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CL2012000314A1 - Compuesto derivado de n1-sustituido-5-fluoro-2-oxopirimidina-1(2h)-carboxamida; composición que lo comprende; y método para el control y prevención de un ataque fúngico en una planta. - Google Patents

Compuesto derivado de n1-sustituido-5-fluoro-2-oxopirimidina-1(2h)-carboxamida; composición que lo comprende; y método para el control y prevención de un ataque fúngico en una planta.

Info

Publication number
CL2012000314A1
CL2012000314A1 CL2012000314A CL2012000314A CL2012000314A1 CL 2012000314 A1 CL2012000314 A1 CL 2012000314A1 CL 2012000314 A CL2012000314 A CL 2012000314A CL 2012000314 A CL2012000314 A CL 2012000314A CL 2012000314 A1 CL2012000314 A1 CL 2012000314A1
Authority
CL
Chile
Prior art keywords
substituted
alkyl
oxopyrimidine
carboxamide
fluoro
Prior art date
Application number
CL2012000314A
Other languages
English (en)
Inventor
Timothy Boebel
Kristy Bryan
Beth Lorsbach
W Owen
Mark Pobanz
Scott Thornburgh
Jeffery Webster
Chenglin Yao
Timothy Martin
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535293&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2012000314(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Publication of CL2012000314A1 publication Critical patent/CL2012000314A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/16—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof the nitrogen atom being part of a heterocyclic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/20—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D239/22—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to ring carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

LA PRESENTE INVENCIÓN SE REFIERE A COMPUESTOS DERIVADOS DE N1-SUSTITUIDO-5-FLUORO-2-OXOPIRIMIDINA-1(2H)-CARBOXAMIDA DE FORMULA I:<br /> EN DONDE; R1 ES H O BENCILO PUEDE ESTAR OPCIONALMENTE SUSTITUIDO CON 1 A 3 R5, R2 ES H O C1-C6 ALQUILO; ALTERNATIVAMENTE, R1 Y R2 SE PUEDEN TOMAR JUNTOS PARA FORMAR=CR11N(R12)R13, R3 ES -C(=O)OR8 O -C(=S)OR8; R5 ES INEPENDIENTEMENTE HALOGENO, C1-C6 ALQUILO O C1-C6 ALCOXI; R8 ES C1-C6 ALQUILO, C2-C6 ALQUELINO, C1-C6 HALOALQUILO, C1-C6 ALCOXIALQUILO, -(CH2)2OH2(C6H5), FENILO O BENCILO EN DONDE CADA UNO DE FENILO O BENCILO PUEDEN ESTAR OPCIONALMENTE SUSTITUIDOS CON 1 A 3 R5, O CON NAFTILO OPCIONALMENTE SUSTITUIDO CON 1 A 3 R5, R11 ES C1-C4 ALQUILO; Y R13 ES C1-C4 ALQUILO. COMPOSICION QUE LO COMPRENDE Y METODO PARA EL CONTROL Y PREVENCION DE UN ATAQUE FUNGICO EN UNA PLANTA.
CL2012000314A 2009-08-07 2012-02-06 Compuesto derivado de n1-sustituido-5-fluoro-2-oxopirimidina-1(2h)-carboxamida; composición que lo comprende; y método para el control y prevención de un ataque fúngico en una planta. CL2012000314A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US23223209P 2009-08-07 2009-08-07

Publications (1)

Publication Number Publication Date
CL2012000314A1 true CL2012000314A1 (es) 2012-10-05

Family

ID=43535293

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2012000314A CL2012000314A1 (es) 2009-08-07 2012-02-06 Compuesto derivado de n1-sustituido-5-fluoro-2-oxopirimidina-1(2h)-carboxamida; composición que lo comprende; y método para el control y prevención de un ataque fúngico en una planta.

Country Status (29)

