AU2001277741A1 - 2-aminopyridine compounds and use thereof as drugs - Google Patents
2-aminopyridine compounds and use thereof as drugsInfo
- Publication number
- AU2001277741A1 AU2001277741A1 AU2001277741A AU2001277741A AU2001277741A1 AU 2001277741 A1 AU2001277741 A1 AU 2001277741A1 AU 2001277741 A AU2001277741 A AU 2001277741A AU 2001277741 A AU2001277741 A AU 2001277741A AU 2001277741 A1 AU2001277741 A1 AU 2001277741A1
- Authority
- AU
- Australia
- Prior art keywords
- drugs
- aminopyridine compounds
- aminopyridine
- compounds
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 150000003930 2-aminopyridines Chemical class 0.000 title 1
- 239000003814 drug Substances 0.000 title 1
- 229940079593 drugs Drugs 0.000 title 1
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2000245056 | 2000-08-11 | ||
JP2000-245056 | 2000-08-11 | ||
PCT/JP2001/006870 WO2002014282A1 (en) | 2000-08-11 | 2001-08-09 | 2-aminopyridine compounds and use thereof as drugs |
Publications (2)
Publication Number | Publication Date |
---|---|
AU2001277741A1 true AU2001277741A1 (en) | 2002-05-23 |
AU2001277741B2 AU2001277741B2 (en) | 2005-12-22 |
Family
ID=18735647
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU7774101A Pending AU7774101A (en) | 2000-08-11 | 2001-08-09 | 2-aminopyridine compounds and use thereof as drugs |
AU2001277741A Ceased AU2001277741B2 (en) | 2000-08-11 | 2001-08-09 | 2-aminopyridine compounds and use thereof as drugs |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU7774101A Pending AU7774101A (en) | 2000-08-11 | 2001-08-09 | 2-aminopyridine compounds and use thereof as drugs |
Country Status (18)
Country | Link |
---|---|
US (1) | US6750232B2 (en) |
EP (1) | EP1308441B1 (en) |
JP (1) | JP4251868B2 (en) |
KR (1) | KR100804111B1 (en) |
CN (1) | CN1446202A (en) |
AT (1) | ATE444752T1 (en) |
AU (2) | AU7774101A (en) |
CA (1) | CA2417846A1 (en) |
DE (1) | DE60140126D1 (en) |
HU (1) | HUP0700086A2 (en) |
IL (2) | IL153995A0 (en) |
MX (1) | MXPA03001136A (en) |
NO (1) | NO325873B1 (en) |
NZ (1) | NZ523998A (en) |
RU (1) | RU2250898C2 (en) |
TW (1) | TWI298064B (en) |
WO (1) | WO2002014282A1 (en) |
ZA (1) | ZA200300482B (en) |
Families Citing this family (50)
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TWI330183B (en) * | 2001-10-22 | 2010-09-11 | Eisai R&D Man Co Ltd | |
BR0306919A (en) | 2002-01-28 | 2004-11-09 | Kyowa Hakko Kogyo Kk | Methods for reducing or suppressing the adverse effectiveness of l-dopa and / or dopamine agonist therapy, and for moderate l-dopa treatment, composition for moderate l-dopa treatment, method for treating parkinson's disease and / or complications. -dopa motors, composition for the treatment of parkinson's disease, and methods for prolonging the effective treatment of parkinson's disease, and for treating movement disorders |
AU2002950853A0 (en) * | 2002-08-19 | 2002-09-12 | Fujisawa Pharmaceutical Co., Ltd. | Aminopyrimidine compound and pharmaceutical use thereof |
US20040067955A1 (en) * | 2002-09-06 | 2004-04-08 | Fujisawa Pharmaceutical Co. Ltd. | Pyridazinone compound and pharmaceutical use thereof |
