl

H

OCF3

33-177

2,2,2-three chloroethyls

H

Me

H

F

H

Seven fluorine sec.-propyls

H

CF3

33-178

2,2,2-three chloroethyls

H

Me

H

F

H

Nine fluoro-2-butyl

H

CF3

33-185

The 2-cyano ethyl

H

Et

H

Cl

H

Seven fluorine sec.-propyls

H

C2F5

33-189

2,2,2-three chloroethyls

H

Me

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

33-191

The n-propyl group

H

Me

H

Cl

H

Pentafluoroethyl group

H

CF3

33-195

The i-propyl group

H

n-Pr

H

Cl

H

Seven fluorine sec.-propyls

H

n-C3F7

33-198

1,3-two chloro-2-propyl group

H

Me

H

Cl

H

Pentafluoroethyl group

H

CF3

33-199

1-chloro-3-fluoro-2-propyl group

H

i-Pr

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

33-203

The i-butyl

H

CH2CH＝CH2

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

33-207

Phenyl

H

Me

Cl

Cl

H

Seven fluorine sec.-propyls

H

CF3

33-209

Ethyl

H

Me

H

Cl

H

Nine fluoro-2-butyl

H

i-C3F7

33-214

The 2-cyano ethyl

H

CN

H

Cl

H

Nine fluoro-2-butyl

H

CF3

33-218

2,2,2-three chloroethyls

H

Me

H

Cl

H

Nine fluoro-2-butyl

H

CF3

33-220

The n-propyl group

H

CH2C≡CH

H

Cl

H

Nine fluoro-2-butyl

H

CF3

33-232

The i-butyl

H

NH2

H

Cl

H

Nine fluoro-2-butyl

H

CF3

33-243

The 2-cyano ethyl

H

Me

H

Br

H

Seven fluorine sec.-propyls

H

C2F5

33-247

2,2,2-three chloroethyls

H

Me

H

Br

H

Seven fluorine sec.-propyls

H

CF3

33-249

The n-propyl group

H

C(O)OMe

H

Br

H

Seven fluorine sec.-propyls

H

CF3

33-254

1,2-two fluoro-2-propyl group

H

Me

H

Br

H

Seven fluorine sec.-propyls

H

n-C3F7

33-260

4,4,4-three fluoro-n-butyl

H

Me

H

Br

H

Seven fluorine sec.-propyls

H

CF3

33-263

Vinyl

H

C(O)C(O)OMe

H

Br

H

Seven fluorine sec.-propyls

H

CF3

33-276

2,2,2-three chloroethyls

H

Me

H

Br

H

Nine fluoro-2-butyl

H

CF3

33-278

The n-propyl group

H

C(O)OEt

H

Br

H

Nine fluoro-2-butyl

H

CF3

33-282

The i-propyl group

H

C(O)Me

H

Br

H

Nine fluoro-2-butyl

H

CF3

33-289

4,4,4-three fluoro-n-butyl

H

Me

H

Br

H

Nine fluoro-2-butyl

H

CF3

33-294

Phenyl

H

C(O)C(O)OEt

H

Br

H

Nine fluoro-2-butyl

H

i-C3F7

33-305

2,2,2-three chloroethyls

H

Me

H

I

H

Seven fluorine sec.-propyls

H

CF3

[table 204]

The 34th table (1)

[table 205]

The 34th table (2)

[table 206]

The 35th table (1)

[table 207]

The 36th table (1)

[table 208]

The 37th table (1)

The compound sequence number

Q 1

R 1

R 2

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

37-1

Phenyl

H

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

37-2

Phenyl

H

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

37-3

Phenyl

H

H

Cl

I

H

Seven fluorine sec.-propyls

H

CF3

37-4

Phenyl

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

37-5

Phenyl

H

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

37-6

Phenyl

H

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

37-7

Phenyl

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

37-8

Phenyl

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

37-9

Phenyl

Me

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

37-10

Phenyl

Me

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

37-11

Phenyl

Me

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

37-12

Phenyl

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

37-13

Phenyl

Me

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

37-14

Phenyl

H

Me

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

37-15

Phenyl

H

Me

H

I

H

Seven fluorine sec.-propyls

H

CF3

37-16

Phenyl

H

Me

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

37-17

Phenyl

H

Me

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

37-18

Phenyl

H

Me

H

Br

H

Nine fluoro-2-butyl

H

CF3

37-19

Phenyl

H

Me

H

CF3

H

Nine fluoro-2-butyl

H

CF3

37-20

Phenyl

Me

Me

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

37-21

Phenyl

Me

Me

H

I

H

Seven fluorine sec.-propyls

H

CF3

37-22

Phenyl

Me

Me

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

37-23

Phenyl

Me

Me

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

37-24

Phenyl

Me

Me

H

Br

H

Nine fluoro-2-butyl

H

CF3

37-25

Phenyl

Me

Me

H

CF3

H

Nine fluoro-2-butyl

H

CF3

37-26

Phenyl

Me

H

H

Br

F

Seven fluorine sec.-propyls

H

OCF3

37-27

Phenyl

H

H

H

I

H

Seven fluorine sec.-propyls

F

CF3

37-28

Phenyl

H

Me

H

CF3

Cl

Seven fluorine sec.-propyls

H

CF3

37-29

Phenyl

H

H

H

Cl

H

Nine fluoro-2-butyl

Cl

OCF3

37-30

Phenyl

H

H

H

Br

Br

Nine fluoro-2-butyl

H

CF3

37-31

Phenyl

H

H

H

I

H

Nine fluoro-2-butyl

I

CF3

37-32

Phenyl

H

H

H

Cl

Me

Nine fluoro-2-butyl

H

CF3

37-33

Phenyl

H

H

H

CF3

H

Nine fluoro-2-butyl

Et

CF3

[table 209]

The 38th table (1)

[table 210]

The 39th table (1)

[table 211]

The 40th table (1)

[table 212]

The 41st table (1)

The compound sequence number

Q 2

R 1

R 2

X 2

Y 1

Y 2

Y 3

Y 4

Y 5

41-1

2,2,2-three chloroethyls

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

41-2

2,2,2-three chloroethyls

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

41-3

2,2,2-three chloroethyls

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

41-4

2,2,2-three chloroethyls

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

41-5

2,2,2-three chloroethyls

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

41-6

2,2,2-three chloroethyls

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

41-7

2,2,2-three chloroethyls

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

41-8

2,2,2-three chloroethyls

Me

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

41-9

2,2,2-three chloroethyls

Me

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

41-10

2,2,2-three chloroethyls

Me

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

41-11

2,2,2-three chloroethyls

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

41-12

2,2,2-three chloroethyls

Me

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

41-13

2,2,2-three chloroethyls

H

Me

H

I

H

Seven fluorine sec.-propyls

H

OCF3

41-14

2,2,2-three chloroethyls

H

Me

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

41-15

2,2,2-three chloroethyls

H

Me

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

41-16

2,2,2-three chloroethyls

H

Me

H

Br

H

Nine fluoro-2-butyl

H

OCF3

41-17

2,2,2-three chloroethyls

H

Me

H

I

H

Nine fluoro-2-butyl

H

CF3

41-18

2,2,2-three chloroethyls

H

Me

H

CF3

H

Nine fluoro-2-butyl

H

CF3

41-19

2,2,2-three chloroethyls

Me

Me

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

41-20

2,2,2-three chloroethyls

Me

Me

H

Br

H

Seven fluorine sec.-propyls

H

CF3

41-21

2,2,2-three chloroethyls

Me

Me

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

41-22

2,2,2-three chloroethyls

Me

Me

H

I

H

Nine fluoro-2-butyl

H

OCF3

41-23

2,2,2-three chloroethyls

Me

Me

H

Cl

H

Nine fluoro-2-butyl

H

CF3

41-24

2,2,2-three chloroethyls

Me

Me

H

CF3

H

Nine fluoro-2-butyl

H

CF3

41-25

2,2,2-three chloroethyls

H

H

H

Br

F

Seven fluorine sec.-propyls

H

OCF3

41-26

2,2,2-three chloroethyls

H

H

H

I

H

Seven fluorine sec.-propyls

Cl

CF3

41-27

2,2,2-three chloroethyls

H

H

H

CF3

Br

Seven fluorine sec.-propyls

H

CF3

41-28

2,2,2-three chloroethyls

H

H

H

I

H

Nine fluoro-2-butyl

I

OCF3

41-29

2,2,2-three chloroethyls

H

H

H

Br

Me

Nine fluoro-2-butyl

H

CF3

41-30

2,2,2-three chloroethyls

H

H

H

CF3

H

Nine fluoro-2-butyl

Et

CF3

41-31

2,2,2-three chloroethyls

H

H

Cl

Br

H

Seven fluorine sec.-propyls

H

CF3

[table 213]

The 42nd table (1)

[table 214]

The 43rd table (1)

The compound sequence number

Q 2

R 1

R 2

X 2

Y 1

Y 2

Y 3

Y 4

Y 5

43-1

2,2,2-three chloroethyls

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

43-2

2,2,2-three chloroethyls

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

43-3

2,2,2-three chloroethyls

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

43-4

2,2,2-three chloroethyls

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

43-5

2,2,2-three chloroethyls

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

43-6

2,2,2-three chloroethyls

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

43-7

2,2,2-three chloroethyls

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

43-8

2,2,2-three chloroethyls

Me

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

43-9

2,2,2-three chloroethyls

Me

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

43-10

2,2,2-three chloroethyls

Me

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

43-11

2,2,2-three chloroethyls

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

43-12

2,2,2-three chloroethyls

Me

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

43-13

2,2,2-three chloroethyls

H

Me

H

I

H

Seven fluorine sec.-propyls

H

OCF3

43-14

2,2,2-three chloroethyls

H

Me

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

43-15

2,2,2-three chloroethyls

H

Me

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

43-16

2,2,2-three chloroethyls

H

Me

H

Br

H

Nine fluoro-2-butyl

H

OCF3

43-17

2,2,2-three chloroethyls

H

Me

H

I

H

Nine fluoro-2-butyl

H

CF3

43-18

2,2,2-three chloroethyls

H

Me

H

CF3

H

Nine fluoro-2-butyl

H

CF3

43-19

2,2,2-three chloroethyls

Me

Me

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

43-20

2,2,2-three chloroethyls

Me

Me

H

Br

H

Seven fluorine sec.-propyls

H

CF3

43-21

2,2,2-three chloroethyls

Me

Me

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

43-22

2,2,2-three chloroethyls

Me

Me

H

I

H

Nine fluoro-2-butyl

H

OCF3

43-23

2,2,2-three chloroethyls

Me

Me

H

Cl

H

Nine fluoro-2-butyl

H

CF3

43-24

2,2,2-three chloroethyls

Me

Me

H

CF3

H

Nine fluoro-2-butyl

H

CF3

43-25

2,2,2-three chloroethyls

H

H

H

Br

F

Seven fluorine sec.-propyls

H

OCF3

43-26

2,2,2-three chloroethyls

H

H

H

I

H

Seven fluorine sec.-propyls

Cl

CF3

43-27

2,2,2-three chloroethyls

H

H

H

CF3

Br

Seven fluorine sec.-propyls

H

CF3

43-28

2,2,2-three chloroethyls

H

H

H

I

H

Nine fluoro-2-butyl

I

OCF3

43-29

2,2,2-three chloroethyls

H

H

H

Br

Me

Nine fluoro-2-butyl

H

CF3

43-30

2,2,2-three chloroethyls

H

H

H

CF3

H

Nine fluoro-2-butyl

Et

CF3

43-31

2,2,2-three chloroethyls

H

H

Cl

Br

H

Seven fluorine sec.-propyls

H

CF3

[table 215]

The 44th table (1)

The compound sequence number

Q 2

R 1

R 2

X 1

Y 1

Y 2

Y 3

Y 4

Y 5

44-1

2,2,2-three chloroethyls

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

44-2

2,2,2-three chloroethyls

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

44-3

2,2,2-three chloroethyls

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

44-4

2,2,2-three chloroethyls

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

44-5

2,2,2-three chloroethyls

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

44-6

2,2,2-three chloroethyls

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

44-7

2,2,2-three chloroethyls

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

44-8

2,2,2-three chloroethyls

Me

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

44-9

2,2,2-three chloroethyls

Me

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

44-10

2,2,2-three chloroethyls

Me

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

44-11

2,2,2-three chloroethyls

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

44-12

2,2,2-three chloroethyls

Me

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

44-13

2,2,2-three chloroethyls

H

Me

H

I

H

Seven fluorine sec.-propyls

H

OCF3

44-14

2,2,2-three chloroethyls

H

Me

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

44-15

2,2,2-three chloroethyls

H

Me

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

44-16

2,2,2-three chloroethyls

H

Me

H

Br

H

Nine fluoro-2-butyl

H

OCF3

44-17

2,2,2-three chloroethyls

H

Me

H

I

H

Nine fluoro-2-butyl

H

CF3

44-18

2,2,2-three chloroethyls

H

Me

H

CF3

H

Nine fluoro-2-butyl

H

CF3

44-19

2,2,2-three chloroethyls

Me

Me

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

44-20

2,2,2-three chloroethyls

Me

Me

H

Br

H

Seven fluorine sec.-propyls

H

CF3

44-21

2,2,2-three chloroethyls

Me

Me

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

44-22

2,2,2-three chloroethyls

Me

Me

H

I

H

Nine fluoro-2-butyl

H

OCF3

44-23

2,2,2-three chloroethyls

Me

Me

H

Cl

H

Nine fluoro-2-butyl

H

CF3

44-24

2,2,2-three chloroethyls

Me

Me

H

CF3

H

Nine fluoro-2-butyl

H

CF3

44-25

2,2,2-three chloroethyls

H

H

H

Br

F

Seven fluorine sec.-propyls

H

OCF3

44-26

2,2,2-three chloroethyls

H

H

H

I

H

Seven fluorine sec.-propyls

Cl

CF3

44-27

2,2,2-three chloroethyls

H

H

H

CF3

Br

Seven fluorine sec.-propyls

H

CF3

44-28

2,2,2-three chloroethyls

H

H

H

I

H

Nine fluoro-2-butyl

I

OCF3

44-29

2,2,2-three chloroethyls

H

H

H

Br

Me

Nine fluoro-2-butyl

H

CF3

44-30

2,2,2-three chloroethyls

H

H

H

CF3

H

Nine fluoro-2-butyl

Et

CF3

44-31

2,2,2-three chloroethyls

H

H

Cl

Br

H

Seven fluorine sec.-propyls

H

CF3

[table 216]

The 45th table (1)

The compound sequence number

Q 2

R 1

R 2

X 1

Y 1

Y 2

Y 3

Y 4

Y 5

45-1

2,2,2-three chloroethyls

H

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

45-2

2,2,2-three chloroethyls

H

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

45-3

2,2,2-three chloroethyls

H

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

45-4

2,2,2-three chloroethyls

H

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

45-5

2,2,2-three chloroethyls

H

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

45-6

2,2,2-three chloroethyls

H

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

45-7

2,2,2-three chloroethyls

Me

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

45-8

2,2,2-three chloroethyls

Me

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

45-9

2,2,2-three chloroethyls

Me

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

45-10

2,2,2-three chloroethyls

Me

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

45-11

2,2,2-three chloroethyls

Me

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

45-12

2,2,2-three chloroethyls

Me

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

45-13

2,2,2-three chloroethyls

H

Me

H

I

H

Seven fluorine sec.-propyls

H

OCF3

45-14

2,2,2-three chloroethyls

H

Me

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

45-15

2,2,2-three chloroethyls

H

Me

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

45-16

2,2,2-three chloroethyls

H

Me

H

Br

H

Nine fluoro-2-butyl

H

OCF3

45-17

2,2,2-three chloroethyls

H

Me

H

I

H

Nine fluoro-2-butyl

H

CF3

45-18

2,2,2-three chloroethyls

H

Me

H

CF3

H

Nine fluoro-2-butyl

H

CF3

45-19

2,2,2-three chloroethyls

Me

Me

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

45-20

2,2,2-three chloroethyls

Me

Me

H

Br

H

Seven fluorine sec.-propyls

H

CF3

45-21

2,2,2-three chloroethyls

Me

Me

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

45-22

2,2,2-three chloroethyls

Me

Me

H

I

H

Nine fluoro-2-butyl

H

OCF3

45-23

2,2,2-three chloroethyls

Me

Me

H

Cl

H

Nine fluoro-2-butyl

H

CF3

45-24

2,2,2-three chloroethyls

Me

Me

H

CF3

H

Nine fluoro-2-butyl

H

CF3

45-25

2,2,2-three chloroethyls

H

H

H

Br

F

Seven fluorine sec.-propyls

H

OCF3

45-26

2,2,2-three chloroethyls

H

H

H

I

H

Seven fluorine sec.-propyls

Cl

CF3

45-27

2,2,2-three chloroethyls

H

H

H

CF3

Br

Seven fluorine sec.-propyls

H

CF3

45-28

2,2,2-three chloroethyls

H

H

H

I

H

Nine fluoro-2-butyl

I

OCF3

45-29

2,2,2-three chloroethyls

H

H

H

Br

Me

Nine fluoro-2-butyl

H

CF3

45-30

2,2,2-three chloroethyls

H

H

H

CF3

H

Nine fluoro-2-butyl

Et

CF3

45-31

2,2,2-three chloroethyls

H

H

Cl

Br

H

Seven fluorine sec.-propyls

H

CF3

[table 217]

The 46th table (1)

[table 218]

The 46th table (2)

The compound sequence number

Q 1

R 1

R 2

A

X 2

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

46-52

Phenyl

H

Me

NH

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

46-53

Phenyl

H

Me

NH

H

H

I

H

Nine fluoro-2-butyl

H

CF3

46-54

Phenyl

H

Me

NH

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

46-55

Phenyl

Me

Me

S

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

46-56

Phenyl

Me

Me

S

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

46-57

Phenyl

Me

Me

S

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

46-58

Phenyl

Me

Me

S

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

46-59

Phenyl

Me

Me

S

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

46-60

Phenyl

Me

Me

S

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

46-61

Phenyl

Me

Me

O

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

46-62

Phenyl

Me

Me

O

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

46-63

Phenyl

Me

Me

O

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

46-64

Phenyl

Me

Me

O

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

46-65

Phenyl

Me

Me

O

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

46-66

Phenyl

Me

Me

O

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

46-67

Phenyl

Me

Me

NH

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

46-68

Phenyl

Me

Me

NH

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

46-69

Phenyl

Me

Me

NH

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

46-70

Phenyl

Me

Me

NH

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

46-71

Phenyl

Me

Me

NH

H

H

I

H

Nine fluoro-2-butyl

H

CF3

46-72

Phenyl

Me

Me

NH

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

46-73

Phenyl

Me

H

S

H

H

Cl

F

Seven fluorine sec.-propyls

H

OCF3

46-74

Phenyl

H

H

S

H

H

Br

H

Seven fluorine sec.-propyls

F

CF3

46-75

Phenyl

H

H

S

H

H

CF3

Cl

Seven fluorine sec.-propyls

H

CF3

46-76

Phenyl

H

H

S

H

H

I

H

Nine fluoro-2-butyl

Cl

OCF3

46-77

Phenyl

H

H

S

H

H

Cl

Br

Nine fluoro-2-butyl

H

CF3

46-78

Phenyl

H

H

S

H

H

CF3

H

Nine fluoro-2-butyl

Br

CF3

46-79

Phenyl

H

H

O

H

H

Br

I

Seven fluorine sec.-propyls

H

OCF3

46-80

Phenyl

Me

H

O

H

H

I

H

Seven fluorine sec.-propyls

I

CF3

46-81

Phenyl

H

H

O

H

H

CF3

Me

Seven fluorine sec.-propyls

H

CF3

46-82

Phenyl

H

H

O

H

H

Cl

H

Nine fluoro-2-butyl

Me

OCF3

46-83

Phenyl

H

H

O

H

H

Br

F

Nine fluoro-2-butyl

F

CF3

46-84

Phenyl

H

H

O

H

H

CF3

Cl

Nine fluoro-2-butyl

Cl

CF3

46-85

Phenyl

H

H

NH

H

H

I

Br

Seven fluorine sec.-propyls

Br

OCF3

46-86

Phenyl

H

H

NH

H

H

Cl

I

Seven fluorine sec.-propyls

I

CF3

46-87

Phenyl

Me

H

NH

H

H

CF3

F

Seven fluorine sec.-propyls

Me

CF3

46-88

Phenyl

H

H

NH

H

H

Br

Cl

Nine fluoro-2-butyl

Me

OCF3

46-89

Phenyl

H

H

NH

H

H

I

Br

Nine fluoro-2-butyl

Me

CF3

46-90

Phenyl

H

H

NH

H

H

CF3

I

Nine fluoro-2-butyl

Me

CF3

[table 219]

The 47th table (1)

The compound sequence number

Q 1

R 1

R 2

A

X 1

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

47-1

Phenyl

H

H

S

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

47-2

Phenyl

H

H

S

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

47-3

Phenyl

H

H

S

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

47-4

Phenyl

H

H

S

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

47-5

Phenyl

H

H

S

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

47-6

Phenyl

H

H

S

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

47-7

Phenyl

H

H

O

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

47-8

Phenyl

H

H

O

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

47-9

Phenyl

H

H

O

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

47-10

Phenyl

H

H

O

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

47-11

Phenyl

H

H

O

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

47-12

Phenyl

H

H

O

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

47-13

Phenyl

H

H

NH

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

47-14

Phenyl

H

H

NH

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

47-15

Phenyl

H

H

NH

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

47-16

Phenyl

H

H

NH

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

47-17

Phenyl

H

H

NH

H

H

I

H

Nine fluoro-2-butyl

H

CF3

47-18

Phenyl

H

H

NH

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

47-19

Phenyl

Me

H

S

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

47-20

Phenyl

Me

H

S

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

47-21

Phenyl

Me

H

S

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

47-22

Phenyl

Me

H

S

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

47-23

Phenyl

Me

H

S

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

47-24

Phenyl

Me

H

S

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

47-25

Phenyl

Me

H

O

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

47-26

Phenyl

Me

H

O

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

47-27

Phenyl

Me

H

O

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

47-28

Phenyl

Me

H

O

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

47-29

Phenyl

Me

H

O

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

47-30

Phenyl

Me

H

O

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

47-31

Phenyl

Me

H

NH

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

47-32

Phenyl

Me

H

NH

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

47-33

Phenyl

Me

H

NH

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

47-34

Phenyl

Me

H

NH

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

[table 220]