Country Link
US (1) US8318758B2 (es)
EP (1) EP2462133B1 (es)
JP (1) JP5818791B2 (es)
KR (1) KR101792286B1 (es)
CN (1) CN102548979B (es)
AU (1) AU2010279408B2 (es)
BR (1) BR112012002807B1 (es)
CA (1) CA2769251C (es)
CL (1) CL2012000314A1 (es)
CO (1) CO6491089A2 (es)
CR (1) CR20120033A (es)
DK (1) DK2462133T3 (es)
EA (1) EA022930B1 (es)
EC (1) ECSP12011651A (es)
ES (1) ES2506169T3 (es)
HK (1) HK1172892A1 (es)
HN (1) HN2012000261A (es)
IL (1) IL217954A (es)
IN (1) IN2012DN00695A (es)
MX (1) MX2012001623A (es)
NI (1) NI201200019A (es)
NZ (1) NZ597638A (es)
PE (1) PE20120689A1 (es)
PL (1) PL2462133T3 (es)
PT (1) PT2462133E (es)
RS (1) RS53658B1 (es)
UA (1) UA106086C2 (es)
WO (1) WO2011017544A1 (es)
ZA (1) ZA201305992B (es)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2769073C (en) * 2009-08-07 2018-07-24 Dow Agrosciences Llc N1-sulfonyl-5-fluoropyrimidinone derivatives
AU2013370490B2 (en) 2012-12-28 2018-05-10 Adama Makhteshim Ltd. N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2H)-carboxamide derivatives
JP6336480B2 (ja) * 2012-12-28 2018-06-06 アダマ・マクテシム・リミテッド １−（置換ベンゾイル）−５−フルオロ−４−イミノ−３−メチル−３，４−ジヒドロピリミジン−２（１ｈ）−オンの誘導体
RU2638556C2 (ru) 2012-12-28 2017-12-14 Адама Мактешим Лтд. Производные n-(замещенного)-5-фтор-4-имино-3-метил-2-оксо-3,4-дигидропиримидин-1(2н)-карбоксилата
RU2644014C2 (ru) 2012-12-31 2018-02-07 Адама Мактешим Лтд. Производные 3-алкил-5-фтор-4-замещенного-имино-3,4-дигидропиримидин-2(н)-она в качестве фунгицидов
US20150183750A1 (en) 2013-12-31 2015-07-02 Dow Agrosciences Llc 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1-(arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
AU2014373850A1 (en) 2013-12-31 2016-08-11 Adama Makhteshim Ltd. Synergistic fungicidal mixtures and compositions for fungal control
WO2016040193A1 (en) 2014-09-08 2016-03-17 Samumed, Llc 3-(1h-imidazo[4,5-c]pyridin-2-yl)-1h-pyrazolo[3,4-b]pyridine and therapeutic uses thereof
KR20180080262A (ko) 2015-11-06 2018-07-11 사뮤메드, 엘엘씨 골관절염의 치료
PL3464285T3 (pl) 2016-06-01 2023-02-06 Biosplice Therapeutics, Inc. Sposób wytwarzania n-(5-(3-(7-(3-fluorofenylo)-3h-imidazo[4,5-c]pirydyn-2-ylo)-1h-indazol-5-ilo)pirydyn-3-ylo)-3-metylobutanoamidu
CA3069619A1 (en) 2017-07-17 2019-02-28 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
KR100482919B1 (ko) * 1996-03-11 2005-10-12 신젠타 파티서페이션즈 아게 살충제로서의피리미딘-4-온유도체
WO2004037159A2 (en) * 2002-10-23 2004-05-06 Obetherapy Biotechnology Compounds, compositions and methods for modulating fat metabolism
ES2566327T3 (es) * 2007-04-27 2016-04-12 Daiichi Sankyo Company, Limited Derivados de anillo aromático de 6 miembros que contiene nitrógeno y productos farmacéuticos que contienen los mismos
ES2456272T3 (es) 2008-08-01 2014-04-21 Dow Agrosciences Llc Uso de 5-fluorocitosina como un fungicida

Also Published As

Publication number Publication date
EP2462133A1 (en) 2012-06-13
RS53658B1 (en) 2015-04-30
CN102548979B (zh) 2015-05-13
JP5818791B2 (ja) 2015-11-18
CO6491089A2 (es) 2012-07-31
DK2462133T3 (en) 2015-01-05
KR20120043069A (ko) 2012-05-03
PL2462133T3 (pl) 2015-03-31
KR101792286B1 (ko) 2017-10-31
ES2506169T3 (es) 2014-10-13
IL217954A0 (en) 2012-03-29
MX2012001623A (es) 2012-04-11
NI201200019A (es) 2012-05-22
AU2010279408B2 (en) 2015-09-10
CR20120033A (es) 2012-03-22
CA2769251C (en) 2018-05-15
NZ597638A (en) 2014-06-27
PT2462133E (pt) 2014-12-26
WO2011017544A1 (en) 2011-02-10
JP2013501726A (ja) 2013-01-17
HN2012000261A (es) 2015-01-05
EP2462133A4 (en) 2013-01-16
BR112012002807A2 (pt) 2015-10-13
EA201270255A1 (ru) 2012-07-30
EA022930B1 (ru) 2016-03-31
IN2012DN00695A (es) 2015-06-19
EP2462133B1 (en) 2014-09-24
PE20120689A1 (es) 2012-06-06
ZA201305992B (en) 2014-10-29
HK1172892A1 (en) 2013-05-03
US8318758B2 (en) 2012-11-27
AU2010279408A1 (en) 2012-02-09
ECSP12011651A (es) 2012-03-30
BR112012002807B1 (pt) 2018-07-10
UA106086C2 (uk) 2014-07-25
CA2769251A1 (en) 2011-02-10
CN102548979A (zh) 2012-07-04
BR112012002807A8 (pt) 2017-07-11
US20110034491A1 (en) 2011-02-10
IL217954A (en) 2016-02-29

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