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AU616819B2 - Beta-amino-boronic acid derivatives - Google Patents

Beta-amino-boronic acid derivatives

Info

Publication number
AU616819B2
AU616819B2 AU45665/89A AU4566589A AU616819B2 AU 616819 B2 AU616819 B2 AU 616819B2 AU 45665/89 A AU45665/89 A AU 45665/89A AU 4566589 A AU4566589 A AU 4566589A AU 616819 B2 AU616819 B2 AU 616819B2
Authority
AU
Australia
Prior art keywords
beta
amino
acid derivatives
boronic acid
boronic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU45665/89A
Other versions
AU4566589A (en
Inventor
Heinz-Werner Kleemann
Dieter Ruppert
Bernward Scholkens
Hansjorg Urbach
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Hoechst AG
Original Assignee
Hoechst AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst AG filed Critical Hoechst AG
Publication of AU4566589A publication Critical patent/AU4566589A/en
Application granted granted Critical
Publication of AU616819B2 publication Critical patent/AU616819B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06191—Dipeptides containing heteroatoms different from O, S, or N

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cardiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Plural Heterocyclic Compounds (AREA)
AU45665/89A 1988-12-01 1989-11-30 Beta-amino-boronic acid derivatives Ceased AU616819B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3840452 1988-12-01
DE3840452A DE3840452A1 (en) 1988-12-01 1988-12-01 (BETA) -amino-boronic acid DERIVATIVES

Publications (2)

Publication Number Publication Date
AU4566589A AU4566589A (en) 1990-06-07
AU616819B2 true AU616819B2 (en) 1991-11-07

Family

ID=6368210

Family Applications (1)

Application Number Title Priority Date Filing Date
AU45665/89A Ceased AU616819B2 (en) 1988-12-01 1989-11-30 Beta-amino-boronic acid derivatives

Country Status (14)

Country Link
EP (1) EP0371467A3 (en)
JP (1) JPH02193997A (en)
KR (1) KR900009663A (en)
AU (1) AU616819B2 (en)
CA (1) CA2004303A1 (en)
DE (1) DE3840452A1 (en)
DK (1) DK605489A (en)
FI (1) FI895718A0 (en)
IL (1) IL92497A0 (en)
NO (1) NO894790L (en)
NZ (1) NZ231578A (en)
PH (1) PH26584A (en)
PT (1) PT92442A (en)
ZA (1) ZA899152B (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU666294B2 (en) * 1990-11-14 1996-02-08 Axis Biochemicals Asa Labelling agents comprising boronic acid conjugates

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0341661A3 (en) * 1988-05-11 1991-05-02 The Du Pont Merck Pharmaceutical Company Peptide-drug compositions containing alpha-aminoboronic acid derivatives
US4983589A (en) * 1989-12-14 1991-01-08 Chevron Research And Technology Company Fungicidal imidazole diphenylaliphaticboranes and derivatives thereof
GB9017694D0 (en) * 1990-08-13 1990-09-26 Sandoz Ltd Improvements in or relating to organic chemistry
US5554728A (en) * 1991-07-23 1996-09-10 Nexstar Pharmaceuticals, Inc. Lipid conjugates of therapeutic peptides and protease inhibitors
US6825169B1 (en) 1991-10-22 2004-11-30 Trustees Of Tufts College Inhibitors of dipeptidyl-aminopeptidase type IV
EP0633881B1 (en) * 1992-03-11 2003-10-29 Narhex Limited Amine derivatives of oxo- and hydroxy-substitued hydrocarbons
US6071895A (en) * 1992-03-11 2000-06-06 Narhex Limited Polar-substituted hydrocarbons
ATE253050T1 (en) 1992-03-11 2003-11-15 Narhex Ltd AMINE DERIVATIVES OF OXO- AND HYDROXY-SUBSTITUTED HYDROCARBONS
US5888992A (en) * 1992-03-11 1999-03-30 Narhex Limited Polar substituted hydrocarbons
US5559256A (en) * 1992-07-20 1996-09-24 E. R. Squibb & Sons, Inc. Aminediol protease inhibitors
US5354491A (en) * 1992-08-14 1994-10-11 The Procter & Gamble Company Liquid detergent compositions containing protease and certain β-aminoalkylboronic acids and esters
EP0655068B1 (en) * 1992-08-14 1997-12-17 The Procter & Gamble Company Process for synthesizing a beta-aminoalkylboronic acid and ester thereof
US5442100A (en) * 1992-08-14 1995-08-15 The Procter & Gamble Company β-aminoalkyl and β-N-peptidylaminoalkyl boronic acids
TR28578A (en) * 1993-08-13 1996-11-04 Procter & Gamble Liquid detergent compositions containing protease and some of -aminoalkylboronic acid and esters.
IL110898A0 (en) * 1993-09-10 1994-11-28 Narhex Australia Pty Ltd Polar-substituted hydrocarbons
US5431842A (en) * 1993-11-05 1995-07-11 The Procter & Gamble Company Liquid detergents with ortho-substituted phenylboronic acids for inhibition of proteolytic enzyme
US5965532A (en) 1996-06-28 1999-10-12 Trustees Of Tufts College Multivalent compounds for crosslinking receptors and uses thereof
US6100234A (en) * 1997-05-07 2000-08-08 Tufts University Treatment of HIV
US6040145A (en) 1997-05-07 2000-03-21 Tufts University Potentiation of the immune response
ES2285785T3 (en) 1997-09-29 2007-11-16 Point Therapeutics, Inc. STIMULATION OF IN VITRO HEMATOPOYETIC CELLS.
CA2331122A1 (en) 1998-05-04 1999-11-11 Point Therapeutics, Inc. Hematopoietic stimulation
US6890904B1 (en) 1999-05-25 2005-05-10 Point Therapeutics, Inc. Anti-tumor agents
CA2862710A1 (en) * 2012-01-09 2013-07-18 University Of Tromso Therapeutic boron-containing compounds

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4537773A (en) * 1983-12-05 1985-08-27 E. I. Du Pont De Nemours And Company α-Aminoboronic acid derivatives
US4499082A (en) * 1983-12-05 1985-02-12 E. I. Du Pont De Nemours And Company α-Aminoboronic acid peptides

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU666294B2 (en) * 1990-11-14 1996-02-08 Axis Biochemicals Asa Labelling agents comprising boronic acid conjugates

Also Published As

Publication number Publication date
NO894790L (en) 1990-06-05
KR900009663A (en) 1990-07-05
CA2004303A1 (en) 1990-06-01
DK605489D0 (en) 1989-11-30
NO894790D0 (en) 1989-11-30
AU4566589A (en) 1990-06-07
PH26584A (en) 1992-08-19
NZ231578A (en) 1992-02-25
EP0371467A3 (en) 1991-04-03
JPH02193997A (en) 1990-07-31
IL92497A0 (en) 1990-08-31
DE3840452A1 (en) 1990-06-07
DK605489A (en) 1990-06-02
EP0371467A2 (en) 1990-06-06
FI895718A0 (en) 1989-11-29
ZA899152B (en) 1990-09-26
PT92442A (en) 1990-06-29

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