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Derks et al., 2021 - Google Patents

Strain-promoted azide–alkyne cycloaddition-based PSMA-targeting ligands for multimodal intraoperative tumor detection of prostate cancer

Derks et al., 2021

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Document ID
9690146898493277818
Author
Derks Y
Rijpkema M
Amatdjais-Groenen H
Loeff C
de Roode K
Kip A
Laverman P
Lütje S
Heskamp S
Lowik D
Publication year
Publication venue
Bioconjugate chemistry

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Snippet

Strain-promoted azide–alkyne cycloaddition (SPAAC) is a straightforward and multipurpose conjugation strategy. The use of SPAAC to link different functional elements to prostate- specific membrane antigen (PSMA) ligands would facilitate the development of a modular …
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