The 47th table (2)

[table 221]

The 48th table (1)

[table 222]

The 48th table (2)

[table 223]

The 49th table (1)

The compound sequence number

Q 2

R 1

R 2

A

X 2

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

49-1

2,2,2-three chloroethyls

H

H

S

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

49-2

2,2,2-three chloroethyls

H

H

S

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

49-3

2,2,2-three chloroethyls

H

H

S

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

49-4

2,2,2-three chloroethyls

H

H

S

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

49-5

2,2,2-three chloroethyls

H

H

S

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

49-6

2,2,2-three chloroethyls

H

H

S

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

49-7

2,2,2-three chloroethyls

H

H

O

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

49-8

2,2,2-three chloroethyls

H

H

O

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

49-9

2,2,2-three chloroethyls

H

H

O

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

49-10

2,2,2-three chloroethyls

H

H

O

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

49-11

2,2,2-three chloroethyls

H

H

O

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

49-12

2,2,2-three chloroethyls

H

H

O

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

49-13

2,2,2-three chloroethyls

H

H

NH

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

49-14

2,2,2-three chloroethyls

H

H

NH

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

49-15

2,2,2-three chloroethyls

H

H

NH

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

49-16

2,2,2-three chloroethyls

H

H

NH

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

49-17

2,2,2-three chloroethyls

H

H

NH

H

H

I

H

Nine fluoro-2-butyl

H

CF3

49-18

2,2,2-three chloroethyls

H

H

NH

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

49-19

2,2,2-three chloroethyls

Me

H

S

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

49-20

2,2,2-three chloroethyls

Me

H

S

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

49-21

2,2,2-three chloroethyls

Me

H

S

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

49-22

2,2,2-three chloroethyls

Me

H

S

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

49-23

2,2,2-three chloroethyls

Me

H

S

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

49-24

2,2,2-three chloroethyls

Me

H

S

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

49-25

2,2,2-three chloroethyls

Me

H

O

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

49-26

2,2,2-three chloroethyls

Me

H

O

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

49-27

2,2,2-three chloroethyls

Me

H

O

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

49-28

2,2,2-three chloroethyls

Me

H

O

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

49-29

2,2,2-three chloroethyls

Me

H

O

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

49-30

2,2,2-three chloroethyls

Me

H

O

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

49-31

2,2,2-three chloroethyls

Me

H

NH

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

49-32

2,2,2-three chloroethyls

Me

H

NH

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

49-33

2,2,2-three chloroethyls

Me

H

NH

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

49-34

2,2,2-three chloroethyls

Me

H

NH

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

49-35

2,2,2-three chloroethyls

Me

H

NH

H

H

I

H

Nine fluoro-2-butyl

H

CF3

[table 224]

The 49th table (2)

[table 225]

The 50th table (1)

The compound sequence number

Q 2

R 1

R 2

A

X 1

X 3

Y 1

Y 2

Y 3

Y 4

Y 5

50-1

2,2,2-three chloroethyls

H

H

S

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

50-2

2,2,2-three chloroethyls

H

H

S

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

50-3

2,2,2-three chloroethyls

H

H

S

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

50-4

2,2,2-three chloroethyls

H

H

S

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

50-5

2,2,2-three chloroethyls

H

H

S

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

50-6

2,2,2-three chloroethyls

H

H

S

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

50-7

2,2,2-three chloroethyls

H

H

O

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

50-8

2,2,2-three chloroethyls

H

H

O

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

50-9

2,2,2-three chloroethyls

H

H

O

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

50-10

2,2,2-three chloroethyls

H

H

O

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

50-11

2,2,2-three chloroethyls

H

H

O

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

50-12

2,2,2-three chloroethyls

H

H

O

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

50-13

2,2,2-three chloroethyls

H

H

NH

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

50-14

2,2,2-three chloroethyls

H

H

NH

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

50-15

2,2,2-three chloroethyls

H

H

NH

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

50-16

2,2,2-three chloroethyls

H

H

NH

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

50-17

2,2,2-three chloroethyls

H

H

NH

H

H

I

H

Nine fluoro-2-butyl

H

CF3

50-18

2,2,2-three chloroethyls

H

H

NH

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

50-19

2,2,2-three chloroethyls

Me

H

S

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

50-20

2,2,2-three chloroethyls

Me

H

S

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

50-21

2,2,2-three chloroethyls

Me

H

S

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

50-22

2,2,2-three chloroethyls

Me

H

S

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

50-23

2,2,2-three chloroethyls

Me

H

S

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

50-24

2,2,2-three chloroethyls

Me

H

S

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

50-25

2,2,2-three chloroethyls

Me

H

O

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

50-26

2,2,2-three chloroethyls

Me

H

O

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

50-27

2,2,2-three chloroethyls

Me

H

O

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

50-28

2,2,2-three chloroethyls

Me

H

O

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

50-29

2,2,2-three chloroethyls

Me

H

O

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

50-30

2,2,2-three chloroethyls

Me

H

O

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

50-31

2,2,2-three chloroethyls

Me

H

NH

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

50-32

2,2,2-three chloroethyls

Me

H

NH

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

50-33

2,2,2-three chloroethyls

Me

H

NH

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

50-34

2,2,2-three chloroethyls

Me

H

NH

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

[table 226]

The 50th table (2)

[table 227]

The 51st table (1)

The compound sequence number

Q 2

R 1

R 2

A

X 1

X 2

Y 1

Y 2

Y 3

Y 4

Y 5

51-1

2,2,2-three chloroethyls

H

H

S

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

51-2

2,2,2-three chloroethyls

H

H

S

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

51-3

2,2,2-three chloroethyls

H

H

S

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

51-4

2,2,2-three chloroethyls

H

H

S

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

51-5

2,2,2-three chloroethyls

H

H

S

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

51-6

2,2,2-three chloroethyls

H

H

S

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

51-7

2,2,2-three chloroethyls

H

H

O

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

51-8

2,2,2-three chloroethyls

H

H

O

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

51-9

2,2,2-three chloroethyls

H

H

O

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

51-10

2,2,2-three chloroethyls

H

H

O

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

51-11

2,2,2-three chloroethyls

H

H

O

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

51-12

2,2,2-three chloroethyls

H

H

O

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

51-13

2,2,2-three chloroethyls

H

H

NH

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

51-14

2,2,2-three chloroethyls

H

H

NH

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

51-15

2,2,2-three chloroethyls

H

H

NH

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

51-16

2,2,2-three chloroethyls

H

H

NH

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

51-17

2,2,2-three chloroethyls

H

H

NH

H

H

I

H

Nine fluoro-2-butyl

H

CF3

51-18

2,2,2-three chloroethyls

H

H

NH

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

51-19

2,2,2-three chloroethyls

Me

H

S

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

51-20

2,2,2-three chloroethyls

Me

H

S

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

51-21

2,2,2-three chloroethyls

Me

H

S

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

51-22

2,2,2-three chloroethyls

Me

H

S

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

51-23

2,2,2-three chloroethyls

Me

H

S

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

51-24

2,2,2-three chloroethyls

Me

H

S

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

51-25

2,2,2-three chloroethyls

Me

H

O

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

51-26

2,2,2-three chloroethyls

Me

H

O

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

51-27

2,2,2-three chloroethyls

Me

H

O

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

51-28

2,2,2-three chloroethyls

Me

H

O

H

H

Cl

H

Nine fluoro-2-butyl

H

OCF3

51-29

2,2,2-three chloroethyls

Me

H

O

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

51-30

2,2,2-three chloroethyls

Me

H

O

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

51-31

2,2,2-three chloroethyls

Me

H

NH

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

51-32

2,2,2-three chloroethyls

Me

H

NH

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

51-33

2,2,2-three chloroethyls

Me

H

NH

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

51-34

2,2,2-three chloroethyls

Me

H

NH

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

51-35

2,2,2-three chloroethyls

Me

H

NH

H

H

I

H

Nine fluoro-2-butyl

H

CF3

[table 228]

The 51st table (2)

The compound sequence number

Q 2

R 1

R 2

A

X 1

X 2

Y 1

Y 2

Y 3

Y 4

Y 5

51-52

2,2,2-three chloroethyls

H

Me

NH

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

51-53

2,2,2-three chloroethyls

H

Me

NH

H

H

I

H

Nine fluoro-2-butyl

H

CF3

51-54

2,2,2-three chloroethyls

H

Me

NH

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

51-55

2,2,2-three chloroethyls

Me

Me

S

H

H

Cl

H

Seven fluorine sec.-propyls

H

OCF3

51-56

2,2,2-three chloroethyls

Me

Me

S

H

H

Br

H

Seven fluorine sec.-propyls

H

CF3

51-57

2,2,2-three chloroethyls

Me

Me

S

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

51-58

2,2,2-three chloroethyls

Me

Me

S

H

H

I

H

Nine fluoro-2-butyl

H

OCF3

51-59

2,2,2-three chloroethyls

Me

Me

S

H

H

Cl

H

Nine fluoro-2-butyl

H

CF3

51-60

2,2,2-three chloroethyls

Me

Me

S

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

51-61

2,2,2-three chloroethyls

Me

Me

O

H

H

Br

H

Seven fluorine sec.-propyls

H

OCF3

51-62

2,2,2-three chloroethyls

Me

Me

O

H

H

I

H

Seven fluorine sec.-propyls

H

CF3

51-63

2,2,2-three chloroethyls

Me

Me

O

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

51-64

2,2,2-three chloroethyls

Me

Me

O

H

H

C?l

H

Nine fluoro-2-butyl

H

OCF3

51-65

2,2,2-three chloroethyls

Me

Me

O

H

H

Br

H

Nine fluoro-2-butyl

H

CF3

51-66

2,2,2-three chloroethyls

Me

Me

O

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

51-67

2,2,2-three chloroethyls

Me

Me

NH

H

H

I

H

Seven fluorine sec.-propyls

H

OCF3

51-68

2,2,2-three chloroethyls

Me

Me

NH

H

H

Cl

H

Seven fluorine sec.-propyls

H

CF3

51-69

2,2,2-three chloroethyls

Me

Me

NH

H

H

CF3

H

Seven fluorine sec.-propyls

H

CF3

51-70

2,2,2-three chloroethyls

Me

Me

NH

H

H

Br

H

Nine fluoro-2-butyl

H

OCF3

51-71

2,2,2-three chloroethyls

Me

Me

NH

H

H

I

H

Nine fluoro-2-butyl

H

CF3

51-72

2,2,2-three chloroethyls

Me

Me

NH

H

H

CF3

H

Nine fluoro-2-butyl

H

CF3

51-73

2,2,2-three chloroethyls

Me

H

S

H

H

Cl

F

Seven fluorine sec.-propyls

H

OCF3

51-74

2,2,2-three chloroethyls

H

H

S

H

H

Br

H

Seven fluorine sec.-propyls

F

CF3

51-75

2,2,2-three chloroethyls

H

H

S

H

H

CF3

Cl

Seven fluorine sec.-propyls

H

CF3

51-76

2,2,2-three chloroethyls

H

H

S

H

H

I

H

Nine fluoro-2-butyl

Cl

OCF3

51-77

2,2,2-three chloroethyls

H

H

S

H

H

Cl

Br

Nine fluoro-2-butyl

H

CF3

51-78

2,2,2-three chloroethyls

H

H

S

H

H

CF3

H

Nine fluoro-2-butyl

Br

CF3

51-79

2,2,2-three chloroethyls

H

H

O

H

H

Br

I

Seven fluorine sec.-propyls

H

OCF3

51-80

2,2,2-three chloroethyls

Me

H

O

H

H

I

H

Seven fluorine sec.-propyls

I

CF3

51-81

2,2,2-three chloroethyls

H

H

O

H

H

CF3

Me

Seven fluorine sec.-propyls

H

CF3

51-82

2,2,2-three chloroethyls

H

H

O

H

H

Cl

H

Nine fluoro-2-butyl

Me

OCF3

51-83

2,2,2-three chloroethyls

H

H

O

H

H

Br

F

Nine fluoro-2-butyl

F

CF3

51-84

2,2,2-three chloroethyls

H

H

O

H

H

CF3

Cl

Nine fluoro-2-butyl

Cl

CF3

51-85

2,2,2-three chloroethyls

H

H

NH

H

H

I

Br

Seven fluorine sec.-propyls

Br

OCF3

51-86

2,2,2-three chloroethyls

H

H

NH

H

H

Cl

I

Seven fluorine sec.-propyls

I

CF3

51-87

2,2,2-three chloroethyls

Me

H

NH

H

H

CF3

F

Seven fluorine sec.-propyls

Me

CF3

51-88

2,2,2-three chloroethyls

H

H

NH

H

H

Br

Cl

Nine fluoro-2-butyl

Me

OCF3

51-89

2,2,2-three chloroethyls

H

H

NH

H

H

I

Br

Nine fluoro-2-butyl

Me

CF3

51-90

2,2,2-three chloroethyls

H

H

NH

H

H

CF3

I

Nine fluoro-2-butyl

Me

CF3

Below, provide the physics value of the representation compound of amide derivatives of the present invention in the 52nd table.Shown here ¹The value that the H-NMR chemical displacement value then obtains as internal standard substance matter for the use tetramethylsilane unless otherwise specified.

[table 229]

The 52nd table (1)

[table 230]

The 52nd table (2)

[table 231]

The 52nd table (3)

[table 232]

The 52nd table (4)

[table 233]

The 52nd table (5)

[table 234]

The 52nd table (6)

[table 235]

The 52nd table (7)

[table 236]

The 52nd table (8)

[table 237]

The 52nd table (9)

[table 238]

The 52nd table (10)

[table 239]

The 52nd table (11)

[table 240]

The 52nd table (12)

[table 241]

The 52nd table (13)

[table 242]

The 52nd table (14)

[table 243]

The 52nd table (15)

[table 244]

The 52nd table (16)

[table 245]

The 52nd table (17)

[table 246]

The 52nd table (18)

[table 247]

The 52nd table (19)

Contain The compounds of this invention and can prevent and kill off following insect effectively with lower concentration: the various Agricultural pests that endanger agricultural garden crop and trees etc. as the noxious organism control agent of effective constituent, people's such as house living environment is brought dysgenic sanitary insect pest, the grain storage pest of the cereal that stores in the harm warehouse etc., the insects of the timber food insect of timber such as harm buildings etc., and under kindred circumstances, take place, and the mite class that endangers, crustaceans, mollusk, harmful organism arbitrarily in the threadworms.

The insects that can use The compounds of this invention to prevent and kill off; The mite class; Crustaceans; Mollusk and threadworms; Particularly for example can enumerate following substances, but be not limited thereto:tea Ji leaf roller (Adoxophyes honmai); Tea olethreutid (Adoxophyes orana faciata); The yellow volume of pears moth (Archips breviplicanus); The little moth of apple moth (Grapholita inopinata); Random line apple skin worm (Archips fuscocupreanus); Oriental fruit months (Grapholita molesta); The long leaf roller of tea (Choristoneura magnanima); Eating-core bean worm (Leguminivora glycinivorella); Mulberry tree leaf roller (Olethreutes mori); The thin moth of apple leaf roll (Caloptilia zachrysa); Peach Eucosmaspp (Argyresthia conjugella); The thin moth of pears (Spulerrina astaurota); Beans steinernema (Matsumuraeses phaseoli); The brown leaf roller of apple (Pandemis heparana); Pears ermine moth (Bucculatrix pyrivorella); Apple leaf miner (Lyonetia clerkella); Peach fruit moth (Carposina niponensis); Crazing lyonetid (Lyonetia prunifoliella malinella); The thin moth of tea (Caloptilia theivora); The little thin moth (Phyllonorycter ringoniella) of diving of gold line; Oranges and tangerines leaf lyonetid (Phyllocnistis citrella); Green onion diamond-back moth (Acrolepiopsis sapporensis); The pseudo-diamond-back moth (Acrolepiopsis suzukiella) of sweet potato; Small cabbage moth (Plutella xylostella); Persimmon is lifted limb moth (Stathmopoda masinissa); Sweet potato sun gelechiid (Helcystogramma triannulella); Pectinophora gossypiella (Pectinophora gossypiella); Peach fruit moth (Carposina sasakii); Striped rice borer (Chilo suppressalis); Cnaphalocrocis medinali (rice leaf roller) (Cnaphalocrocis medinalis); Cacac moth (Ephestia elutella); Dichocrocis punctiferalis (Conogethes punctiferalis); The wild snout moth's larva (Diaphania indica) of melon thin, tough silk; Beanpod phycitid (Etiella zinckenella); The wild snout moth's larva (Glyphodes pyloalis) of mulberry thin, tough silk; Some snout moth's larvas (Scirpophaga incertulas); Oeobia undalis (Hellula undalis); Ostrinia furnacalis (Ostrinia furnacalis); The wild snout moth's larva (Ostrinia scapulalis) of beans stalk; Crambid (Parapediasia teterrella); Rice hesperiidae (Parnara guttata); Large white butterfly (Pieris brassicae); Cabbage butterfly (Pieris rapae crucivora); Papilio xuthus Linnaeus (Papilio xuthus); Big bridging worm (Ascotis selenaria); Soybean noctuid (Pseudoplusia includens); Euproctis pseudoconspersa (Euproctis pseudoconspersa); Gypsymoth (Lymantria dispar); Revolve orgyia antiqua (Orgyia thyellina); Autumn curtain moth (Hyphantria cunea); Peculiar prestige moths attracted by lamplight (Lemyra imparilis); Withered leaf noctuid (Adris tyrannus); Hickie is tired of noctuid (Aedia leucomelas); Ball dish noctuid (Agrotis ipsilon); Turnip noctuid (Agrotis segetum); Stain three-spotted phytometra (Autographa nigrisigna); Three-spotted phytometra (Ctenoplusia agnata); Codling moth (Cydla pomonella); Bollworm (Helicoverpa armigera); Tobacco budworm (Helicoverpa assulta); The real noctuid (Helicoverpa zea) of paddy; Heliothis virescens (Heliothis virescens); Pyrausta nubilalis (Hubern). (Ostrinia nubilalis); Lopper worm (Mamestra brassicae); Mythimna separata (Mythimna separata); Sesamia inferens (Sesamia inferens); Rice green caterpillar (Naranga aenescens); South spodoptera (Spodoptera eridania); Beet armyworm (Spodoptera exigua); Noctuid (Spodoptera frugiperda) is coveted on the meadow; Sea spodoptera (Spodoptera littoralis); Prodenia litura (Spodoptera litura); Light sword line spodoptera (Spodoptera depravata); Cabbage looper (Trichoplusia ni); Grape certain kind of berries fruit moth (Endopiza viteana); Tomato hawkmoth (Manduca quinquemaculata); Maduca sexta lepidopterous insects such as (Manduca sexta);

Grape Ah jassids (Arboridia apicalis), black chest two Room leafhopper (Balclutha saltuella), 2 cicadellids (Epiacanthus stramineus), broad bean Empoasca spp (Empoasca fabae), Empoasca nipponica, pass through smaller green leaf hopper (Empoasca onukii) greatly, plate well smaller green leaf hopper (Empoasca sakaii), Macrosteles striifrons, rice green leafhopper (Nephotettix cinctinceps), Psuedatomoscelis seriatus, small brown rice planthopper (Laodelphax striatella), brown paddy plant hopper (Nilaparvata lugens), white backed planthopper (Sogatella furcifera), oranges and tangerines wood louse (Diaphorina citri), pear sucker (Psylla pyrisuga), citrus spiny white fly (Aleurocanthus spiniferus), Bemisia argentifolii (Bemisia argentifolii), tobacco aleyrodid (Bemisia tabaci), oranges and tangerines aleyrodid (Dialeurodes citri), Trialeurodes vaporariorum Westwood (Trialeurodes vaporariorum), grape white fly (Trialeurodes vittata) (Aleurolobus taonabae), grape phylloxera (Viteus vitifolii), radish aphid (Lipaphis erysimi), cotten aphid (Aphis gossypii), spiraea aphid (Aphis spiraecola), black peach aphid (Myzus persicae), black citrus aphid (Toxoptera aurantii), giant mealy bug (Drosicha corpulenta), icerya purchasi (Icerya purchasi), the continuous mealybug (Phenacoccus solani) of short-tube lycoris, citrus giant coccid (Pulvinaria aurantii), tangerine stern line mealybug (Planococcus citri), citrus circle scale insect (Pseudaonidia duplex), rattan stern line mealybug (Planococcus kuraunhiae), Kang Shi powder scale insect (Pseudococcus comstocki), pears circle scale insect (Comstockaspis perniciosa), ceroplastes (Ceroplastes ceriferus), ceroplastes rubens (Ceroplastes rubens), California red scale (Aonidiella aurantii), tea place shield scale insect (Fiorinia theae), tree peony net armored scale (Pseudaonidia paeoniae), white mulberry scale (Pseudaulacaspis pentagona), the white a red-spotted lizard of plum (Pseudaulacaspis prunicola), winged euonymus is sloughed off armored scale (Unaspis euonymi), arrowhead scale (Unaspis yanonensis), bed bug (Cimex lectularius), spot palpus stinkbug (Dolycoris baccarum), wrinkle cabbage bug (Eurydema rugosum), north two star stinkbugs (Eysarcoris aeneus), Japan two star stinkbugs (Eysarcoris lewisi), black abdomen stinkbug (Eysarcoris ventralis), blue or green stinkbug (Glaucias subpunctatus), tea wing stinkbug (Halyomorpha halys), black palpus green rice stinkbug (Nezara antennata), Nezara viridula smaragdula Fabricius. (Nezara viridula), ancient piece of jade, round, flat and with a hole in its centre stinkbug (Piezodorus hybneri), amber stinkbug (Plautia crossota), scotinophora lurida (Scotinophora lurida), rice spiny coreid (Cletus punctiger), China's Leptocorisa spp (Leptocorisa chinensis), rod honeybee coried (Riptortus clavatus), Radix Dauci Sativae coried (Rhopalus msculatus), sugarcane chinch bug (Cavelerius saccharivorus), cucurbit chinch bug (Togo hemipterus), red cotton bug (Dysdercus cingulatus), cuckoo hat lace bug (Stephanitis pyrioides), Halticus insularis, America tarnished plant bug (Lygus lineolaris), the narrow fleahopper in siberian (Stenodema sibiricum), red fine fleahopper (Stenotus rubrovittatus), rice leaf insect hemipterans such as (Trigonotylus caelestialium);

