[go: up one dir, main page]
More Web Proxy on the site http://driver.im/

BR9609964A - Formulação sólida estável de sal de enalaprila e processo para preparação da mesma - Google Patents

Formulação sólida estável de sal de enalaprila e processo para preparação da mesma

Info

Publication number
BR9609964A
BR9609964A BR9609964A BR9609964A BR9609964A BR 9609964 A BR9609964 A BR 9609964A BR 9609964 A BR9609964 A BR 9609964A BR 9609964 A BR9609964 A BR 9609964A BR 9609964 A BR9609964 A BR 9609964A
Authority
BR
Brazil
Prior art keywords
enalapril
preparing
solid formulation
stable solid
water
Prior art date
Application number
BR9609964A
Other languages
English (en)
Inventor
Bernard Charles Sherman
Original Assignee
Bernard Charles Sherman
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=24034300&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR9609964(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bernard Charles Sherman filed Critical Bernard Charles Sherman
Publication of BR9609964A publication Critical patent/BR9609964A/pt

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/401—Proline; Derivatives thereof, e.g. captopril
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/55—Protease inhibitors
    • A61K38/556—Angiotensin converting enzyme inhibitors
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2009—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Vascular Medicine (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Inorganic Chemistry (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
  • Pyrrole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
BR9609964A 1995-08-04 1996-07-30 Formulação sólida estável de sal de enalaprila e processo para preparação da mesma BR9609964A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US08/511,297 US5573780A (en) 1995-08-04 1995-08-04 Stable solid formulation of enalapril salt and process for preparation thereof
PCT/CA1996/000513 WO1997005881A1 (en) 1995-08-04 1996-07-30 Stable solid formulation of enalapril salt and process for preparation thereof

Publications (1)

Publication Number Publication Date
BR9609964A true BR9609964A (pt) 1999-02-02

Family

ID=24034300

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9609964A BR9609964A (pt) 1995-08-04 1996-07-30 Formulação sólida estável de sal de enalaprila e processo para preparação da mesma

Country Status (14)

Country Link
US (2) US5573780A (pt)
EP (4) EP1442746A1 (pt)
JP (1) JP3290994B2 (pt)
AT (1) ATE288271T1 (pt)
AU (1) AU697696C (pt)
BR (1) BR9609964A (pt)
CA (1) CA2166001C (pt)
DE (4) DE04078149T1 (pt)
DK (1) DK0841930T3 (pt)
ES (4) ES2245275T1 (pt)
IL (1) IL123185A (pt)
NZ (1) NZ313576A (pt)
RU (1) RU2161970C2 (pt)
WO (1) WO1997005881A1 (pt)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5573780A (en) * 1995-08-04 1996-11-12 Apotex Usa Inc. Stable solid formulation of enalapril salt and process for preparation thereof
ES2125198B1 (es) * 1997-05-13 1999-11-16 Vita Invest Sa Asociacion a dosis fija de un inhibidor de la enzima convertidora de angiotensina y de un antagonista de los canales de calcio, procedimiento para su preparacion y su utilizacion para el tratamiento de enfermees cardiovasculares.
US6296871B1 (en) * 1998-04-12 2001-10-02 Ranbaxy Laboratories Limited Stable solid pharmaceutical compositions containing enalapril maleate
US6153223A (en) * 1998-06-05 2000-11-28 Watson Pharmaceuticals, Inc. Stabilized pharmaceutical compositions
NZ333206A (en) 1998-12-08 2000-07-28 Bernard Charles Sherman Solid pharmaceutical compositions comprising a stable magnesium salt of quinapril that acts as a ACE (Angiotensin Converting Enzyme) inhibitor
US6637359B1 (en) * 1998-12-15 2003-10-28 Maritrans Inc. System and method for internally fitting a new inner hull to an existing outer hull to form a rebuilt double hull vessel
US6555551B1 (en) 1999-08-31 2003-04-29 Mutual Pharmaceutical Co., Inc. Stable formulations of ACE inhibitors, and methods for preparation thereof
US6764694B1 (en) * 1999-08-31 2004-07-20 Mutual Pharmaceutical Co., Inc. Stable formulations of ACE inhibitors, and methods for preparation thereof
US20030225124A1 (en) * 1999-08-31 2003-12-04 Spiridon Spireas Stable formulations of ACE inhibitors, and methods for preparation thereof
US20040157911A1 (en) * 1999-08-31 2004-08-12 Spiridon Spireas Storage-stable and bio-stable formulations of ace inhibitors, and methods for preparation thereof
AU2003235579A1 (en) * 2002-01-15 2003-07-30 Delta Hf. Formulations of quinapril and related ace inhibitors
US20030215526A1 (en) * 2002-03-08 2003-11-20 Scott Stofik Stable formulations of angiotensin converting enzyme (ACE) inhibitors
SI1948224T1 (sl) 2005-11-17 2014-07-31 Silverstone Pharma Est. Stabilna formulacija amorfnih perindoprilnih soli, postopek za njihovo pripravo, posebno industrijsko pripravo, in njihova uporaba pri zdravljenju hipertenzije
EA027787B1 (ru) 2010-06-23 2017-09-29 Крка, Товарна Здравил, Д.Д., Ново Место Пероральные лекарственные формы, содержащие лерканидипин и эналаприл и их фармацевтически приемлемые соли
SI2654729T1 (sl) 2010-12-24 2016-08-31 Krka, D.D., Novo Mesto Homogene farmacevtske oralne dozirne oblike, ki obsegajo lerkanidipin in enalapril ali njune farmacevtsko sprejemljive soli skupaj z organsko kislino
CN109350733A (zh) * 2018-06-08 2019-02-19 山东理工职业学院 一种马来酸依那普利片剂的制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL58849A (en) * 1978-12-11 1983-03-31 Merck & Co Inc Carboxyalkyl dipeptides and derivatives thereof,their preparation and pharmaceutical compositions containing them
US4743450A (en) * 1987-02-24 1988-05-10 Warner-Lambert Company Stabilized compositions
YU48602B (sh) * 1991-11-25 1998-12-23 Krka Tovarna Zdravil P.O. Postupak za dobijanje stabilne formulacije soli enalaprila
WO1994001093A1 (en) * 1992-07-09 1994-01-20 Merck & Co., Inc. Controlled porosity osmotic enalapril pump
US5573780A (en) * 1995-08-04 1996-11-12 Apotex Usa Inc. Stable solid formulation of enalapril salt and process for preparation thereof

