BR9505899A - Tienopiridonas processo para sua preparação processo para a produção farmacêutica preparação farmacêutica e uso - Google Patents
Tienopiridonas processo para sua preparação processo para a produção farmacêutica preparação farmacêutica e usoInfo
- Publication number
- BR9505899A BR9505899A BR9505899A BR9505899A BR9505899A BR 9505899 A BR9505899 A BR 9505899A BR 9505899 A BR9505899 A BR 9505899A BR 9505899 A BR9505899 A BR 9505899A BR 9505899 A BR9505899 A BR 9505899A
- Authority
- BR
- Brazil
- Prior art keywords
- preparation
- pharmaceutical
- thienopyridones
- production
- pharmaceutical production
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/06—Antianaemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Pain & Pain Management (AREA)
- Psychiatry (AREA)
- Hematology (AREA)
- Hospice & Palliative Care (AREA)
- Cardiology (AREA)
- Diabetes (AREA)
- Anesthesiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE4444815A DE4444815A1 (de) | 1994-12-15 | 1994-12-15 | Thienopyridone |
CN95120906.XA CN1133843A (zh) | 1994-12-15 | 1995-12-19 | 噻吩并吡啶酮 |
Publications (1)
Publication Number | Publication Date |
---|---|
BR9505899A true BR9505899A (pt) | 1998-01-06 |
Family
ID=37698014
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR9505899A BR9505899A (pt) | 1994-12-15 | 1995-12-14 | Tienopiridonas processo para sua preparação processo para a produção farmacêutica preparação farmacêutica e uso |
Country Status (17)
Country | Link |
---|---|
US (1) | US5602144A (pt) |
EP (1) | EP0717044A1 (pt) |
JP (1) | JPH08239387A (pt) |
CN (1) | CN1133843A (pt) |
AU (1) | AU703603B2 (pt) |
BR (1) | BR9505899A (pt) |
CA (1) | CA2165129A1 (pt) |
CZ (1) | CZ319395A3 (pt) |
DE (1) | DE4444815A1 (pt) |
FI (1) | FI956024L (pt) |
HU (1) | HUT75091A (pt) |
NO (1) | NO955075L (pt) |
PL (1) | PL311838A1 (pt) |
RU (1) | RU2155766C2 (pt) |
SK (1) | SK157195A3 (pt) |
TR (1) | TR199501562A2 (pt) |
ZA (1) | ZA9510671B (pt) |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2440760C (en) * | 2001-03-14 | 2010-02-09 | Matthias Gerlach | Substituted pyrazolopyrimidines and thiazolopyrimidines used as analgesics |
GB0124848D0 (en) * | 2001-10-16 | 2001-12-05 | Celltech R&D Ltd | Chemical compounds |
US7119205B2 (en) * | 2003-05-16 | 2006-10-10 | Abbott Laboratories | Thienopyridones as AMPK activators for the treatment of diabetes and obesity |
SE0401578D0 (sv) * | 2004-06-18 | 2004-06-18 | Active Biotech Ab | Novel compounds |
EP1754483A1 (en) | 2005-08-18 | 2007-02-21 | Merck Sante | Use of thienopyridone derivatives as AMPK activators and pharmaceutical compositions containing them |
CN101998853B (zh) | 2008-04-11 | 2015-02-11 | 默克专利有限公司 | 作为amp-活化的蛋白激酶(ampk)激活剂的噻吩并吡啶酮衍生物 |
ES2388485T3 (es) * | 2008-05-05 | 2012-10-15 | Merck Patent Gmbh | Derivados de tienopiridona como activadores de proteína quinasa activada por AMP (AMPK) |
US8691849B2 (en) * | 2008-09-02 | 2014-04-08 | Janssen Pharmaceuticals, Inc. | 3-azabicyclo[3.1.0]hexyl derivatives as modulators of metabotropic glutamate receptors |
EP2679591A1 (en) | 2012-06-29 | 2014-01-01 | Poxel | Thienopyridone derivatives useful as activators of AMPK |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ZA903588B (en) * | 1989-05-16 | 1991-02-27 | Merrell Dow Pharma | Excitatory amino acid antagonists |
