BRPI0411537A - derivados de lincomicina que possuem atividade antibacteriana - Google Patents
derivados de lincomicina que possuem atividade antibacterianaInfo
- Publication number
- BRPI0411537A BRPI0411537A BRPI0411537-6A BRPI0411537A BRPI0411537A BR PI0411537 A BRPI0411537 A BR PI0411537A BR PI0411537 A BRPI0411537 A BR PI0411537A BR PI0411537 A BRPI0411537 A BR PI0411537A
- Authority
- BR
- Brazil
- Prior art keywords
- antibacterial activity
- derivatives
- lincomycin derivatives
- lincomycin
- compounds
- Prior art date
Links
- OJMMVQQUTAEWLP-KIDUDLJLSA-N lincomycin Chemical class CN1C[C@H](CCC)C[C@H]1C(=O)N[C@H]([C@@H](C)O)[C@@H]1[C@H](O)[C@H](O)[C@@H](O)[C@@H](SC)O1 OJMMVQQUTAEWLP-KIDUDLJLSA-N 0.000 title abstract 4
- 230000000844 anti-bacterial effect Effects 0.000 title abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 2
- 241000894006 Bacteria Species 0.000 abstract 1
- 239000004599 antimicrobial Substances 0.000 abstract 1
- 230000015572 biosynthetic process Effects 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 230000003389 potentiating effect Effects 0.000 abstract 1
- 238000003786 synthesis reaction Methods 0.000 abstract 1
Classifications
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Abstract
"DERIVADOS DE LINCOMICINA QUE POSSUEM ATIVIDADE ANTIBACTERIANA". São revelados derivados de lincomicina. Esses derivados lincomicina apresentam atividade antibacteriana. Como os compostos da presente invenção apresentam potentes atividades contra bactérias, incluindo organismos gram-positivos, eles são agentes antimicrobianos úteis. São também revelados métodos de síntese e de uso dos compostos.
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US47950203P | 2003-06-17 | 2003-06-17 | |
US10/642,807 US7164011B2 (en) | 2002-08-15 | 2003-08-15 | Lincomycin derivatives possessing antibacterial activity |
PCT/US2003/025820 WO2004016632A2 (en) | 2002-08-15 | 2003-08-15 | Lincomycin derivatives possessing antibacterial activity |
US10/777,455 US7199105B2 (en) | 2002-08-15 | 2004-02-11 | Lincomycin derivatives possessing antibacterial activity |
PCT/US2004/019497 WO2005007665A2 (en) | 2003-06-17 | 2004-06-17 | Lincomycin derivatives possessing antibacterial activity |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0411537A true BRPI0411537A (pt) | 2006-08-01 |
Family
ID=36717101
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0411537-6A BRPI0411537A (pt) | 2003-06-17 | 2004-06-17 | derivados de lincomicina que possuem atividade antibacteriana |
Country Status (2)
Country | Link |
---|---|
JP (1) | JP2007528360A (pt) |
BR (1) | BRPI0411537A (pt) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2007516172A (ja) * | 2003-06-17 | 2007-06-21 | ビキュロン・ファーマシューティカルズ・インコーポレイテッド | 抗菌活性を有する新規リンコマイシン誘導体 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3496163A (en) * | 1965-02-08 | 1970-02-17 | Upjohn Co | 7-halo-7-deoxylincomycins and process for preparing the same |
US3435025A (en) * | 1966-03-18 | 1969-03-25 | Upjohn Co | 7-deoxylincomycin and analogs and isomers thereof and process for making the same |
US3549615A (en) * | 1968-10-17 | 1970-12-22 | Upjohn Co | Lincomycin derivatives and process for producing the same |
ZA806438B (en) * | 1979-11-23 | 1981-10-28 | Upjohn Co | Analogs of lincomycin and clindamycin |
-
2004
- 2004-06-17 JP JP2006517386A patent/JP2007528360A/ja active Pending
- 2004-06-17 BR BRPI0411537-6A patent/BRPI0411537A/pt not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
JP2007528360A (ja) | 2007-10-11 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application fees: dismissal - article 86 of industrial property law |
Free format text: REFERENTE A 6A E 7A ANUIDADES. |
|
B08K | Lapse as no evidence of payment of the annual fee has been furnished to inpi (acc. art. 87) |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2129 DE 25/10/2011. |