Bronze different beetle (Anomala cuprea), Ji cockchafer (Anomala rufocuprea), little blue and white cockchafer (Gametis jucunda), pitch seven cheek cockchafers (Heptophylla picea), beans cockchafer (Popillia japonica), colorado potato beetles (Lepinotarsa decemlineata), mexican bean ladybird (Epilachna varivestis), Ipomoea batatas comb pawl click beetle (Melanotus fortnumi), multitudinous comb pawl Pleonomus (Melanotus tamsuyensis), cigarette beetle (Lasioderma serricorne), Lyctus brunneus Stephens (Lyctusbrunneus), blastophagus piniperda (Tomicus piniperda), lesser grain borer (Rhizopertha dominica), Epuraea domina, mexican bean ladybird (Epilachna varivestis), potato ladybug (Epilachna vigntioctopunctata), tenebrio molitor (Tenebrio molitor), red flour beetle (Tribolium castaneum), longicorn beetle (Anoplophora malasiaca), Monochamus alternatus (Monochamus alternatus), yellow star longicorn (Psacothea hilaris), grape borer (Xylotrechus pyrrhoderus) (Xylotrechus pyrrhoderus), Callosobruchus chinensis (Callosobruchus chinensis), aulacophora femoralis (Aulacophora femoralis), rice leaf beetles (Oulema oryzae) Chard dish flea beetle (Chaetocnema concinna), cucumber point chrysomelid (Diabrotica undecimpunctata), corn root leaf A (Diabrotica virgifera), north corn rootworm (Diabrotica barberi), yellow bar leaf flea (Phyllotreta striolata), the narrow chest flea beetle of eggplant (Psylliodes angusticollis), peach real image (Rhynchites heros), cylas formicarius (Cylas formicarius), Mexico's cotton boll resembles (Anthonomus grandis), rice resembles (Echinocnemus squameus), west India sweet potato resembles (Euscepes postfasciatus), alfalfa leaf resembles (Hypera postica), rice water weevil (Lissohoptrus oryzophilus), vine black ear beak resembles (Otiorhynchus sulcatus), grain weevil (Sitophilus granarius), sitophilus zea-mais (Sitophilus zeamais), Sphenophorus venatus vestitus, blue or green wing rove beetle coleopterons such as (Paederus fuscipes);

Total homopterous insect such as flower thrips (Frankliniella intonsa), golden thistle horse (Thrips flavus), west flower thrips (Frankliniella occidentalis), greenhouse thrips (Heliothrips haemorrhoidalis), tea golden thistle horse (Scirtothrips dorsalis), southern golden thistle horse (Thrips palmi), onion thrips (Thrips tabaci), Ponticulothrips diospyrosi,

Asphondylia yushimai, wheat midge (Sitodiplosis mosellana), melon trypetid (Bactrocera cucurbitae), citrus fruit fly (Bactrocera dorsalis), Mediterranean fruitfly (Ceratitis capitata), hydrellia griseola (Hydrellia griseola), cherry fruit bat (Drosophila suzukii), rice stem maggot (Agromyza oryzae), the color fly (Chromatomyia horticola) of diving of pea, tomato liriomyza bryoniae (Liriomyza bryoniae), green onion liriomyza bryoniae (Liriomyza chinensis), vegetables liriomyza bryoniae (Liriomyza sativae), African chrysanthemum liriomyza bryoniae (Liriomyza trifolii), delia platura (Delia platura), onion fly (Delia antique), Xiao lamb's-quarters spring fly (Pegomya cunicularia), Rhagoletis pomonella (Rhagoletis pomonella), wheat cecidomyiia (Mayetiola destructor), housefly (Musca domestica), tatukira (Stomoxys calcitrans), sheep hippoboscid (Melophagus ovinus), bomb fly (Hypoderma bovis), heel fly (Hypoderma lineatum), Oestrus ovis (Oestrus ovis), glossina morsitans (Glossina palpalis, Glossina morsitans), Prosimulium yezoensis, horsefly (Tabanus trigonus), hickie moth buffalo gnat (Telmatoscopus albipunctatus), Leptoconops nipponensis, culex pipiens pollens (Culex pipiens pallens), Aedes Aegypti (Aedes aegypti), Asia tiger mosquito (Aedes albopicutus), dipteral insects such as Anopheles hyracanus sinesis;

Apethymus kuri, Xinjiang cabbage sawfly (Athalia rosae), rose three joint sawflies (Arge pagana), pine and cypress Neodiprion spp (Neodiprion sertifer), Chinese chestnut cynipid (Dryocosmus kuriphilus), army antenna (Eciton burchelli, Eciton schmitti), Japanese hunchbacked ant (Camponotus japonicus), Vespa magnifiac (Sonan). (Vespa mandarina), bull ant (Myrmecia spp.), red fire ant class (Solenopsis spp.), little red ant hymenopterans such as (Monomorium pharaonis),

Yellow face oily calabash (Teleogryllus emma), east mole cricket (Gryllotalpa orientalis), migratory locusts (Locusta migratoria), rice grasshopper (Oxya yezoensis), desert locust orthopterans such as (Schistocerca gregaria),

The white Onychiurus arcticus of dish (Onychiurus folsomi), arctic Onychiurus arcticus (Onychiurus sibiricus), yellow star sminthurid Chaetonotoidea insects such as (Bourletiella hortensis),

Peroplaneta fluligginosa (Periplaneta fuliginosa), the big Lian (Periplaneta japonica) of Japan, Groton bug (Blattella germanica), the non-Lian in America (Periplaneta Americana), etc. the Dictyoptera insect,

Taiwan formosanes (Coptotermes formosanus), the northern reticulitermes flavipe that dwells (Reticulitermes speratus), blackwing subterranean isoptera insects such as (Odontotermes formosanus),

Cat flea (Ctenocephalidae felis), dog flea (Ctenocephalides canis), chicken flea (Echidnophaga gallinacea), Pulex irritans (Pulex irritans), Xanthopsyllacheopis isoptera insects such as (Xenopsylla cheopis),

Corpus luteum poultry louse (Menacanthus stramineus), ox bird lice Mallophaga insects such as (Bovicola bovis),

Ox louse (Haematopinus eurysternus), haematopinus suis (Haematopinus suis), Linognathus vituli (Linognathus vituli), solenoptes capillatus Anoplura insects such as (Solenopotes capillatus),

Primrose herbivore mite (Phytonemus pallidus), Polyphagotarsonemus latus Banks (Polyphagotarsonemus latus), double leaf tarsonemid mite dust mite classes such as (Tarsonemus bilobatus),

Penthaleus erythrocephalus, wheat leaf pawl mite (Penthaleus major) etc. walk the mite class,

Zhen Kaji unguiculus mite (Oligonychus shinkajii), panonychus citri (Panonychus citri), mulberry Panonychus citri (Panonychus mori), panonychus ulmi (Panonychus ulmi), kamisawa tetranychus (Tetranychus kanzawai), T.urticae Koch spider mite kinds such as (Tetranychus urticae),

Tea point leaf segment tick (Acaphylla theavagrans), turmeric goitre mite (Aceria tulipae), tomato peronium goitre mite (Aculops lycopersici), tangerine peronium goitre mite (Aculops pelekassi), Si Shi thorn goitre mite (Aculus schlechtendali), Eriophyes chibaensis, tangerine wrinkle leaf Aculus goitre mite classes such as (Phyllocoptruta oleivora),

Luo Bingen mite (Rhizoglyphus robini), the corrosion junket mite (Tyrophagus putrescentiae), seemingly eat junket mite flour mite classes such as (Tyrophagus similis),

Ya Shi watt of mite watt mite classes such as (Varroa jacobsoni),

Boophilus microplus (Boophilus microplus), brown dog tick (Rhipicephalus sanguineus), haemaphysalis longicornis (Haemaphysalis longicornis), haemaphysalis flava (Haemophysalis flava), haemaphysalis campanulata (Haemophysalis campanulata), ixodes ovatus (Ixodes ovatus), ixodes persulcatus (Ixodes persulcatus), flower tick (Amblyomma spp.), leather tick tick classes such as (Dermacentor spp.),

Dog Ji chela mite (Cheyletiella yasguri), cat Ji chela mite cheyletid mite classes such as (Cheyletiella blakei),

Dog demodicid mite (Demodex canis), cat demodicid mite demodicid mite classes such as (Demodex cati),

Sheep itch mite itch mite classes such as (Psoroptes ovis),

Itch mite (Sarcoptes scabiei), cat back of the body anus mite (Notoedres cati), knee mite itch mite classes such as (Knemidocoptes spp.),

Armadillidum vulgare crustaceans such as (Armadillidium vulgare),

Fushou spiral shell (Pomacea canaliculata), African Snail (Achatina fulica), two-wire slug (Meghimatium bilineatum), Limax Valentiana, snail (Acusta despecta sieboldiana), Japanese soil snail snailss such as (Euhadra peliomphala),

Coffee Pratylenchidae (Prathylenchus coffeae), Cobb root (Prathylenchus penetrans), wounded or disabled Pratylenchidae (Prathylenchus vulnus), globodera rostochiensis (Globodera rostochiensis), soybean Cyst nematode (Heterodera glycines), north root knot nematode (Meloidogyne hapla), Meloidogyne incognita (Meloidogyne incognita), aphelenchoides besseyi (Aphelenchoides besseyi), pine wood nematode threadwormss such as (Bursaphelenchus xylophilus) etc.

As the noxious organism control agent of effective constituent above-mentioned harmful crops of infringement wet crop, dry crop, fruit tree, vegetables, other crops and flowers etc. had significant preventive effect with The compounds of this invention, therefore take place according to prediction the period of harmful organism, before harmful organism is taken place or confirm moment of generation harmful organism, paddy field water, cauline leaf or soil to paddy field, dry land, fruit tree, vegetables, other crops, flowers etc. are handled, and can access the effect as noxious organism control agent of the present invention thus.

As the noxious organism control agent of effective constituent the grain storage pest that produces etc. had significant preventive effect with The compounds of this invention in the harvesting product is preserved.That is, in order to The compounds of this invention as the noxious organism control agent of effective constituent to the place of retention of harvesting product or harvesting product spray, smear, be coated with, dipping, powder clothing, stifling fumigation or pressurization are injected etc., and results backs (postharvest) handle gets final product.

In addition, will be applicable to plant seed as the noxious organism control agent of effective constituent, and can prevent thus by the caused infringement of the insect that produces in the plant after planting with The compounds of this invention.Promptly, will be as the noxious organism control agent of effective constituent directly or suitably dilution or such as water so that its outstanding turbid form with The compounds of this invention, with the significant quantity of prevent and kill off insect pests to plant seed spray, smear, processing such as dipping or powder clothing, The compounds of this invention is contacted with plant seed gets final product.

So-called plant seed, be meant store plant seedlings germinate required nutritive ingredient, on agricultural, be used to the material of breeding.For example, can enumerate the kind ball etc. of the napiform root such as kind taro, edible lily, turmeric of the seed of corn, soybean, red bean, cotton, paddy rice, sugar beet, wheat, barley, Sunflower Receptacle, tomato, cucumber, eggplant, spinach, Kidney bean, pumpkin, sugarcane, tobacco leaf, sweet green pepper and Canadian rape etc. or taro, potato, sweet potato, Betel Ze etc. or Chinese onion etc.

As the noxious organism control agent of effective constituent Diptera pest (culex pipiens pollens, player whose turn comes next mosquito, midge, housefly, butterfly fly, horsefly etc.), guiding principle wing order insect sanitary insect pests such as (Groton bug, Peroplaneta fluligginosa, the non-Lian in America etc.) had significant preventive effect with The compounds of this invention.

As the noxious organism control agent of effective constituent termite, Lyctus brunneus Stephens, lesser grain borer, death watch beetle, longicorn timber such as (Cerambycidae) are eaten insect with The compounds of this invention and have significant preventive effect, by the timber of soil or buildings etc. is handled, can prevent and kill off above-mentioned timber food insect.

The compounds of this invention shows preventive effect to various harmful organisms; demonstrate the effect of the useful crop of protection; simultaneously demonstrate preventive effect, therefore have and make the effect of huge contribution reducing carrying capacity of environment as sterilant or acaricidal excellence with low medication amount.And The compounds of this invention also can show excellent preventive effect by mixing with other insecticide for agricultural or horticultural use, miticide, nematocides, sterilant, weedicide, plant-growth regulator, biological pesticide etc. to use.

When using The compounds of this invention, usually can mix with suitable solid carrier or liquid vehicle, and then add tensio-active agent as required, penetrant, spreader-sticker (spreader), thickening material, frostproofer, tackiness agent, anti-hard caking agent, disintegrating agent, defoamer, sanitas and decomposition prevent agent etc., make following formulation arbitrarily and be used for practicality, described formulation is solution (soluble concentrate), emulsion (emulsifiable concentrate), wettable powder (wettable powder), water solvent (water soluble powder), water dispersion granule (water dispersible granule), water-soluble granular formulation (water soluble granule), clouding agent (suspension concentrate), emulsifiable concentrate (concentrated emulsion), suspension emulsion (suspoemulsion), micro emulsion (microemulsion), pulvis (dustable powder), granule (granule) tablet (tablet) and emulsifying property gelifying agent (emulsifiable gel) etc.In addition, consider, supply in the preparation inclosure water-soluble capsule that can also above-mentioned any formulation and the water soluble package bodies such as bag of water-solubility membrane from the viewpoint that laborsavingization and security improve.

Can be in solid or the liquid any as the inert support that can use in the present invention, as the material that can form solid inert carrier, can enumerate for example soyflour, grain flour, wood powder, tree bark powder, the saw powder, tobacco leaf stem powder, walnut shell flour, chaff, cellulose powder, residue after the plant milk extract extraction, pulverize synthetic polymers such as synthetic resins, clay class (kaolin for example, wilkinite, acidic white earth etc.), talcs (talcum for example, pyrophyllite etc.), silica-based (diatomite for example, silica sand, mica, white carbon(ink) [is also referred to as moisture micro mist silicon, the synthetic high dispersive silicic acid of moisture silicic acid, according to the difference of product, have to contain the product of Calucium Silicate powder as main component.]), chemical fertilizer, compost etc. such as inorganic mineral powder, sulphur ammonium, phosphorus ammonium, ammonium nitrate, urea, ammonium chloride such as activated carbon, sulphur powder, float stone, sintering diatomite, brick crushed material, flying dust, sand, lime carbonate, calcium phosphate, above-mentioned carrier can use separately, perhaps also can use with the form of the mixture more than two kinds.

As the material that can become the liquid inert support, except that the material that itself has solvent nature, can also select not have solvent nature, but the effect by auxiliary agent makes effective constituent compound dispersive material, for example can enumerate the following carrier of enumerating as typical example, following carrier can use separately or use with the form of the mixture more than 2 kinds, water for example, alcohols (for example, methyl alcohol, ethanol, Virahol, butanols, ethylene glycol etc.), ketone (acetone for example, methyl ethyl ketone, methyl iso-butyl ketone (MIBK), diisobutyl ketone, pimelinketone etc.), ethers (ether for example, dioxane, cellosolve, Di Iso Propyl Ether, tetrahydrofuran (THF) etc.), aliphatic hydrocarbon (kerosene (kerosene) for example, the mineral wet goods), aromatic hydrocarbon based (benzene for example, toluene, dimethylbenzene, solvent naphtha, alkylnaphthalene etc.), halogenated hydrocarbon (methylene dichloride for example, chloroform, tetracol phenixin, chlorobenzene etc.), ester class (ethyl acetate for example, butylacetate, ethyl propionate, diisobutyl phthalate, dibutyl phthalate, dioctyl phthalate (DOP) etc.), amides (dimethyl formamide for example, diethylformamide, N,N-DIMETHYLACETAMIDE etc.), nitrile (for example acetonitrile etc.).

Above-mentioned solid and liquid vehicle can use separately also and can use simultaneously more than 2 kinds.

As tensio-active agent, can enumerate for example Voranol EP 2001, polyxyethylated (list or two) phenyl ether, polyoxyethylene is (single, two or three) styryl phenyl ether, polyoxyethylene polyoxypropylene block copolymer, polyoxyethylene fatty acid (list or two) ester, sorbitan fatty(acid)ester, the polyoxyethylene sorbitan fatty acid ester, the Viscotrol C ethylene oxide adduct, ethylene glycol (acetylene glycol), acetylene alcohol, the ethylene oxide adduct of ethylene glycol, nonionic surfactants such as the ethylene oxide adduct of acetylene alcohol and alkyl glucoside, alkyl sulfuric ester salt, alkylbenzene sulfonate, Sulfite lignin, alkyl sulfo succinate, naphthalenesulfonate, sulfonated alkyl naphathalene, the salt of the formaldehyde condensation products of naphthene sulfonic acid, the salt of the formaldehyde condensation products of alkyl naphthalene sulfonic acid, Voranol EP 2001 sulfuric acid or phosphate ester salt, polyoxyethylene (list or two) alkyl phenyl ether sulfuric acid or phosphate ester salt, polyoxyethylene is (single, two or three) styryl phenyl ether sulfuric acid or phosphate ester salt, polycarboxylate (for example, polyacrylate, the multipolymer that polymaleic acid salt and toxilic acid and alkene form etc.) and anionic surfactant such as poly styrene sulfonate, cationic surfactant such as alkylamine salt and alkyl quaternary ammonium salts, amphotericses such as amino acid pattern and betaine type, polysiloxane-based tensio-active agent and fluorine class tensio-active agent.

The content of above-mentioned tensio-active agent is not particularly limited, and is with respect to 100 weight parts preparation of the present invention, preferred usually in the scope of 0.05～20 weight part.In addition, above-mentioned tensio-active agent can use separately or use simultaneously more than 2 kinds.

In order to prevent and kill off various insects, with it directly or suitably dilution or make it become outstanding turbid form such as water, with prevent and kill off disease effectively amount be used to predict the crop that produces this insect or use and get final product at the position of not wishing to take place.Its usage quantity according to various factors for example bearing status, the insect of purpose, object insect, crop occurence tendency, weather, envrionment conditions, formulation, application process, use the place, use and change in period etc., expect that usually effective constituent uses with 0.0001～5000ppm, the concentration that is preferably 0.01～1000ppm.In addition, the amount of application of every 10a is counted 1～300g with effective constituent usually.

The effective constituent amount of compound of the present invention, when being 5～90 weight %, water dispersion granule when being 0.1～20 weight % and suspensoid when being 3～90 weight %, granule when being 5～50 weight %, wettable powder when generally, being 0.1～20 weight %, emulsion during pulvis is 3～90 weight %.On the other hand, the amount of the carrier in each formulation generally is 80～99.9 weight % during pulvis when being 10～90 weight %, granule when being 40～95 weight %, wettable powder when being 60～99.9 weight %, emulsion, is 10～90 weight % when being 10～95 weight %, water dispersion granule when reaching suspensoid.In addition, the amount of auxiliary agent is 0.1～20 weight % during pulvis when being 0.1～20 weight %, water dispersion granule when being 0.1～20 weight % and suspensoid when being 0.1～20 weight %, granule when being 1～20 weight %, wettable powder when being 0.1～20 weight %, emulsion generally.

In addition, when using The compounds of this invention, also can mix when preparation or when scattering as required and use with the weedicide of other kinds, various sterilant, miticide, nematocides, sterilant, plant-growth regulator, synergistic agent, fertilizer, soil improvement agent etc. as agricultural chemicals.

Whole documents of putting down in writing in this specification sheets, patent application, and technical specification, with as with reference to each document, patent application, and the technology regulations specifically and the degree of situation about introducing respectively in the same manner, as with reference to introducing in this specification sheets.

[embodiment]

By following examples representational embodiment of the present invention is described, but the present invention is not limited to this.In the present embodiment, DMF represents N, and dinethylformamide, THF represent that tetrahydrofuran (THF), IPE represent that isopropyl ether, DMI represent 1, and 3-dimethyl-2-imidazolone, DMSO represent dimethyl sulfoxide (DMSO).

" % " is not quality criteria when in addition, having specified otherwise.

＜embodiment 1 〉

The preparation of N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-fluoro-3-(N-methyl-benzamide base) benzamide (compound sequence number 7-1574).

<1-1>

The preparation of 4-(perfluoropropane-2-yl)-2-(trifluoromethyl) aniline

100g (0.608mol) 2-(trifluoromethyl) aniline, 131g (0.639mol) 85% V-Brite B, 20.9g (0.0608mol) 4-butyl ammonium hydrogen sulfate are packed in the mixing solutions of 1500ml ethyl acetate, 1500ml water, add 53.9g (0.639mol) sodium bicarbonate.Splash into 198g (0.669mol) seven fluorine isopropyl iodides under the room temperature, stirring at room 6 hours.Behind the separatory, the solvent of removing organic layer, the 500ml ethyl acetate of packing into are distilled in decompression down.Splash into 160g (0.608mol) 4M hydrogenchloride/ethyl acetate solution, stirring at room is after 30 minutes, and 5 ℃ were stirred 1 hour.After the filtration, water, saturated sodium bicarbonate aqueous solution after the wash filtrate, are used anhydrous magnesium sulfate drying successively, and decompression distillation down removes and desolvates.Residue obtained with silica gel column chromatography (expansion solvent; Hexane: ethyl acetate=10: 1) refining, prepare 60.0g (yield 30%) title compound thus.

¹H-NMR(CDCl ₃，ppm)δ4.49(2H，broad-s)，6.81(1H，d，J＝8.3Hz)，7.48(1H，d，J＝8.3Hz)，7.64(1H，s).

