CA2000479A1 - Vasopermeability-enhancing conjugates - Google Patents
Vasopermeability-enhancing conjugatesInfo
- Publication number
- CA2000479A1 CA2000479A1 CA2000479A CA2000479A CA2000479A1 CA 2000479 A1 CA2000479 A1 CA 2000479A1 CA 2000479 A CA2000479 A CA 2000479A CA 2000479 A CA2000479 A CA 2000479A CA 2000479 A1 CA2000479 A1 CA 2000479A1
- Authority
- CA
- Canada
- Prior art keywords
- species
- vasoactive
- disclosed
- agent
- linked
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Landscapes
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Abstract
Conjugates having a clinically useful delivery vehicle linked to a biologically active species which acts to increase vascular permeability and expand blood volume at or in proximity to the tumor site are disclosed. the vehicle-linked species may be, for example, a vasoactive agent, a substance that recruits or amplifies a vasoactive species, a drug, or a pharmaceutical compound. Suitable biological species comprises peptides, lipids, carbohydrates, or their derivatives. Chemical or recombinant DNA methods suitable for linking the species to the vehicles are indicated. A therapy is disclosed which comprises administering the vasoactive conjugate and delivering a diagnostic agent or a therapeutic agent at an optimal time thereafter, when tumor vasculature is maximally affected.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US25551388A | 1988-10-11 | 1988-10-11 | |
US255,513 | 1988-10-11 |
Publications (2)
Publication Number | Publication Date |
---|---|
CA2000479A1 true CA2000479A1 (en) | 1990-04-11 |
CA2000479C CA2000479C (en) | 2000-06-20 |
Family
ID=22968671
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA002000479A Expired - Lifetime CA2000479C (en) | 1988-10-11 | 1989-10-11 | Vasopermeability-enhancing conjugates |
Country Status (1)
Country | Link |
---|---|
CA (1) | CA2000479C (en) |
-
1989
- 1989-10-11 CA CA002000479A patent/CA2000479C/en not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
CA2000479C (en) | 2000-06-20 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
EEER | Examination request | ||
MKEX | Expiry |