OA07356A - Substituted 3,4-Diamino-1,2,5-thiadiazoles possessing histamine H2 receptor antagonist activity. - Google Patents

Substituted 3,4-Diamino-1,2,5-thiadiazoles possessing histamine H2 receptor antagonist activity.

Info

Publication number: OA07356A
Authority: OA; OAPI
Prior art keywords: thiadiazoles; histamine; diamino; possessing; substituted
Prior art date: 1982-03-29

Application number

OA57955A

Other languages

French (fr)

Inventor

Ronnie Ray Crenshaw

Original Assignee

Bristol Myers Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1982-03-29

Filing date

1983-03-29

Publication date

1984-08-31

1983-03-29 Application filed by Bristol Myers Co filed Critical Bristol Myers Co

1984-08-31 Publication of OA07356A publication Critical patent/OA07356A/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/01—Five-membered rings
- C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
- C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
- C07D285/10—1,2,5-Thiadiazoles; Hydrogenated 1,2,5-thiadiazoles
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/01—Five-membered rings
- C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
- C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
- C07D285/06—1,2,3-Thiadiazoles; Hydrogenated 1,2,3-thiadiazoles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
Furan Compounds (AREA)
Pyridine Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Heterocyclic Compounds Containing Sulfur Atoms (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Hydrogenated Pyridines (AREA)
Pyrrole Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

OA57955A 1982-03-29 1983-03-29 Substituted 3,4-Diamino-1,2,5-thiadiazoles possessing histamine H2 receptor antagonist activity. OA07356A (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US36320782A	1982-03-29	1982-03-29

Publications (1)

Publication Number	Publication Date
OA07356A true OA07356A (en)	1984-08-31

Family

ID=23429274

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
OA57955A OA07356A (en)	1982-03-29	1983-03-29	Substituted 3,4-Diamino-1,2,5-thiadiazoles possessing histamine H2 receptor antagonist activity.

Country Status (30)

Country	Link
JP (2)	JPS58180477A (en)
KR (1)	KR880002209B1 (en)
AT (1)	AT386599B (en)
AU (2)	AU557577B2 (en)
BE (1)	BE896291A (en)
CH (2)	CH660880A5 (en)
CS (2)	CS250240B2 (en)
DD (2)	DD210909A5 (en)
DE (1)	DE3311281A1 (en)
DK (2)	DK166677B1 (en)
ES (3)	ES520982A0 (en)
FR (2)	FR2542741B1 (en)
GB (2)	GB2117769B (en)
GR (1)	GR78524B (en)
HU (2)	HU188742B (en)
IE (1)	IE55596B1 (en)
IL (1)	IL68259A0 (en)
IT (1)	IT1164633B (en)
LU (1)	LU84716A1 (en)
MY (1)	MY8700942A (en)
NL (1)	NL8301063A (en)
NO (1)	NO163055C (en)
NZ (1)	NZ203726A (en)
OA (1)	OA07356A (en)
PT (1)	PT76459B (en)
SE (2)	SE461040B (en)
SU (2)	SU1419518A3 (en)
YU (1)	YU44849B (en)
ZA (1)	ZA832154B (en)
ZW (1)	ZW7683A1 (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
AU2222083A (en) *	1982-12-14	1984-06-21	Smith Kline & French Laboratories Limited	Pyridine derivatives
US4593039A (en) *	1984-04-02	1986-06-03	Merck & Co., Inc.	1-aryloxy-3-(substituted aminoalkylamino)-2-propanols
US4644006A (en) *	1984-06-22	1987-02-17	Bristol-Myers Company	Substituted 3,4-diamino-1,2,5-thiadiazoles having histamine H2 -receptor antagonist activity
JPH0622828B2 (en) *	1986-06-30	1994-03-30	フアナツク株式会社	Direct pressure type mold clamping mechanism
EP4196793A1 (en)	2020-08-11	2023-06-21	Université de Strasbourg	H2 blockers targeting liver macrophages for the prevention and treatment of liver disease and cancer

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3018289A (en) *	1960-02-10	1962-01-23	Wyandotte Chemicals Corp	Process for preparing oxamidines
GB1595291A (en) *	1976-09-21	1981-08-12	Smith Kline French Lab	Pyrimidone and thiopyrimidone derivatives
FI76795C (en) *	1979-09-04	1988-12-12	Bristol Myers Co	Process for the preparation of novel, therapeutically useful 3,4-disubstituted 1,2,5-thiadiazole-1-oxides and -1,1-dioxides and novel intermediates
EP0040696B1 (en) *	1980-04-30	1986-08-27	Merck & Co. Inc.	Aminothiadiazoles as gastric secretion inhibitors
AU2222083A (en) *	1982-12-14	1984-06-21	Smith Kline & French Laboratories Limited	Pyridine derivatives