BRPI0415863A (en) * | 2003-10-27 | 2007-01-09 | Astellas Pharma Inc | pyrazine derivatives and their pharmaceutical uses |
ES2241496B1 (en) * | 2004-04-15 | 2006-12-01 | Almirall Prodesfarma, S.A. | NEW DERIVATIVES OF PIRIDINA. |
EP1807396B1 (en) * | 2004-10-29 | 2013-06-26 | Merck Sharp & Dohme Corp. | 2-aminopyridine compounds useful as beta-secretase inhibitors for the treatment of alzheimer's disease |
DE102004061288A1 (en) * | 2004-12-14 | 2006-06-29 | Schering Ag | New 3-amino-pyrazolo(3,4b)pyridine derivatives are protein tyrosine kinases inhibitors useful e.g. for treating hyperproliferation of body cells, neurodegenerative disease, blood vessel disease and angiogenic disease |
MX2007014114A (en) | 2005-05-10 | 2008-03-14 | Intermune Inc | Pyridone derivatives for modulating stress-activated protein kinase system. |
WO2007011760A2 (en) * | 2005-07-15 | 2007-01-25 | Kalypsys, Inc. | Inhibitors of mitotic kinesin |
ES2270715B1 (en) * | 2005-07-29 | 2008-04-01 | Laboratorios Almirall S.A. | NEW DERIVATIVES OF PIRAZINA. |
ES2274712B1 (en) * | 2005-10-06 | 2008-03-01 | Laboratorios Almirall S.A. | NEW IMIDAZOPIRIDINE DERIVATIVES. |
ES2273599B1 (en) | 2005-10-14 | 2008-06-01 | Universidad De Barcelona | COMPOUNDS FOR THE TREATMENT OF HEADPHONE FIBRILATION. |
TWI417095B (en) | 2006-03-15 | 2013-12-01 | Janssen Pharmaceuticals Inc | 1,4-disubstituted 3-cyano-pyridone derivatives and their use as positive allosteric modulators of mglur2-receptors |
US20080009623A1 (en) * | 2006-07-06 | 2008-01-10 | Eisai R&D Management Co., Ltd. | Pyrimidine compounds |
ES2303776B1 (en) * | 2006-12-29 | 2009-08-07 | Laboratorios Almirall S.A. | DERIVATIVES OF 5-PHENYL-6-PIRIDIN-4-IL-1,3-DIHIDRO-2H-IMIDAZO (4,5-B) PIRIDIN-2-ONA USEFUL AS ANTAGONISTS OF ADENOSINE A2B RECEIVER. |
TW200845978A (en) | 2007-03-07 | 2008-12-01 | Janssen Pharmaceutica Nv | 3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives |
TW200900065A (en) | 2007-03-07 | 2009-01-01 | Janssen Pharmaceutica Nv | 3-cyano-4-(4-pyridinyloxy-phenyl)-pyridin-2-one derivatives |
ES2356032T3 (en) | 2007-09-14 | 2011-04-04 | Ortho-Mcneil-Janssen Pharmaceuticals, Inc. | 4-PHENYL-3,4,5,6-TETRAHIDRO-2H, 1'H- [1,4 '] BIPIRIDINIL-2'-ONAS 1,3'-DISUSTITUTED. |
EA014100B1 (en) * | 2008-02-21 | 2010-08-30 | Общество С Ограниченной Ответственностью "Валексфарм" | 2,4-diaminopyridine derivatives, pharmaceutical composition, medicament based thereon for treating and preventing diseases and disorders caused by nmda-receptors hyperactivation and/or as stimulators of cognitive function and method of treatment |
ES2567283T3 (en) * | 2008-06-03 | 2016-04-21 | Intermune, Inc. | Compounds and methods to treat inflammatory and fibrotic disorders |
CN102232074B (en) | 2008-11-28 | 2014-12-03 | 奥梅-杨森制药有限公司 | Indole and benzoxazine derivatives as modulators of metabotropic glutamate receptors |
BRPI1010831A2 (en) | 2009-05-12 | 2016-04-05 | Addex Pharmaceuticals Sa | 1,2,4-triazolo [4,3-a] pyridine derivatives and their as positive allosteric modulators of mglur2 receptors |
