NO325501B1 - Piperazinforbindelser, anvendelse og fremstilling derav, samt farmasoytisk preparat. - Google Patents

Piperazinforbindelser, anvendelse og fremstilling derav, samt farmasoytisk preparat. Download PDF

Info

Publication number: NO325501B1
Authority: NO; Norway
Prior art keywords: compound; pharmaceutical preparation; patient; treatment; disorders
Prior art date: 2000-11-28

Application number

NO20032390A

Other languages

English (en)

Norwegian (no)

Other versions

NO20032390L (no

NO20032390D0 (no

Inventor

Michael Gerard Kelly

Wayne Everett Childers

Sharon Joy Rosenzweig-Lipson

Original Assignee

Wyeth Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-11-28

Filing date

2003-05-27

Publication date

2008-05-26

2003-05-27 Application filed by Wyeth Corp filed Critical Wyeth Corp

2003-05-27 Publication of NO20032390D0 publication Critical patent/NO20032390D0/no

2003-07-22 Publication of NO20032390L publication Critical patent/NO20032390L/no

2008-05-26 Publication of NO325501B1 publication Critical patent/NO325501B1/no

Links

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Classifications

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- C07—ORGANIC CHEMISTRY
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- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
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- A61P25/36—Opioid-abuse
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Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Psychiatry (AREA)
Addiction (AREA)
Pain & Pain Management (AREA)
Endocrinology (AREA)
Psychology (AREA)
Reproductive Health (AREA)
Cardiology (AREA)
Hospice & Palliative Care (AREA)
Diabetes (AREA)
Nutrition Science (AREA)
Heart & Thoracic Surgery (AREA)
Gynecology & Obstetrics (AREA)
Anesthesiology (AREA)
Urology & Nephrology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Plural Heterocyclic Compounds (AREA)

NO20032390A 2000-11-28 2003-05-27 Piperazinforbindelser, anvendelse og fremstilling derav, samt farmasoytisk preparat. NO325501B1 (no)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US25330100P	2000-11-28	2000-11-28
US29781401P	2001-06-13	2001-06-13
PCT/US2001/043160 WO2002044142A2 (en)	2000-11-28	2001-11-27	Piperazine derivatives, their preparation and their use for treating central nervous system (cns) disorders

Publications (3)

Publication Number	Publication Date
NO20032390D0 NO20032390D0 (no)	2003-05-27
NO20032390L NO20032390L (no)	2003-07-22
NO325501B1 true NO325501B1 (no)	2008-05-26

Family

ID=26943115

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20032390A NO325501B1 (no)	2000-11-28	2003-05-27	Piperazinforbindelser, anvendelse og fremstilling derav, samt farmasoytisk preparat.

Country Status (25)

Country	Link
US (3)	US6469007B2 (xx)
EP (1)	EP1339406B1 (xx)
JP (1)	JP4198989B2 (xx)
KR (1)	KR100835552B1 (xx)
CN (1)	CN100352437C (xx)
AR (1)	AR035603A1 (xx)
AT (1)	ATE269078T1 (xx)
AU (2)	AU2002237654B2 (xx)
BR (1)	BR0115609A (xx)
CA (1)	CA2428039C (xx)
DE (1)	DE60103927T2 (xx)
DK (1)	DK1339406T3 (xx)
EA (1)	EA005925B1 (xx)
ES (1)	ES2222401T3 (xx)
HK (1)	HK1057864A1 (xx)
HU (1)	HUP0400551A2 (xx)
IL (1)	IL156098A0 (xx)
MX (1)	MXPA03004677A (xx)
NO (1)	NO325501B1 (xx)
NZ (1)	NZ526150A (xx)
PL (1)	PL363219A1 (xx)
PT (1)	PT1339406E (xx)
TR (1)	TR200401546T4 (xx)
TW (1)	TWI224102B (xx)
WO (1)	WO2002044142A2 (xx)

