AU2001262318A1 - Acylphenyl urea derivatives, methods for the production thereof and use thereof as a medicament - Google Patents

Acylphenyl urea derivatives, methods for the production thereof and use thereof as a medicament

Info

Publication number: AU2001262318A1
Authority: AU; Australia
Prior art keywords: acylphenyl; medicament; production; methods; urea derivatives
Prior art date: 2000-06-09
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

AU2001262318A

Other versions

AU2001262318B2 (en

Inventor

Karl-Heinz Baringhaus

Hans-Joerg Burger

Elisabeth Defossa

Andreas Herling

Thomas Klabunde

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Sanofi Aventis Deutschland GmbH

Original Assignee

Sanofi Aventis Deutschland GmbH

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-06-09

Filing date

2001-05-26

Publication date

2002-03-07

2001-04-04 Priority claimed from DE2001116768 external-priority patent/DE10116768A1/en

2001-05-26 Application filed by Sanofi Aventis Deutschland GmbH filed Critical Sanofi Aventis Deutschland GmbH

2001-05-26 Priority claimed from PCT/EP2001/006030 external-priority patent/WO2001094300A1/en

2002-03-07 Publication of AU2001262318A1 publication Critical patent/AU2001262318A1/en

2005-09-08 Application granted granted Critical

2005-09-08 Publication of AU2001262318B2 publication Critical patent/AU2001262318B2/en

2005-12-15 Assigned to SANOFI-AVENTIS DEUTSCHLAND GMBH reassignment SANOFI-AVENTIS DEUTSCHLAND GMBH Request for Assignment Assignors: AVENTIS PHARMA DEUTSCHLAND GMBH

2021-05-26 Anticipated expiration legal-status Critical

Status Ceased legal-status Critical Current

Applications Claiming Priority (5)

Application Number	Priority Date	Filing Date	Title
DE10028175.3		2000-06-09
DE10028175		2000-06-09
DE2001116768 DE10116768A1 (en)	2001-04-04	2001-04-04	Hypoglycemic medicaments useful for treating type II diabetes contain new or known N-aroyl-N'-phenyl-urea derivatives which are glycogen phosphorylase a inhibitors
DE10116768.7		2001-04-04
PCT/EP2001/006030 WO2001094300A1 (en)	2000-06-09	2001-05-26	Acylphenyl urea derivatives, methods for the production thereof and use thereof as a medicament

Publications (2)

Publication Number	Publication Date
AU2001262318A1 true AU2001262318A1 (en)	2002-03-07
AU2001262318B2 AU2001262318B2 (en)	2005-09-08

Family

ID=26005991

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
AU2001262318A Ceased AU2001262318B2 (en)	2000-06-09	2001-05-26	Acylphenyl urea derivatives, methods for the production thereof and use thereof as a medicament
AU6231801A Pending AU6231801A (en)	2000-06-09	2001-05-26	Acylphenyl urea derivatives, methods for the production thereof and use thereof as a medicament

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
AU6231801A Pending AU6231801A (en)	2000-06-09	2001-05-26	Acylphenyl urea derivatives, methods for the production thereof and use thereof as a medicament

Country Status (28)

Country	Link
US (1)	US6506778B2 (en)
EP (1)	EP1294682B1 (en)
JP (1)	JP4510372B2 (en)
KR (1)	KR20030007934A (en)
CN (1)	CN1280266C (en)
AR (1)	AR030230A1 (en)
AT (1)	ATE265424T1 (en)
AU (2)	AU2001262318B2 (en)
BR (1)	BR0111457A (en)
CA (1)	CA2411082A1 (en)
CZ (1)	CZ20024003A3 (en)
DE (1)	DE50102147D1 (en)
DK (1)	DK1294682T3 (en)
EE (1)	EE200200634A (en)
ES (1)	ES2215902T3 (en)
HK (1)	HK1056715A1 (en)
HR (1)	HRP20020968A2 (en)
HU (1)	HUP0301749A2 (en)
IL (1)	IL153273A0 (en)
MX (1)	MXPA02011458A (en)
NO (1)	NO20025879L (en)
NZ (1)	NZ523034A (en)
PL (1)	PL359178A1 (en)
PT (1)	PT1294682E (en)
SK (1)	SK17252002A3 (en)
TR (1)	TR200401029T4 (en)
WO (1)	WO2001094300A1 (en)
YU (1)	YU91002A (en)

