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BR0210407A - Composto, composição farmacêutica, uso de um composto e método de tratamento de um distúrbio ou de uma doença de corpo animal vivo, incluindo um humano - Google Patents

Composto, composição farmacêutica, uso de um composto e método de tratamento de um distúrbio ou de uma doença de corpo animal vivo, incluindo um humano

Info

Publication number
BR0210407A
BR0210407A BR0210407-5A BR0210407A BR0210407A BR 0210407 A BR0210407 A BR 0210407A BR 0210407 A BR0210407 A BR 0210407A BR 0210407 A BR0210407 A BR 0210407A
Authority
BR
Brazil
Prior art keywords
compound
human
disorder
pharmaceutical composition
animal body
Prior art date
Application number
BR0210407-5A
Other languages
English (en)
Inventor
Mario Rottlonder
Ejner Knud Moltzen
Ivan Mikkelsen
Thomas Ruhland
Kim Andersen
Christian Krog-Jensen
Original Assignee
Lundbeck & Co As H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H
Publication of BR0210407A publication Critical patent/BR0210407A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Nutrition Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)

Abstract

"COMPOSTO, COMPOSIçãO FARMACêUTICA, USO DE UM COMPOSTO E MéTODO DE TRATAMENTO DE UM DISTúRBIO OU DE UMA DOENçA DE CORPO ANIMAL VIVO, INCLUINDO UM HUMANO". Um derivado heteroarilado possuindo a fórmula (I) Os compostos da invenção são considerados úteis para o tratamento de distúrbios afetivos tais como distúrbio de ansiedade geral, distúrbio de pânico, distúrbio compulsivo obsessivo, depressão, fobia social e distúrbios de alimentação, e distúrbios neurológicos tal como psicose.
BR0210407-5A 2001-06-29 2002-06-27 Composto, composição farmacêutica, uso de um composto e método de tratamento de um distúrbio ou de uma doença de corpo animal vivo, incluindo um humano BR0210407A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DKPA200101037 2001-06-29
PCT/DK2002/000436 WO2003002552A1 (en) 2001-06-29 2002-06-27 Novel indole derivatives

Publications (1)

Publication Number Publication Date
BR0210407A true BR0210407A (pt) 2004-08-17

Family

ID=8160599

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0210407-5A BR0210407A (pt) 2001-06-29 2002-06-27 Composto, composição farmacêutica, uso de um composto e método de tratamento de um distúrbio ou de uma doença de corpo animal vivo, incluindo um humano

Country Status (28)

Country Link
US (1) US7342015B2 (pt)
EP (1) EP1399434B1 (pt)
JP (1) JP2004535448A (pt)
KR (1) KR20040019027A (pt)
CN (1) CN100338058C (pt)
AR (1) AR034658A1 (pt)
AT (1) ATE304007T1 (pt)
AU (1) AU2002344950B2 (pt)
BG (1) BG108538A (pt)
BR (1) BR0210407A (pt)
CA (1) CA2451229C (pt)
CZ (1) CZ2004155A3 (pt)
DE (1) DE60206043T2 (pt)
DK (1) DK1399434T3 (pt)
EA (1) EA006104B1 (pt)
ES (1) ES2247347T3 (pt)
HK (1) HK1069579A1 (pt)
HU (1) HUP0400834A2 (pt)
IL (1) IL158830A0 (pt)
IS (1) IS2431B (pt)
MX (1) MXPA03011766A (pt)
NO (1) NO326513B1 (pt)
NZ (1) NZ529461A (pt)
PL (1) PL366520A1 (pt)
SK (1) SK642004A3 (pt)
UA (1) UA74651C2 (pt)
WO (1) WO2003002552A1 (pt)
ZA (1) ZA200308848B (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA75407C2 (en) * 2001-06-29 2006-04-17 Lundbeck & Co As H Heteroaryl derivatives of pyridine and pyrimidine, pharmaceutical composition and use thereof
WO2006056600A1 (en) 2004-11-26 2006-06-01 Janssen Pharmaceutica N.V. Isoxazoline-indole derivatives with an improved antipsychotic and anxiolytic a ivity
AR055203A1 (es) * 2005-08-31 2007-08-08 Otsuka Pharma Co Ltd Derivados de benzotiofeno con propiedades antipsicoticas
JP4785881B2 (ja) * 2007-02-27 2011-10-05 大塚製薬株式会社 医薬
CN116554145A (zh) * 2022-01-29 2023-08-08 江苏恩华药业股份有限公司 芳烷基-4-(1h)吲哚基哌嗪衍生物、其制备方法和应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0900792B1 (en) * 1997-09-02 2003-10-29 Duphar International Research B.V Piperazine and piperidine derivatives as 5-HT1A and dopamine D2-receptor (ant)agonists
WO1999055672A2 (en) * 1998-04-29 1999-11-04 American Home Products Corporation Antipsychotic indolyl derivatives
AR027134A1 (es) * 1999-12-30 2003-03-12 Lundbeck & Co As H Derivados de indol.
UA75407C2 (en) * 2001-06-29 2006-04-17 Lundbeck & Co As H Heteroaryl derivatives of pyridine and pyrimidine, pharmaceutical composition and use thereof

Also Published As

Publication number Publication date
UA74651C2 (en) 2006-01-16
ZA200308848B (en) 2006-02-22
MXPA03011766A (es) 2004-04-02
ES2247347T3 (es) 2006-03-01
KR20040019027A (ko) 2004-03-04
BG108538A (bg) 2005-01-31
DE60206043D1 (de) 2005-10-13
NO20035672L (no) 2003-12-18
US7342015B2 (en) 2008-03-11
EA006104B1 (ru) 2005-08-25
JP2004535448A (ja) 2004-11-25
WO2003002552A1 (en) 2003-01-09
HK1069579A1 (en) 2005-05-27
EA200400104A1 (ru) 2004-04-29
NO20035672D0 (no) 2003-12-18
SK642004A3 (en) 2004-05-04
EP1399434A1 (en) 2004-03-24
US20060258678A1 (en) 2006-11-16
ATE304007T1 (de) 2005-09-15
CA2451229C (en) 2009-02-10
CN1529703A (zh) 2004-09-15
HUP0400834A2 (hu) 2004-08-30
IL158830A0 (en) 2004-05-12
PL366520A1 (en) 2005-02-07
CN100338058C (zh) 2007-09-19
NZ529461A (en) 2005-09-30
IS7022A (is) 2003-11-10
NO326513B1 (no) 2008-12-22
AR034658A1 (es) 2004-03-03
DE60206043T2 (de) 2006-06-29
EP1399434B1 (en) 2005-09-07
DK1399434T3 (da) 2005-12-12
AU2002344950B2 (en) 2008-04-03
CA2451229A1 (en) 2003-01-09
IS2431B (is) 2008-10-15
CZ2004155A3 (cs) 2004-07-14

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Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B15K Others concerning applications: alteration of classification

Free format text: ALTERADA DA INT.CL: C07D 401/12, C07D 403/12, A61K 31/497, A61K 31/506

Ipc: C07D 401/12 (2011.01), C07D 403/12 (2011.01), A61K

B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 8A E 9A ANUIDADE(S).

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO RPI 2108 DE 31/05/2011.