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AT230379B - Process for the preparation of 2,4-diamino-5-arylmethylpyrimidines - Google Patents

Process for the preparation of 2,4-diamino-5-arylmethylpyrimidines

Info

Publication number
AT230379B
AT230379B AT656060A AT656060A AT230379B AT 230379 B AT230379 B AT 230379B AT 656060 A AT656060 A AT 656060A AT 656060 A AT656060 A AT 656060A AT 230379 B AT230379 B AT 230379B
Authority
AT
Austria
Prior art keywords
arylmethylpyrimidines
diamino
preparation
Prior art date
Application number
AT656060A
Other languages
German (de)
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27258299&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=AT230379(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Wellcome Found filed Critical Wellcome Found
Application granted granted Critical
Publication of AT230379B publication Critical patent/AT230379B/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/44—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D317/46—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 ortho- or peri-condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C07D317/48—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring
    • C07D317/50—Methylenedioxybenzenes or hydrogenated methylenedioxybenzenes, unsubstituted on the hetero ring with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to atoms of the carbocyclic ring
    • C07D317/60—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyridine Compounds (AREA)
AT656060A 1959-09-03 1960-08-29 Process for the preparation of 2,4-diamino-5-arylmethylpyrimidines AT230379B (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB3010259A GB957797A (en) 1959-09-03 1959-09-03 Method for making 2,4-diamino-5-arylmethylpyrimidines and intermediates therefor
GB3956059 1959-11-20
GB2410160 1960-07-11

Publications (1)

Publication Number Publication Date
AT230379B true AT230379B (en) 1963-12-10

Family

ID=27258299

Family Applications (1)

Application Number Title Priority Date Filing Date
AT656060A AT230379B (en) 1959-09-03 1960-08-29 Process for the preparation of 2,4-diamino-5-arylmethylpyrimidines

Country Status (7)

Country Link
AT (1) AT230379B (en)
CH (1) CH418338A (en)
DE (2) DE1445176C3 (en)
FI (1) FI42960B (en)
GB (1) GB957797A (en)
IT (1) IT1061608B (en)
MY (1) MY6600061A (en)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT385033B (en) * 1981-06-26 1988-02-10 Egyt Gyogyszervegyeszeti Gyar METHOD FOR PRODUCING 2,4-DIAMINO-5 (3 ', 4', 5'-TRIMETHOXY-BENZYL) -PYRIMIDINE
AT387961B (en) * 1981-06-26 1989-04-10 Egyt Gyogyszervegyeszeti Gyar METHOD FOR PRODUCING ALPHA- (3,4,5-TRIMETHOXYBENZYL)-BETA- (2ALKOXY | THOXY) -ACRYLNITRILES

