CL2018002930A1 - (+)-azasetron para uso en el tratamiento de desórdenes de oído. - Google Patents
(+)-azasetron para uso en el tratamiento de desórdenes de oído.Info
- Publication number
- CL2018002930A1 CL2018002930A1 CL2018002930A CL2018002930A CL2018002930A1 CL 2018002930 A1 CL2018002930 A1 CL 2018002930A1 CL 2018002930 A CL2018002930 A CL 2018002930A CL 2018002930 A CL2018002930 A CL 2018002930A CL 2018002930 A1 CL2018002930 A1 CL 2018002930A1
- Authority
- CL
- Chile
- Prior art keywords
- azasetron
- treatment
- ear disorders
- disorders
- ear
- Prior art date
Links
- 229950005951 azasetron Drugs 0.000 title abstract 2
- 208000032625 disorder of ear Diseases 0.000 title abstract 2
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/538—1,4-Oxazines, e.g. morpholine ortho- or peri-condensed with carbocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Zoology (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
LA PRESENTE INVENCIÓN SE REFIERE A (+)-AZASETRÓN, O UNA SAL Y/O SOLVATO FARMACÉUTICAMENTE ACEPTABLE DEL MISMO, PARA TRATAR TRASTORNOS DEL OÍDO.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201662322690P | 2016-04-14 | 2016-04-14 | |
EP16180192 | 2016-07-19 |
Publications (1)
Publication Number | Publication Date |
---|---|
CL2018002930A1 true CL2018002930A1 (es) | 2019-02-15 |
Family
ID=65588799
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CL2018002930A CL2018002930A1 (es) | 2016-04-14 | 2018-10-12 | (+)-azasetron para uso en el tratamiento de desórdenes de oído. |
Country Status (18)
Country | Link |
---|---|
US (2) | US11612605B2 (es) |
EP (1) | EP4335508A3 (es) |
JP (1) | JP7158723B2 (es) |
CN (1) | CN109310698B (es) |
AU (1) | AU2023202897B2 (es) |
CL (1) | CL2018002930A1 (es) |
DK (1) | DK3442537T3 (es) |
ES (1) | ES2975016T3 (es) |
FI (1) | FI3442537T3 (es) |
HR (1) | HRP20240453T1 (es) |
HU (1) | HUE066000T2 (es) |
IL (1) | IL262305B (es) |
MX (1) | MX384045B (es) |
NZ (1) | NZ747201A (es) |
PL (1) | PL3442537T3 (es) |
RS (1) | RS65379B1 (es) |
SI (1) | SI3442537T1 (es) |
ZA (1) | ZA201806894B (es) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP6994765B2 (ja) * | 2015-05-18 | 2022-02-10 | センソリオン | 難聴の処置のためのセトロンファミリーのカルシニューリン阻害剤 |
Family Cites Families (23)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4695578A (en) | 1984-01-25 | 1987-09-22 | Glaxo Group Limited | 1,2,3,9-tetrahydro-3-imidazol-1-ylmethyl-4H-carbazol-4-ones, composition containing them, and method of using them to treat neuronal 5HT function disturbances |
US5360800A (en) | 1987-09-03 | 1994-11-01 | Glaxo Group Limited | Tetrahydro-1H-pyrido[4,3-b]indol-1-one derivatives |
CA1304082C (en) | 1987-10-22 | 1992-06-23 | Tetsuya Tahara | Benzoxazine compounds and pharmaceutical use thereof |
GB9423511D0 (en) | 1994-11-22 | 1995-01-11 | Glaxo Wellcome Inc | Compositions |
GB0009914D0 (en) | 2000-04-20 | 2000-06-07 | Metris Therapeutics Limited | Device |
GB0104554D0 (en) | 2001-02-23 | 2001-04-11 | Glaxo Group Ltd | New uses |
US20030044356A1 (en) | 2001-04-20 | 2003-03-06 | Jin Auh | Composition for nasal solution sprays having effective component of 1,2,3,9-tetrahydro-9-methyl-3-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-carbazol-4-one) |
WO2003071986A2 (en) | 2002-02-22 | 2003-09-04 | Control Delivery Systems, Inc. | Method for treating otic disorders |
GB0213869D0 (en) | 2002-06-17 | 2002-07-31 | Arakis Ltd | The treatment of pain |
PL378369A1 (pl) | 2003-01-13 | 2006-04-03 | Dynogen Pharmaceuticals, Inc. | Sposób leczenia mdłości, wymiotów, nudności lub ich dowolnej kombinacji |
TWI355936B (en) | 2003-02-18 | 2012-01-11 | Helsinn Healthcare Sa | Uses of palonosetron hydrochloride |