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US6432826B1 (en) *	1999-11-29	2002-08-13	Applied Materials, Inc.	Planarized Cu cleaning for reduced defects
US20060287335A1 (en) *	2000-11-28	2006-12-21	Wyeth	Serotonergic agents for treating sexual dysfunction
US20060223824A1 (en) *	2000-11-28	2006-10-05	Wyeth	Serotonergic agents
DK1408976T5 (da)	2001-07-20	2011-01-10	Psychogenics Inc	Behandling af ADHD (Attention deficit hyperactivity disorder)
RU2315762C2 (ru)	2002-03-12	2008-01-27	Уайт	Способ синтеза хиральных n-арилпиперазинов
BR0308347A (pt)	2002-03-12	2005-01-25	Wyeth Corp	Processo para fabricação de piperazinas 1,4-dissubstituìdas quirais
US7091349B2 (en)	2002-03-12	2006-08-15	Wyeth	Process for synthesizing N-aryl piperazines with chiral N′-1-[benzoyl(2-pyridyl)amino]-2-propane substitution
US7361773B2 (en)	2002-03-12	2008-04-22	Wyeth	Preparation of N1-(2'-pyridyl)-1,2-propanediamine sulfamic acid and its use in the synthesis of biologically active piperazines
GB0219961D0 (en) *	2002-08-28	2002-10-02	Pfizer Ltd	Oxytocin inhibitors
US20040192730A1 (en) *	2003-03-13	2004-09-30	Dynogen Pharmaceuticals, Inc.	Methods of using compounds with combined 5-HT1A and SSRI activities as-needed to treat sexual dysfunction
US20070099931A1 (en) *	2004-03-19	2007-05-03	Wyeth	Pharmaceutical dosage forms and compositions
US20050215561A1 (en) *	2004-03-19	2005-09-29	Krishnendu Ghosh	Pharmaceutical dosage forms and compositions
US20050209245A1 (en) *	2004-03-19	2005-09-22	Wyeth	Process for preparing N-aryl-piperazine derivatives
KR100646337B1 (ko) *	2004-06-30	2006-11-23	주식회사 롯데기공	보일러의 누수 감지방법
DE602005021534D1 (de) *	2004-10-15	2010-07-08	Us Gov Health & Human Serv	Amphipathische helixförmige multidomänenpeptide und verfahren zu deren anwendung
TW200700413A (en) *	2005-03-01	2007-01-01	Wyeth Corp	Crystalline and amorphous 4-cyano-n-{(2r)-2-[4-(2,3-dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-propyl}-n-pyridin-2-yl-benzamide hydrochloride
TW200800959A (en) *	2005-06-10	2008-01-01	Wyeth Corp	Piperazine-piperidine antagonists and agonists of the 5-HT1a receptor
EP1893617A1 (en) *	2005-06-17	2008-03-05	Wyeth a Corporation of the State of Delaware	Tricyclic compounds useful as serotonin inhibitors and 5-ht1a agonists and antagonists
EP1993527A4 (en) *	2006-01-26	2009-08-05	Univ Rochester	INHIBITION OF AMYLOID BETA PEPTIDE / RAGE INTERACTION AT BLOOD BRAIN BARRIER
TW200808740A (en) *	2006-06-09	2008-02-16	Wyeth Corp	Succinate salts of 6-methoxy-8-[4-(1-(5-fluoro)-quinolin-8-yl-piperidin-4-yl)-piperazin-1-yl]-quinoline and crystalline forms thereof
TW200811144A (en) *	2006-06-09	2008-03-01	Wyeth Corp	Crystalline forms of 6-methoxy-8-[4-(1-(5-fluoro)-quinolin-8-yl-piperidin-4-yl)-piperazin-1-yl]-quinoline
TW200808741A (en) *	2006-06-09	2008-02-16	Wyeth Corp	6-methoxy-8-[4-(1-(5-fluoro)-quinolin-8-yl-piperidin-4-yl)-piperazin-1-yl]-quinoline hydrochloric acid salts
CL2007003410A1 (es) *	2006-11-28	2008-04-11	Wyeth Corp	Compuestos derivados de 5-fluoro-8-{4-[4-(6-metoxiquinolin-8-il)piperazin-1-il]piperidin-1-il}quinolina; procedimiento de preparacion; compuestos intermediarios; procedimiento de preparacion; composicion farmaceutica; y uso en el tratamiento de trast
TW200901974A (en) *	2007-01-16	2009-01-16	Wyeth Corp	Compounds, compositions, and methods of making and using them
WO2009129263A1 (en) *	2008-04-15	2009-10-22	The Government Of The Usa As Represented By The Secretary Of The Department Of Health & Human Serv.	Peptides promoting lipid efflux via abca1 and activating a lipoprotein lipase

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IL101722A (en)	1991-05-02	1996-05-14	Wyeth John & Brother Ltd	History of piperazine, their preparation and pharmaceutical preparations containing them
GB9514901D0 (en)	1995-07-20	1995-09-20	American Home Prod	Piperazine derivatives

