AU2001288617A1 - Methods for forming combinatorial libraries combining amide bond formation with epoxide opening - Google Patents
Methods for forming combinatorial libraries combining amide bond formation with epoxide openingInfo
- Publication number
- AU2001288617A1 AU2001288617A1 AU2001288617A AU8861701A AU2001288617A1 AU 2001288617 A1 AU2001288617 A1 AU 2001288617A1 AU 2001288617 A AU2001288617 A AU 2001288617A AU 8861701 A AU8861701 A AU 8861701A AU 2001288617 A1 AU2001288617 A1 AU 2001288617A1
- Authority
- AU
- Australia
- Prior art keywords
- methods
- amide bond
- bond formation
- combinatorial libraries
- epoxide opening
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
- C07D303/02—Compounds containing oxirane rings
- C07D303/12—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms
- C07D303/18—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms by etherified hydroxyl radicals
- C07D303/20—Ethers with hydroxy compounds containing no oxirane rings
- C07D303/22—Ethers with hydroxy compounds containing no oxirane rings with monohydroxy compounds
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
- C07D303/02—Compounds containing oxirane rings
- C07D303/36—Compounds containing oxirane rings with hydrocarbon radicals, substituted by nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
- C07D303/02—Compounds containing oxirane rings
- C07D303/38—Compounds containing oxirane rings with hydrocarbon radicals, substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C40—COMBINATORIAL TECHNOLOGY
- C40B—COMBINATORIAL CHEMISTRY; LIBRARIES, e.g. CHEMICAL LIBRARIES
- C40B40/00—Libraries per se, e.g. arrays, mixtures
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US23012200P | 2000-09-05 | 2000-09-05 | |
| US60/230,122 | 2000-09-05 | ||
| PCT/US2001/027226 WO2002020436A2 (en) | 2000-09-05 | 2001-08-31 | Methods for forming combinatorial libraries combining amide bond formation with epoxide opening |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AU2001288617A1 true AU2001288617A1 (en) | 2002-03-22 |
Family
ID=22864027
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AU2001288617A Abandoned AU2001288617A1 (en) | 2000-09-05 | 2001-08-31 | Methods for forming combinatorial libraries combining amide bond formation with epoxide opening |
Country Status (3)
| Country | Link |
|---|---|
| US (1) | US20020077491A1 (en) |
| AU (1) | AU2001288617A1 (en) |
| WO (1) | WO2002020436A2 (en) |
Families Citing this family (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MY151199A (en) | 2001-11-02 | 2014-04-30 | Rigel Pharmaceuticals Inc | Substituted diphenyl heterocycles useful for treating hcv infection |
| MXPA04012959A (en) * | 2002-06-29 | 2005-05-16 | Zentaris Gmbh | Arylcarbonylpiperazines and heteroarylcarbonylpiperazines and the use thereof for treating benign and malignant tumour diseases. |
| WO2004018463A2 (en) | 2002-08-23 | 2004-03-04 | Rigel Pharmaceuticals, Inc. | Pyridyl substituted heterocycles useful for treating or preventing hcv infection |
| JP2007521252A (en) * | 2003-04-11 | 2007-08-02 | エスジーエックス ファーマシューティカルズ，インコーポレイティド | Compound library and drug discovery method |
| WO2004099164A1 (en) | 2003-05-02 | 2004-11-18 | Rigel Pharmaceuticals, Inc. | Substituted diphenyl isoxazoles, pyrazoles and oxadiazoles useful for treating hcv infection |
| US7326790B2 (en) | 2003-05-02 | 2008-02-05 | Rigel Pharmaceuticals, Inc. | Diphenylisoxazole compounds and hydro isomers thereof |
| US7220745B2 (en) | 2003-05-15 | 2007-05-22 | Rigel Pharmaceuticals | Heterocyclic compounds useful to treat HCV |
| US8373000B2 (en) * | 2003-06-30 | 2013-02-12 | Johnson & Johnson Vision Care, Inc. | Process for the production of bis(trimethylsilyloxy)silylalkylglycerol methacrylates |
| US6933401B2 (en) * | 2003-06-30 | 2005-08-23 | Frank Molock | Process for the production of vicinal diesters from epoxides |
| WO2005049065A2 (en) | 2003-11-19 | 2005-06-02 | Rigel Pharmaceuticals, Inc. | Synergistic combinations of dihaloacetamide with interferon or ribavirin for treatment hcv infections |
| US7514434B2 (en) | 2004-02-23 | 2009-04-07 | Rigel Pharmaceuticals, Inc. | Heterocyclic compounds having an oxadiazole moiety and hydro isomers thereof |
| CA2606106A1 (en) | 2005-05-02 | 2007-03-08 | Rigel Pharmaceuticals, Inc. | Heterocyclic anti-viral compounds comprising metabolizable moieties and their uses |
| JP5070797B2 (en) * | 2005-12-08 | 2012-11-14 | Ｊｎｃ株式会社 | Lateral oxirane compound and polymer thereof |
| JP2011148762A (en) * | 2009-12-22 | 2011-08-04 | Jnc Corp | Polymerizable liquid crystal compound, polymerizable liquid crystal composition and anisotropic polymer |
| PT3752501T (en) | 2018-02-13 | 2023-07-12 | Gilead Sciences Inc | Pd-1/pd-l1 inhibitors |
| EP3781556A1 (en) | 2018-04-19 | 2021-02-24 | Gilead Sciences, Inc. | Pd-1/pd-l1 inhibitors |
| AU2019301811B2 (en) | 2018-07-13 | 2022-05-26 | Gilead Sciences, Inc. | PD-1/PD-L1 inhibitors |
| EP3870566A1 (en) | 2018-10-24 | 2021-09-01 | Gilead Sciences, Inc. | Pd-1/pd-l1 inhibitors |
| CN118191186B (en) * | 2024-05-16 | 2024-07-23 | 西南林业大学 | Extraction method and application of sulfonamide antibiotics in water body |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6207861B1 (en) * | 1998-01-05 | 2001-03-27 | Neogenesis, Inc. | Method for producing and screening mass coded combinatorial libraries for drug discovery and target validation |
-
2001
- 2001-08-31 AU AU2001288617A patent/AU2001288617A1/en not_active Abandoned
- 2001-08-31 US US09/943,852 patent/US20020077491A1/en not_active Abandoned
- 2001-08-31 WO PCT/US2001/027226 patent/WO2002020436A2/en active Application Filing
Also Published As
| Publication number | Publication date |
|---|---|
| WO2002020436A2 (en) | 2002-03-14 |
| US20020077491A1 (en) | 2002-06-20 |
| WO2002020436A3 (en) | 2003-01-09 |
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