RAVIDA et al. - Google Patents
SYNTHESIS AND ELABORATION OF MONO-AND OLIGO-SACCHARIDESRAVIDA et al.
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- 11514613131246051911
- Author
- RAVIDA M
- DE NAPOLI L
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The extreme mildness of the above mentioned promoting systems is demonstrated by the syntheses of novel glycoconjugates with pharmacological activity. 17β-Estradiol and derivatives thereof are regioselectively glycosylated in order to improve their …
- 238000003786 synthesis reaction 0 title abstract description 98
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- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/02—Acyclic radicals, not substituted by cyclic structures
- C07H15/04—Acyclic radicals, not substituted by cyclic structures attached to an oxygen atom of the saccharide radical
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- C07H13/02—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids by carboxylic acids
- C07H13/04—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids by carboxylic acids having the esterifying carboxyl radicals attached to acyclic carbon atoms
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- C07H15/14—Acyclic radicals, not substituted by cyclic structures attached to a sulfur, selenium or tellurium atom of a saccharide radical
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- C07H13/12—Compounds containing saccharide radicals esterified by carbonic acid or derivatives thereof, or by organic acids, e.g. phosphonic acids by acids having the group -X-C(=X)-X-, or halides thereof, in which each X means nitrogen, oxygen, sulfur, selenium or tellurium, e.g. carbonic acid, carbamic acid
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