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Schulman et al., 2012 - Google Patents

Local anesthetic pharmacology

Schulman et al., 2012

Document ID
15393778834372439146
Author
Schulman J
Strichartz G
Publication year
Publication venue
Principles of pharmacology: the pathophysiologic basis of drug therapy

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Snippet

INTRODUCTION The word anesthesia comes directly from the Greek:“an" meaning without, and “aisthesis” meaning feeling or sensation. Local anesthetics (LAs) are a set of locally applied chemicals, with similar molecular structures, that can both inhibit the perception of …
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine, rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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    • A61K31/445—Non condensed piperidines, e.g. piperocaine
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    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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