AR029618A1 - Compuestos de amida , procedimientos para prepararlos, las composiciones farmaceuticas que los contienen y el uso de dichos compuestos para la fabricacion de medicamentos - Google Patents
Compuestos de amida , procedimientos para prepararlos, las composiciones farmaceuticas que los contienen y el uso de dichos compuestos para la fabricacion de medicamentosInfo
- Publication number
- AR029618A1 AR029618A1 ARP000100793A ARP000100793A AR029618A1 AR 029618 A1 AR029618 A1 AR 029618A1 AR P000100793 A ARP000100793 A AR P000100793A AR P000100793 A ARP000100793 A AR P000100793A AR 029618 A1 AR029618 A1 AR 029618A1
- Authority
- AR
- Argentina
- Prior art keywords
- compounds
- pharmaceutical compositions
- compositions containing
- medicines
- procedures
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
- C07C233/64—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings
- C07C233/65—Carboxylic acid amides having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atoms of the carboxamide groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C275/00—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
- C07C275/28—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
- C07C275/30—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by halogen atoms, or by nitro or nitroso groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
- C07D217/02—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines
- C07D217/06—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with only hydrogen atoms or radicals containing only carbon and hydrogen atoms, directly attached to carbon atoms of the nitrogen-containing ring; Alkylene-bis-isoquinolines with the ring nitrogen atom acylated by carboxylic or carbonic acids, or with sulfur or nitrogen analogues thereof, e.g. carbamates
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
- C07C2601/16—Systems containing only non-condensed rings with a six-membered ring the ring being unsaturated
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2602/00—Systems containing two condensed rings
- C07C2602/02—Systems containing two condensed rings the rings having only two atoms in common
- C07C2602/04—One of the condensed rings being a six-membered aromatic ring
- C07C2602/10—One of the condensed rings being a six-membered aromatic ring the other ring being six-membered, e.g. tetraline
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Psychiatry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Hydrogenated Pyridines (AREA)
- Pyridine Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Se describen compuestos de amida de la formula (1), en donde R1, R2 y R3 tienen los significados dados en la descripcion de la solicitud; X es CH o N, Y es un enlace simple o -NH-, y Q es -C(O)- y las sales de los mismos. También se describen los métodos para preparar dichos compuestos, las composiciones farmacéuticas que los contienen y el uso de dichos compuestos para la preparacion de medicamentos. Los compuestos de la presente son utiles como medicamentos para tratar y/o prevenir la amnesia y la demencia en mamíferos.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
AUPP8912A AUPP891299A0 (en) | 1999-02-26 | 1999-02-26 | New 6-membered cyclic compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
AR029618A1 true AR029618A1 (es) | 2003-07-10 |
Family
ID=3813111
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP000100793A AR029618A1 (es) | 1999-02-26 | 2000-02-24 | Compuestos de amida , procedimientos para prepararlos, las composiciones farmaceuticas que los contienen y el uso de dichos compuestos para la fabricacion de medicamentos |
Country Status (19)
Country | Link |
---|---|
EP (1) | EP1159258B1 (es) |
JP (1) | JP4089159B2 (es) |
KR (1) | KR100620406B1 (es) |
CN (1) | CN1170814C (es) |
AR (1) | AR029618A1 (es) |
AT (1) | ATE282022T1 (es) |
AU (2) | AUPP891299A0 (es) |
BR (1) | BR0010225A (es) |
CA (1) | CA2371827C (es) |
DE (1) | DE60015732T2 (es) |
DK (1) | DK1159258T3 (es) |
ES (1) | ES2226775T3 (es) |
HK (1) | HK1044934B (es) |
HU (1) | HUP0200116A3 (es) |
PT (1) | PT1159258E (es) |