MY153913A (en) | 2009-05-12 | 2015-04-15 | Janssen Pharmaceuticals Inc | 7-aryl-1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors |
MY161325A (en) | 2009-05-12 | 2017-04-14 | Janssen Pharmaceuticals Inc | 1, 2, 4-triazolo[4,3-a]pyridine derivatives and their use for the treatment or prevention of neurological and psychiatric disorders |
ES2552455T3 (en) | 2010-11-08 | 2015-11-30 | Janssen Pharmaceuticals, Inc. | 1,2,4-Triazolo [4,3-a] pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors |
WO2012062751A1 (en) | 2010-11-08 | 2012-05-18 | Janssen Pharmaceuticals, Inc. | 1,2,4-TRIAZOLO[4,3-a]PYRIDINE DERIVATIVES AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS |
ES2552879T3 (en) | 2010-11-08 | 2015-12-02 | Janssen Pharmaceuticals, Inc. | 1,2,4-Triazolo [4,3-a] pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors |
JP6215315B2 (en) * | 2012-06-12 | 2017-10-18 | アッヴィ・インコーポレイテッド | Pyridinone and pyridazinone derivatives |
AR092742A1 (en) | 2012-10-02 | 2015-04-29 | Intermune Inc | ANTIFIBROTIC PYRIDINONES |
BR112015007182A2 (en) * | 2012-10-05 | 2017-07-04 | Rigel Pharmaceuticals Inc | gdf-8 inhibitors |
TWI644899B (en) | 2013-02-04 | 2018-12-21 | 健生藥品公司 | Flap modulators |
EP2951170B1 (en) | 2013-02-04 | 2018-10-24 | Janssen Pharmaceutica NV | Flap modulators |
JO3368B1 (en) | 2013-06-04 | 2019-03-13 | Janssen Pharmaceutica Nv | 6,7-DIHYDROPYRAZOLO[1,5-a]PYRAZIN-4(5H)-ONE COMPOUNDS AND THEIR USE AS NEGATIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS |
ES2784489T3 (en) * | 2013-06-27 | 2020-09-28 | Lg Chemical Ltd | Biaryl derivatives as GPR120 agonists |
JO3367B1 (en) | 2013-09-06 | 2019-03-13 | Janssen Pharmaceutica Nv | 1,2,4-TRIAZOLO[4,3-a]PYRIDINE COMPOUNDS AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS |
EP3080132A4 (en) | 2013-12-10 | 2017-08-02 | AbbVie Inc. | Bromodomain inhibitors |
KR20200126026A (en) | 2014-01-21 | 2020-11-05 | 얀센 파마슈티카 엔.브이. | Combinations comprising positive allosteric modulators or orthosteric agonists of metabotropic glutamatergic receptor subtype 2 and their use |
EP3431106B1 (en) | 2014-01-21 | 2020-12-30 | Janssen Pharmaceutica NV | Combinations comprising positive allosteric modulators of metabotropic glutamatergic receptor subtype 2 and their use |
CN103804312B (en) * | 2014-02-17 | 2016-04-20 | 四川百利药业有限责任公司 | Aza cyclic cpds and its production and use |
EP3126362B1 (en) | 2014-04-02 | 2022-01-12 | Intermune, Inc. | Anti-fibrotic pyridinones |
ES2580702B1 (en) * | 2015-02-25 | 2017-06-08 | Palobiofarma, S.L. | 2-Aminopyridine derivatives as adenosine A2b receptor antagonists and MT3 melatonin receptor ligands |
JP2017149663A (en) * | 2016-02-24 | 2017-08-31 | 株式会社Lttバイオファーマ | Irritable bowel syndrome therapeutic agent |
MX2020003732A (en) * | 2017-09-28 | 2021-06-29 | Cstone Pharmaceuticals Suzhou Co Ltd | Fused ring derivative as a. |
JP7474709B2 (en) * | 2018-02-27 | 2024-04-25 | インサイト・コーポレイション | Imidazopyrimidines and triazolopyrimidines as A2A/A2B inhibitors |
CN110240593A (en) * | 2018-03-09 | 2019-09-17 | 四川科伦博泰生物医药股份有限公司 | Substituted aromatic amines compound and its preparation method and application |