1983
- 1983-03-25 ES ES520982A patent/ES520982A0/en active Granted
- 1983-03-25 NL NL8301063A patent/NL8301063A/en not_active Application Discontinuation
- 1983-03-25 ZA ZA832154A patent/ZA832154B/en unknown
- 1983-03-25 FR FR838304934A patent/FR2542741B1/en not_active Expired
- 1983-03-25 ZW ZW76/83A patent/ZW7683A1/en unknown
- 1983-03-28 PT PT76459A patent/PT76459B/en not_active IP Right Cessation
- 1983-03-28 NZ NZ203726A patent/NZ203726A/en unknown
- 1983-03-28 LU LU84716A patent/LU84716A1/en unknown
- 1983-03-28 AU AU12907/83A patent/AU557577B2/en not_active Ceased
- 1983-03-28 SU SU833568849A patent/SU1419518A3/en active
- 1983-03-28 SE SE8301725A patent/SE461040B/en not_active IP Right Cessation
- 1983-03-28 GB GB08308518A patent/GB2117769B/en not_active Expired
- 1983-03-28 DE DE19833311281 patent/DE3311281A1/en not_active Withdrawn
- 1983-03-28 IL IL68259A patent/IL68259A0/en not_active IP Right Cessation
- 1983-03-28 HU HU831040A patent/HU188742B/en not_active IP Right Cessation
- 1983-03-28 NO NO831100A patent/NO163055C/en unknown
- 1983-03-28 DK DK141383A patent/DK166677B1/en not_active IP Right Cessation
- 1983-03-28 BE BE0/210417A patent/BE896291A/en not_active IP Right Cessation
- 1983-03-28 HU HU854071A patent/HU196386B/en not_active IP Right Cessation
- 1983-03-28 GR GR70903A patent/GR78524B/el unknown
- 1983-03-28 IT IT48005/83A patent/IT1164633B/en active
- 1983-03-28 IE IE686/83A patent/IE55596B1/en not_active IP Right Cessation
- 1983-03-29 CH CH575/86A patent/CH660880A5/en not_active IP Right Cessation
- 1983-03-29 DD DD83249300A patent/DD210909A5/en not_active IP Right Cessation
- 1983-03-29 CS CS841958A patent/CS250240B2/en unknown
- 1983-03-29 CS CS832191A patent/CS250229B2/en unknown
- 1983-03-29 JP JP58051740A patent/JPS58180477A/en active Granted
- 1983-03-29 YU YU744/83A patent/YU44849B/en unknown
- 1983-03-29 CH CH1749/83A patent/CH655111A5/en not_active IP Right Cessation
- 1983-03-29 DD DD83260707A patent/DD219768A5/en not_active IP Right Cessation
- 1983-03-29 OA OA57955A patent/OA07356A/en unknown
- 1983-03-29 AT AT0111083A patent/AT386599B/en not_active IP Right Cessation
- 1983-03-29 KR KR1019830001283A patent/KR880002209B1/en not_active IP Right Cessation
- 1983-11-30 ES ES527686A patent/ES527686A0/en active Granted
- 1983-11-30 ES ES527685A patent/ES527685A0/en active Granted
1984
- 1984-06-08 SU SU843750493A patent/SU1355123A3/en active
- 1984-12-31 GB GB08432809A patent/GB2149406B/en not_active Expired
1986
- 1986-09-30 AU AU63272/86A patent/AU586037B2/en not_active Ceased
1987
- 1987-05-22 FR FR878707197A patent/FR2597867B1/en not_active Expired
- 1987-11-25 SE SE8704689A patent/SE464302B/en not_active IP Right Cessation
- 1987-12-30 MY MY942/87A patent/MY8700942A/en unknown
1992
- 1992-06-18 DK DK92811A patent/DK81192D0/en not_active Application Discontinuation
1993
- 1993-04-16 JP JP5124585A patent/JPH06135925A/en active Pending