<1-2>

The preparation of 2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) aniline

100g (0.273mol) 4-(perfluoropropane-2-yl)-2-(trifluoromethyl) aniline is packed among the 500mlDMF into 52.1g (0.287mol) the N-bromo-succinimide of in batches packing into through 30 minutes.60 ℃ are stirred after 2 hours down, are cooled to room temperature, enter in the 2000ml water.Behind ethyl acetate extraction, clean with saturated aqueous common salt, use anhydrous magnesium sulfate drying.Distillation is except that desolvating down in decompression, and the residue obtained silica gel column chromatography of using (launches solvent; Hexane: ethyl acetate=20: 1) refining, prepare 89.0g (yield 80%) title compound thus.

¹H-NMR(CDCl ₃，ppm)δ5.03(2H，broad-s)，7.61(1H，s)，7.79(1H，s).

<1-3>

The preparation of N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-chloro-3-nitrobenzamide

2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) aniline 3.60g (8.82mmol) is packed among the 20ml dehydration THF, be cooled to-70 ℃ under the nitrogen atmosphere.Splash into 4.85ml (9.70mmol) 2.0M lithium diisopropylamine hexane solution, then, splash into 2.34g (10.7mmol) be dissolved among the 5ml dehydration THF, by 2-chloro-3-nitrobenzoic acid and the synthetic acyl chlorides of thionyl chloride ,-70 ℃ are stirred after 30 minutes stirring at room 30 minutes down.After entering in the aqueous ammonium chloride solution, use ethyl acetate extraction, use anhydrous magnesium sulfate drying.Distillation is except that desolvating down in decompression, and the residue obtained silica gel column chromatography of using (launches solvent; Hexane: ethyl acetate=10: 1 → 8: 2 → 3: 1) refining, prepare 1.76g (yield: title compound 34%) thus.

¹H-NMR(CDCl ₃，ppm)δ7.61(1H，t，J＝7.8Hz)，7.67(1H，broad-s)，7.93-7.97(3H，m)，8.18(1H，broad-s).

<1-4>

The preparation of N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-fluoro-3-nitrobenzamide

Under the nitrogen gas stream, add 2.40g (41.3mmol) Potassium monofluoride (spraying drying thing) in the 50ml of N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-chloro-3-nitrobenzamide 4.89g (8.27mmol) dehydration DMF solution, 130 ℃ were stirred 10 hours down.Add ethyl acetate, hexane, water in the reaction solution, behind the separatory, water, clean organic layer, use anhydrous magnesium sulfate drying with saturated aqueous common salt.Distillation is except that desolvating down in decompression, and the residue obtained silica gel column chromatography of using (launches solvent; Hexane: ethyl acetate=10: 1) refining, prepare 0.940g (yield 20%) title compound thus.

¹H-NMR(CDCl ₃，ppm)δ7.53(1H，t，J＝7.3Hz)，7.93(1H，broad-s)，8.17-8.18(2H，m)，8.28-8.32(1H，m)，8.44-8.48(1H，m).

<1-5>

The preparation of 3-amino-N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-fluorobenzamide

0.940g (1.63mmol) N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-fluoro-3-nitrobenzamide, 0.960g (5.05mmol) tin protochloride (anhydrous) are added in the 10ml ethanol, add 1.02ml (9.78mmol) concentrated hydrochloric acid then and stirred 4 hours down at 60 ℃.Adding aqueous sodium hydroxide solution adjusting pH in the reaction solution is 10, the insolubles that uses the diatomite filtering to separate out.Filtration gleanings on the diatomite is cleaned with ethyl acetate.Use ethyl acetate extraction filtrate, use 20% aqueous sodium hydroxide solution, saturated aqueous common salt to clean organic layer after, use anhydrous magnesium sulfate drying.Distillation is except that desolvating down in decompression, and the residue obtained silica gel column chromatography of using (launches solvent; Hexane: ethyl acetate=4: 1) refining, prepare 0.930g (yield 99%) title compound thus.

¹H-NMR(CDCl ₃，ppm)δ3.93(2H，broad-s)，6.99-7.04(1H，m)，7.11(1H，t，J＝7.8Hz)，7.47-7.49(1H，m)，7.91(1H，s)，8.14(1H，s)，8.28(1H，d，J＝14.6Hz).

<1-6>

The preparation of N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-fluoro-3-(methylamino) benzamide

0.930g (1.71mmol) 3-amino-N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-fluorobenzamide is added in the 5ml vitriol oil, and 40 ℃ drip 10ml 37% formalin down.Reaction solution is poured in the frozen water, after use aqueous sodium hydroxide solution adjusting pH is 10, added ethyl acetate extraction.After using 20% aqueous sodium hydroxide solution, saturated aqueous common salt to clean organic layer, use anhydrous magnesium sulfate drying.Distillation is except that desolvating down in decompression, and the residue obtained silica gel column chromatography of using (launches solvent; Hexane: ethyl acetate=8: 1) refining, prepare 0.690g (yield 72%) title compound thus.

¹H-NMR(CDCl ₃，ppm)δ2.94(3H，s)，4.14(1H，broad-s)，6.88-6.93(1H，m)，7.18(1H，t，J＝7.8Hz)，7.37-7.41(1H，m)，7.90(1H，s)，8.13(1H，s)，8.27(1H，d，J＝14.6Hz).

[1-7]

The preparation of N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-fluoro-3-(N-methyl-benzamide base) benzamide (compound sequence number 7-1574)

Add 0.460g (3.30mmol) Benzoyl chloride in the 5ml THF solution of 1.54g (2.75mmol) N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-fluoro-3-(methylamino) benzamide, 0.330g (4.13mmol) pyridine, 60 ℃ were stirred 5 hours down.Add entry, ethyl acetate in the reaction solution, behind 1M hydrochloric acid, saturated sodium bicarbonate aqueous solution, saturated aqueous common salt cleaning organic layer, use anhydrous magnesium sulfate drying.Distillation is except that desolvating down in decompression, and the residue obtained silica gel column chromatography of using (launches solvent; Hexane: ethyl acetate=8: 1) refining, clean the gained solid with IPE, prepare 1.45g (yield 80%) title compound thus.

¹H-NMR(CDCl ₃，ppm)δ3.50(3H，s)，6.99-7.33(6H，m)，7.43-7.45(1H，m)，7.90(1H，s)，7.97-8.06(2H，m)，8.13(1H，s).

＜embodiment 2 〉

The preparation of 2-chloro-N-(3-(2,6-two bromo-4-(perfluoropropane-2-yl) phenyl amino formyl radical)-2-fluorophenyl) niacinamide (compound sequence number 6-1140)

<2-1>

The preparation of 4-(perfluoropropane-2-yl) aniline

100g (1.02mol) aniline, 230g (1.12mol) 85% V-Brite B, 35.1g (0.100mol) 4-butyl ammonium hydrogen sulfate are packed in the mixing solutions of 1500ml t-butyl methyl ether, 1500ml water, add 94.7g (1.12mol) sodium bicarbonate.Room temperature splashes into 350g (1.12mol) seven fluorine isopropyl iodides, stirring at room 6 hours.Behind the separatory, behind 1M hydrochloric acid, water, saturated sodium bicarbonate aqueous solution cleaning organic layer, use anhydrous sodium sulfate drying.Decompression is distilled down to remove and is desolvated the 500ml ethyl acetate of packing into.Splash into 255g (1.02mol) 4M hydrogenchloride/ethyl acetate solution, stirring at room 30 minutes also stirred 1 hour under 5 ℃.Leach the solid of separating out, solid is packed in the 1000ml ethyl acetate,, be adjusted to pH8～9, carry out separatory adding the 1000ml saturated sodium bicarbonate aqueous solution below 20 ℃.Behind the anhydrous sodium sulfate drying organic layer, decompression distillation down prepares 188g (yield 71%) title compound thus except that desolvating.

¹H-NMR(CDCl ₃，ppm)δ3.92(2H，broad-s)，6.69-6.74(2H，m)，7.35(2H，d，J＝9.3Hz).

<2-2>

2, the preparation of 6-two bromo-4-(perfluoropropane-2-yl) aniline

216g (0.802mol) 4-(perfluoropropane-2-yl) aniline is packed among the 863mlDMF, be cooled to 5 ℃.285g (1.60mol) the N-bromo-succinimide of in batches packing into through 1 hour.After the stirring at room 1 hour, stirred 2 hours down at 37 ℃.After entering in the 2000ml water, use the 2000ml ethyl acetate extraction, clean with the 1000ml saturated aqueous common salt.Behind anhydrous magnesium sulfate drying, decompression is distilled down to remove and is desolvated.Residue obtained with silica gel column chromatography (expansion solvent; Hexane: ethyl acetate=20: 1) refining, prepare 304g (yield 90%) title compound thus.

¹H-NMR(CDCl ₃，ppm)δ4.88(2H，broad-s)，7.59(2H，s).

<2-3>

The preparation of 2-chloro-N-(2,6-two bromo-4-(perfluoropropane-2-yl) phenyl)-3-nitrobenzamide

According to the method for the 1-3 of embodiment 1, by 2,6-two bromo-4-(perfluoropropane-2-yl) aniline prepares title compound.

¹H-NMR(CDCl ₃，ppm)δ7.58(1H，t，J＝7.8Hz)，7.66(1H，broad-s)，7.90(2H，s)，7.93(1H，dd，J＝1.5，7.8Hz)，7.98(1H，d，J＝7.8Hz).

<2-4>

The preparation of N-(2,6-two bromo-4-(perfluoropropane-2-yl) phenyl)-2-fluoro-3-nitrobenzamide

Method according to the 1-4 of embodiment 1 prepares title compound by 2-chloro-N-(2,6-two bromo-4-(perfluoropropane-2-yl) phenyl)-3-nitrobenzamide.

¹H-NMR(CDCl ₃，ppm)δ7.51-7.55(1H，m)，7.90(2H，s)，8.16(1H，d，J＝11.7Hz)，8.27-8.31(1H，m)，8.48(1H，t，J＝6.3Hz).

<2-5>

The preparation of 3-amino-N-(2,6-two bromo-4-(perfluoropropane-2-yl) phenyl)-2-fluorobenzamide

Method according to the 1-5 of embodiment 1 prepares title compound by N-(2,6-two bromo-4-(perfluoropropane-2-yl) phenyl)-2-fluoro-3-nitrobenzamide.

¹H-NMR(CDCl ₃，ppm)δ3.93(2H，broad-s)，6.99-7.04(1H，m)，7.11(1H，t，J＝7.8Hz)，7.47-7.49(1H，m)，7.91(1H，s)，8.14(1H，s)，8.28(1H，d，J＝14.6Hz).

<2-6>

The preparation of 2-chloro-N-(3-(2,6-two bromo-4-(perfluoropropane-2-yl) phenyl amino formyl radical)-2-fluorophenyl) niacinamide (compound sequence number 6-1140)

Method according to the 1-7 of embodiment 1 prepares title compound by 3-amino-N-(2,6-two bromo-4-(perfluoropropane-2-yl) phenyl)-2-fluorobenzamide and 2-chloronicotinoyl chloride.

¹H-NMR(CDCl ₃，ppm)δ7.40-7.49(2H，m)，7.89(2H，s)，7.94-7.96(1H，m)，8.13(1H，d，J＝12.7Hz)，8.32-8.34(1H，m)，8.57-8.59(1H，m)，8.67-8.71(1H，m)，8.75(1H，broad-s).

＜embodiment 3 〉

The preparation of 3-benzoylamino-2-fluoro-N-(4-(perfluoropropane-2-yl)-2,6-two (trifluoromethyl) phenyl) benzamide (compound sequence number 6-2110)

<3-1>

2, the preparation of 6-two iodo-4-(perfluoropropane-2-yl) aniline

Under 5 ℃, add 2.16g (22.0mmol) vitriol oil in the 50ml ethanolic soln of the 4-that in the 2-1 of embodiment 2, obtains (perfluoropropane-2-yl) aniline 5.74g (22.0mmol).Reaction solution is warming up to room temperature, adds 10.0g (44.0mmol) N-iodo succimide and stirred 3 hours.Reaction solution is injected saturated sodium bicarbonate aqueous solution to neutralize.The crystallization that filtration is separated out, water carries out drying after cleaning, and prepares 9.00g (yield 80%) title compound thus.

¹H-NMR(CDCl ₃，ppm)δ4.95(2H，broad-s)，7.79(2H，s).

<3-2>

The preparation of 2-chloro-N-(2,6-two iodo-4-(perfluoropropane-2-yl) phenyl)-3-nitrobenzamide

To 2, add 20.6g (94.0mmol) 2-chloro-3-nitrobenzoyl chloride in the 100ml DMI solution of 6-two iodo-4-(perfluoropropane-2-yl) aniline 40.0g (78.0mmol) and stirred 3 hours down at 135 ℃.Be cooled to room temperature, reaction solution is injected 1000ml water.Add the 1000ml ethyl acetate and extract, water is used anhydrous magnesium sulfate drying after cleaning organic layer.Underpressure distillation removes and desolvates, and the residue with hexane cleaning gained prepares 56.2g (yield 99%) title compound thus.

¹H-NMR(CDCl ₃，ppm)δ7.58(1H，t，J＝8.3Hz)，7.70(1H，d，J＝3.4Hz)，7.93(1H，dd，J＝1.5，6.3Hz)，8.08-8.10(1H，m)，8.13(2H，s).

<3-3>

The preparation of N-(2,6-two iodo-4-(perfluoropropane-2-yl) phenyl)-2-fluoro-3-nitrobenzamide

Method according to the 1-4 of embodiment 1 prepares title compound by 2-chloro-N-(2,6-two iodo-4-(perfluoropropane-2-yl) phenyl)-3-nitrobenzamide.

1H-NMR(CDCl3，ppm)δ7.52-7.55(1H，m)，8.12-8.18(3H，m)，8.29-8.32(1H，m)，8.48-8.51(1H，m).

<3-4>

The preparation of 3-amino-N-(2,6-two iodo-4-(perfluoropropane-2-yl) phenyl)-2-fluorobenzamide

Method according to the 1-5 of embodiment 1 prepares title compound by N-(2,6-two iodo-4-(perfluoropropane-2-yl) phenyl)-2-fluoro-3-nitrobenzamide.

¹H-NMR(CDCl ₃，ppm)δ3.93(2H，broad-s)，6.99-7.04(1H，m)，7.08(1H，t，J＝7.8Hz)，7.39-7.43(1H，m)，8.10(2H，s)，8.72(1H，d，J＝11.2Hz).

<3-5>

The preparation of 3-benzoylamino-N-(2,6-two iodo-4-(perfluoropropane-2-yl) phenyl)-2-fluorobenzamide (compound sequence number 6-1260)

Method according to the 1-7 of embodiment 1 prepares title compound by 3-amino-N-(2,6-two iodo-4-(perfluoropropane-2-yl) phenyl)-2-fluorobenzamide.

¹H-NMR(CDCl ₃，ppm)δ7.39(1H，t，J＝7.8Hz)，7.52-7.57(4H，m)，7.60-7.63(2H，m)，7.93-7.94(4H，m)，8.70(1H，t，J＝6.3Hz).

<3-6>

The preparation of 3-benzoylamino-2-fluoro-N-(4-(perfluoropropane-2-yl)-2,6-two (trifluoromethyl) phenyl) benzamide (compound sequence number 6-2110)

The 50mlDMF solution of 1.95g (2.59mmol) 3-benzoylamino-N-(2,6-two iodo-4-(perfluoropropane-2-yl) phenyl)-2-fluorobenzamide, 0.10g (0.520mmol) cupric iodide, 1.24g (6.48mmol) fluorosulfonyl difluoroacetic acid methyl esters was stirred 6 hours down at 100 ℃.After reaction solution is cooled to room temperature, add 10ml water, 100ml ethyl acetate, carry out diatomite filtration.Behind the organic layer of water, saturated sodium bicarbonate aqueous solution wash filtrate, use anhydrous magnesium sulfate drying.Underpressure distillation removes and desolvates, and is residue obtained with silica gel column chromatography (expansion solvent; Hexane: ethyl acetate=1: 1) refining, the solid with hexane cleaning gained prepares 0.840g (yield 51%) title compound thus.

¹H-NMR(CDCl ₃，ppm)δ7.36-7.40(1H，m)，7.53-7.64(3H，m)，7.84-7.97(1H，m)，7.92-7.94(2H，m)，8.04-8.07(1H，m)，8.08-8.13(1H，m)，8.20(2H，s)，8.68-8.72(1H，m).

＜embodiment 4 〉

The preparation of N-(2,6-two bromo-4-(perfluorinated butane-2-yl) phenyl)-2-fluoro-3-(N-methyl-benzamide base) benzamide (compound sequence number 7-1182)

<4-1>

The preparation of 4-(perfluorinated butane-2-yl) aniline

Use the reaction vessel of shading, 4.90g (52.6mmol) aniline, 10.1g (58.0mmol) 85% V-Brite B, 1.90g (5.77mmol) 4-butyl ammonium hydrogen sulfate are packed in the mixing solutions of 150ml t-butyl methyl ether, 150ml water, add 4.84g (57.6mmol) sodium bicarbonate.Splash into 20.0g (57.8mmol) nine fluoro-s-butyl iodides under the room temperature, stirring at room 5 hours.Separate to obtain organic phase, clean 2 times with the aqueous hydrochloric acid of 2mol/L after, clean with saturated aqueous common salt, sodium bicarbonate aqueous solution, saturated aqueous common salt.Behind the anhydrous magnesium sulfate drying organic layer, underpressure distillation removes and desolvates, and prepares 8.32g (yield 51%) title compound thus.

¹H-NMR(CDCl ₃，ppm)δ3.92(2H，broad-s)，6.72(2H，d，J＝8.8Hz)，7.34(2H，d，J＝8.8Hz).

<4-2>

2, the preparation of 6-two bromo-4-(perfluorinated butane-2-yl) aniline

Method according to the 2-2 of embodiment 2 prepares title compound by 4-(perfluorinated butane-2-yl) aniline.

¹H-NMR(CDCl ₃，ppm)δ4.89(2H，broad-s)，7.57(2H，s).

<4-3>

The preparation of 2-chloro-N-(2,6-two bromo-4-(perfluorinated butane-2-yl) phenyl)-3-nitrobenzamide

Add 9.90g (21.1mmol) 2 in 27ml DMI, 6-two bromo-4-(perfluorinated butane-2-yl) aniline, 4.60g (20.9mmol) 2-chloro-3-nitrobenzoyl chloride stirred 4 hours down at 140 ℃.Add entry and ethyl acetate in reaction soln, extracted organic phase is cleaned with 1mol/L aqueous sodium hydroxide solution, saturated aqueous common salt, and behind anhydrous magnesium sulfate drying, underpressure distillation removes and desolvates.Residue obtained with silica gel column chromatography (expansion solvent; Hexane: ethyl acetate=20: 1 → 10: 1 → 5: 1 → 3: 1) refining, prepare 5.44g (yield 40%) title compound thus.

¹H-NMR(CDCl ₃，ppm)δ7.52-7.61(2H，m)，7.89(2H，s)，7.94(1H，dd，J＝1.5，8.3Hz)，7.99(1H，d，J＝7.8Hz).

<4-4>

The preparation of N-(2,6-two bromo-4-(perfluorinated butane-2-yl) phenyl)-2-fluoro-3-nitrobenzamide

In 108ml DMSO, add 5.44g (8.34mmol) 2-chloro-N-(2,6-two bromo-4-(perfluorinated butane-2-yl) phenyl)-3-nitrobenzamide, 4.90g (84.3mmol) Potassium monofluoride (spraying drying thing), stirred 2 hours down at 145 ℃.In frozen water, inject reaction soln, make it separate out crystallization, filter the crystallization of gained and clean with hexane.(launch solvent with silica gel column chromatography; Hexane: ethyl acetate=5: the 1) crystallization of refining gained prepares 2.42g (yield 46%) title compound thus.

¹H-NMR(CDCl ₃，ppm)δ7.53-7.54(1H，m)，7.89(2H，s)，8.17(1H，d，J＝12.2Hz)，8.29-8.30(1H，m)，8.48-8.49(1H，m).

<4-5>

The preparation of 3-amino-N-(2,6-two bromo-4-(perfluorinated butane-2-yl) phenyl)-2-fluorobenzamide

Method according to the 1-5 of embodiment 1 prepares title compound by N-(2,6-two bromo-4-(perfluorinated butane-2-yl) phenyl)-2-fluoro-3-nitrobenzamide.

¹H-NMR(CDCl ₃，ppm)δ3.92(2H，broad-s)，6.99-7.04(1H，m)，7.11-7.12(1H，m)，7.48-7.52(1H，m)，7.86(2H，s)，8.22(1H，d，J＝14.1Hz).

<4-6>

The preparation of N-(2,6-two bromo-4-(perfluorinated butane-2-yl) phenyl)-2-fluoro-3-(methylamino) benzamide

Method according to the 1-6 of embodiment 1 prepares title compound by 3-amino-N-(2,6-two bromo-4-(perfluorinated butane-2-yl) phenyl)-2-fluorobenzamide.

¹H-NMR(CDCl ₃，ppm)δ2.95(3H，s)，4.14(1H，broad-s)，6.91-6.92(1H，m)，7.17-7.21(1H，m)，7.39-7.43(1H，m)，7.85(2H，s)，8.21(1H，d，J＝14.1Hz).

<4-7>

The preparation of N-(2,6-two bromo-4-(perfluorinated butane-2-yl) phenyl)-2-fluoro-3-(N-methyl-benzamide base) benzamide (compound sequence number 7-1182)

Method according to the 1-7 of embodiment 1 prepares title compound by N-(2,6-two bromo-4-(perfluorinated butane-2-yl) phenyl)-2-fluoro-3-(methylamino) benzamide.

¹H-NMR(CDCl ₃，ppm)δ3.51(3H，s)，7.22-7.44(7H，m)，7.85(2H，s)，8.00-8.03(2H，m).

＜embodiment 5 〉

The preparation of N-(2-bromo-6-(perfluor ethyl)-4-(perfluoropropane-2-yl) phenyl)-3-(4-cyano group benzoylamino)-2-fluorobenzamide (compound sequence number 6-5911)

<5-1>

The preparation of 2-(perfluor ethyl)-4-(perfluoropropane-2-yl) aniline

According to the method for the 1-1 of embodiment 1, by the 4-that obtains among the embodiment 2-1 (perfluoropropane-2-yl) aniline and 1,1,2,2,2-pentafluoroethyl group iodine prepares title compound.