RU (1) | RU2211215C2 (es) |
TR (1) | TR200102494T2 (es) |
TW (1) | TWI225856B (es) |
WO (1) | WO2000051970A1 (es) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1133230A4 (en) | 1998-11-23 | 2004-05-26 | Bonnie M Davis | DOSAGE FORMULAS FOR ACETYLCHOLINESTERASE INHIBITORS |
KR100437105B1 (ko) | 1998-12-24 | 2004-06-23 | 얀센 파마슈티카 엔.브이. | 방출 조절형 갈란타민 조성물 |
PE20020870A1 (es) | 2001-02-13 | 2002-11-18 | Aventis Pharma Gmbh | 6,7,8,9-tetrahidro-5h-benzocicloheptenil aminas aciladas |
PE20020856A1 (es) * | 2001-02-13 | 2002-11-11 | Aventis Pharma Gmbh | 1,2,3,4-tetrahidronaftil aminas aciladas |
TWI241190B (en) | 2001-02-13 | 2005-10-11 | Aventis Pharma Gmbh | 4-Fluoro-N-indan-2-yl benzamide and its use as pharmaceutical |
TWI243164B (en) | 2001-02-13 | 2005-11-11 | Aventis Pharma Gmbh | Acylated indanyl amines and their use as pharmaceuticals |
JP2005526137A (ja) | 2002-05-17 | 2005-09-02 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | アミノテトラリン−誘動尿素のバニロイドvr1受容体調節剤 |
CA2535036C (en) | 2003-08-06 | 2015-11-24 | Senomyx, Inc. | Novel flavors, flavor modifiers, tastants, taste enhancers, umami or sweet tastants, and/or enhancers and use thereof |
TWI548352B (zh) | 2006-04-21 | 2016-09-11 | 賽諾米克斯公司 | 包含高度鮮味風味劑之可食用組合物及其製造方法 |
EP2025674A1 (de) | 2007-08-15 | 2009-02-18 | sanofi-aventis | Substituierte Tetrahydronaphthaline, Verfahren zu ihrer Herstellung und ihre Verwendung als Arzneimittel |
TW201040154A (en) | 2009-02-13 | 2010-11-16 | Sanofi Aventis | Novel substituted indanes, process for preparation thereof and use thereof as a medicament |
WO2023176554A1 (ja) * | 2022-03-14 | 2023-09-21 | 国立大学法人東北大学 | 認知機能改善剤 |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR8287M (es) * | 1968-12-31 | 1970-11-09 | ||
US4797419A (en) * | 1986-11-03 | 1989-01-10 | Warner-Lambert Company | Method of treating the symptoms of senile cognitive decline employing di- or trisubstituted urea cholinergic agents |
EP0306375A1 (fr) * | 1987-08-07 | 1989-03-08 | Synthelabo | Dérivés de[(pipéridinyl-4)méthyl]-2 tétrahydro-1,2,3,4 isoquinoléine, leur préparation et leur application en thérapeutique |
CA1340113C (en) * | 1988-05-24 | 1998-11-03 | Magid A. Abou-Gharbia | Aryl-and heteroaryl piperazinyl carboxamides having central nervous system activity |
JPH06107544A (ja) * | 1992-09-29 | 1994-04-19 | Taisho Pharmaceut Co Ltd | コリン作動性神経不全の改善・治療薬 |
JPH06298732A (ja) * | 1993-02-16 | 1994-10-25 | Taisho Pharmaceut Co Ltd | インドール誘導体 |
-
1999
- 1999-02-26 AU AUPP8912A patent/AUPP891299A0/en not_active Abandoned
-
2000
- 2000-02-03 DK DK00902080T patent/DK1159258T3/da active
- 2000-02-03 WO PCT/JP2000/000601 patent/WO2000051970A1/en active IP Right Grant
- 2000-02-03 PT PT00902080T patent/PT1159258E/pt unknown
- 2000-02-03 KR KR1020017010325A patent/KR100620406B1/ko not_active IP Right Cessation
- 2000-02-03 BR BR0010225-3A patent/BR0010225A/pt not_active Application Discontinuation
- 2000-02-03 TR TR2001/02494T patent/TR200102494T2/xx unknown
- 2000-02-03 ES ES00902080T patent/ES2226775T3/es not_active Expired - Lifetime
- 2000-02-03 DE DE60015732T patent/DE60015732T2/de not_active Expired - Lifetime
- 2000-02-03 AT AT00902080T patent/ATE282022T1/de not_active IP Right Cessation
- 2000-02-03 HU HU0200116A patent/HUP0200116A3/hu unknown
- 2000-02-03 JP JP2000602198A patent/JP4089159B2/ja not_active Expired - Fee Related
- 2000-02-03 CN CNB008043035A patent/CN1170814C/zh not_active Expired - Fee Related
- 2000-02-03 CA CA002371827A patent/CA2371827C/en not_active Expired - Fee Related
- 2000-02-03 AU AU23257/00A patent/AU766655B2/en not_active Ceased
- 2000-02-03 EP EP00902080A patent/EP1159258B1/en not_active Expired - Lifetime
- 2000-02-03 RU RU2001126120/04A patent/RU2211215C2/ru not_active IP Right Cessation
- 2000-02-14 TW TW089102410A patent/TWI225856B/zh not_active IP Right Cessation
- 2000-02-24 AR ARP000100793A patent/AR029618A1/es unknown
-
2002
- 2002-09-10 HK HK02106646.3A patent/HK1044934B/zh not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
ATE282022T1 (de) | 2004-11-15 |
KR20010102140A (ko) | 2001-11-15 |
CN1170814C (zh) | 2004-10-13 |
