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MX2009009133A - Composiciones medicinales mejoradas que comprenden buprenorfina y naloxona. - Google Patents

Composiciones medicinales mejoradas que comprenden buprenorfina y naloxona.

Info

Publication number
MX2009009133A
MX2009009133A MX2009009133A MX2009009133A MX2009009133A MX 2009009133 A MX2009009133 A MX 2009009133A MX 2009009133 A MX2009009133 A MX 2009009133A MX 2009009133 A MX2009009133 A MX 2009009133A MX 2009009133 A MX2009009133 A MX 2009009133A
Authority
MX
Mexico
Prior art keywords
naloxone
buprenorphine
medicinal compositions
improved medicinal
composition
Prior art date
Application number
MX2009009133A
Other languages
English (en)
Inventor
Christopher Bourne Chapleo
Neil Hyde
Original Assignee
Reckitt Benckiser Healthcare
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Reckitt Benckiser Healthcare filed Critical Reckitt Benckiser Healthcare
Publication of MX2009009133A publication Critical patent/MX2009009133A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/485Morphinan derivatives, e.g. morphine, codeine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

Se proporciona una composición para el tratamiento de dolor en pacientes humanos en donde dicha composición comprende buprenorfina a naloxona en una relación en peso de 2.1:1 a 8:1, la cantidad de buprenorfina y naloxona es adecuada para proporcionar analgesia, la composición está en una forma de dosificación transdérmica o transmucósica. También se proporciona un método y uso relacionado.
MX2009009133A 2007-03-01 2008-02-15 Composiciones medicinales mejoradas que comprenden buprenorfina y naloxona. MX2009009133A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB0703967A GB2447015A (en) 2007-03-01 2007-03-01 Analgesic composition comprising a specific ratio of buprenorphine and naltrexone
PCT/GB2008/000523 WO2008104737A1 (en) 2007-03-01 2008-02-15 Improved medicinal compositions comprising buprenorphine and naloxone

Publications (1)

Publication Number Publication Date
MX2009009133A true MX2009009133A (es) 2009-09-03

Family

ID=37965734

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2009009133A MX2009009133A (es) 2007-03-01 2008-02-15 Composiciones medicinales mejoradas que comprenden buprenorfina y naloxona.

Country Status (16)

Country Link
US (1) US20100168147A1 (es)
EP (1) EP2114453A1 (es)
JP (1) JP2010520185A (es)
KR (1) KR20090115863A (es)
CN (2) CN101622013A (es)
AR (1) AR065581A1 (es)
AU (1) AU2008220573A1 (es)
BR (1) BRPI0807905A2 (es)
CA (1) CA2678675A1 (es)
CL (1) CL2008000610A1 (es)
GB (1) GB2447015A (es)
MX (1) MX2009009133A (es)
PE (1) PE20081874A1 (es)
TW (1) TW200836738A (es)
WO (1) WO2008104737A1 (es)
ZA (1) ZA200905691B (es)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2658585C (en) 2006-07-21 2011-03-01 Biodelivery Sciences International, Inc. Transmucosal delivery devices with enhanced uptake
CN102056578A (zh) * 2008-06-23 2011-05-11 生物递送科学国际公司 多向粘膜给药装置及使用方法
US8475832B2 (en) 2009-08-07 2013-07-02 Rb Pharmaceuticals Limited Sublingual and buccal film compositions
MX352959B (es) 2011-08-18 2017-12-15 Biodelivery Sciences Int Inc Dispositivos mucoadhesivos resistentes al abuso para el suministro de buprenorfina.
RS62505B1 (sr) 2011-09-19 2021-11-30 Orexo Ab Sublingvalne tablete otporne na zloupotrebu koje sadrže buprenorfin i nalokson
US9901539B2 (en) 2011-12-21 2018-02-27 Biodelivery Sciences International, Inc. Transmucosal drug delivery devices for use in chronic pain relief
US20140275148A1 (en) * 2013-03-15 2014-09-18 Novus Pharma LLC Orally administrable, self-supporting dissolving film dosage forms
WO2015095644A1 (en) 2013-12-20 2015-06-25 AntiOP, Inc. Intranasal naloxone compositions and methods of making and using same
US9561177B2 (en) 2014-03-14 2017-02-07 Adapt Pharma Limited Nasal drug products and methods of their use
US9480644B2 (en) 2014-03-14 2016-11-01 Opiant Pharmaceuticals, Inc. Nasal drug products and methods of their use
US10085937B2 (en) 2014-03-14 2018-10-02 Adapt Pharma Limited Nasal drug products and methods of their use
WO2015136373A1 (en) 2014-03-14 2015-09-17 Lightlake Therapeutics Inc. Nasal drug products and methods of their use
US20250144015A1 (en) 2023-11-06 2025-05-08 Extrovis Ag Pharmaceutical Compositions

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4457933A (en) * 1980-01-24 1984-07-03 Bristol-Myers Company Prevention of analgesic abuse
GB8332556D0 (en) * 1983-12-06 1984-01-11 Reckitt & Colmann Prod Ltd Analgesic compositions
JP2001526229A (ja) * 1997-12-22 2001-12-18 ユーロ−セルティーク,エス.エイ. オピオイド投薬剤形の乱用を防止する方法
AR031682A1 (es) 1999-11-19 2003-10-01 Reckitt Benckiser Helthcare Uk Composiciones farmaceuticas
US20050191340A1 (en) * 2002-08-09 2005-09-01 Gruenenthal Gmbh Opioid-receptor antagonists in transdermal systems having buprenorphine
ATE367155T1 (de) * 2002-08-09 2007-08-15 Gruenenthal Gmbh Opiod-rezeptor-antagonisten in transdermalen systemen mit buprenorphin
EP1584335A3 (en) * 2004-04-05 2006-02-22 Laboratorios Del Dr. Esteve, S.A. Active substance combination comprising a carbinol composition and an opioid
US8236751B2 (en) * 2007-03-07 2012-08-07 The Johns Hopkins University Methods of increasing muscle mass using follistatin-like related gene (FLRG)

Also Published As

Publication number Publication date
AU2008220573A1 (en) 2008-09-04
ZA200905691B (en) 2010-10-27
TW200836738A (en) 2008-09-16
CL2008000610A1 (es) 2008-09-05
CN102670610A (zh) 2012-09-19
BRPI0807905A2 (pt) 2014-06-17
CN101622013A (zh) 2010-01-06
JP2010520185A (ja) 2010-06-10
WO2008104737A1 (en) 2008-09-04
KR20090115863A (ko) 2009-11-09
US20100168147A1 (en) 2010-07-01
GB2447015A (en) 2008-09-03
GB0703967D0 (en) 2007-04-11
PE20081874A1 (es) 2009-01-26
CA2678675A1 (en) 2008-09-04
AR065581A1 (es) 2009-06-17
EP2114453A1 (en) 2009-11-11

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