¹H-NMR(CDCl ₃，ppm)δ4.56(2H，broad-s)，6.79(1H，d，J＝8.8Hz)，7.47(1H，d，J＝8.8Hz)，7.53(1H，s).

<5-2>

The preparation of 2-bromo-6-(perfluor ethyl)-4-(perfluoropropane-2-yl) aniline

Method according to the 1-2 of embodiment 1 prepares title compound by 2-(perfluor ethyl)-4-(perfluoropropane-2-yl) aniline.

¹H-NMR(CDCl ₃，ppm)δ5.14(2H，broad-s)，7.58(1H，s)，7.81(1H，s).

<5-3>

The preparation of N-(2-bromo-6-(perfluor ethyl)-4-(perfluoropropane-2-yl) phenyl)-2-chloro-3-nitrobenzamide

Method according to the 4-3 of embodiment 4 prepares title compound by 2-bromo-6-(perfluor ethyl)-4-(perfluoropropane-2-yl) aniline.

¹H-NMR(CDCl ₃，ppm)δ7.56-7.61(1H，m)，7.73(1H，s)，7.88(1H，d，J＝1.5Hz)，7.92-7.98(2H，m)，8.21(1H，s).

<5-4>

The preparation of N-(2-bromo-6-(perfluor ethyl)-4-(perfluoropropane-2-yl) phenyl)-2-fluoro-3-nitrobenzamide

Method according to the 1-4 of embodiment 1 prepares title compound by N-(2-bromo-6-(perfluor ethyl)-4-(perfluoropropane-2-yl) phenyl)-2-chloro-3-nitrobenzamide.

APCI-MS?m/z(M+1)：626

<5-5>

The preparation of 3-amino-N-(2-bromo-6-(perfluor ethyl)-4-(perfluoropropane-2-yl) phenyl)-2-fluorobenzamide

Method according to the 1-5 of embodiment 1 prepares title compound by N-(2-bromo-6-(perfluor ethyl)-4-(perfluoropropane-2-yl) phenyl)-2-fluoro-3-nitrobenzamide.

¹H-NMR(CDCl ₃，ppm)δ3.92(2H，broad-s)，6.99-7.04(1H，m)，7.05-7.18(1H，m)，7.46-7.51(1H，m)，7.85(1H，broad-s)，8.17(1H，broad-s)，8.34(1H，d，J＝15.1Hz).

<5-6>

The preparation of N-(2-bromo-6-(perfluor ethyl)-4-(perfluoropropane-2-yl) phenyl)-3-(4-cyano group benzoylamino)-2-fluorobenzamide (compound sequence number 6-5911)

Method according to the 1-7 of embodiment 1 prepares title compound by 3-amino-N-(2-bromo-6-(perfluor ethyl)-4-(perfluoropropane-2-yl) phenyl)-2-fluorobenzamide and 4-cyano-benzoyl chloride.

¹H-NMR(CDCl ₃，ppm)δ7.41(1H，t，J＝8.3Hz)，7.84-7.87(3H，m)，7.91-7.95(1H，m)，8.03-8.05(2H，m)，8.10(1H，broad-s)，8.17-8.20(2H，m)，8.63-8.67(1H，m).

＜embodiment 6 〉

The preparation of N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-6-(N-methyl-benzamide base) pyridine carboxamide (compound sequence number 17-1103)

<6-1>

The preparation of N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-6-chloropyridine methane amide

Method according to the 1-3 of embodiment 1 prepares title compound by 2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) aniline that obtains among the 1-2 with 2-chloropyridine-6-formic acid and the synthetic 2-chloropyridine of thionyl chloride-6-formyl chloride and embodiment 1.

¹H-NMR(CDCl ₃，ppm)δ7.59(1H，d，J＝7.3Hz)，7.90-7.93(2H，m)，8.14(1H，s)，8.20-8.24(1H，m)，9.60(1H，s).

<6-2>

The preparation of N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-6-(methylamino) pyridine carboxamide

5ml 1 to N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-6-chloropyridine methane amide 0.100g (0.180mmol), add 0.00600g (0.0360mmol) copper sulfate, 0.140g (1.80mmol) 40% aqueous methylamine solution in the 4-dioxane solution, under air-proof condition, stirred 3 hours down for 80 ℃ at oil bath temperature.Make reaction solution return to room temperature and make it open, add entry, ethyl acetate, water, saturated aqueous common salt clean organic layer, use anhydrous magnesium sulfate drying.Underpressure distillation removes and desolvates, and is residue obtained with silica gel column chromatography (expansion solvent; Hexane: ethyl acetate=2: 1) refining, prepare 0.0700g (yield 69%) title compound thus.

¹H-NMR(CDCl ₃，ppm)δ2.64(3H，s)，3.79(1H，broad-s)，7.56-7.60(1H，m)，7.87-7.93(2H，m)，8.14-8.15(1H，m)，8.20-8.23(1H，m)，9.60(1H，s).

<6-3>

The preparation of N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-6-(N-methyl-benzamide base) pyridine carboxamide (compound sequence number 17-1103)

Method according to the 1-7 of embodiment 1 prepares title compound by N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-6-(methylamino) pyridine carboxamide.

¹H-NMR(CDCl ₃，ppm)δ3.65(3H，s)，7.28-7.41(6H，m)，7.77(1H，t，J＝7.8Hz)，7.91(1H，s)，8.00-8.02(1H，m)，8.14(1H，s)，9.39(1H，s).

＜embodiment 7 〉

The preparation of N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-(2-fluoro-N-methyl-benzamide base) thiazole-4-carboxamide (compound sequence number 27-628)

<7-1>

The preparation of thiazolamine-4-formic acid

In the 40ml aqueous solution of thiazolamine-4-formic acid ethyl ester 4.00g (23.2mmol), add 1.86g (46.5mmol) sodium hydroxide, stirring at room 5 hours.Adding concentrated hydrochloric acid adjusting pH in the reaction solution is 1, and the crystallization that leaching is separated out prepares 2.84g (yield 85%) title compound thus.

¹H-NMR(CDCl ₃，ppm)δ7.18(2H，broad-s)，7.38(1H，s).

Do not detect the proton of carboxylic acid.

<7-2>

The preparation of 2-diuril azoles-4-formic acid

To the 30ml 1 of 2.84g (19.7mmol) thiazolamine-4-formic acid, add the 50ml concentrated hydrochloric acid in the 4-dioxane solution, be cooled to 0 ℃, at 0～5 ℃ of 10ml aqueous solution that drips 2.04g (29.6mmol) Sodium Nitrite down.After under 0 ℃ reaction solution being stirred 2 hours, 2.93g (29.6mmol) cupric chloride of in batches packing into makes reaction solution return to stirring at room 8 hours.In reaction solution, add entry, ethyl acetate, use ethyl acetate extraction 4 times.Behind saturated aqueous common salt cleaning organic layer, use anhydrous magnesium sulfate drying.Underpressure distillation removes and desolvates, and prepares 1.77g (yield 55%) title compound thus.

¹H-NMR(DMSO-d ₆，ppm)δ8.41(1H，s).

Do not detect the proton of carboxylic acid.

<7-3>

The preparation of N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-chlorine thiazole-4-carboxamide

Method according to the 4-3 of embodiment 4 prepares title compound by 2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) aniline that obtains among the 1-2 with 2-diuril azoles-4-formic acid and the synthetic 2-diuril azoles of thionyl chloride-4-carbonyl chlorine and embodiment 1.

¹H-NMR(CDCl ₃，ppm)δ7.91(1H，s)，8.13(1H，s)，8.19(1H，s)，8.82(1H，s).

<7-4>

The preparation of N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-(methylamino) thiazole-4-carboxamide

Method according to the 6-2 of embodiment 6 prepares title compound by N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-chlorine thiazole-4-carboxamide.

¹H-NMR(CDCl ₃，ppm)δ3.03(3H，s)，5.11-5.12(1H，m)，7.50(1H，s)，7.88(1H，s)，8.11(1H，s)，8.99(1H，s).

<7-5>

The preparation of N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-(2-fluoro-N-methyl-benzamide base) thiazole-4-carboxamide (compound sequence number 27-628)

Method according to the 1-7 of embodiment 1 prepares title compound by N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-(methylamino) thiazole-4-carboxamide and 2-fluorobenzoyl chloride.

¹H-NMR(CDCl ₃，ppm)δ3.67(3H，s)，6.99-7.24(1H，m)，7.29-7.35(1H，m)，7.52-7.59(2H，m)，7.90(1H，s)，8.06(1H，s)，8.14(1H，s)，9.08(1H，s).

＜embodiment 8 〉

2-fluoro-3-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl (methyl) carboxylamine 2,2, the preparation of 2-three chloro-ethyl esters (compound sequence number 12-864)

<8-1>

The preparation of 4-(perfluorinated butane-2-yl)-2-(trifluoromethyl) aniline

Method according to the 1-1 of embodiment 1 under the shading reaction conditions, prepares title compound by 2-(trifluoromethyl) aniline and nine fluoro-s-butyl iodides.

¹H-NMR(CDCl ₃，ppm)δ4.49(2H，broad-s)，6.81(1H，d，J＝8.8Hz)，7.47(1H，d，J＝8.8Hz)，7.61(1H，s).

<8-2>

The preparation of 2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) aniline

In 100mL ethanol, add 17.0g (44.8mmol) 4-(perfluorinated butane-2-yl)-2-(trifluoromethyl) aniline, at ice-cold 5.28g (53.8mmol) vitriol oil, 12.6g (55.8mmol) the N-iodo succimide of adding down, stirring at room stirred 4 hours down for 1 hour 30 minutes, 40 ℃.In reaction soln, add the 4M aqueous sodium hydroxide solution, behind the neutralization reaction solution, add ethyl acetate, extracted organic phase.Clean organic phase with saturated aqueous common salt, behind anhydrous magnesium sulfate drying, underpressure distillation removes and desolvates.Residue obtained with silica gel column chromatography (expansion solvent; Hexane: ethyl acetate=10: 1) refining, prepare 14.6g (yield 65%) title compound thus.

¹H-NMR(CDCl ₃，ppm)δ5.04(2H，broad-s)，7.62(1H，s)，7.97(1H，s).

<8-3>

The preparation of 2-chloro-N-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl)-3-nitrobenzamide

Method according to the 4-3 of embodiment 4 prepares title compound by 2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) aniline.

¹H-NMR(CDCl ₃，ppm)δ7.60-7.61(1H，m)，7.77(1H，s)，7.89-7.96(2H，m)，8.03-8.04(1H，m)，8.38(1H，s).

<8-4>

The preparation of 2-fluoro-N-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl)-3-nitrobenzamide

Method according to the 1-4 of embodiment 1 prepares title compound by 2-chloro-N-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl)-3-nitrobenzamide.

¹H-NMR(CDCl ₃，ppm)δ7.53-7.54(1H，m)，7.95(1H，s)，8.24-8.32(2H，m)，8.36(1H，s)，8.44-8.48(1H，m).

<8-5>

The preparation of 3-amino-2-fluoro-N-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl) benzamide

Method according to the 1-5 of embodiment 1 prepares title compound by 2-fluoro-N-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl)-3-nitrobenzamide.

¹H-NMR(CDCl ₃，ppm)δ3.93(2H，broad-s)，7.02-7.03(1H，m)，7.11-7.13(1H，m)，7.47-7.51(1H，m)，7.92(1H，s)，8.31-8.34(2H，m).

<8-6>

The preparation of 2-fluoro-N-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl)-3-(methylamino) benzamide

Method according to the 1-6 of embodiment 1 prepares title compound by 3-amino-2-fluoro-N-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl) benzamide.

¹H-NMR(CDCl ₃，ppm)δ2.95-2.96(3H，m)，4.15(1H，broad-s)，6.91-6.93(1H，m)，7.19-7.20(1H，m)，7.38-7.42(1H，m)，7.92(1H，s)，8.32(1H，d，J＝14.1Hz)，8.34(1H，s).

<8-7>

2-fluoro-3-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl (methyl) carboxylamine 2,2, the preparation of 2-three chloro-ethyl esters (compound sequence number 12-864)

According to the method for the 1-7 of embodiment 1, by 2-fluoro-N-(2-iodo-4-(perfluorinated butane-2-yl)-6-(trifluoromethyl) phenyl)-3-(methylamino) benzamide and 2,2,2-trichlorine ethoxy carbonyl chlorine prepares title compound.

¹H-NMR(CDCl ₃，ppm)δ3.40(3H，s)，4.74(2H，broad-s)，7.37(1H，t，J＝7.8Hz)，7.52-7.58(1H，m)，7.93(1H，s)，8.12-8.15(1H，m)，8.28-8.34(2H，m).

＜embodiment 9 〉

The preparation of N-(2-chloro-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-cyano group-3-(4-cyano group-N-methyl-benzamide base) benzamide (compound sequence number 2-491)

<9-1>

The preparation of 2-chloro-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) aniline

According to the method for the 1-2 of embodiment 1, the 4-that obtains among the 1-1 by embodiment 1 (perfluoropropane-2-yl)-2-(trifluoromethyl) aniline and N-neoprene imide prepare title compound.

¹H-NMR(CDCl ₃，ppm)δ4.97(2H，broad-s)，7.57(1H，s)，7.64(1H，s).

<9-2>

The preparation of N-(2-chloro-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-iodo-3-nitrobenzamide

According to the method for the 1-3 of embodiment 1, by preparing title compound with 4-iodo-3-nitrobenzoic acid and the synthetic 4-iodo-of thionyl chloride 3-nitrobenzoyl chloride and 2-chloro-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) aniline.

¹H-NMR(CDCl ₃，ppm)δ7.52-7.81(2H，m)，7.89(1H，s)，8.00(1H，s)，8.25(1H，d，J＝8.3Hz)，8.38(1H，d，J＝1.9Hz).

<9-3>

The preparation of 3-amino-N-(2-chloro-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-iodobenzene methane amide

Method according to the 1-5 of embodiment 1 prepares title compound by N-(2-chloro-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-iodo-3-nitrobenzamide.

¹H-NMR(CDCl ₃，ppm)δ4.35(2H，s)，6.92(1H，dd，J＝1.9，8.3Hz)，7.29(1H，d，J＝1.9Hz)，7.60(1H，s)，7.79(1H，d，J＝8.3Hz)，7.86(1H，s)，7.97(1H，s).

<9-4>

The preparation of N-(2-chloro-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-iodo-3-(methylamino) benzamide

Method according to the 1-6 of embodiment 1 prepares title compound by 3-amino-N-(2-chloro-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-iodobenzene methane amide.

¹H-NMR(CDCl ₃，ppm)δ2.97(3H，s)，4.46(1H，broad-s)，6.89(1H，dd，J＝1.9，8.3Hz)，7.07(1H，d，J＝1.9Hz)，7.65(1H，s)，7.80(1H，d，J＝8.3Hz)，7.86(1H，s)，7.97(1H，s).

<9-5>

The preparation of N-(2-chloro-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-cyano group-3-(methylamino) benzamide

In 10mL DMF, add 0.350g (0.560mmol) N-(2-chloro-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-iodo-3-(methylamino) benzamide, 0.200g (2.25mmol) cupric cyanide (I), stirred 1 hour 30 minutes down at 140 ℃.In reaction soln, inject saturated aqueous sodium thiosulfate, make the reaction quenching thus after, separate to obtain organic layer with ethyl acetate, clean with saturated aqueous common salt.Behind the anhydrous magnesium sulfate drying organic layer, underpressure distillation removes and desolvates.Residue obtained with silica gel column chromatography (expansion solvent; Hexane: ethyl acetate=5: 1 → 3: 1) refining, prepare 0.250g (yield 86%) title compound thus.

¹H-NMR(CDCl ₃，ppm)δ3.01(1/2*3H，s)，3.03(1/2*3H，s)，4.89(1/2 ₁H，s)，4.90(1/2 ₁H，s)，7.80(1H，dd，J＝1.5，8.3Hz)，7.21-7.22(1H，m)，7.54(1H，d，J＝8.3Hz)，7.67(1H，s)，7.88(1H，s)，7.99(1H，s).

<9-6>

The preparation of N-(2-chloro-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-cyano group-3-(4-cyano group-N-methyl-benzamide base) benzamide (compound sequence number 2-491)

Method according to the 1-7 of embodiment 1 prepares title compound by N-(2-chloro-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-cyano group-3-(methylamino) benzamide and 4-cyano-benzoyl chloride.

¹H-NMR(CDCl ₃，ppm)δ3.81(3H，broad-s)，7.52-7.84(8H，m)，7.89(1H，s)，8.00(1H，s).

＜embodiment 10 〉

The preparation of N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical)-6-cyano group-2-fluorophenyl)-6-chloro niacinamide (compound sequence number 1-1968)

<10-1>

N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-cyano group-2, the preparation of 3-difluorobenzamide

To 0.840g (4.59mmol) 4-cyano group-2, add 1 DMF, 0.470ml (5.51mmol) oxalyl chloride among the dichloromethane solution 10ml of 3-difluoro-benzoic acid, stirred 1 hour under the room temperature.Underpressure distillation is removed the 4-cyano group-2 of the gained that desolvates, the 3-difluoro benzoyl chloride is added among the DMI solution 5ml of 2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) the aniline 1.56g (3.83mmol) that obtains among the 1-2 of embodiment 1, and 130 ℃ were stirred 5 hours down.Add entry, ethyl acetate in the reaction solution, behind saturated sodium bicarbonate aqueous solution, saturated aqueous common salt cleaning organic layer, use anhydrous magnesium sulfate drying.Underpressure distillation removes and desolvates, with residue silica gel column chromatography (the expansion solvent of gained; Hexane: ethyl acetate=1: 0 → 10: 1) refining, prepare 0.58g (yield 27%) title compound thus.

¹H-NMR(CDCl ₃，ppm)δ7.52-7.62(1H，m)，7.92-7.94(1H，m)，8.02-8.06(1H，m)，8.13-8.16(2H，m).

<10-2>

The preparation of 3-amino-N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-cyano group-2-fluorobenzamide

To N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-cyano group-2, add the 49.0mg volatile salt among the DMSO solution 5ml of 3-difluorobenzamide, 100 ℃ were stirred 5 hours down.Add entry, ethyl acetate in the reaction solution, water is used anhydrous magnesium sulfate drying after cleaning organic layer.Underpressure distillation removes and desolvates, and (launches solvent with residue obtained with silica gel column chromatography; Hexane: ethyl acetate=8: 1 → 4: 1) refining, prepare 0.30g (yield 51%) title compound thus.

¹H-NMR(CDCl ₃，ppm)δ4.71(2H，broad-s)，7.35-7.39(1H，m)，7.40-7.44(1H，m)，7.92(1H，s)，8.12-8.15(2H，m).

<10-3>

The preparation of N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical)-6-cyano group-2-fluorophenyl)-6-chloro niacinamide (compound sequence number 1-1968)

In the DMI solution 0.200ml of 0.0500g (0.0877mol) 3-amino-N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-cyano group-2-fluorobenzamide, add 0.0308g (0.175mmol) 6-chloronicotinoyl chloride, stirred 6 hours down at 130 ℃.Add entry, ethyl acetate in the reaction solution, behind 1M hydrochloric acid, saturated sodium bicarbonate aqueous solution, saturated aqueous common salt cleaning organic layer, use anhydrous magnesium sulfate drying.Underpressure distillation removes and desolvates, and (launches solvent with residue obtained with silica gel column chromatography; Hexane: ethyl acetate=2: 1) refining, prepare 0.0100g (yield 16%) title compound thus.

¹H-NMR(CDCl ₃，ppm)δ7.54(1H，d，J＝8.8Hz)，7.72(1H，d，J＝8.8Hz)，7.93(1H，s)，8.09(1H，s)，8.17-8.18(2H，m)，8.27(1H，dd，J＝2.4Hz8.8Hz)，8.38(1H，d，J＝10.8Hz)，8.98(1H，d，J＝2.4Hz).

＜embodiment 11 〉

The preparation of 3-(4-cyano group benzoylamino)-N-(2,6-two iodo-4-(perfluorinated butane-2-yl) phenyl) benzamide (compound sequence number 6-79)

<11-1>

2, the preparation of 6-two iodo-4-(perfluorinated butane-2-yl) aniline

According to the method for the 3-1 of embodiment 3, the 4-that obtains among the 4-1 by embodiment 4 (perfluorinated butane-2-yl) aniline prepares title compound.

¹H-NMR(CDCl ₃，ppm)δ4.95(2H，broad-s)，7.78(2H，s).

<11-2>

The preparation of N-(2,6-two iodo-4-(perfluorinated butane-2-yl) phenyl)-3-nitrobenzamide

According to the method for the 4-3 of embodiment 4, by 2,6-two iodo-4-(perfluorinated butane-2-yl) aniline and 3-nitrobenzoyl chloride prepare title compound.

¹H-NMR(CDCl ₃，ppm)δ7.74(1H，t，J＝8.0Hz)，8.11(2H，s)，8.42(1H，d，J＝7.6Hz)，8.46(1H，d，J＝8.4Hz)，8.90(1H，d，J＝12.4Hz)，8.92(1H，s).

<11-3>

The preparation of 3-amino-N-(2,6-two iodo-4-(perfluorinated butane-2-yl) phenyl) benzamide

Method according to the 1-5 of embodiment 1 prepares title compound by N-(2,6-two iodo-4-(perfluorinated butane-2-yl) phenyl)-3-nitrobenzamide.

¹H-NMR(CDCl ₃，ppm)δ5.39(2H，broad-s)，6.89-6.93(1H，m)，7.29-7.31(3H，m)，7.68(1H，s)，8.08(2H，s).

<11-4>

The preparation of 3-(4-cyano group benzoylamino)-N-(2,6-two iodo-4-(perfluorinated butane-2-yl) phenyl) benzamide (compound sequence number 6-79)

Method according to the 1-7 of embodiment 1 prepares title compound by 3-amino-N-(2,6-two iodo-4-(perfluorinated butane-2-yl) phenyl) benzamide and 4-cyano-benzoyl chloride.

¹H-NMR(CDCl ₃，ppm)δ7.58(1H，t，J＝8.2Hz)，7.79-7.83(3H，m)，7.97(2H，s)，8.01(2H，d，J＝8.0Hz)，8.09(2H，s)，8.18(1H，s)，8.29(1H，s).