AUPP891299A0 (en) | 1999-03-25 |
RU2211215C2 (ru) | 2003-08-27 |
PT1159258E (pt) | 2005-02-28 |
AU2325700A (en) | 2000-09-21 |
CA2371827A1 (en) | 2000-09-08 |
HUP0200116A2 (hu) | 2002-05-29 |
TWI225856B (en) | 2005-01-01 |
EP1159258A1 (en) | 2001-12-05 |
CA2371827C (en) | 2008-06-10 |
HUP0200116A3 (en) | 2002-11-28 |
JP2002538132A (ja) | 2002-11-12 |
JP4089159B2 (ja) | 2008-05-28 |
KR100620406B1 (ko) | 2006-09-13 |
TR200102494T2 (tr) | 2002-01-21 |
WO2000051970A1 (en) | 2000-09-08 |
HK1044934B (zh) | 2005-06-03 |
AU766655B2 (en) | 2003-10-23 |
EP1159258B1 (en) | 2004-11-10 |
DK1159258T3 (da) | 2005-02-14 |
CN1341095A (zh) | 2002-03-20 |
DE60015732T2 (de) | 2005-03-31 |
ES2226775T3 (es) | 2005-04-01 |
DE60015732D1 (de) | 2004-12-16 |
HK1044934A1 (en) | 2002-11-08 |
BR0010225A (pt) | 2002-01-22 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
AR017182A1 (es) | Compuestos de aminotiazol, inhibidores de las kinasas dependientes de ciclinas y las composiciones farmaceuticas que los contienen. | |
HU895609D0 (en) | Process for the preparation of novel 1,4-diazepine derivatives and pharmaceutical compositions containing such compounds | |
NO905572D0 (no) | Fremgangsmaate for fremstilling av peptidforbindelser. | |
ES2058527T3 (es) | Derivados de pirimidina condensados procedimiento y compuestos intermedios para su preparacion y composiciones farmaceuticas que los contienen. | |
AR018634A1 (es) | Derivados de benzo(b)tiepin-1,1,-dioxido, procedimiento para su preparacion, medicamentos conteniendo estos compuestos, procedimiento para la preparacion de medicamentos y su empleo para la preparacion de medicamentos. | |
BR9908764A (pt) | Composto e seus sais farmaceuticamente aceitáveis ou ésteres hidrolisáveis in vivo, uso destes, processo para prepará-los, e, composição farmacêutica | |
AR029383A1 (es) | Moleculas pequenas, los intermediarios para su sintesis, las composiciones farmaceuticas que las contienen y su uso para preparar un medicamento destinado al tratamiento o la profilaxis de enfermedades inflamatorias o mediadas por celulas inmunes | |
FI941987A (fi) | Uudet aminohappojohdannaiset, menetelmät niiden valmistamiseksi ja näitä yhdisteitä sisältävät farmaseuttiset koostumukset | |
ATE103812T1 (de) | Zusammensetzung zur behandlung von ischaemischen stoerungen in organen. | |
ES2123039T3 (es) | Nuevas 3-(hidroxi-bencilidenil)-indolin-2-onas, su procedimiento de preparacion y composiciones farmaceuticas que las contienen. | |
AR029618A1 (es) | Compuestos de amida , procedimientos para prepararlos, las composiciones farmaceuticas que los contienen y el uso de dichos compuestos para la fabricacion de medicamentos | |
MY129176A (en) | Tetrahydro gamma-carbolines | |
JPS5665869A (en) | Novel 22hydroxyalkyll3*4*55trihydroxyypiperidine compound* its manufacture and drug | |
NO892295L (no) | Fremgangsmaate for fremstilling av nye cefemforbindelser. | |
DE3882679D1 (de) | Kardiovaskulaer aktive verbindungen. | |
MX9306394A (es) | Derivados de benzofurano, proceso para su preparacion y composicion farmaceutica que los contiene | |
ES2094324T3 (es) | Nuevos derivados de pirrolidina, su procedimiento de preparacion y las composiciones farmaceuticas que los contienen. | |
NO905245L (no) | Fremgangsmaate for fremstilling av terapeutisk aktive heterocykliske forbindelser. | |
EA200101204A1 (ru) | Новые бициклические соединения аминопиразинона, способ их получения и содержащие их фармацевтические композиции | |
UA50722C2 (uk) | Нітробензаміди, спосіб їх одержання (варіанти), фармацевтична композиція | |
EA200100343A3 (ru) | Новые гетероциклоалкилбензоциклобутановые и гетероарилбензоциклобутановые производные, способ их получения и содержащие их фармацевтические композиции | |
FI903511A0 (fi) | Pyrrolo (2,1-b) tiazolderivat. | |
TH6029A (th) | อนุพันธ์ของควิโนลิเนียม และไอโซควิโนลิเนียมที่ควบแน่น | |
MX9405283A (es) | Empleo de las fenalquilaminas para la fabricacion de medicamentos paradisminuir el colesterol y los medicamentos que las incluyen. | |
TH17758A (th) | สารเคมี |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
FB | Suspension of granting procedure |