US20040204466A1 (en) | 2003-04-14 | 2004-10-14 | Orchid Chemicals And Pharmaceuticals Ltd. | Treatment of bronchial asthma using 5-HT3 receptor antagonists |
US20070265329A1 (en) | 2006-05-12 | 2007-11-15 | Devang Shah T | Methods for the prevention of acute and delayed chemotherapy-induced nausea and vomiting (CINV) |
EP2244735A4 (en) | 2007-10-02 | 2011-02-23 | Avaxia Biologics Inc | ANTIBODY THERAPY FOR USE IN THE DIGESTIVE TUBE |
MX2011000545A (es) | 2008-07-14 | 2011-02-24 | Otonomy Inc | Composiciones de liberacion controlada para la modulacion de apoptosis y metodos para el tratamiento de trastornos oticos. |
EP2253316B1 (en) * | 2009-05-20 | 2013-08-14 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Serotonin 5-HT3 receptor antagonists for use in the treatment or prevention of an inner ear pathology with vestibular deficits |
KR101779991B1 (ko) | 2009-05-20 | 2017-09-19 | 인쎄름 (엥스띠뛰 나씨오날 드 라 쌍떼 에 드 라 흐쉐르슈 메디깔) | 병소성 전정 질환을 치료하기 위한 세로토닌 5-ht3 수용체 길항제의 용도 |
CN101786963B (zh) | 2010-03-03 | 2013-05-08 | 山东众诚药业股份有限公司 | 阿扎司琼中间体的合成方法 |
JP2015511242A (ja) | 2012-02-23 | 2015-04-16 | インセルム(インスティチュート ナショナル デ ラ サンテ エ デ ラリシェルシェ メディカル) | 病変性前庭障害の治療に使用するカルシニューリン阻害剤 |
JP6289460B2 (ja) | 2012-07-16 | 2018-03-07 | コーネル ユニヴァーシティー | 難聴を治療するためのニコチンアミドリボシド |
CN105682639B (zh) * | 2013-07-31 | 2021-02-05 | 兰色制药医药工业股份有限公司 | 口腔可分散膜 |
CN104557906A (zh) | 2015-01-21 | 2015-04-29 | 扬子江药业集团四川海蓉药业有限公司 | 一种盐酸阿扎司琼的制备方法 |
JP6994765B2 (ja) | 2015-05-18 | 2022-02-10 | センソリオン | 難聴の処置のためのセトロンファミリーのカルシニューリン阻害剤 |
-
2017
- 2017-04-14 DK DK17717441.4T patent/DK3442537T3/da active
- 2017-04-14 CN CN201780036585.4A patent/CN109310698B/zh active Active
- 2017-04-14 NZ NZ747201A patent/NZ747201A/en unknown
- 2017-04-14 SI SI201731500T patent/SI3442537T1/sl unknown
- 2017-04-14 HU HUE17717441A patent/HUE066000T2/hu unknown
- 2017-04-14 ES ES17717441T patent/ES2975016T3/es active Active
- 2017-04-14 PL PL17717441.4T patent/PL3442537T3/pl unknown
- 2017-04-14 EP EP23220392.7A patent/EP4335508A3/en not_active Withdrawn
- 2017-04-14 FI FIEP17717441.4T patent/FI3442537T3/fi active
- 2017-04-14 JP JP2018553953A patent/JP7158723B2/ja active Active
- 2017-04-14 RS RS20240412A patent/RS65379B1/sr unknown
- 2017-04-14 US US16/093,911 patent/US11612605B2/en active Active
- 2017-04-14 HR HRP20240453TT patent/HRP20240453T1/hr unknown
- 2017-04-14 MX MX2018012587A patent/MX384045B/es unknown
-
2018
- 2018-10-11 IL IL262305A patent/IL262305B/en unknown
- 2018-10-12 CL CL2018002930A patent/CL2018002930A1/es unknown
- 2018-10-16 ZA ZA2018/06894A patent/ZA201806894B/en unknown
-
2023
- 2023-03-13 US US18/182,511 patent/US20230226071A1/en active Pending
- 2023-05-09 AU AU2023202897A patent/AU2023202897B2/en active Active
Also Published As
Publication number | Publication date |
---|---|
RS65379B1 (sr) | 2024-04-30 |
MX2018012587A (es) | 2019-03-07 |
AU2023202897A1 (en) | 2023-05-25 |
IL262305A (en) | 2018-11-29 |
ZA201806894B (en) | 2023-03-29 |
MX384045B (es) | 2025-03-14 |
ES2975016T3 (es) | 2024-07-02 |
SI3442537T1 (sl) | 2024-05-31 |
HRP20240453T1 (hr) | 2024-06-21 |
HUE066000T2 (hu) | 2024-06-28 |
PL3442537T3 (pl) | 2024-07-15 |
EP4335508A3 (en) | 2024-07-10 |
DK3442537T3 (da) | 2024-03-25 |
JP2019513780A (ja) | 2019-05-30 |
FI3442537T3 (fi) | 2024-04-04 |
NZ747201A (en) | 2023-02-24 |
CN109310698B (zh) | 2021-12-24 |
EP4335508A2 (en) | 2024-03-13 |
JP7158723B2 (ja) | 2022-10-24 |
US20190083503A1 (en) | 2019-03-21 |
US20230226071A1 (en) | 2023-07-20 |
AU2023202897B2 (en) | 2025-01-30 |
IL262305B (en) | 2022-03-01 |
US11612605B2 (en) | 2023-03-28 |
CN109310698A (zh) | 2019-02-05 |
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