Also Published As

Publication number Publication date
ES2264912T1 (es) 2007-02-01
EP1637142A2 (en) 2006-03-22
EP1442746A1 (en) 2004-08-04
EP1527780A1 (en) 2005-05-04
CA2166001A1 (en) 1996-12-05
DE04076118T1 (de) 2005-02-10
EP1637142A3 (en) 2008-04-02
AU697696C (en) 2006-04-06
AU697696B2 (en) 1998-10-15
JP3290994B2 (ja) 2002-06-10
DE69616072T2 (de) 2009-09-10
ES2236741T3 (es) 2005-07-16
EP0841930A1 (en) 1998-05-20
RU2161970C2 (ru) 2001-01-20
ATE288271T1 (de) 2005-02-15
AU6608496A (en) 1997-03-05
DE69616072D1 (de) 2001-11-22
JPH10511103A (ja) 1998-10-27
IL123185A0 (en) 1998-09-24
IL123185A (en) 2001-08-08
WO1997005881A1 (en) 1997-02-20
NZ313576A (en) 1999-05-28
US5690962A (en) 1997-11-25
ES2223315T1 (es) 2005-03-01
DE04078149T1 (de) 2005-12-29
CA2166001C (en) 2005-12-27
US5573780A (en) 1996-11-12
ES2245275T1 (es) 2006-01-01
DE05076813T1 (de) 2006-11-30
EP0841930B1 (en) 2005-02-02
DK0841930T3 (da) 2005-04-25

Similar Documents

Publication Publication Date Title
BR9609964A (pt) Formulação sólida estável de sal de enalaprila e processo para preparação da mesma
TR200000832A2 (tr) Sıkıştırılmış kalıp cisimleri için yoğunlaştırılmış patlayıcı taneler.
DK0774949T3 (da) Klæbemiddel til tandproteser
DK0801559T3 (da) Fremgangsmåde til fremstilling af orale doseringsformer indeholdende et beta-lactam antibiotikum
AU2145192A (en) Solid, storage-stable, germicidal, pre-iodine composition
ES2184452T3 (es) Preparacion farmaceutica que contiene levotiroxina de sodio.
ES2058288T3 (es) Composiciones de ibuprofen secadas por atomizacion.
TW344662B (en) A process for preparing a freeze dried thiotepa composition
EA199900193A1 (ru) Грануляты, содержащие водорастворимое соединение и целлюлозу
WO2002011740A3 (en) 'slow release' pharmaceutical compositions comprising lithium carbonate
TR200200995T2 (tr) 7-amino-3-metksimetil-3-sefem-4-karbosilik asitin hazırlanmasına yönelik proses.
PT989994E (pt) Derivados de estreptograminas, a sua preparacao e as composicoes que os contem
ATE275577T1 (de) Quinapril magnesium enthaltende, pharmazeutisch wirksame zusammensetzung
BR0110310A (pt) Dispersão sólida, processo para sua produção e preparado farmacêutico contendo a mesma
DK1117365T3 (da) Vedhæftningsmiddel til tandproteser
JPS5740573A (en) Water-soluble sizing composition
KR920003967A (ko) 젬피브로질 제제
RU94046203A (ru) Способ получения 5-дихлорацетил-3,3,6-триметил-9-оксо-1,5-диазабицикло[4,3,0]нонана
UY24851A1 (es) Derivados de ácidos n-acil-alfa-aminados
RU99104271A (ru) Состав для химического расширения каналов
RU95122428A (ru) Способ получения синтетического дубителя
RU96121905A (ru) Применение водных растворов солей l-триптофана и l-треонина
RU97114057A (ru) Способ подготовки стекольной шихты
RU97100111A (ru) Пластификатор тампонажных растворов
JPS52133902A (en) Novel antibiotic substance sf-1771-b and its preparation

Legal Events

Date Code Title Description
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]