＜embodiment 12 〉

The preparation of N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethoxy) phenyl amino formyl radical)-2-fluorophenyl)-2-chloro niacinamide (compound sequence number 6-5908)

<12-1>

The preparation of 4-(perfluoropropane-2-yl)-2-(trifluoromethoxy) aniline

Method according to the 1-1 of embodiment 1 prepares title compound by the 2-trifluoro-methoxyaniline.

¹H-NMR(CDCl ₃，ppm)δ4.19(2H，broad-s)，6.86(1H，d，J＝8.8Hz)，7.30(1H，d，J＝8.8Hz)，7.36(1H，s).

<12-2>

The preparation of 2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethoxy) aniline

Method according to the 1-2 of embodiment 1 prepares title compound by 4-(perfluoropropane-2-yl)-2-(trifluoromethoxy) aniline.

¹H-NMR(CDCl ₃，ppm)δ4.65(2H，broad-s)，7.33(1H，s)，7.71(1H，s).

<12-3>

The preparation of N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethoxy) phenyl)-2-chloro-3-nitrobenzamide

Method according to the 1-3 of embodiment 1 prepares title compound by 2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethoxy) aniline.

¹H-NMR(CDCl ₃，ppm)δ7.49-7.61(3H，m)，7.80-7.96(3H，m).

<12-4>

The preparation of N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethoxy) phenyl)-2-fluoro-3-nitrobenzamide

Method according to the 1-4 of embodiment 1 prepares title compound by N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethoxy) phenyl)-2-chloro-3-nitrobenzamide.

¹H-NMR(CDCl ₃，ppm)δ7.53(1H，t，J＝7.8Hz)，7.60(1H，broad-s)，7.89(1H，d，J＝1.5Hz)，8.07(1H，broad-d，J＝12.7Hz)，8.29-8.30(1H，m)，8.43-8.47(1H，m).

<12-5>

The preparation of 3-amino-N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethoxy) phenyl)-2-fluorobenzamide

Method according to the 1-5 of embodiment 1 prepares title compound by N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethoxy) phenyl)-2-fluoro-3-nitrobenzamide.

¹H-NMR(CDCl ₃，ppm)δ3.92(2H，broad-s)，6.99-7.04(1H，m)，7.11(1H，t，J＝7.8Hz)，7.45-7.49(1H，m)，7.57(1H，broad-s)，7.87(1H，d，J＝2.0Hz)，8.14(1H，d，J＝14.2Hz).

<12-6>

The preparation of N-(3-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethoxy) phenyl amino formyl radical)-2-fluorophenyl)-2-chloro niacinamide (compound sequence number 6-5908)

Method according to the 1-7 of embodiment 1 prepares title compound by 3-amino-N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethoxy) phenyl)-2-fluorobenzamide and 2-chloronicotinoyl chloride.

¹H-NMR(CDCl ₃，ppm)δ7.39-7.49(2H，m)，7.59(1H，s)，7.88-7.94(2H，m)，8.07(1H，d，J＝12.2Hz)，8.31-8.33(1H，m)，8.57-8.58(1H，m)，8.60-8.70(1H，m)，8.74(1H，broad-s).

＜embodiment 13 〉

The preparation of 3-benzoylamino-N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-fluorobenzamide (compound sequence number 6-3348)

<13-1>

The preparation of N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-fluoro-3-nitrobenzamide

Method according to the 1-3 of embodiment 1 prepares title compound by the 2-bromo-4-that obtains among the 1-2 with 4-fluoro-3-nitrobenzoic acid and the synthetic 4-fluoro-of thionyl chloride 3-nitrobenzoyl chloride and embodiment 1 (perfluoropropane-2-yl)-6-(trifluoromethyl) aniline.

¹H-NMR(CDCl ₃，ppm)δ7.47-7.50(1H，m)，7.92(2H，d，J＝5.9Hz)，8.16(1H，s)，8.23-8.28(1H，m)，8.65-8.67(1H，m).

<13-2>

The preparation of 3-amino-N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-fluorobenzamide

Method according to the 1-5 of embodiment 1 prepares title compound by N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-fluoro-3-nitrobenzamide.

APCI-MS?m/z(M+1)：546

<13-3>

The preparation of 3-benzoylamino-N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-fluorobenzamide (compound sequence number 6-3348)

Method according to the 1-7 of embodiment 1 prepares title compound by 3-amino-N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-fluorobenzamide.

¹H-NMR(CDCl ₃，ppm)δ7.29-7.34(1H，m)，7.53-7.65(3H，m)，7.80-7.84(1H，m)，7.90-7.92(3H，m)，8.14(1H，broad-s)，8.20(1H，d，J＝2.9Hz)，8.25(1H，broad-s)，9.10(1H，dd，J＝1.9，7.3Hz).

＜embodiment 14 〉

The preparation (compound sequence number 6-460) of 2-chloro-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) niacinamide

<14-1>

The preparation of 2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) aniline

According to the method for the 8-2 of embodiment 8, the 4-that obtains among the 1-1 by embodiment 1 (perfluoropropane-2-yl)-2-(trifluoromethyl) aniline and N-iodo succimide prepare title compound.

¹H-NMR(CDCl ₃，ppm)δ5.04(2H，broad-s)，7.64(1H，s)，7.99(1H，s).

<14-2>

The preparation of N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-nitrobenzamide

Method according to the 4-3 of embodiment 4 prepares title compound by 2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) aniline and 3-nitrobenzoyl chloride.

¹H-NMR(CDCl ₃，ppm)δ7.76-7.80(2H，m)，7.97(1H，s)，8.28-8.30(1H，m)，8.37(1H，s)，8.49-8.52(1H，m)，8.78(1H，s).

<14-3>

The preparation of 3-amino-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide

Method according to the 1-5 of embodiment 1 prepares title compound by N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-nitrobenzamide.

¹H-NMR(CDCl ₃，ppm)δ3.89(2H，broad-s)，6.89-6.92(1H，m)，7.23-7.32(3H，m)，7.68(1H，s)，7.93(1H，s)，8.34-8.36(1H，m).

<14-4>

The preparation (compound sequence number 6-460) of 2-chloro-N-(3-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl amino formyl radical) phenyl) niacinamide

Method according to the 1-7 of embodiment 1 prepares title compound by 3-amino-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide and 2-chloronicotinoyl chloride.

¹H-NMR(CDCl ₃，ppm)δ7.43-7.46(1H，m)，7.58(1H，t，J＝7.8Hz)，7.77(1H，d，J＝7.8Hz)，7.91-7.95(2H，m)，8.01(1H，s)，8.24(1H，dd，J＝2.0，7.8Hz)，8.28(1H，s)，8.36(1H，s)，8.41(1H，s)，8.54-8.56(1H，m).

＜embodiment 15 〉

The preparation of 2-fluoro-3-(4-fluoro-N-methyl-benzamide base)-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide (compound sequence number 7-1733)

<15-1>

The preparation of 2-chloro-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-nitrobenzamide

According to the method for the 4-3 of embodiment 4, the 2-iodo-4-that obtains among the 14-1 by embodiment 14 (perfluoropropane-2-yl)-6-(trifluoromethyl) aniline and 2-chloro-3-nitrobenzoyl chloride prepare title compound.

¹H-NMR(CDCl ₃，ppm)δ7.60(1H，t，J＝7.8Hz)，7.76(1H，s)，7.94(1H，dd，J＝1.5，7.8Hz)，7.97(1H，s)，8.03(1H，dd，J＝1.5，7.8Hz)，8.39(1H，s).

<15-2>

The preparation of 2-fluoro-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-nitrobenzamide

Method according to the 1-4 of embodiment 1 prepares title compound by 2-chloro-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-nitrobenzamide.

¹H-NMR(CDCl ₃，ppm)δ7.51-7.55(1H，m)，7.97(1H，s)，8.23(1H，d，J＝12.2Hz)，8.28-8.32(1H，m)，8.37(1H，s)，8.44-8.48(1H，m).

<15-3>

The preparation of 3-amino-2-fluoro-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide

Method according to the 1-5 of embodiment 1 prepares title compound by 2-fluoro-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-nitrobenzamide.

¹H-NMR(CDCl ₃，ppm)δ3.92(2H，broad-s)，7.02-7.04(1H，m)，7.11(1H，t，J＝7.8Hz)，7.47-7.52(1H，m)，7.94(1H，s)，8.30-8.35(2H，m).

<15-4>

The preparation of 2-fluoro-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-(methylamino) benzamide

Method according to the 1-6 of embodiment 1 prepares title compound by 3-amino-2-fluoro-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide.

¹H-NMR(CDCl ₃，ppm)δ2.95(3H，s)，4.15(1H，broad-s)，6.90(1H，t，J＝8.2Hz)，7.19(1H，t，J＝7.8Hz)，7.40(1H，t，J＝7.8Hz)，7.92(1H，s)，8.30(1H，s)，8.34(1H，s).

<15-5>

The preparation of 2-fluoro-3-(4-fluoro-N-methyl-benzamide base)-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl) benzamide (compound sequence number 7-1733)

Method according to the 1-7 of embodiment 1 prepares title compound by 2-fluoro-N-(2-iodo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-(methylamino) benzamide and 4-fluorobenzoyl chloride.

¹H-NMR(CDCl ₃，ppm)δ3.50(3H，s)，6.91(2H，s)，6.93-7.35(3H，m)，7.46(1H，t，J＝7.0Hz)，7.93(1H，s)，8.01-8.10(1H，m)，8.13(1H，broad-s)，8.34(1H，s).

＜embodiment 16 〉

The preparation of N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-fluoro-N-methyl-3-(N-methyl-benzamide base) benzamide (compound sequence number 9-2164)

Add 0.00900g (0.230mmol) sodium hydride (60%inoil) among the DMF solution 5ml of the 0.100g that in the 1-7 of embodiment 1, obtains (0.150mmol) N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-2-fluoro-3-(N-methyl-benzamide base) benzamide, stirred 40 minutes under the room temperature.Add 0.0300g (0.180mmol) methyl iodide in the reaction solution, under uniform temp, stirred 6 hours.Add entry, ethyl acetate in the reaction solution, water, saturated aqueous common salt clean organic layer, use anhydrous magnesium sulfate drying.Underpressure distillation removes and desolvates, and is residue obtained with silica gel column chromatography (expansion solvent; Hexane: ethyl acetate=4: 1) refining, prepare the 0.106g title compound thus quantitatively.

¹H-NMR(CDCl ₃，ppm)δ2.18-2.19(3H，m)，3.48(3H，s)，7.21-7.25(4H，m)，7.32-7.40(4H，m)，7.92(1H，s)，8.13(1H，s).

＜embodiment 17 〉

The preparation of N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-(4-cyano group benzoylamino)-N-methyl-benzamide (compound sequence number 8-289)

<17-1>

The preparation of N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-nitrobenzamide

According to the method for the 4-3 of embodiment 4,2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) aniline and the 3-nitrobenzoyl chloride that are obtained by the 1-2 of embodiment 1 prepare title compound.

¹H-NMR(CDCl ₃，ppm)δ7.75-7.79(2H，m)，7.94(1H，s)，8.17(1H，d，J＝1.0Hz)，8.28(1H，dd，J＝1.5，7.8Hz)，8.48-8.51(1H，m)，8.76-8.77(1H，m).

<17-2>

The preparation of N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-N-methyl-3-nitro benzamide

According to the method for embodiment 16, prepare title compound by N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-nitrobenzamide.

¹H-NMR(CDCl ₃，ppm)δ3.28(1/2*3H，s)，3.44(1/2*3H，s)，7.41(1/2*1H，t，J＝7.8Hz)，7.71-7.76(2/2*1H，m)，7.84(1/2*1H，s)，7.93-7.95(1/2*1H，m)，7.98(1/2*1H，s)，8.07-8.09(2/2*1H，m)，8.14-8.16(1/2*1H，m)，8.19(1/2*1H，s)，8.39-8.41(1/2*1H，m)，8.45-8.46(1/2*1H，m).

<17-3>

The preparation of 3-amino-N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-N-methyl-benzamide

Method according to the 1-5 of embodiment 1 prepares title compound by N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-N-methyl-3-nitro benzamide.

¹H-NMR(CDCl ₃，ppm)δ3.24(3/4*3H，s)，3.37(1/4*3H，s)，3.80(2H，broad-s)，6.47(1/4*1H，d，J＝7.8Hz)，6.54-6.57(1/4*1H，m)，6.78-6.84(5/4*1H，m)，6.86(3/4*1H，t，J＝2.0Hz)，6.96(3/4*1H，d，J＝7.8Hz)，7.23-7.27(3/4*1H，m)，7.79(1/4*1H，s)，7.94(3/4*1H，s)，8.00(1/4*1H，s)，8.15(3/4*1H，s).

<17-4>

The preparation of N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-3-(4-cyano group benzoylamino)-N-methyl-benzamide (compound sequence number 8-289)

According to the 1-7 method of embodiment 1, prepare title compound by 3-amino-N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-N-methyl-benzamide and 4-cyano-benzoyl chloride.

¹H-NMR(CDCl ₃，ppm)δ3.26(2/3*3H，s)，3.38(1/3*3H，s)，7.08-7.09(1/3*1H，m)，7.12-7.14(1/3*1H，m)，7.32(2/3*1H，d，J＝7.8Hz)，7.45-7.49(3/3*1H，m)，7.72-7.76(9/3*1H，m)，7.83(1/3*1H，s)，7.85-7.89(4/3*1H，m)，7.95(2/3*1H，s)，7.98-8.00(4/3*1H，m)，8.04(2/3*1H，d，J＝6.3Hz)，8.16(2/3*1H，s)，8.57(2/3*1H，s).

＜embodiment 18 〉

The preparation of 3-benzoylamino-N-(2-bromo-4-(perfluor ethyl)-6-(trifluoromethyl) phenyl) benzamide (compound sequence number 6-5913)

<18-1>

The preparation of 4-(perfluor ethyl)-2-(trifluoromethyl) aniline

In the aqueous solution 40ml of 7.04g (40.4mmol) 85% V-Brite B, 3.40g (40.4mmol) sodium bicarbonate, add 13.6g (33.7mmol) 2-(trifluoromethyl) aniline and 40ml DMF.Add 11.2g (45.5mmol) 1,1,2,2 in this reaction solution, the 50ml DMF solution of 2-pentafluoroethyl group iodine (DMF being cooled to-30 ℃ and make 1,1,2,2, the dissolving of 2-pentafluoroethyl group iodine) in the autoclave of packing into, stirred 9 hours down at 110 ℃.After placing a night under the room temperature, in reaction solution, add entry, ethyl acetate, use ethyl acetate extraction.Water, saturated sodium bicarbonate aqueous solution, saturated aqueous common salt clean organic layer.Behind the anhydrous sodium sulfate drying organic layer, underpressure distillation removes and desolvates, and (launches solvent with residue obtained with silica gel column chromatography; Hexane: ethyl acetate=10: 1 → 5: 1) refining, prepare 1.95g (yield 21%) title compound thus.

¹H-NMR(CDCl ₃，ppm)δ4.53(2H，broad-s)，6.81(1H，d，J＝8.3Hz)，7.48(1H，d，J＝8.3Hz)，7.63(1H，broad-s).

<18-2>

The preparation of 2-bromo-4-(perfluor ethyl)-6-(trifluoromethyl) aniline

Method according to the 1-2 of embodiment 1 prepares title compound by 4-(perfluor ethyl)-2-(trifluoromethyl) aniline.

¹H-NMR(CDCl ₃，ppm)δ5.08(2H，broad-s)，7.62(1H，s)，7.80(1H，s).

<18-3>

The preparation of N-(2-bromo-4-(perfluor ethyl)-6-(trifluoromethyl) phenyl)-3-nitrobenzamide

In the pyridine solution 20ml of 2.50g (6.99mmol) 2-bromo-4-(perfluor ethyl)-6-(trifluoromethyl) aniline, add 2.72g (14.7mmol) 3-nitrobenzoyl chloride, stirred 12 hours down at 100 ℃.Add entry, ethyl acetate in the reaction solution, use ethyl acetate extraction.Clean organic layer with 1M hydrochloric acid, saturated sodium bicarbonate aqueous solution, saturated aqueous common salt.Behind the anhydrous sodium sulfate drying organic layer, decompression distillation down adds THF, aqueous sodium hydroxide solution except that desolvating in the residue that obtains, stirred 8 hours under the room temperature.With the above-mentioned dry reaction liquid that similarly extracts, underpressure distillation removes and desolvates, and (launches solvent with residue obtained with silica gel column chromatography; Hexane: ethyl acetate=7: 1 → 5: 1) refining, prepare 0.202g (yield 6%) title compound thus.

¹H-NMR(CDCl ₃，ppm)δ7.75(1H，s)，7.78(1H，t，J＝7.8Hz)，7.94(1H，s)，8.17(1H，s)，8.29-8.30(1H，m)，8.50-8.52(1H，m)，8.78(1H，t，J＝2.0Hz).

<18-4>

The preparation of 3-amino-N-(2-bromo-4-(perfluor ethyl)-6-(trifluoromethyl) phenyl) benzamide

Method according to the 1-5 of embodiment 1 prepares title compound by N-(2-bromo-4-(perfluor ethyl)-6-(trifluoromethyl) phenyl)-3-nitrobenzamide.

¹H-NMR(CDCl ₃，ppm)δ3.89(2H，broad-s)，6.90-6.92(1H，m)，7.23-7.32(3H，m)，7.64(1H，s)，7.90(1H，s)，8.13(1H，s).

<18-5>

The preparation of 3-benzoylamino-N-(2-bromo-4-(perfluor ethyl)-6-(trifluoromethyl) phenyl) benzamide (compound sequence number 6-5913)

Method according to the 1-7 of embodiment 1 prepares title compound by 3-amino-N-(2-bromo-4-(perfluor ethyl)-6-(trifluoromethyl) phenyl) benzamide.

¹H-NMR(CDCl ₃，ppm)δ7.51-7.62(4H，m)，7.72(1H，dd，J＝1.5，7.8Hz)，7.89-8.00(6H，m)，8.14(1H，s)，8.27(1H，t，J＝2.0Hz).

＜embodiment 19 〉

The preparation of 3-benzoylamino-N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-cyano group benzamide (compound sequence number 1-627)

<19-1>

The preparation of N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-fluoro-3-nitrobenzamide

Method according to the 4-3 of embodiment 4 prepares title compound by the 2-bromo-4-that obtains among the 1-2 with 4-fluoro-3-nitrobenzoic acid and the synthetic 4-fluoro-of thionyl chloride 3-nitrobenzoyl chloride and embodiment 1 (perfluoropropane-2-yl)-6-(trifluoromethyl) aniline.

¹H-NMR(CDCl ₃，ppm)δ7.47-7.50(1H，m)，7.92(2H，d，J＝5.9Hz)，8.16(1H，s)，8.23-8.28(1H，m)，8.65-8.67(1H，m).

<19-2>

The preparation of N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-cyano group-3-nitrobenzamide

In the DMF solution 5ml of 0.500g (0.870mmol) N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-fluoro-3-nitrobenzamide, add 0.0639g (1.31mmol) sodium cyanide, stirred 10 hours under the room temperature.Add entry, ethyl acetate in the reaction solution, use ethyl acetate extraction.Clean organic layer with 10% aqueous sodium hydroxide solution, saturated aqueous common salt.Behind the anhydrous sodium sulfate drying organic layer, underpressure distillation removes and desolvates, and with residue obtained refining with silica gel column chromatography, prepares 0.0500g (yield 10%) title compound thus.

¹H-NMR(CDCl ₃，ppm)δ7.80(1H，s)，7.96(1H，s)，8.12-8.14(1H，m)，8.18(1H，s)，8.36(1H，dd，J＝2.0，8.3Hz)，8.84(1H，d，J＝1.5Hz).

<19-3>

The preparation of 3-amino-N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-cyano group benzamide

Method according to the 1-5 of embodiment 1 prepares title compound by N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-cyano group-3-nitrobenzamide.

¹H-NMR(CDCl ₃，ppm)δ4.68(2H，broad-s)，7.18(1H，dd，J＝1.9，8.3Hz)，7.29(1H，s)，7.52-7.55(1H，m)，7.68(1H，s)，7.92(1H，s)，8.14(1H，d，J＝1.5Hz).

<19-4>

The preparation of 3-benzoylamino-N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-cyano group benzamide (compound sequence number 1-627)

Method according to the 1-7 of embodiment 1 prepares title compound by 3-amino-N-(2-bromo-4-(perfluoropropane-2-yl)-6-(trifluoromethyl) phenyl)-4-cyano group benzamide.

¹H-NMR(CDCl ₃，ppm)δ7.56-7.59(3H，m)，7.64-7.66(1H，m)，7.80-7.87(2H，m)，7.94-7.97(2H，m)，8.16(1H，s)，8.46(1H，s)，8.57(1H，s)，9.16(1H，s).

Next, provide and contain the formulation example of The compounds of this invention, but the present invention is not limited to this as effective constituent.Need to prove, in the formulation example, part expression weight part.

＜formulation example 1 〉

The The compounds of this invention of 20 parts of general formulas (1) expression, 10 parts of polyoxyethylene styryl phenyl ethers, 70 parts of dimethylbenzene homogeneous mixing are obtained emulsion.

＜formulation example 2 〉

The compounds of this invention, 2 parts of sodium lauryl sulphate, 2 parts of dialkyl sulfosuccinates, 1 part of beta-naphthalenesulfonic-acid formaldehyde condensation compound sodium salt, 85 parts of diatomite homogeneous of 10 parts of general formulas (1) expression are mixed and obtain wettable powder.

＜formulation example 3 〉

The The compounds of this invention of 0.3 part of general formula (1) expression, 0.3 part of white carbon(ink) homogeneous are mixed, add 99.2 parts of clays, 0.2 part of DRILESS A (three are total to the Agro system), homogeneous is pulverized and is mixed, and obtains pulvis.

＜formulation example 4 〉

After the The compounds of this invention of 3 parts of general formulas (1) expressions, 1.5 parts of polyoxyethylene polyoxypropylene condensess, 3 parts of carboxymethyl celluloses, 64.8 parts of clays, 27.7 parts of talcum homogeneous are pulverized and mix, add the mixing and granulating and drying of entry and obtain granule.

