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MX2016013684A - Composicion farmaceutica que contiene derivado de hidantoina. - Google Patents

Composicion farmaceutica que contiene derivado de hidantoina.

Info

Publication number
MX2016013684A
MX2016013684A MX2016013684A MX2016013684A MX2016013684A MX 2016013684 A MX2016013684 A MX 2016013684A MX 2016013684 A MX2016013684 A MX 2016013684A MX 2016013684 A MX2016013684 A MX 2016013684A MX 2016013684 A MX2016013684 A MX 2016013684A
Authority
MX
Mexico
Prior art keywords
pharmaceutical composition
containing pharmaceutical
hydantoin derivative
formula
hydantoin
Prior art date
Application number
MX2016013684A
Other languages
English (en)
Other versions
MX371090B (es
Inventor
Kitamura Hidetomo
Tamura Tatsuya
Noda Horoshi
Original Assignee
Chugai Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chugai Pharmaceutical Co Ltd filed Critical Chugai Pharmaceutical Co Ltd
Publication of MX2016013684A publication Critical patent/MX2016013684A/es
Publication of MX371090B publication Critical patent/MX371090B/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41661,3-Diazoles having oxo groups directly attached to the heterocyclic ring, e.g. phenytoin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41881,3-Diazoles condensed with other heterocyclic ring systems, e.g. biotin, sorbinil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5355Non-condensed oxazines and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/04Drugs for skeletal disorders for non-specific disorders of the connective tissue
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Immunology (AREA)
  • Biomedical Technology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Una composición farmacéutica para inducir una acción de absorción del hueso y/o cartílago, que incluye como un componente eficaz de la misma un compuesto indicado por la fórmula general (1) o una sal farmacológicamente aceptable del mismo (en la fórmula, R1, R2, R3, y R4 son como se definen en las Reivindicaciones).
MX2016013684A 2014-06-09 2014-06-09 Composicion farmaceutica que contiene derivado de hidantoina. MX371090B (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/JP2014/065262 WO2015189901A1 (ja) 2014-06-09 2014-06-09 ヒダントイン誘導体含有医薬組成物

Publications (2)

Publication Number Publication Date
MX2016013684A true MX2016013684A (es) 2017-01-20
MX371090B MX371090B (es) 2020-01-16

Family

ID=54833033

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2016013684A MX371090B (es) 2014-06-09 2014-06-09 Composicion farmaceutica que contiene derivado de hidantoina.

Country Status (10)

Country Link
US (1) US9993462B2 (es)
EP (1) EP3153166B1 (es)
KR (2) KR102266021B1 (es)
CN (2) CN106572994B (es)
AU (1) AU2014397042B2 (es)
BR (1) BR112016003511B8 (es)
CA (1) CA2949023C (es)
MX (1) MX371090B (es)
RU (1) RU2701168C2 (es)
WO (2) WO2015189901A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SG11201504204XA (en) * 2012-12-10 2015-07-30 Chugai Pharmaceutical Co Ltd Hydantoin derivative
BR112021001170A2 (pt) * 2018-07-30 2021-04-27 Chugai Seiyaku Kabushiki Kaisha dispersão sólida de derivado de hidantoína

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH1135470A (ja) 1997-07-23 1999-02-09 Teijin Ltd ビタミンd3誘導体を含有する副甲状腺ホルモン産生促進剤
CA2353924A1 (en) 1998-12-11 2000-06-22 F. Hoffmann-La Roche Ag Cyclic hydrazine derivatives as tnf-alpha inhibitors
US20050101574A1 (en) 2000-08-30 2005-05-12 Seiichi Ishizuka Parathyroid hormone production inhibitors containing vitamin d3 derivatives
JP2004518635A (ja) 2000-10-26 2004-06-24 ファイザー・プロダクツ・インク スピロ−ピリミジン−2,4,6−トリオンメタロプロテイナーゼ阻害剤
SE0100902D0 (sv) 2001-03-15 2001-03-15 Astrazeneca Ab Compounds
AR038658A1 (es) 2001-06-15 2005-01-26 Novartis Ag Derivados de 4-aril-2(1h) quinazolinona y 4-aril-quinazolina 2-sustituidas, un proceso para su preparacion, composiciones farmaceuticas y el uso de dichos derivados para la preparacion de un medicamento
EP1713815A4 (en) 2004-02-11 2009-03-11 Smithkline Beecham Corp PTH AGONISTS
WO2005077918A1 (en) 2004-02-11 2005-08-25 Smithkline Beecham Corporation Pth agonists
CA2582593A1 (en) 2004-10-07 2006-04-20 Merck & Co., Inc. Cgrp receptor antagonists
WO2007135417A1 (en) 2006-05-19 2007-11-29 James Black Foundation Benzotriazepinone derivatives
US20070299072A1 (en) * 2006-06-20 2007-12-27 Wyeth Kv1.5 potassium channel inhibitors
TW200831080A (en) * 2006-12-15 2008-08-01 Irm Llc Compounds and compositions as inhibitors of cannabinoid receptor 1 activity
ATE486058T1 (de) * 2007-06-07 2010-11-15 Hoffmann La Roche Prolinamidderivate als nk3-antagonisten
WO2009074575A2 (en) 2007-12-10 2009-06-18 Novartis Ag Organic compounds
US7981904B2 (en) 2008-03-20 2011-07-19 Takeda Pharmaceutical Company Limited Acetyl CoA carboxylase inhibitors
WO2010045229A2 (en) 2008-10-13 2010-04-22 University Of Rochester Protecting and repairing cartilage and musculoskeletal soft tissues
JP5671453B2 (ja) 2009-04-28 2015-02-18 中外製薬株式会社 スピロイミダゾロン誘導体
SG11201504204XA (en) * 2012-12-10 2015-07-30 Chugai Pharmaceutical Co Ltd Hydantoin derivative

Also Published As

Publication number Publication date
CN106535892B (zh) 2020-09-18
BR112016003511B8 (pt) 2023-10-03
CN106572994B (zh) 2020-09-18
AU2014397042A1 (en) 2016-02-11
RU2701168C2 (ru) 2019-09-25
EP3153166A1 (en) 2017-04-12
EP3153166B1 (en) 2022-08-03
WO2015189901A1 (ja) 2015-12-17
CA2949023A1 (en) 2015-12-17
US20170112812A1 (en) 2017-04-27
CN106535892A (zh) 2017-03-22
BR112016003511B1 (pt) 2022-11-08
EP3153166A4 (en) 2018-01-17
CA2949023C (en) 2021-10-12
KR102382331B1 (ko) 2022-04-01
AU2014397042B2 (en) 2020-04-09
MX371090B (es) 2020-01-16
BR112016003511A2 (es) 2017-08-01
RU2016113896A3 (es) 2018-07-18
RU2016113896A (ru) 2018-07-18
KR20170010354A (ko) 2017-01-31
KR102266021B1 (ko) 2021-06-16
BR112016003511A8 (pt) 2018-01-30
CN106572994A (zh) 2017-04-19
KR20170010439A (ko) 2017-01-31
WO2015190451A1 (ja) 2015-12-17
US9993462B2 (en) 2018-06-12

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