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Jordi et al., 1992 - Google Patents

Asymmetric synthesis of pyrrolo [2, 1-b][1, 3, 4] thiadiazepine derivatives

Jordi et al., 1992

Document ID
7378421922184837141
Author
Jordi B
Angel P
Santiago G
Lluís A
Aurelio S
Ortiz J
Publication year
Publication venue
Tetrahedron

External Links

Snippet

The asymmetric synthesis of compound 2, with potential ACE inhibitory activity, is reported. The key intermediaet 3 contains the novel heterocyclic nucleus pyrrolo [2, 1-b][1, 3, 4] thiadiazepine. This compound has been prepared through a sequence involving pyrrole …
Continue reading at www.sciencedirect.com (other versions)

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    • C07D207/04Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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