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3485840A (en) * 1964-11-12 1969-12-23 Hoffmann La Roche 2,4-diamino - 5 - (2',4',5'-substituted benzyl) pyrimidines,intermediates and processes
US3855265A (en) * 1969-03-06 1974-12-17 Burroughs Wellcome Co 5-benzyl pyrimidines intermediates therefore, and method
US3998814A (en) 1969-03-06 1976-12-21 Burroughs Wellcome Co. Process for preparing β-amino-α-benzylacrylonitriles
US3852276A (en) * 1969-03-06 1974-12-03 Burroughs Wellcome Co 5-benzyl pyrimidines intermediate therefore, and method
US3950378A (en) * 1969-03-06 1976-04-13 Burroughs Wellcome Co. Preparation of β-anilino-α-benzylacrylonitriles
DE2065367C2 (en) * 1969-03-06 1985-04-04 The Wellcome Foundation Ltd., London Process for the preparation of 2,4-diamino-5-benzylpyrimidines
US3991050A (en) * 1969-03-06 1976-11-09 Burroughs Wellcome Co. Preparation of β-Amino-α-benzylacrylonitriles
GB1261455A (en) * 1969-03-06 1972-01-26 Burroughs Wellcome Co Improvements in or relating to substituted acrylonitriles
US4052553A (en) * 1969-03-06 1977-10-04 Burroughs Wellcome Co. 5-benzyl pyrimidines intermediates therefore, and method
DE2051871A1 (en) * 1969-05-16 1971-11-18 The Wellcome Foundation Ltd., London Beta-amino-alpha-aryloxymethylacrylonitrile - and 2,4-diamino-5-benzylpyrimidine derivs. useful as antibacterial agents
BR6915082D0 (en) 1969-05-16 1973-03-08 Wellcome Found PROCESS OF PREPARATION OF BENZYL-PYRIMIDINES
BE789904A (en) * 1971-10-12 1973-04-10 Wellcome Found ORGANIC SYNTHESIS PROCESSES
BE792096A (en) * 1971-12-01 1973-05-30 Hoffmann La Roche NEW BENZYLPYRIMIDINES
US4039543A (en) 1974-12-24 1977-08-02 Hoffmann-La Roche Inc. Benzylpyrimidines
CH624943A5 (en) * 1977-02-04 1981-08-31 Hoffmann La Roche
DE2720771C3 (en) 1977-05-09 1979-11-29 Ludwig Heumann & Co Gmbh, 8500 Nuernberg 2,4-Diamino-5- (33-dimethoxy-4thioalkyl-benzyD-pyrimidines, process for their preparation and pharmaceuticals containing these compounds
EP0046856A3 (en) * 1980-08-29 1982-07-28 Hüls Troisdorf Aktiengesellschaft Process for preparing 4-amino-2-mercapto-pyrimidines
US4438267A (en) 1980-11-11 1984-03-20 Daluge Susan M Monoheteroring compounds and their use
AT384023B (en) * 1980-11-11 1987-09-25 Wellcome Found METHOD FOR PRODUCING NEW 2,4-DIAMINO-5- (SUBST.) PYRIMIDINES AND THEIR SALTS, N-OXIDES AND N-ACYL DERIVATIVES
DK190983A (en) * 1982-05-01 1983-11-02 Wellcome Found 2,4-DIAMINO-5- (SUBSTITUTED) PYRIMIDINES, PROCEDURES FOR THEIR PREPARATION AND INTERMEDIATES
US4587341A (en) * 1982-05-07 1986-05-06 Burroughs Wellcome Co. 2,4-diamino-5-(1,2,3,4-tetrahydro-(substituted or unsubstituted)-6-quinolylmethyl)pyrimidines, useful as antimicrobials
DE3603577A1 (en) * 1986-02-06 1987-08-13 Joachim K Prof Dr Seydel NEW SUBSTITUTED 2,4-DIAMINO-5-BENZYLPYRIMIDINE, THEIR PRODUCTION AND USE THEREOF AS A MEDICINE WITH ANTIBACTERIAL EFFECTIVENESS
FI895821A0 (en) * 1988-12-07 1989-12-05 Wellcome Found PHARMACEUTICAL ACTIVE CNS FOERENINGAR.

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AT385033B (en) * 1981-06-26 1988-02-10 Egyt Gyogyszervegyeszeti Gyar METHOD FOR PRODUCING 2,4-DIAMINO-5 (3 ', 4', 5'-TRIMETHOXY-BENZYL) -PYRIMIDINE
AT387961B (en) * 1981-06-26 1989-04-10 Egyt Gyogyszervegyeszeti Gyar METHOD FOR PRODUCING ALPHA- (3,4,5-TRIMETHOXYBENZYL)-BETA- (2ALKOXY | THOXY) -ACRYLNITRILES

Also Published As

Publication number Publication date
IT1061608B (en) 1983-04-30
DE1445176C3 (en) 1974-04-25
MY6600061A (en) 1966-12-31
FI42960B (en) 1970-09-02
GB957797A (en) 1964-05-13
DE1445176A1 (en) 1968-10-17
DE1303727B (en) 1976-02-05
CH418338A (en) 1966-08-15
DE1445176B2 (en) 1973-09-06

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