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ATE164839T1 - Retrovirale proteaseinhibitoren - Google Patents

Retrovirale proteaseinhibitoren

Info

Publication number
ATE164839T1
ATE164839T1 AT92901068T AT92901068T ATE164839T1 AT E164839 T1 ATE164839 T1 AT E164839T1 AT 92901068 T AT92901068 T AT 92901068T AT 92901068 T AT92901068 T AT 92901068T AT E164839 T1 ATE164839 T1 AT E164839T1
Authority
AT
Austria
Prior art keywords
protease inhibitors
retroviral protease
inhibitors
retroviral
protease
Prior art date
Application number
AT92901068T
Other languages
English (en)
Inventor
Michael Clare
Gary Anthony Decrescenzo
John Nicholas Freskos
Daniel Paul Getman
Robert Martin Heintz
Ko-Chung Lin
Richard August Mueller
Kathryn Lea Reed
John Jeffrey Talley
Michael Lawrence Vazquez
Eric Tak Sun
Original Assignee
Monsanto Co
Searle & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Monsanto Co, Searle & Co filed Critical Monsanto Co
Application granted granted Critical
Publication of ATE164839T1 publication Critical patent/ATE164839T1/de

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    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
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    • C07K5/06Dipeptides
    • C07K5/06191Dipeptides containing heteroatoms different from O, S, or N
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/17Amides, e.g. hydroxamic acids having the group >N—C(O)—N< or >N—C(S)—N<, e.g. urea, thiourea, carmustine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
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    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
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    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/216Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acids having aromatic rings, e.g. benactizyne, clofibrate
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AT92901068T 1990-11-19 1991-11-18 Retrovirale proteaseinhibitoren ATE164839T1 (de)

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AT97105350T ATE296624T1 (de) 1990-11-19 1991-11-18 Retrovirusprotease inhibitoren
AT92900449T ATE170169T1 (de) 1990-11-19 1991-11-18 Retrovirale protease inhibitoren
AT97105351T ATE296626T1 (de) 1990-11-19 1991-11-18 Retrovirusprotease inhibitoren
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AT97105351T ATE296626T1 (de) 1990-11-19 1991-11-18 Retrovirusprotease inhibitoren
AT97105352T ATE296625T1 (de) 1990-11-19 1991-11-18 Retrovirusprotease inhibitoren

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ATE296626T1 (de) 2005-06-15
AU661667B2 (en) 1995-08-03
ATE170169T1 (de) 1998-09-15
ES2243960T3 (es) 2005-12-01
DE69133463D1 (de) 2005-07-07
EP0558630B1 (de) 1998-04-08
ZA919162B (en) 1993-08-19
IL100084A0 (en) 1992-08-18
PT99552A (pt) 1994-01-31
DK0815856T3 (da) 2005-10-03
CA2096525C (en) 2005-02-08
EP0813868A3 (de) 1998-03-18
DE69129235D1 (de) 1998-05-14
DE69130070D1 (de) 1998-10-01
MX9102137A (es) 1994-03-31
WO1992008701A1 (en) 1992-05-29
ES2243959T3 (es) 2005-12-01
ES2059295T3 (es) 1998-06-01
ZA919163B (en) 1993-05-19
EP0815856A2 (de) 1998-01-07
DE69133464T2 (de) 2006-05-18
EP0558630A1 (de) 1993-09-08
EP0813868A2 (de) 1997-12-29
PT99554A (pt) 1992-10-30
ES2059293T3 (es) 1998-12-16
JPH06502860A (ja) 1994-03-31
ATE296624T1 (de) 2005-06-15
ES2059295T1 (es) 1994-11-16
PT99553A (pt) 1992-10-30
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ZA919161B (en) 1993-08-19
CA2096409C (en) 2005-02-08
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DE69129235T2 (de) 1998-11-12
ATE296625T1 (de) 2005-06-15
WO1992008688A1 (en) 1992-05-29
EP0815856B1 (de) 2005-06-01
EP0813868B1 (de) 2005-06-01
HU9301447D0 (en) 1993-11-29
DE69130070T2 (de) 1999-04-29
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MX9102136A (es) 1994-01-31
ZA919160B (en) 1993-08-19
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