＜formulation example 5 〉

After The compounds of this invention, 3 parts of beta-naphthalenesulfonic-acid formaldehyde condensation compound sodium salts, 1 part of triphenyl vinyl phenol, 5 parts of propylene glycol, 0.5 part of silicon defoamer, 33.5 parts of water of 10 parts of general formulas (1) expressions are fully mixed, mix once more with material and to obtain suspensoid 0.3 part of xanthan gum, 46.7 parts of water mixing gained.

＜formulation example 6 〉

After the The compounds of this invention of 20 parts of general formulas (1) expressions, 6 parts of naphthalene sulfonic acidformaldehyde condensation product metal-salts, 1 part of dialkyl sulfosuccinate succsinic acid metal-salt, 73 parts of lime carbonate homogeneous are pulverized and mix, add the mixing and granulating and drying of entry and obtain water dispersion granule.

When using the preparation of above-mentioned gained,, or do not dilute, directly scatter 1～10000 times of above-mentioned preparation dilute with water.

Next, the availability for as the noxious organism control agent of The compounds of this invention specify in following test example, but the present invention is not limited to this.

＜test example 1 〉

Insecticidal test to prodenia litura (Spodopteralitura)

Dipping Caulis et Folium Brassicae capitatae leaf is 30 seconds in the soup that test compound is modulated to normality, air-dry after, put into the polyethylene cup of the 7cm that has laid filter paper, put into prodenia litura 2 instar larvaes.Be placed in 25 ℃ of thermostatic chambers " Invest, Then Investigate " life and death borer population on the 6th.Carry out in 52 modes that connect system in 1 district.

Need to prove that compound as a comparison uses the international disclosed following compound (A) in No. 2005/073165 specification sheets that discloses.

The result of above-mentioned test, following compound has shown the dead worm rate more than 70% in concentration during for 1ppm, and the sequence number of described compound is: 1-470,1-491,1-513,1-627,1-1925,2-491,6-38,6-39,6-45,6-46,6-47,6-57,6-60,6-71,6-72,6-78,6-79,6-80,6-90,6-93,6-111,6-147,6-268,6-269,6-270,6-271,6-272,6-288,6-289,6-290,6-293,6-300,6-304,6-306,6-311,6-346,6-347,6-348,6-349,6-366,6-367,6-368,6-382,6-389,6-424,6-425,6-426,6-427,6-428,6-444,6-445,6-446,6-448,6-449,6-450,6-452,6-453,6-460,6-461,6-467,6-502,6-503,6-504,6-505,6-522,6-523,6-524,6-538,6-545,6-804,6-824,6-825,6-840,6-1104,6-1105,6-1106,6-1107,6-1124,6-1125,6-1126,6-1140,6-1147,6-1182,6-1183,6-1184,6-1185,6-1202,6-1203,6-1204,6-1218,6-1225,6-1260,6-1261,6-1262,6-1263,6-1280,6-1281,6-1282,6-1296,6-1303,6-1338,6-1339,6-1340,6-1341,6-1358,6-1359,6-1360,6-1374,6-1381,6-1574,6-1575,6-1576,6-1577,6-1594,6-1595,6-1596,6-1610,6-1617,6-1652,6-1653,6-1654,6-1655,6-1672,6-1673,6-1674,6-1688,6-1695,6-1730,6-1731,6-1732,6-1733,6-1734,6-1750,6-1751,6-1752,6-1754,6-1755,6-1766,6-1773,6-1808,6-1809,6-1810,6-1811,6-1828,6-1829,6-1830,6-1851,6-2110,6-3348,6-3384,6-5902,6-5903,6-5904,6-5905,6-5906,6-5907,6-5908,6-5909,6-5910,6-5911,6-5912,7-38,7-39,7-45,7-46,7-47,7-57,7-60,7-71,7-72,7-78,7-79,7-80,7-90,7-93,7-132,7-147,7-268,7-269,7-270,7-271,7-285,7-286,7-288,7-289,7-290,7-299,7-300,7-301,7-303,7-304,7-305,7-311,7-346,7-347,7-348,7-349,7-366,7-367,7-368,7-382,7-389,7-424,7-425,7-426,7-427,7-428,7-444,7-445,7-446,7-449,7-460,7-467,7-502,7-504,7-505,7-522,7-523,7-538,7-804,7-824,7-825,7-840,7-948,7-969,7-984,7-1104,7-1105,7-1106,7-1107,7-1124,7-1125,7-1126,7-1140,7-1147,7-1182,7-1183,7-1184,7-1185,7-1202,7-1203,7-1204,7-1218,7-1225,7-1260,7-1261,7-1262,7-1263,7-1280,7-1281,7-1282,7-1296,7-1303,7-1338,7-1339,7-1340,7-1341,7-1358,7-1359,7-1360,7-1374,7-1381,7-1417,7-1574,7-1575,7-1576,7-1577,7-1594,7-1595,7-1596,7-1605,7-1606,7-1608,7-1610,7-1616,7-1617,7-1638,7-1639,7-1645,7-1652,7-1672,7-1673,7-1730,7-1731,7-1732,7-1733,7-1750,7-1751,7-1752,7-1764,7-1766,7-1773,7-1794,7-1808,7-1809,7-1810,7-1811,7-1828,7-1829,7-1844,7-1851,7-3348,7-3369,7-3384,7-5902,7-5903,7-5904,7-5905,7-5906,7-5907,7-5910,8-268,8-288,8-289,8-304,8-804,8-824,8-840,9-270,9-290,9-291,9-306,9-2164,9-2322,11-777,11-835,12-777,12-835,12-864,27-627,27-663.

In addition, following compound has shown the dead worm rate more than 70% in concentration during for 10ppm, and the sequence number of described compound is 1-506,1-1968,2-513,2-518,6-454,6-5913,6-5914,7-316,7-5911,7-5912,7-5908,7-5909,17-1103,27-628.

On the other hand, compound (A) is when concentration is 10ppm, and dead worm rate is below 50%.

＜test example 2 〉

Insecticidal test to small cabbage moth (Plutellaxylostella)

Dipping Caulis et Folium Brassicae capitatae leaf is 30 seconds in the soup that test compound is modulated to normality, air-dry after, add in the polyethylene cup of the 7cm that has laid filter paper, put into small cabbage moth 3 instar larvaes.Be placed in 25 ℃ of thermostatic chambers " Invest, Then Investigate " life and death borer population on the 6th.Carry out in 52 modes that connect system in 1 district.

Need to prove that compound uses above-claimed cpd (A) as a comparison.

The result of above-mentioned test, following compound has shown the dead worm rate more than 70% in concentration during for 1ppm, and the sequence number of described compound is 1-491,1-513,1-627,1-1925,1-1968,2-491,2-513,6-38,6-39,6-45,6-46,6-47,6-57,6-71,6-72,6-78,6-79,6-80,6-90,6-111,6-147,6-268,6-270,6-271,6-272,6-288,6-289,6-290,6-293,6-300,6-304,6-306,6-346,6-347,6-348,6-349,6-366,6-367,6-368,6-382,6-389,6-424,6-425,6-426,6-427,6-428,6-444,6-445,6-446,6-449,6-450,6-453,6-460,6-461,6-467,6-502,6-503,6-504,6-505,6-522,6-523,6-524,6-538,6-545,6-804,6-824,6-825,6-840,6-1104,6-1105,6-1106,6-1107,6-1124,6-1125,6-1126,6-1140,6-1147,6-1182,6-1183,6-1184,6-1185,6-1202,6-1203,6-1204,6-1218,6-1225,6-1260,6-1261,6-1262,6-1263,6-1280,6-1281,6-1282,6-1296,6-1303,6-1338,6-1339,6-1340,6-1341,6-1358,6-1359,6-1360,6-1374,6-1381,6-1574,6-1575,6-1576,6-1577,6-1594,6-1595,6-1596,6-1610,6-1617,6-1652,6-1653,6-1654,6-1655,6-1672,6-1673,6-1674,6-1688,6-1695,6-1730,6-1731,6-1732,6-1733,6-1734,6-1750,6-1751,6-1752,6-1754,6-1755,6-1766,6-1773,6-1808,6-1809,6-1810,6-1811,6-1828,6-1829,6-1830,6-1851,6-2110,6-3348,6-3384,6-5903,6-5904,6-5905,6-5906,6-5907,6-5908,6-5909,6-5910,6-5911,6-5912,7-38,7-39,7-45,7-46,7-47,7-57,7-60,7-71,7-72,7-78,7-79,7-80,7-90,7-93,7-132,7-147,7-268,7-271,7-286,7-288,7-289,7-290,7-299,7-300,7-301,7-303,7-304,7-305,7-311,7-346,7-347,7-348,7-349,7-366,7-367,7-368,7-382,7-389,7-424,7-425,7-426,7-427,7-428,7-444,7-445,7-446,7-449,7-460,7-467,7-502,7-504,7-505,7-522,7-523,7-538,7-824,7-840,7-948,7-969,7-984,7-1104,7-1105,7-1106,7-1107,7-1124,7-1125,7-1126,7-1140,7-1147,7-1182,7-1183,7-1184,7-1185,7-1202,7-1203,7-1204,7-1218,7-1225,7-1260,7-1261,7-1262,7-1263,7-1280,7-1281,7-1282,7-1296,7-1303,7-1338,7-1339,7-1340,7-1341,7-1358,7-1359,7-1360,7-1374,7-1381,7-1417,7-1574,7-1575,7-1576,7-1577,7-1594,7-1595,7-1596,7-1605,7-1606,7-1608,7-1610,7-1616,7-1617,7-1638,7-1639,7-1645,7-1652,7-1672,7-1673,7-1730,7-1731,7-1732,7-1733,7-1750,7-1751,7-1752,7-1764,7-1766,7-1773,7-1794,7-1808,7-1809,7-1810,7-1811,7-1828,7-1829,7-1844,7-1851,7-3348,7-3369,7-3384,7-5902,7-5903,7-5904,7-5905,7-5906,7-5907,7-5909,7-5910,8-268,8-288,8-289,8-304,8-824,9-270,9-290,9-291,9-306,9-2164,9-2322,11-777,11-835,12-777,12-835,12-864.

In addition, following compound has shown the dead worm rate more than 70% in concentration during for 10ppm, and the sequence number of described compound is 1-470,1-506,2-518,6-60,6-93,6-269,6-311,6-448,6-452,6-454,6-5913,6-5914,7-269,7-270,7-285,7-316,7-804,7-825,7-5908,7-5911,7-5912,8-804,8-840,17-1103,27-627,27-628,27-663.

On the other hand, compound (A) dead worm rate when concentration is 10ppm is below 50%.

＜test example 3 〉

Insecticidal test to tea Ji leaf roller (Adoxophyeshonmai)

The artificial diet thinly sliced of dipping are 30 seconds in the soup that test compound is modulated to normality, air-dry after, add in the polyethylene cup of 7cm, put into tea Ji leaf roller 2 instar larvaes.Be placed in 25 ℃ of thermostatic chambers " Invest, Then Investigate " life and death borer population on the 6th.Carry out in 52 modes that connect system in 1 district.

Need to prove that compound uses above-claimed cpd (A) as a comparison.

The result of above-mentioned test, following compound demonstrates dead worm rate more than 70% during for 1ppm in concentration, and the sequence number of described compound is 6-72,6-80,6-90,6-347,6-348,6-349,6-366,6-382,6-427,6-446,6-449,6-460,6-503,6-504,6-505,6-522,6-524,6-538,6-1106,6-1182,6-1202,6-1260,6-1262,6-1263,6-1341,6-1358,6-1574,6-1576,6-1594,6-1596,6-1652,6-1654,6-1655,6-1672,6-1674,6-1688,6-1730,6-1732,6-1733,6-1750,6-1809,6-1811,6-1828,6-1830,7-348,7-366,7-382,7-502,7-505,7-522,7-538,7-1106,7-1202,7-1262,7-1280,7-1303,7-1338,7-1358,7-1574,7-1576,7-1594,7-1605,7-1652,7-1730,7-1732,7-1733,7-1750,7-1764,7-1808,7-1809,7-1810,7-1811.

In addition, following compound concentrations has shown the dead worm rate more than 70% during for 10ppm, and the sequence number of described compound is 6-271,6-367,6-389,6-426,6-523,6-1104,6-1577,6-1695,6-1851,6-2110,7-424,7-444,7-523,7-1104,7-1124,7-1260,7-1263,7-1577,7-1616,7-1731,7-1773,7-1851.

On the other hand, compound (A) dead worm rate when concentration is 10ppm is below 50%.

＜test example 4 〉

Insecticidal test to the long leaf roller of tea (Choristoneuramagnanima)

The artificial diet thinly sliced of dipping are 30 seconds in the soup that test compound is modulated to normality, air-dry after, add in the polyethylene cup of 7cm, put into long leaf roller 2 instar larvaes of tea.Be placed in 25 ℃ of thermostatic chambers " Invest, Then Investigate " life and death borer population on the 6th.Carry out in 52 modes that connect system in 1 district.

Need to prove that compound uses above-claimed cpd (A) as a comparison.

The result of above-mentioned test, following compound has shown the dead worm rate more than 70% during for 1ppm in concentration, the sequence number of described compound is 6-72,6-80,6-90,6-271,6-349,6-366,6-367,6-426,6-427,6-1104,6-1106,6-1182,6-1260,6-1263,6-1358,6-1574,6-1577,6-1595,6-1596,6-1652,6-1654,6-1655,6-1672,6-1673,6-1674,6-1695,6-1730,6-1732,6-1733,6-1750,6-1751,6-1809,6-1811,6-1828,6-1829,6-1830,6-1851,7-90,7-348,7-366,7-382,7-389,7-444,7-502,7-504,7-505,7-523,7-1104,7-1106,7-1107,7-1124,7-1125,7-1260,7-1262,7-1263,7-1280,7-1281,7-1303,7-1358,7-1359,7-1574,7-1576,7-1577,7-1594,7-1595,7-1605,7-1616,7-1617,7-1652,7-1730,7-1732,7-1733,7-1750,7-1764,7-1773,7-1808,7-1809,7-1810,7-1811,7-1829,7-1851

Following compound has shown the dead worm rate more than 70% in concentration during for 10ppm, and the sequence number of described compound is 6-382,6-446,6-460,6-2110,7-424,7-538,7-1606.

On the other hand, compound (A) dead worm rate when concentration is 10ppm is below 50%.

＜test example 5 〉

Insecticidal test to bollworm (Helicoverpa armigera)

Dipping Caulis et Folium Brassicae capitatae blade (cabbage leaf disk) is 30 seconds in the soup that test compound is modulated to normality, and is air-dry.Add blade (leaf disk) in having laid 6 hole plastic cups of filter paper, 12 instar larvae is put in per 1 hole.Be placed in 25 ℃ of thermostatic chambers " Invest, Then Investigate " life and death borer population on the 3rd.Carry out in 52 modes that connect system in 1 district.

Need to prove that compound uses above-claimed cpd (A) as a comparison.

The result of above-mentioned test, following compound has shown the dead worm rate more than 70% in concentration during for 1ppm, and the sequence number of described compound is 6-72,6-80,6-90,6-271,6-347,6-348,6-349,6-366,6-367,6-382,6-389,6-426,6-427,6-446,6-449,6-460,6-503,6-504,6-505,6-522,6-523,6-524,6-538,6-1104,6-1106,6-1260,6-1262,6-1263,6-1281,6-1341,6-1358,6-1359,6-1574,6-1576,6-1577,6-1594,6-1595,6-1596,6-1652,6-1654,6-1655,6-1672,6-1673,6-1674,6-1695,6-1730,6-1732,6-1733,6-1750,6-1751,6-1808,6-1809,6-1811,6-1828,6-1829,6-1830,6-1851,6-2110,7-90,7-348,7-366,7-382,7-389,7-424,7-444,7-502,7-505,7-522,7-523,7-538,7-1106,7-1107,7-1125,7-1262,7-1263,7-1280,7-1303,7-1338,7-1358,7-1359,7-1574,7-1576,7-1577,7-1594,7-1595,7-1605,7-1606,7-1616,7-1617,7-1652,7-1730,7-1731,7-1732,7-1733,7-1750,7-1751,7-1764,7-1773,7-1808,7-1809,7-1810,7-1811,7-1829,7-1851.

In addition, the compound sequence number is that the compound of 7-1104 has shown the dead worm rate more than 70% during for 10ppm in concentration.

On the other hand, compound (A) dead worm rate when concentration is 10ppm is below 50%.

＜test example 6 〉

Insecticidal test to small brown rice planthopper (Laodelphaxstriatellus)

Preparation is modulated to the acetone soln of normality with test compound, and 2.5ml intersperses among on the rice seedling with this acetone soln, air-dry after, add and put into the diameter 3cm of water, the Glass tubing of high 13cm, put into small brown rice planthopper 3 instar larvaes and cover lid.Be placed in 25 ℃ of thermostatic chambers " Invest, Then Investigate " life and death borer population on the 6th.Carry out in 10 2 modes that connect system in 1 district.

The result of above-mentioned test, following compound has shown the dead worm rate more than 70% in concentration during for 100ppm, and the sequence number of described compound is 1-491,1-627,2-491,6-39,6-45,6-47,6-57,6-71,6-72,6-79,6-80,6-90,6-147,6-268,6-269,6-270,6-271,6-290,6-304,6-306,6-311,6-346,6-347,6-368,6-382,6-425,6-427,6-444,6-445,6-446,6-460,6-461,6-503,6-1104,6-1106,6-1107,6-1124,6-1126,6-1140,6-1147,6-1182,6-1183,6-1184,6-1185,6-1202,6-1203,6-1204,6-1218,6-1225,6-1260,6-1261,6-1262,6-1263,6-1280,6-1281,6-1282,6-1296,6-1303,6-1338,6-1339,6-1340,6-1341,6-1358,6-1359,6-1360,6-1374,6-1381,6-1574,6-1575,6-1576,6-1577,6-1594,6-1595,6-1596,6-1610,6-1617,6-1652,6-1653,6-1654,6-1655,6-1672,6-1673,6-1674,6-1688,6-1695,6-1730,6-1731,6-1732,6-1733,6-1734,6-1750,6-1751,6-1752,6-1754,6-1766,6-1773,6-1808,6-1809,6-1810,6-1811,6-1828,6-1829,6-1830,6-1851,6-2110,6-3348,6-3384,6-5903,6-5904,6-5905,6-5906,6-5907,6-5908,6-5909,6-5910,6-5911,6-5914,7-47,7-57,7-90,7-268,7-285,7-286,7-288,7-289,7-301,7-303,7-304,7-305,7-311,7-316,7-346,7-348,7-368,7-382,7-389,7-424,7-426,7-427,7-444,7-445,7-446,7-460,7-467,7-538,7-825,7-840,7-948,7-984,7-1104,7-1105,7-1106,7-1107,7-1124,7-1125,7-1126,7-1140,7-1147,7-1182,7-1183,7-1184,7-1185,7-1202,7-1203,7-1204,7-1218,7-1225,7-1260,7-1261,7-1262,7-1263,7-1280,7-1281,7-1282,7-1296,7-1303,7-1338,7-1339,7-1340,7-1341,7-1358,7-1359,7-1360,7-1374,7-1381,7-1417,7-1574,7-1575,7-1576,7-1577,7-1594,7-1595,7-1596,7-1605,7-1606,7-1608,7-1610,7-1616,7-1617,7-1638,7-1639,7-1645,7-1652,7-1672,7-1673,7-1730,7-1731,7-1732,7-1733,7-1750,7-1751,7-1752,7-1764,7-1766,7-1773,7-1794,7-1808,7-1809,7-1810,7-1811,7-1828,7-1829,7-1844,7-1851,7-3348,7-3369,7-5902,7-5903,7-5904,7-5906,7-5907,7-5909,7-5912,8-289,8-304,8-840,9-270,9-290,9-291,9-306,9-2164,9-2322,12-835,12-864.

＜test example 7 〉

Insecticidal test to housefly (Muscadomestica)

Preparation is modulated to the acetone soln of normality with test compound, and this acetone soln 1ml is splashed in the Petri dish of diameter 9cm, air-dry after, put into housefly female insect and cover lid.Be placed in 25 ℃ of thermostatic chambers " Invest, Then Investigate " life and death borer population on the 1st.Carry out in 52 modes that connect system in 1 district.

The result of above-mentioned test, following compound has shown the dead worm rate more than 70% in concentration during for 100ppm, and the sequence number of described compound is 1-1925,1-1968,6-39,6-47,6-72,6-272,6-293,6-346,6-347,6-348,6-366,6-368,6-382,6-389,6-426,6-427,6-428,6-450,6-452,6-453,6-460,6-503,6-504,6-505,6-522,6-523,6-524,6-538,6-1105,6-1107,6-1124,6-1125,6-1126,6-1147,6-1184,6-1204,6-1218,6-1260,6-1281,6-1338,6-1341,6-1358,6-1359,6-1360,6-1374,6-1575,6-1576,6-1577,6-1594,6-1596,6-1617,6-1652,6-1672,6-1673,6-1695,6-1730,6-1731,6-1732,6-1733,6-1734,6-1750,6-1751,6-1752,6-1773,6-1808,6-1809,6-1810,6-1811,6-1828,6-1829,6-1830,6-1851,6-2110,6-5905,7-39,7-57,7-90,7-268,7-346,7-348,7-349,7-366,7-367,7-368,7-382,7-389,7-424,7-428,7-444,7-446,7-449,7-504,7-522,7-538,7-1104,7-1105,7-1106,7-1107,7-1126,7-1262,7-1280,7-1282,7-1296,7-1303,7-1338,7-1340,7-1358,7-1359,7-1360,7-1381,7-1417,7-1574,7-1575,7-1576,7-1577,7-1596,7-1652,7-1731,7-1732,7-1733,7-1750,7-1752,7-1764,7-1766,7-1730,7-1773,7-1794,7-1808,7-1809,7-1810,7-1811,7-1828,7-1829,7-1851,9-2164,9-2322,11-777,11-835,12-777,12-835,12-864,17-1103,27-627.