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DE10225635C1 (en) *	2002-06-07	2003-12-24	Aventis Pharma Gmbh	N-benzoylureido-cinnamic acid derivatives, process for their preparation and their use
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NZ537603A (en)	2002-07-12	2006-09-29	Sanofi Aventis Deutschland	Heterocyclically substituted benzoylureas, method for their production and their use as medicaments
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DE10246434B4 (en) *	2002-10-04	2005-08-04	Aventis Pharma Deutschland Gmbh	Carboxyalkoxy-substituted acyl-carboxyphenyl-urea derivatives and their use as pharmaceuticals
US20040157922A1 (en) *	2002-10-04	2004-08-12	Aventis Pharma Deutschland Gmbh	Carboxyalkoxy-substituted acyl-carboxyphenylurea derivatives and their use as medicaments
US7179941B2 (en) *	2003-01-23	2007-02-20	Sanofi-Aventis Deutschland Gmbh	Carbonylamino-substituted acyl phenyl urea derivatives, process for their preparation and their use
DE10302452B4 (en) *	2003-01-23	2005-02-24	Aventis Pharma Deutschland Gmbh	Carbonylamino-substituted acyl-phenyl-urea derivatives, processes for their preparation and their use
US7196114B2 (en) *	2003-02-17	2007-03-27	Sanofi-Aventis Deutschland Gmbh	Substituted 3-(benzoylureido) thiophene derivatives, processes for preparing them and their use
DE10306502B4 (en) *	2003-02-17	2005-03-17	Aventis Pharma Deutschland Gmbh	Substituted 3- (benzoylureido) thiophene derivatives and medicaments containing them
US7148246B2 (en)	2003-02-27	2006-12-12	Sanofi-Aventis Deutschland Gmbh	Cycloalkyl derivatives having bioisosteric carboxylic acid groups, processes for their preparation and their use as pharmaceuticals
DE10308351A1 (en) *	2003-02-27	2004-11-25	Aventis Pharma Deutschland Gmbh	1,3-substituted cycloalkyl derivatives having acidic, usually heterocyclic groups, processes for their preparation and their use as medicaments
DE10308355A1 (en) *	2003-02-27	2004-12-23	Aventis Pharma Deutschland Gmbh	Aryl-cycloalkyl-substituted alkanoic acid derivatives, process for their preparation and their use as medicaments
DE10308352A1 (en)	2003-02-27	2004-09-09	Aventis Pharma Deutschland Gmbh	Branched side chain arylcycloalkyl derivatives, process for their preparation and their use as medicaments
DE10308353A1 (en)	2003-02-27	2004-12-02	Aventis Pharma Deutschland Gmbh	Diarylcycloalkyl derivatives, processes for their preparation and their use as medicines
DE10309929B4 (en) *	2003-03-07	2006-02-23	Sanofi-Aventis Deutschland Gmbh	Substituted benzoylureidopyridyl-piperidine and -pyrrolidine-carboxylic acid derivatives, process for their preparation and their use
US7501440B2 (en)	2003-03-07	2009-03-10	Sanofi-Aventis Deutschland Gmbh	Substituted benzoylureidopyridylpiperidine-and-pyrrolidinecarboxylic acid derivatives, processes for preparing them and their use
DE10335092B3 (en)	2003-08-01	2005-02-03	Aventis Pharma Deutschland Gmbh	Substituted benzoylureido-o-benzoylamides, process for their preparation and their use
US7241787B2 (en)	2004-01-25	2007-07-10	Sanofi-Aventis Deutschland Gmbh	Substituted N-cycloexylimidazolinones, process for their preparation and their use as medicaments
EP1586573B1 (en)	2004-04-01	2007-02-07	Sanofi-Aventis Deutschland GmbH	Oxadiazolones, processes for their preparation and their use as pharmaceuticals
US7963448B2 (en) *	2004-12-22	2011-06-21	Cognex Technology And Investment Corporation	Hand held machine vision method and apparatus
JP2008536932A (en) *	2005-04-18	2008-09-11	サイード・アール・カーン	Tubulin polymerization inhibitors: design and synthesis of bonzoylphenylurea (BPU) sulfur analogues
WO2006126695A1 (en) *	2005-05-23	2006-11-30	Japan Tobacco Inc.	Pyrazole compound and therapeutic agent for diabetes comprising the same
DE102005026762A1 (en)	2005-06-09	2006-12-21	Sanofi-Aventis Deutschland Gmbh	Azolopyridin-2-one derivatives as inhibitors of lipases and phospholipases
PE20110235A1 (en)	2006-05-04	2011-04-14	Boehringer Ingelheim Int	PHARMACEUTICAL COMBINATIONS INCLUDING LINAGLIPTIN AND METMORPHINE
WO2008062739A1 (en) *	2006-11-20	2008-05-29	Japan Tobacco Inc.	Pyrazoles and use thereof as drugs
US8969514B2 (en)	2007-06-04	2015-03-03	Synergy Pharmaceuticals, Inc.	Agonists of guanylate cyclase useful for the treatment of hypercholesterolemia, atherosclerosis, coronary heart disease, gallstone, obesity and other cardiovascular diseases
US9616097B2 (en)	2010-09-15	2017-04-11	Synergy Pharmaceuticals, Inc.	Formulations of guanylate cyclase C agonists and methods of use
EP4424697A2 (en)	2013-06-05	2024-09-04	Bausch Health Ireland Limited	Ultra-pure agonists of guanylate cyclase c, method of making and using same
WO2016030534A1 (en)	2014-08-29	2016-03-03	Tes Pharma S.R.L.	INHIBITORS OF α-AMINO-β-CARBOXYMUCONIC ACID SEMIALDEHYDE DECARBOXYLASE
AU2017342083A1 (en)	2016-10-14	2019-04-11	Tes Pharma S.R.L.	Inhibitors of alpha-amino-beta-carboxymuconic acid semialdehyde decarboxylase
CN113302189A (en)	2018-11-20	2021-08-24	Tes制药有限责任公司	Inhibitors of alpha-amino-beta-carboxyadipimic acid semialdehyde decarboxylating enzyme