CN111018858B (en) * | 2018-10-10 | 2022-11-18 | 复旦大学 | Heterocyclic derivative and preparation method and application thereof |
EP3904348A4 (en) * | 2018-12-28 | 2022-10-19 | Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd. | Aminopyridine compound, preparation method therefor and use thereof |
CN111035638A (en) * | 2019-06-24 | 2020-04-21 | 南开大学 | A medicine containing adenosine A1/A2AReceptor-selective adenosine A1Receptor antagonists |
WO2022150349A1 (en) * | 2021-01-06 | 2022-07-14 | The Penn State Research Foundation | Methods and materials for treating bone loss |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DD287260A5 (en) * | 1989-08-29 | 1991-02-21 | Akademie Der Wissenschaften Der Ddr,De | PROCESS FOR PREPARING 6-SUBSTITUTED 2-AMINO-3-CYAN-5- (PYRID-4-YL) -PYRIDINES |
DE4117802A1 (en) * | 1991-05-30 | 1992-12-03 | Berlin Chemie Ag | New 2-amino-pyridin-3-carbo:nitrile derivs. - used for treatment of human cytomegalovirus |
US5686470A (en) | 1995-02-10 | 1997-11-11 | Weier; Richard M. | 2, 3-substituted pyridines for the treatment of inflammation |
DE69821132T2 (en) * | 1997-10-27 | 2004-10-21 | Takeda Chemical Industries Ltd | 1,3-THIAZOLE AS ADENOSINE A3 RECEPTOR ANTAGONISTS FOR TREATING ASTHMA, ALLERGIES AND DIABETES |
JP3990061B2 (en) | 1998-01-05 | 2007-10-10 | エーザイ・アール・アンド・ディー・マネジメント株式会社 | Purine derivatives and adenosine A2 receptor antagonists as preventive and therapeutic agents for diabetes |
US6030969A (en) | 1998-04-09 | 2000-02-29 | Abbott Laboratories | 5,6,7-trisubstituted-4-aminopyrido[2,3-D] pyrimidine compounds |
-
2001
- 2001-08-09 CN CN01814043A patent/CN1446202A/en active Pending
- 2001-08-09 AT AT01955633T patent/ATE444752T1/en not_active IP Right Cessation
- 2001-08-09 EP EP01955633A patent/EP1308441B1/en not_active Expired - Lifetime
- 2001-08-09 JP JP2002519425A patent/JP4251868B2/en not_active Expired - Fee Related
- 2001-08-09 WO PCT/JP2001/006870 patent/WO2002014282A1/en active IP Right Grant
- 2001-08-09 KR KR1020037001943A patent/KR100804111B1/en not_active IP Right Cessation
- 2001-08-09 US US10/333,689 patent/US6750232B2/en not_active Expired - Fee Related
- 2001-08-09 IL IL15399501A patent/IL153995A0/en active IP Right Grant
- 2001-08-09 NZ NZ523998A patent/NZ523998A/en unknown
- 2001-08-09 CA CA002417846A patent/CA2417846A1/en not_active Abandoned
- 2001-08-09 AU AU7774101A patent/AU7774101A/en active Pending
- 2001-08-09 HU HU0700086A patent/HUP0700086A2/en unknown
- 2001-08-09 DE DE60140126T patent/DE60140126D1/en not_active Expired - Lifetime
- 2001-08-09 RU RU2003106397/04A patent/RU2250898C2/en not_active IP Right Cessation
- 2001-08-09 AU AU2001277741A patent/AU2001277741B2/en not_active Ceased
- 2001-08-09 MX MXPA03001136A patent/MXPA03001136A/en active IP Right Grant
- 2001-08-10 TW TW090119669A patent/TWI298064B/en not_active IP Right Cessation
-
2003
- 2003-01-16 IL IL153995A patent/IL153995A/en not_active IP Right Cessation
- 2003-01-17 ZA ZA200300482A patent/ZA200300482B/en unknown
- 2003-02-07 NO NO20030637A patent/NO325873B1/en not_active IP Right Cessation
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