＜test example 8 〉

Insecticidal test to Groton bug (Blattellagermanica)

Preparation is modulated to the acetone soln of normality with test compound, and this acetone soln 1ml is splashed in the Petri dish of diameter 9cm, air-dry after, put into Groton bug male insect and cover lid.Be placed in 25 ℃ of thermostatic chambers " Invest, Then Investigate " life and death borer population on the 1st.Carry out in 52 modes that connect system in 1 district.

The result of above-mentioned test, following compound has shown the dead worm rate more than 70% when concentration 100ppm, the sequence number of described compound is 1-1925,6-39,6-47,6-346,6-347,6-367,6-368,6-382,6-389,6-426,6-427,6-503,6-538,6-1105,6-1106,6-1107,6-1124,6-1125,6-1126,6-1147,6-1184,6-1204,6-1218,6-1280,6-1296,6-1338,6-1358,6-1359,6-1575,6-1576,6-1577,6-1594,6-1595,6-1596,6-1610,6-1617,6-1730,6-1731,6-1732,6-1733,6-1750,6-1751,6-1752,6-1773,6-1811,6-5905,7-57,7-268,7-305,7-347,7-349,7-367,7-382,7-389,7-424,7-444,7-446,7-502,7-505,7-538,7-1104,7-1105,7-1106,7-1107,7-1125,7-1126,7-1261,7-1262,7-1280,7-1282,7-1296,7-1303,7-1381,7-1574,7-1575,7-1576,7-1577,7-1594,7-1595,7-1596,7-1617,7-1731,7-1732,7-1733,7-1750,7-1752,7-1766,7-1773,7-1851.

＜test example 9 〉

The insecticidal test of player whose turn comes next mosquito (Culex pipiens molestus) over the ground

Test compound is modulated to the acetone soln of normality, above-mentioned acetone soln 1ml is splashed in the Petri dish of diameter 9cm, air-dry after, put into ground player whose turn comes next mosquito adult and cover lid.Be placed in 25 ℃ of thermostatic chambers, handle " Invest, Then Investigate " life and death borer population on the 1st.Carry out in 52 modes that connect system in 1 district.

The result of above-mentioned test, compound sequence number are that the compound of 7-424,7-1574,7-1577,7-1730,7-1732,7-1733 has shown the dead worm rate more than 70% during for 1000ppm in concentration.

＜test example 10 〉

Insecticidal test to Taiwan formosanes (Coptotermesformosanus)

Preparation is modulated to the acetone soln of normality with test compound, this acetone soln 20 μ l is splashed in the filter paper that adds the diameter 2.6mm in the polypropylene tube, air-dry after, add the water of 20 μ l, put into Taiwan formosanes and cover lid.Be placed in 28 ℃ of thermostatic chambers, handle " Invest, Then Investigate " life and death borer population on the 5th.Carry out in 10 2 modes that connect system in 1 district.

The result of above-mentioned test, following compound has shown the dead worm rate more than 70% in concentration during for 30ppm, and the sequence number of described compound is 6-460,6-1260,6-1652,7-268,7-424,7-1104,7-1574,7-1577,7-1730,7-1732,7-1733.

Utilizability on the industry

According to the present invention, can provide novel amide derivatives. This amide derivatives shows superior efficacy in the Pesticidal activity, the value height on the industry.

Claims (19)

1. the amide derivatives of following general formula (1) expression,

In the general formula (1),

A represents carbon atom, Sauerstoffatom, nitrogen-atoms, oxidized nitrogen-atoms or sulphur atom,

Necessary non-metallic atom group when K is illustrated in 2 carbon atoms with A and A bonding and forms cyclic linker group, described cyclic linker group is from benzene, pyridine, N-pyridine oxide, pyrimidine, pyrazine, pyridazine, triazine, pyrroles, pyrazoles, imidazoles, oxazole, isoxazole, thiazole, isothiazole, furans, thiophene, oxadiazole, thiadiazoles or triazole;

X represents hydrogen atom, halogen atom, the C1-C6 alkyl, the C1-C6 haloalkyl, the C3-C9 cycloalkyl, the C3-C9 halogenated cycloalkyl, the C2-C6 alkenyl, the C2-C6 halogenated alkenyl, the C2-C6 alkynyl, C2-C6 halo alkynyl, the C1-C6 alkoxyl group, the C1-C6 halogenated alkoxy, the C2-C6 alkenyl oxy, the C2-C6 halogenated alkenyl oxy, C2-C6 alkynyloxy base, C2-C6 halo alkynyloxy base, the C3-C9 cycloalkyloxy, C3-C9 halo cycloalkyloxy, C1-C6 alkyl sulfenyl, C1-C6 haloalkyl sulfenyl, the C1-C6 alkyl sulphinyl, C1-C6 haloalkyl sulfinyl, the C1-C6 alkyl sulphonyl, the C1-C6 halogenated alkyl sulfonyl, C1-C6 alkyl sulphonyl oxygen base, C1-C6 halogenated alkyl sulfonyl oxygen base, the C2-C7 alkyl-carbonyl, the C2-C7 halogenated alkyl carbonyl, the C3-C7 alkenyl carbonyl, C3-C7 halogenated alkenyl carbonyl, C3-C7 alkynyl carbonyl, C3-C7 halo alkynyl carbonyl, the C4-C10 naphthene base carbonyl, C4-C10 halogenated cycloalkyl carbonyl, C2-C7 alkyl-carbonyl oxygen base, C2-C7 halogenated alkyl carbonyl oxygen base, aryl carbonyl oxygen base, the C2-C7 alkoxy carbonyl, the C2-C7 halo alkoxy carbonyl, C3-C7 alkenyl oxy carbonyl, C3-C7 halogenated alkenyl oxy carbonyl, C3-C7 alkynyloxy base carbonyl, C3-C7 halo alkynyloxy base carbonyl, C4-C10 cycloalkyl oxy carbonyl, C4-C10 halogenated cycloalkyl oxygen base carbonyl, the C2-C7 alkyl-carbonyl-amino, C2-C7 halogenated alkyl carbonyl amino, the C2-C7 alkoxycarbonyl amino, C2-C7 halo alkoxy carbonyl amino, the C2-C7 alkoxy-carbonyl oxy, C2-C7 halo alkoxy carbonyl oxygen base, aryl-amino-carbonyl, amino, formamyl, cyano group, hydroxyl, Pentafluorosulfanyl, the C1-C6 alkylamino, C1-C6 haloalkyl amino, the C2-C6 alkenyl amino, C2-C6 halogenated alkenyl amino, C2-C6 alkynyl amino, C2-C6 halo alkynyl amino, the C3-C9 cycloalkyl amino, C3-C9 halogenated cycloalkyl amino, the C2-C7 alkyl amino-carbonyl, C2-C7 haloalkyl aminocarboxyl, C3-C7 alkenyl amino carbonyl, C3-C7 halogenated alkenyl aminocarboxyl, C3-C7 alkynyl aminocarboxyl, C3-C7 halo alkynyl aminocarboxyl, C4-C10 cycloalkyl amino carbonyl, C4-C10 halogenated cycloalkyl aminocarboxyl, phenyl, or heterocyclic radical, when having a plurality of X, each X can be same to each other or different to each other;

N represents 0～4 integer;

T represents-C (=G ₁)-Q ₁, or-C (=G ₁)-G ₂Q ₂

G ₁And G ₂Represent Sauerstoffatom or sulphur atom respectively independently,

Q ₁And Q ₂Expression:

Hydrogen atom,

The C1-C6 alkyl,

The C1-C6 haloalkyl,

The C2-C6 alkenyl,

The C2-C6 halogenated alkenyl,

The C2-C6 alkynyl,

C2-C6 halo alkynyl,

The C3-C9 cycloalkyl,

The C3-C9 halogenated cycloalkyl,

Benzyl,

Can have substituent phenyl,

Naphthyl,

Maybe can have substituent heterocyclic radical;

Y ₁And Y ₅Represent halogen atom, C1-C6 halogenated alkoxy or C1-C3 haloalkyl respectively independently,

Y ₂And Y ₄Represent hydrogen atom, halogen atom or C1-C4 alkyl respectively independently,

Y ₃Expression C2-C5 haloalkyl;

Need to prove Q ₁And Q ₂In, the substituting group that can have substituent phenyl and can have a substituent heterocyclic radical represents to be selected from the substituting group more than 1 in the following radicals, described group is: halogen atom, the C1-C6 alkyl, the C1-C6 haloalkyl, the C3-C9 cycloalkyl, the C3-C9 halogenated cycloalkyl, the C2-C6 alkenyl, the C2-C6 halogenated alkenyl, the C2-C6 alkynyl, C2-C6 halo alkynyl, the C1-C6 alkoxyl group, the C1-C6 halogenated alkoxy, the C2-C6 alkenyl oxy, the C2-C6 halogenated alkenyl oxy, C2-C6 alkynyloxy base, C2-C6 halo alkynyloxy base, the C3-C9 cycloalkyloxy, C3-C9 halo cycloalkyloxy, C1-C6 alkyl sulfenyl, C1-C6 haloalkyl sulfenyl, the C1-C6 alkyl sulphinyl, C1-C6 haloalkyl sulfinyl, the C1-C6 alkyl sulphonyl, the C1-C6 halogenated alkyl sulfonyl, the C2-C7 alkyl-carbonyl, the C2-C7 halogenated alkyl carbonyl, the C3-C7 alkenyl carbonyl, C3-C7 halogenated alkenyl carbonyl, C3-C7 alkynyl carbonyl, C3-C7 halo alkynyl carbonyl, the C4-C10 naphthene base carbonyl, C4-C10 halogenated cycloalkyl carbonyl, C2-C7 alkyl-carbonyl oxygen base, C2-C7 halogenated alkyl carbonyl oxygen base, C1-C6 alkyl sulphonyl oxygen base, C1-C6 halogenated alkyl sulfonyl oxygen base, the C2-C7 alkoxy carbonyl, the C2-C7 halo alkoxy carbonyl, C3-C7 alkenyl oxy carbonyl, C3-C7 halogenated alkenyl oxy carbonyl, C3-C7 alkynyloxy base carbonyl, C3-C7 halo alkynyloxy base carbonyl, C4-C10 cycloalkyl oxy carbonyl, C4-C10 halogenated cycloalkyl oxygen base carbonyl, the C2-C7 alkyl-carbonyl-amino, C2-C7 halogenated alkyl carbonyl amino, the C2-C7 alkoxycarbonyl amino, C2-C7 halo alkoxy carbonyl amino, the C1-C6 alkylamino, C1-C6 haloalkyl amino, the C2-C6 alkenyl amino, C2-C6 halogenated alkenyl amino, C2-C6 alkynyl amino, C2-C6 halo alkynyl amino, the C3-C9 cycloalkyl amino, C3-C9 halogenated cycloalkyl amino, the C2-C7 alkyl amino-carbonyl, C2-C7 haloalkyl aminocarboxyl, C3-C7 alkenyl amino carbonyl, C3-C7 halogenated alkenyl aminocarboxyl, C3-C7 alkynyl aminocarboxyl, C3-C7 halo alkynyl aminocarboxyl, C4-C10 cycloalkyl amino carbonyl, C4-C10 halogenated cycloalkyl aminocarboxyl, amino, formamyl, cyano group, nitro, hydroxyl, Pentafluorosulfanyl, can have substituent phenyl, and can have substituent heterocyclic radical, when having 2 above substituting groups, each substituting group can be the same or different;

And then, X, Q ₁, and Q ₂In heterocyclic radical represent pyridyl, N-pyridine oxide base, pyrimidyl, pyrazinyl, pyridazinyl, furyl, thienyl, oxazolyl, isoxazolyl, oxadiazole base, thiazolyl, isothiazolyl, thiadiazolyl group, pyrryl, imidazolyl, triazolyl, pyrazolyl or tetrazyl;

G ₃Expression Sauerstoffatom or sulphur atom;

R ₁And R ₂Represent hydrogen atom respectively independently; Sauerstoffatom; halogen atom; hydroxyl; nitro; nitroso-group; trimethyl silyl; t-butyldimethylsilyl; cyano group; amino; can have substituent C1-C6 alkyl; can have substituent C1-C6 haloalkyl; the C2-C7 alkyl-carbonyl; the C2-C7 halogenated alkyl carbonyl; can have substituent C2-C6 alkenyl; can have substituent C2-C6 halogenated alkenyl; can have substituent C2-C6 alkynyl; can have substituent C2-C6 halo alkynyl; the C2-C7 alkoxy carbonyl; the C2-C7 halo alkoxy carbonyl; C3-C7 alkenyl oxy carbonyl; C3-C7 halogenated alkenyl oxy carbonyl; C3-C7 alkynyloxy base carbonyl; C3-C7 halo alkynyloxy base carbonyl; phenyloxycarbonyl; the C2-C7 alkyl amino-carbonyl; C2-C7 haloalkyl aminocarboxyl; C2-C7 alkyl-carbonyl oxygen base; C2-C7 halogenated alkyl carbonyl oxygen base; benzoyl; the C1-C6 alkoxyl group; the C1-C6 halogenated alkoxy; C1-C6 alkyl sulfenyl; C1-C6 haloalkyl sulfenyl; the C1-C6 alkyl sulphinyl; C1-C6 haloalkyl sulfinyl; the C1-C6 alkyl sulphonyl; the C1-C6 halogenated alkyl sulfonyl; benzenesulfonyl; the benzyl alkylsulfonyl; benzyl; or-C (=O) C (=O) R ₇, in the formula, R ₇Expression C1-C6 alkyl, C1-C6 haloalkyl, C1-C6 alkoxyl group or C1-C6 halogenated alkoxy;

But the amide derivatives that does not comprise above-mentioned general formula (1) expression is any one the situation in following (A)～(I):

(A) in the above-mentioned general formula (1), K necessary non-metallic atom group when forming the cyclic linker group from pyridine at 2 carbon atoms, Y with A and A bonding ₁Be halogen atom, Y ₅Be the C1-C6 halogenated alkoxy, T is-C (=G ₁)-Q ₁

(B) in the above-mentioned general formula (1), K is necessary non-metallic atom group when 2 carbon atoms with A and A bonding form cyclic linker group, described cyclic linker group is from pyrroles, pyrazoles, imidazoles, oxazole, isoxazole, thiazole, isothiazole, furans, thiophene, oxadiazole, thiadiazoles or triazole, Y ₁And Y ₅Be halogen atom independently respectively, T is-C (=G ₁)-G ₂Q ₂

(C) in the above-mentioned general formula (1), K is necessary non-metallic atom group when 2 carbon atoms with A and A bonding form cyclic linker group, described cyclic linker group is from pyrroles, pyrazoles, imidazoles, oxazole, isoxazole, thiazole, isothiazole, furans, thiophene, oxadiazole, thiadiazoles or triazole, and T is-C (=G ₁)-Q ₁, Y ₁Be halogen atom, Y ₅Be halogen atom or halogenated alkoxy;

(D) amide compound of following general formula (2) expression,

In the general formula (2), Y ₂～Y ₄, Q ₁, G ₁, G ₃, R ₁, and R ₂With the Y in the general formula (1) ₂～Y ₄, Q ₁, G ₁, G ₃, R ₁, and R ₂The difference synonym, Y ₁Be halogen atom, Y ₅Be the C1-C2 halogenated alkoxy;

(E) in the above-mentioned general formula (2), Y ₁And Y ₅Be halogen atom, X is hydrogen atom, Y ₃Be the C2-C3 haloalkyl;

(F) amide derivatives of following general formula (3) expression,

In the general formula (3), Y ₁And Y ₅Be halogen atom independently respectively, X ₁And X ₃Be hydrogen atom or fluorine atom independently respectively, Q ₁With the Q in the general formula (1) ₁Synonym, R ₁Be hydrogen atom or methyl, Y ₃Be the C3-C4 perfluoroalkyl;

(G) amide derivatives of following general formula (4) expression,

In the general formula (4), X ₁Be fluorine atom, X ₂, X ₃, and X ₄Be hydrogen atom, Y ₁And Y ₅Differ from one another, be bromine atoms or trifluoromethoxy, Y ₂And Y ₄Be hydrogen atom, Y ₃Be seven fluorine sec.-propyls, Q ₁Be phenyl or 2-chloropyridine-3-base, R ₁And R ₂Differ from one another, be hydrogen atom or methyl,

Perhaps X ₁Be fluorine atom, X ₂, X ₃, and X ₄Be hydrogen atom, Y ₁And Y ₅Be bromine atoms, Y ₂And Y ₄Be hydrogen atom, Y ₃Be pentafluoroethyl group, Q ₁Be 2-fluorophenyl, R ₁And R ₂Be hydrogen atom or methyl independently respectively;

(H) amide derivatives of following general formula (5) expression,

In the general formula (5), Y ₁And Y ₅Be halogen atom independently respectively, X ₁Be hydrogen atom or fluorine atom, Q ₂Be 2,2,2-three chloroethyls and 3,3,3-three fluoro-n-propyl group, Y ₃Be the C2-C4 haloalkyl;

(I) amide derivatives of following general formula (6) expression,

In the general formula (6), Y ₁And Y ₅Be halogen atom independently respectively, Q ₂With the Q in the general formula (1) ₂Synonym, R ₁Be hydrogen atom or methyl, Y ₃Be the C3-C4 haloalkyl.

2. amide compound as claimed in claim 1, with following general formula (7) expression,

In the general formula (7), n is 4, X, Y ₁～Y ₅, Q ₁, G ₁, G ₃, R ₁, and R ₂With X, the Y in the general formula (1) ₁～Y ₅, Q ₁, G ₁, G ₃, R ₁, and R ₂The difference synonym.

3. amide derivatives as claimed in claim 2, with following general formula (8) expression,

In the general formula (8), Q ₁Expression can have substituent phenyl maybe can have substituent pyridyl;

X ₁, X ₂, X ₃, and X ₄Represent hydrogen atom or fluorine atom respectively independently;

R ₁And R ₂Represent hydrogen atom or C1-C3 alkyl respectively independently;

Y ₁And Y ₅Represent halogen atom, C1-C3 halogenated alkoxy or C1-C3 haloalkyl respectively independently, Y ₂And Y ₄Represent hydrogen atom, halogen atom or C1-C4 alkyl, Y respectively independently ₃Expression C3-C4 haloalkyl;

Wherein, Y ₁And Y ₅When being halogen atom simultaneously, X ₁And X ₂In at least one side be fluorine atom; In addition, Y ₁Or Y ₅During for the C1-C3 halogenated alkoxy, X ₂Be fluorine atom.

4. amide derivatives as claimed in claim 3, wherein,

In the above-mentioned general formula (8), Y ₃Be the C3-C4 perfluoroalkyl.

5. amide derivatives as claimed in claim 4, wherein,

In the above-mentioned general formula (8), Y ₁And Y ₅Be chlorine atom, bromine atoms, iodine atom, trifluoromethoxy, trifluoromethyl or pentafluoroethyl group independently respectively, Y ₂And Y ₄Be hydrogen atom.

6. amide derivatives as claimed in claim 5, wherein,

In the above-mentioned general formula (8), X ₁And X ₂Be hydrogen atom or fluorine atom independently respectively, X ₃And X ₄Be hydrogen atom.

7. amide derivatives as claimed in claim 6, wherein,

In the above-mentioned general formula (8), R ₁And R ₂Be hydrogen atom or methyl independently respectively.

8. amide derivatives as claimed in claim 7, wherein,

In the above-mentioned general formula (8), Q ₁For having substituent phenyl or the pyridyl that is selected from halogen atom, C1 haloalkyl, nitro and the cyano group.

9. amide derivatives as claimed in claim 8, wherein,

In the above-mentioned general formula (8), Q ₁In above-mentioned substituent quantity be 1 or 2.

10. amide derivatives as claimed in claim 2, wherein,

In the above-mentioned general formula (7), Y ₃Be C2-C4 perfluoroalkyl, Y ₂And Y ₄Be hydrogen atom, Y ₁And Y ₅Be halogen atom or C1-C3 haloalkyl, Y ₁And Y ₅In the either party be the C1-C3 haloalkyl.

11. amide derivatives as claimed in claim 10, wherein,

In the above-mentioned general formula (7), 4 X are hydrogen atom, halogen atom or cyano group respectively independently.

12. amide derivatives as claimed in claim 1, with following general formula (9) expression,

In the general formula (9), n is 4, X, Y ₁～Y ₅, Q ₂, G ₁～G ₃, R ₁, and R ₂With X, the Y in the general formula (1) ₁～Y ₅, Q ₂, G ₁～G ₃, R ₁, and R ₂The difference synonym.

13. amide derivatives as claimed in claim 12, in the above-mentioned general formula (9), Y ₃Be C2-C4 perfluoroalkyl, Y ₂And Y ₄Be hydrogen atom, Y ₁And Y ₅Be halogen atom or C1-C3 haloalkyl, Y ₁, Y ₅In the either party be the C1-C3 haloalkyl.

14. amide derivatives as claimed in claim 13, in the above-mentioned general formula (9), 4 X are hydrogen atom, halogen atom or cyano group respectively independently.

15. amide derivatives as claimed in claim 1, in the above-mentioned general formula (1), K is necessary non-metallic atom group when 2 carbon atoms with A and A bonding form cyclic linker group, and described cyclic linker group is from pyridine, N-pyridine oxide, pyrimidine, pyrazine, pyridazine, triazine, pyrroles, pyrazoles, imidazoles, oxazole, isoxazole, thiazole, isothiazole, furans, thiophene, oxadiazole, thiadiazoles or triazole.

16. amide derivatives as claimed in claim 15, wherein,

In the above-mentioned general formula (1), Y ₃Be C2-C4 perfluoroalkyl, Y ₂And Y ₄Be hydrogen atom, Y ₁And Y ₅Be halogen atom or C1-C3 haloalkyl, Y ₁And Y ₅In the either party be the C1-C3 haloalkyl.

17. amide derivatives as claimed in claim 16, wherein,

In the above-mentioned general formula (1), K is necessary non-metallic atom group when 2 carbon atoms with A and A bonding form cyclic linker group, and described cyclic linker group is from pyridine, N-pyridine oxide, pyrroles, thiazole, furans or thiophene.

18. a noxious organism control agent, contain claim 1 to the claim 17 at least a kind in each described amide derivatives as effective constituent.

19. the method for control of a harmful organism is used for harmful organism with the described noxious organism control agent of claim 18.