US5112821A (en) * | 1989-05-16 | 1992-05-12 | Merrell Dow Pharmaceuticals Inc. | Excitatory amino acid antagonists which are certain thienopyridives |
US5026700A (en) * | 1989-05-16 | 1991-06-25 | Merrell Dow Pharmaceuticals | Certain quinolines and thienopyridines as excitatory amino acid antagonists |
GB9022785D0 (en) * | 1990-10-19 | 1990-12-05 | Merck Sharp & Dohme | Therapeutic agents |
US5129864A (en) * | 1991-02-27 | 1992-07-14 | Dayco Products, Inc. | Tensioner for a power transmission belt and method of making the same |
US5219864A (en) * | 1991-03-12 | 1993-06-15 | Kyowa Hakko Kogyo Co., Ltd. | Thienopyridine derivatives |
US5155115A (en) * | 1991-03-12 | 1992-10-13 | Kyowa Hakko Kogyo Co., Ltd. | Thienopyridine derivatives |
JPH05134373A (ja) * | 1991-11-14 | 1993-05-28 | Konica Corp | 新規な写真用カプラー |
DE4227747A1 (de) * | 1992-08-21 | 1994-02-24 | Basf Ag | Heteroaromatisch kondensierte Hydroxypyridoncarbonsäureamide, deren Herstellung und Verwendung |
-
1994
- 1994-12-15 DE DE4444815A patent/DE4444815A1/de not_active Withdrawn
-
1995
- 1995-12-01 CZ CZ953193A patent/CZ319395A3/cs unknown
- 1995-12-02 EP EP95119009A patent/EP0717044A1/de not_active Withdrawn
- 1995-12-07 AU AU40292/95A patent/AU703603B2/en not_active Ceased
- 1995-12-07 RU RU95121158/04A patent/RU2155766C2/ru active
- 1995-12-12 TR TR95/01562A patent/TR199501562A2/xx unknown
- 1995-12-13 CA CA002165129A patent/CA2165129A1/en not_active Abandoned
- 1995-12-14 ZA ZA9510671A patent/ZA9510671B/xx unknown
- 1995-12-14 US US08/572,750 patent/US5602144A/en not_active Expired - Lifetime
- 1995-12-14 NO NO955075A patent/NO955075L/no not_active Application Discontinuation
- 1995-12-14 FI FI956024A patent/FI956024L/fi unknown
- 1995-12-14 BR BR9505899A patent/BR9505899A/pt not_active Application Discontinuation
- 1995-12-14 HU HU9503582A patent/HUT75091A/hu unknown
- 1995-12-14 PL PL95311838A patent/PL311838A1/xx unknown
- 1995-12-15 SK SK1571-95A patent/SK157195A3/sk unknown
- 1995-12-15 JP JP7347097A patent/JPH08239387A/ja active Pending
- 1995-12-19 CN CN95120906.XA patent/CN1133843A/zh active Pending
Also Published As
Publication number | Publication date |
---|---|
FI956024A7 (fi) | 1996-06-16 |
ZA9510671B (en) | 1996-07-11 |
HU9503582D0 (en) | 1996-02-28 |
US5602144A (en) | 1997-02-11 |
FI956024L (fi) | 1996-06-16 |
PL311838A1 (en) | 1996-06-24 |
EP0717044A1 (de) | 1996-06-19 |
NO955075D0 (no) | 1995-12-14 |
AU4029295A (en) | 1996-06-20 |
HUT75091A (en) | 1997-04-28 |
RU2155766C2 (ru) | 2000-09-10 |
FI956024A0 (fi) | 1995-12-14 |
SK157195A3 (en) | 1996-07-03 |
NO955075L (no) | 1996-06-17 |
CA2165129A1 (en) | 1996-06-16 |
JPH08239387A (ja) | 1996-09-17 |
AU703603B2 (en) | 1999-03-25 |
DE4444815A1 (de) | 1996-06-20 |
CN1133843A (zh) | 1996-10-23 |
TR199501562A2 (tr) | 1996-07-21 |
CZ319395A3 (en) | 1996-07-17 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FB36 | Technical and formal requirements: requirement - article 36 of industrial property law | ||
FA8 | Dismissal: dismissal - article 36, par. 1 of industrial property law |