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Kwiatkowska et al., 2009 - Google Patents

Arginine vasopressin and its analogues–The influence of position 2 modification with 3, 3-diphenylalanine enantiomers. Highly potent V2 agonists

Kwiatkowska et al., 2009

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Document ID
6620765182921636941
Author
Kwiatkowska A
Sobolewski D
Prahl A
Borovičková L
Slaninová J
Lammek B
Publication year
Publication venue
European journal of medicinal chemistry

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Eleven new analogues of arginine vasopressin (AVP) modified in position 2 by 3, 3-diphenyl- l-alanine or its d-enantiomer (Dip or d-Dip) were synthesized and pharmacologically evaluated for their pressor, antidiuretic and in vitro uterotonic activities. Both the Dip and d …
Continue reading at www.academia.edu (PDF) (other versions)

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