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ZA793186B (en) *	1978-07-06	1981-02-25	Duphar Int Res	New urea and thiourea compounds, method of preparing the new compounds, as well as insecticidal compositions on the basis of these compounds
DE3478573D1 (en) *	1983-09-01	1989-07-13	Duphar Int Res	Benzoyl urea derivatives having anti-tumor activity
JPS60237056A (en) *	1984-05-08	1985-11-25	Ishihara Sangyo Kaisha Ltd	N-benzoyl-n'-phenylurea based compound and insecticide containing same
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DE3504749A1 (en) *	1985-02-08	1986-08-14	Schering AG, 1000 Berlin und 4709 Bergkamen	Acyl ureas, insecticidal agents containing these compounds, and processes for their preparation
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2001
- 2001-05-26 NZ NZ523034A patent/NZ523034A/en unknown
- 2001-05-26 MX MXPA02011458A patent/MXPA02011458A/en active IP Right Grant
- 2001-05-26 AT AT01936399T patent/ATE265424T1/en not_active IP Right Cessation
- 2001-05-26 EE EEP200200634A patent/EE200200634A/en unknown
- 2001-05-26 KR KR1020027016791A patent/KR20030007934A/en not_active Application Discontinuation
- 2001-05-26 CA CA002411082A patent/CA2411082A1/en not_active Abandoned
- 2001-05-26 AU AU2001262318A patent/AU2001262318B2/en not_active Ceased
- 2001-05-26 CZ CZ20024003A patent/CZ20024003A3/en unknown
- 2001-05-26 PT PT01936399T patent/PT1294682E/en unknown
- 2001-05-26 ES ES01936399T patent/ES2215902T3/en not_active Expired - Lifetime
- 2001-05-26 HU HU0301749A patent/HUP0301749A2/en unknown
- 2001-05-26 IL IL15327301A patent/IL153273A0/en unknown
- 2001-05-26 EP EP01936399A patent/EP1294682B1/en not_active Expired - Lifetime
- 2001-05-26 PL PL01359178A patent/PL359178A1/en not_active Application Discontinuation
- 2001-05-26 CN CNB018108016A patent/CN1280266C/en not_active Expired - Fee Related
- 2001-05-26 DK DK01936399T patent/DK1294682T3/en active
- 2001-05-26 SK SK1725-2002A patent/SK17252002A3/en unknown
- 2001-05-26 TR TR2004/01029T patent/TR200401029T4/en unknown
- 2001-05-26 WO PCT/EP2001/006030 patent/WO2001094300A1/en active IP Right Grant
- 2001-05-26 YU YU91002A patent/YU91002A/en unknown
- 2001-05-26 JP JP2002501817A patent/JP4510372B2/en not_active Expired - Fee Related
- 2001-05-26 BR BR0111457-3A patent/BR0111457A/en not_active IP Right Cessation
- 2001-05-26 AU AU6231801A patent/AU6231801A/en active Pending
- 2001-05-26 DE DE50102147T patent/DE50102147D1/en not_active Expired - Lifetime
- 2001-06-07 AR ARP010102735A patent/AR030230A1/en unknown
- 2001-06-08 US US09/875,901 patent/US6506778B2/en not_active Expired - Lifetime
2002
- 2002-12-06 NO NO20025879A patent/NO20025879L/en not_active Application Discontinuation
- 2002-12-06 HR HR20020968A patent/HRP20020968A2/en not_active Application Discontinuation
2003
- 2003-12-11 HK HK03109010A patent/HK1056715A1/en not_active IP Right Cessation

Publication	Publication Date	Title
AU2001262318A1 (en)	2002-03-07	Acylphenyl urea derivatives, methods for the production thereof and use thereof as a medicament
AU6231801A (en)	2001-12-17	Acylphenyl urea derivatives, methods for the production thereof and use thereof as a medicament
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AU2002219174A1 (en)	2002-09-05	Quinazoline derivatives, medicaments containing said compounds, their utilization and method for the production thereof
ZA200305498B (en)	2004-05-07	Xanthine derivative, production and use thereof as a medicament.
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AU2001284021A1 (en)	2002-03-13	Quinazoline derivatives, medicaments containing these compounds, their use, and methods for the production thereof
AU2003282094A1 (en)	2004-06-15	Novel dihydroxy-methylphenyl derivatives, method for the production and use thereof as medicaments
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SI1294682T1 (en)	2004-10-31	Acylphenyl urea derivatives, methods for the production thereof and use thereof as a medicament
AU2002333449A1 (en)	2003-06-05	C2-substituted indane-1-ols and their derivatives, method for their production and their use as medicaments
AU2002336983A1 (en)	2003-06-05	C2-disubstituted Indane-1-ones and their derivatives, method for their production and their use as medicaments