Also Published As

Publication number	Publication date
IT8348005A0 (en)	1983-03-28
FR2597867B1 (en)	1989-12-08
ES8404683A1 (en)	1984-05-16
NZ203726A (en)	1986-05-09
GB2149406B (en)	1986-01-02
ZW7683A1 (en)	1984-01-04
AU6327286A (en)	1987-01-08
IL68259A0 (en)	1983-06-15
DK166677B1 (en)	1993-06-28
LU84716A1 (en)	1983-12-05
ES8505978A1 (en)	1985-06-16
PT76459A (en)	1983-04-01
AT386599B (en)	1988-09-12
KR840004095A (en)	1984-10-06
ATA111083A (en)	1988-02-15
NO831100L (en)	1983-09-30
AU1290783A (en)	1983-10-06
FR2542741B1 (en)	1989-12-08
DK141383A (en)	1983-09-30
GR78524B (en)	1984-09-27
ES527686A0 (en)	1985-06-16
ES8505977A1 (en)	1985-06-16
GB2117769B (en)	1985-08-29
IE830686L (en)	1983-09-29
ES527685A0 (en)	1985-06-16
SE8301725L (en)	1983-11-25
CS250240B2 (en)	1987-04-16
SU1355123A3 (en)	1987-11-23
SE464302B (en)	1991-04-08
NO163055B (en)	1989-12-18
AU557577B2 (en)	1986-12-24
SE8704689L (en)	1987-11-25
YU44849B (en)	1991-04-30
SE461040B (en)	1989-12-18
PT76459B (en)	1986-03-11
DE3311281A1 (en)	1983-11-24
YU74483A (en)	1986-02-28
FR2542741A1 (en)	1984-09-21
SE8704689D0 (en)	1987-11-25
DD210909A5 (en)	1984-06-27
ES520982A0 (en)	1984-05-16
CS250229B2 (en)	1987-04-16
BE896291A (en)	1983-09-28
JPS58180477A (en)	1983-10-21
DK81192A (en)	1992-06-18
GB8432809D0 (en)	1985-02-06
HU196386B (en)	1988-11-28
DD219768A5 (en)	1985-03-13
KR880002209B1 (en)	1988-10-18
IT1164633B (en)	1987-04-15
GB2117769A (en)	1983-10-19
GB2149406A (en)	1985-06-12
GB8308518D0 (en)	1983-05-05
AU586037B2 (en)	1989-06-29
ZA832154B (en)	1983-12-28
HU188742B (en)	1986-05-28
CH660880A5 (en)	1987-05-29
MY8700942A (en)	1987-12-31
IE55596B1 (en)	1990-11-21
FR2597867A1 (en)	1987-10-30
DK141383D0 (en)	1983-03-28
SU1419518A3 (en)	1988-08-23
NO163055C (en)	1990-03-28
DK81192D0 (en)	1992-06-18
CH655111A5 (en)	1986-03-27
JPH0568472B2 (en)	1993-09-29
SE8301725D0 (en)	1983-03-28
JPH06135925A (en)	1994-05-17
NL8301063A (en)	1983-10-17

Publication	Publication Date	Title
ATE30023T1 (en)	1987-10-15	LEUKOTRIAN ANTAGONISTS.
FI834202A (en)	1984-05-19	SLANGFORMIGT LIVSMEDELSHOELJE, I SYNNERHET KORVSKINN MED FOERBAETTRAD AVSKALBARHET.
DE3574665D1 (en)	1990-01-18	GLUTAMATE RECEPTOR INHIBITANT.
FI854957A (en)	1986-06-25	BENTONIT INNEHAOLLANDE, MJUKGOERANDE, FLYTANDE TVAETTMEDEL FOER TEXTILER.
DE3485456D1 (en)	1992-02-27	PHOTO RECEPTOR.
OA07356A (en)	1984-08-31	Substituted 3,4-Diamino-1,2,5-thiadiazoles possessing histamine H2 receptor antagonist activity.
ZA783141B (en)	1979-06-27	Histamine h2 receptor antagonists
DE3578233D1 (en)	1990-07-19	PHOTO RECEPTOR.
OA08039A (en)	1987-01-31	Substituted 3,4-diamido-1,2,5-thiadiazoles exhibiting histamine H2 receptor antagonist activity.
IT8321317A0 (en)	1983-05-26	VEHICLE SEAT, FOR AT LEAST TWO PEOPLE.
ES516395A0 (en)	1983-06-16	"KNITTING LATCH FOR FLAT KNITTING".
NO843726L (en)	1985-03-22	2,5-DISUBSTITUTED-4 (3H) -PYRIMIDONES WITH HISTAMINE H2 RECEPTOR ANTAGONIST EFFECT
ES515054A0 (en)	1983-05-01	"PROCEDURE FOR THE PREPARATION OF 2-AMINO-5-MERCAPTO-1,3,4-TIADIAZOLES".
DE69004827D1 (en)	1994-01-13	Alpha-adrenergic receptor antagonists.
Welch	1983	The Geomorphology of the Strawberry Creek Basin, Central Alberta
IT8320738A0 (en)	1983-04-22	PROCEDURE FOR PRODUCING 2,3-DIHYDRO-2,2-DIMETHYL-7-BENZOPURANOL.
ES265348Y (en)	1983-07-01	"HEAD-TERMINAL, FOR TUBULAR ELEMENTS OF METALLIC STRUCTURES".
ES266710Y (en)	1983-10-16	"BUCKET FEEDER".
ES263615Y (en)	1983-10-16	"SEAT".
IE810940L (en)	1981-10-28	17-substituted-6-desoxy-7,8-dihydro-6ó-methylnoroxymorphone¹narcotic antagonists
IT1209497B (en)	1989-08-30	PROCEDURE FOR PREVENTING PHOTOTOXIC REACTIONS.
ATE19775T1 (en)	1986-05-15	AMINOPYRIMIDINONE DERIVATIVES USABLE AS HISTAMINE H1 ANTAGONISTS.
TR21881A (en)	1985-10-03	SOME 2. (2-SUBSTITUTED BENZOIL) -1,3-SIKLOHEKSANADIONS
ATE30018T1 (en)	1987-10-15	LEUKOTRIAN ANTAGONISTS.
IT8223991A0 (en)	1982-10-29	NEW 2,2-DISOSTITUTED 2,3-DIHYDRO-1,4-BENZODIOXINES WITH HYPOTENSIVE ACTIVITY.