2001
- 2001-11-13 US US10/010,575 patent/US6469007B2/en not_active Expired - Fee Related
- 2001-11-27 DK DK01986458T patent/DK1339406T3/da active
- 2001-11-27 AU AU2002237654A patent/AU2002237654B2/en not_active Ceased
- 2001-11-27 CN CNB018196853A patent/CN100352437C/zh not_active Expired - Fee Related
- 2001-11-27 TW TW090129285A patent/TWI224102B/zh not_active IP Right Cessation
- 2001-11-27 JP JP2002546512A patent/JP4198989B2/ja not_active Expired - Fee Related
- 2001-11-27 NZ NZ526150A patent/NZ526150A/en unknown
- 2001-11-27 DE DE60103927T patent/DE60103927T2/de not_active Expired - Lifetime
- 2001-11-27 TR TR2004/01546T patent/TR200401546T4/xx unknown
- 2001-11-27 CA CA2428039A patent/CA2428039C/en not_active Expired - Fee Related
- 2001-11-27 AT AT01986458T patent/ATE269078T1/de not_active IP Right Cessation
- 2001-11-27 AR ARP010105502A patent/AR035603A1/es not_active Application Discontinuation
- 2001-11-27 PL PL01363219A patent/PL363219A1/xx not_active Application Discontinuation
- 2001-11-27 WO PCT/US2001/043160 patent/WO2002044142A2/en active IP Right Grant
- 2001-11-27 ES ES01986458T patent/ES2222401T3/es not_active Expired - Lifetime
- 2001-11-27 AU AU3765402A patent/AU3765402A/xx active Pending
- 2001-11-27 HU HU0400551A patent/HUP0400551A2/hu unknown
- 2001-11-27 IL IL15609801A patent/IL156098A0/xx unknown
- 2001-11-27 EA EA200300619A patent/EA005925B1/ru not_active IP Right Cessation
- 2001-11-27 EP EP01986458A patent/EP1339406B1/en not_active Expired - Lifetime
- 2001-11-27 KR KR1020037007064A patent/KR100835552B1/ko not_active IP Right Cessation
- 2001-11-27 MX MXPA03004677A patent/MXPA03004677A/es active IP Right Grant
- 2001-11-27 BR BR0115609-8A patent/BR0115609A/pt not_active Application Discontinuation
- 2001-11-27 PT PT01986458T patent/PT1339406E/pt unknown
2002
- 2002-08-14 US US10/218,251 patent/US6586436B2/en not_active Expired - Fee Related
2003
- 2003-05-20 US US10/441,536 patent/US7026320B2/en not_active Expired - Fee Related
- 2003-05-27 NO NO20032390A patent/NO325501B1/no not_active IP Right Cessation
2004
- 2004-02-04 HK HK04100730A patent/HK1057864A1/xx not_active IP Right Cessation

Also Published As

Publication number	Publication date
US6586436B2 (en)	2003-07-01
US6469007B2 (en)	2002-10-22
AU2002237654B2 (en)	2005-07-28
NO20032390L (no)	2003-07-22
DE60103927D1 (de)	2004-07-22
TR200401546T4 (tr)	2004-09-21
US20030022901A1 (en)	2003-01-30
WO2002044142A3 (en)	2002-08-08
JP4198989B2 (ja)	2008-12-17
KR20030051879A (ko)	2003-06-25
HUP0400551A2 (en)	2006-02-28
EP1339406B1 (en)	2004-06-16
WO2002044142A2 (en)	2002-06-06
CA2428039C (en)	2011-08-09
MXPA03004677A (es)	2003-09-05
AU3765402A (en)	2002-06-11
ATE269078T1 (de)	2004-07-15
PL363219A1 (en)	2004-11-15
BR0115609A (pt)	2003-11-11
EP1339406A2 (en)	2003-09-03
US20020107254A1 (en)	2002-08-08
HK1057864A1 (en)	2004-04-23
JP2004520289A (ja)	2004-07-08
DE60103927T2 (de)	2005-06-23
US20030216408A1 (en)	2003-11-20
NZ526150A (en)	2004-11-26
KR100835552B1 (ko)	2008-06-09
US7026320B2 (en)	2006-04-11
CN1477961A (zh)	2004-02-25
DK1339406T3 (da)	2004-09-27
PT1339406E (pt)	2004-10-29
TWI224102B (en)	2004-11-21
CN100352437C (zh)	2007-12-05
EA200300619A1 (ru)	2003-10-30
NO20032390D0 (no)	2003-05-27
ES2222401T3 (es)	2005-02-01
EA005925B1 (ru)	2005-08-25
AR035603A1 (es)	2004-06-16
IL156098A0 (en)	2003-12-23
CA2428039A1 (en)	2002-06-06

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SK10222001A3 (sk)	2002-03-05	Morfolinobenzamidové soli
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US20040127543A1 (en)	2004-07-01	Antidepressant cycloalkylamine derivatives of 2,3-dihydro-1,4-benzodioxan
ZA200304994B (en)	2004-10-04	Piperazine derivatives, their preparation and their use for treating central nervous systems (CNS) disorders.
JP2010534705A (ja)	2010-11-11	Ｈ１受容体のアンタゴニストとして有用なスピロ化合物
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