ATE544766T1 - Verfahren zur synthese von paliperidon - Google Patents

Verfahren zur synthese von paliperidon

Info

Publication number: ATE544766T1
Authority: AT; Austria
Prior art keywords: paliperidone; synthesis; purification; invention describes; improved process
Prior art date: 2009-07-13

Application number

AT09009122T

Other languages

English (en)

Inventor

Milos Ruzic

Anica Pecavar

Darja Prudic

Igor Plaper

Andrej Klobcar

Jernej Hvala

Miha Plevnik

Original Assignee

Krka

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2009-07-13

Filing date

2009-07-13

Publication date

2012-02-15

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41050429&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ATE544766(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2009-07-13 Application filed by Krka filed Critical Krka

2012-02-15 Application granted granted Critical

2012-02-15 Publication of ATE544766T1 publication Critical patent/ATE544766T1/de

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Neurology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Biomedical Technology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Neurosurgery (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Psychiatry (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

AT09009122T 2009-07-13 2009-07-13 Verfahren zur synthese von paliperidon ATE544766T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
EP09009122A EP2275423B9 (de)	2009-07-13	2009-07-13	Verfahren zur Synthese von Paliperidon

Publications (1)

Publication Number	Publication Date
ATE544766T1 true ATE544766T1 (de)	2012-02-15

Family

ID=41050429

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT09009122T ATE544766T1 (de)	2009-07-13	2009-07-13	Verfahren zur synthese von paliperidon

Country Status (4)

Country	Link
EP (2)	EP2275423B9 (de)
AT (1)	ATE544766T1 (de)
SI (2)	SI2275423T1 (de)
WO (1)	WO2011006638A1 (de)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO2012035554A1 (en) *	2010-09-14	2012-03-22	Megafine Pharma (P) Ltd.	An improved process for the preparation of highly pure paliperidone
AU2012264476B2 (en)	2011-05-30	2016-12-08	Cipla Limited	Process for the preparation of paliperidone

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE3148379A1 (de)	1981-12-07	1983-06-09	Hunter Douglas Industries B.V., 3008 Rotterdam	"lamellenjalousie mit vertikalen lamellen"
US4804663A (en)	1985-03-27	1989-02-14	Janssen Pharmaceutica N.V.	3-piperidinyl-substituted 1,2-benzisoxazoles and 1,2-benzisothiazoles
CA2000786C (en)	1988-11-07	1999-01-26	Cornelus G. M. Janssen	3-piperidinyl-1,2-benzisoxazoles
US5158952A (en)	1988-11-07	1992-10-27	Janssen Pharmaceutica N.V.	3-[2-[4-(6-fluoro-1,2-benzisoxozol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9 tetrahydro-9-hydroxy-2-methyl-4H-pyrido [1,2-a]pyrimidin-4-one, compositions and method of use
FR2654104B1 (fr)	1989-11-07	1992-01-03	Adir	Nouveaux derives du 1,2-benzisoxazole, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent.
EP1922319A2 (de)	2006-08-14	2008-05-21	Teva Pharmaceutical Industries Ltd.	Reines paliperidon und verfahren zu dessen herstellung
DE202007018473U1 (de)	2006-08-14	2008-08-07	Teva Pharmaceutical Industries Ltd.	9-Hydroxy-Risperidon (Paliperidon)
US7820816B2 (en)	2006-08-23	2010-10-26	Teva Pharmaceutical Industries Ltd.	Process for the synthesis of CMHTP and intermediates thereof
EP1924583A2 (de)	2006-08-23	2008-05-28	Teva Pharmaceutical Industries Ltd.	Verfahren zur herstellung von cmhtp und zwischenprodukte dafür
WO2009010988A1 (en)	2007-07-19	2009-01-22	Natco Pharma Limited	An improved, industrially viable process for the preparation of high purity paliperidone
WO2009045489A2 (en)	2007-10-03	2009-04-09	Teva Pharmaceutical Industries Ltd.	Process for the synthesis of cmhtp, a paliperidone intermediate
EP2195318A2 (de)	2007-10-09	2010-06-16	Cipla Limited	Verfahren zur herstellung von paliperidon und pharmazeutisch akzeptable salze daraus sowie zwischenprodukte zur verwendung in den verfahren

2009
- 2009-07-13 AT AT09009122T patent/ATE544766T1/de active
- 2009-07-13 SI SI200930239T patent/SI2275423T1/sl unknown
- 2009-07-13 EP EP09009122A patent/EP2275423B9/de active Active
2010
- 2010-07-13 SI SI201031073T patent/SI2454256T1/sl unknown
- 2010-07-13 EP EP10732311.5A patent/EP2454256B1/de not_active Revoked
- 2010-07-13 WO PCT/EP2010/004258 patent/WO2011006638A1/en active Application Filing

Also Published As

Publication number	Publication date
EP2275423B8 (de)	2012-06-20
EP2275423B9 (de)	2012-08-15
EP2454256A1 (de)	2012-05-23
SI2275423T1 (sl)	2012-06-29
EP2454256B1 (de)	2015-09-16
WO2011006638A1 (en)	2011-01-20
EP2275423B1 (de)	2012-02-08
EP2275423A1 (de)	2011-01-19
SI2454256T1 (sl)	2016-01-29

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