ATE421964T1 - Radioaktiv markierte antagonisten des neuropeptid y y5-rezeptors - Google Patents
Radioaktiv markierte antagonisten des neuropeptid y y5-rezeptorsInfo
- Publication number
- ATE421964T1 ATE421964T1 AT02750193T AT02750193T ATE421964T1 AT E421964 T1 ATE421964 T1 AT E421964T1 AT 02750193 T AT02750193 T AT 02750193T AT 02750193 T AT02750193 T AT 02750193T AT E421964 T1 ATE421964 T1 AT E421964T1
- Authority
- AT
- Austria
- Prior art keywords
- neuropeptide
- receptor
- radioactively labeled
- antagonists
- labeled antagonists
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K51/00—Preparations containing radioactive substances for use in therapy or testing in vivo
- A61K51/02—Preparations containing radioactive substances for use in therapy or testing in vivo characterised by the carrier, i.e. characterised by the agent or material covalently linked or complexing the radioactive nucleus
- A61K51/04—Organic compounds
- A61K51/041—Heterocyclic compounds
- A61K51/044—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
- A61K51/0459—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having six-membered rings with two nitrogen atoms as the only ring hetero atoms, e.g. piperazine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/05—Isotopically modified compounds, e.g. labelled
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Optics & Photonics (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- Physics & Mathematics (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Oscillators With Electromechanical Resonators (AREA)
- Steroid Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US30749901P | 2001-07-24 | 2001-07-24 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE421964T1 true ATE421964T1 (de) | 2009-02-15 |
Family
ID=23190036
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT02750193T ATE421964T1 (de) | 2001-07-24 | 2002-07-19 | Radioaktiv markierte antagonisten des neuropeptid y y5-rezeptors |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US6939966B2 (de) |
| EP (1) | EP1470129B1 (de) |
| JP (1) | JP4554202B2 (de) |
| AT (1) | ATE421964T1 (de) |
| CA (1) | CA2454228C (de) |
| DE (1) | DE60231062D1 (de) |
| WO (1) | WO2003010175A2 (de) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6803372B2 (en) * | 1999-08-20 | 2004-10-12 | Banyu Pharmaceutical Co., Ltd. | Spiro compounds |
| EA006964B1 (ru) * | 2001-08-07 | 2006-06-30 | Баниу Фармасьютикал Ко., Лтд. | Спиросоединения |
| WO2006082497A1 (en) * | 2005-02-01 | 2006-08-10 | Ge Healthcare Limited | Method for the use of [11c] carbon monoxide in labeling synthesis of 11c-labelled compounds by thermally induced free radical carbonylation |
| US7834031B2 (en) * | 2005-09-29 | 2010-11-16 | Merck Sharp & Dohme Corp. | Radiolabeled glycine transporter inhibitors |
| CN101918408A (zh) | 2007-11-30 | 2010-12-15 | 惠氏有限责任公司 | 作为磷酸二酯酶10的抑制剂的芳基和杂芳基稠合的咪唑并[1,5-a]吡嗪 |
| WO2010101247A1 (ja) | 2009-03-05 | 2010-09-10 | 塩野義製薬株式会社 | Ｎｐｙ ｙ５受容体拮抗作用を有するシクロヘキサン誘導体 |
| WO2010138833A1 (en) | 2009-05-29 | 2010-12-02 | Wyeth | SUBSTITUTED IMIDAZO[1,5-a]QUINOXALINES AS INHIBITORS OF PHOSPHODIESTERASE 10 |
| JP2012196144A (ja) | 2009-08-03 | 2012-10-18 | Ajinomoto Co Inc | ビブリオ属細菌を用いたｌ−リジンの製造法 |
| CA2799708A1 (en) | 2010-05-21 | 2011-11-24 | Pfizer Inc. | 2-phenyl benzoylamides |
| US20120039804A1 (en) * | 2010-06-04 | 2012-02-16 | Philippe Diaz | Novel Tricyclic Modulators of Cannabinoid Receptors |
| JP2014513923A (ja) | 2011-03-04 | 2014-06-19 | ファイザー・インク | Ｅｄｎ３様ペプチドおよびその使用 |
| JP6740051B2 (ja) * | 2016-07-26 | 2020-08-12 | キヤノンメディカルシステムズ株式会社 | 超音波診断装置、医用画像処理装置及び医用画像処理プログラム |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5569742A (en) * | 1994-06-22 | 1996-10-29 | The Salk Institute For Biological Studies | Centrally truncated NPY cyclic peptides |
| TWI279402B (en) * | 1999-08-20 | 2007-04-21 | Banyu Pharma Co Ltd | Spiro compounds having NPY antagonistic activities and agents containing the same |
-
2002
- 2002-07-19 AT AT02750193T patent/ATE421964T1/de not_active IP Right Cessation
- 2002-07-19 CA CA2454228A patent/CA2454228C/en not_active Expired - Fee Related
- 2002-07-19 US US10/484,551 patent/US6939966B2/en not_active Expired - Fee Related
- 2002-07-19 EP EP02750193A patent/EP1470129B1/de not_active Expired - Lifetime
- 2002-07-19 DE DE60231062T patent/DE60231062D1/de not_active Expired - Lifetime
- 2002-07-19 WO PCT/US2002/023044 patent/WO2003010175A2/en active Application Filing
- 2002-07-19 JP JP2003515534A patent/JP4554202B2/ja not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| JP4554202B2 (ja) | 2010-09-29 |
| US6939966B2 (en) | 2005-09-06 |
| EP1470129B1 (de) | 2009-01-28 |
| WO2003010175A2 (en) | 2003-02-06 |
| EP1470129A2 (de) | 2004-10-27 |
| WO2003010175A3 (en) | 2004-05-27 |
| US20040192705A1 (en) | 2004-09-30 |
| CA2454228C (en) | 2011-03-22 |
| CA2454228A1 (en) | 2003-02-06 |
| JP2005501830A (ja) | 2005-01-20 |
| EP1470129A4 (de) | 2007-08-01 |
| DE60231062D1 (de) | 2009-03-19 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |