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PL2069332T3 - Związki azetydynowe jako antagoniści receptorów oreksynowych - Google Patents

Związki azetydynowe jako antagoniści receptorów oreksynowych

Info

Publication number
PL2069332T3
PL2069332T3 PL07826034T PL07826034T PL2069332T3 PL 2069332 T3 PL2069332 T3 PL 2069332T3 PL 07826034 T PL07826034 T PL 07826034T PL 07826034 T PL07826034 T PL 07826034T PL 2069332 T3 PL2069332 T3 PL 2069332T3
Authority
PL
Poland
Prior art keywords
receptor antagonists
orexin receptor
azetidine compounds
compounds
azetidine
Prior art date
Application number
PL07826034T
Other languages
English (en)
Inventor
Hamed Aissaoui
Christoph Boss
Markus Gude
Ralf Koberstein
Thierry Sifferlen
Original Assignee
Actelion Pharmaceuticals Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Actelion Pharmaceuticals Ltd filed Critical Actelion Pharmaceuticals Ltd
Publication of PL2069332T3 publication Critical patent/PL2069332T3/pl

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    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K31/397—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
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PL07826034T 2006-08-15 2007-08-15 Związki azetydynowe jako antagoniści receptorów oreksynowych PL2069332T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IB2006052814 2006-08-15
EP07826034A EP2069332B1 (en) 2006-08-15 2007-08-15 Azetidine compounds as orexin receptor antagonists
PCT/IB2007/053244 WO2008020405A2 (en) 2006-08-15 2007-08-15 Azetidine compounds as orexin receptor antagonists

Publications (1)

Publication Number Publication Date
PL2069332T3 true PL2069332T3 (pl) 2011-07-29

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Application Number Title Priority Date Filing Date
PL07826034T PL2069332T3 (pl) 2006-08-15 2007-08-15 Związki azetydynowe jako antagoniści receptorów oreksynowych

Country Status (15)

Country Link
US (1) US7994336B2 (pl)
EP (1) EP2069332B1 (pl)
JP (1) JP2010500401A (pl)
KR (1) KR101113626B1 (pl)
CN (1) CN101506199A (pl)
AT (1) ATE500250T1 (pl)
AU (1) AU2007285371A1 (pl)
BR (1) BRPI0715893A2 (pl)
CA (1) CA2659299A1 (pl)
DE (1) DE602007012910D1 (pl)
ES (1) ES2360376T3 (pl)
MX (1) MX2009001432A (pl)
PL (1) PL2069332T3 (pl)
RU (1) RU2447070C2 (pl)
WO (1) WO2008020405A2 (pl)

Families Citing this family (37)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2350460T3 (es) * 2006-09-29 2011-01-24 Actelion Pharmaceuticals Ltd. Derivados de 3-aza-biciclo[3.1.0]hexano.
CN101568533A (zh) 2006-12-01 2009-10-28 埃科特莱茵药品有限公司 3-异芳基(氨基或酰胺基)-1-(联苯或苯基噻唑基)羰基哌啶衍生物食欲素受体抑制剂
CL2007003827A1 (es) * 2006-12-28 2008-09-26 Actelion Pharmaceuticals Ltd Compuestos derivados de n-(2-aza-biciclo(3.1.0)hex-3-ilmetil)amida; y su uso para prevenir o tratar la depresion, neurosis, esquizofrenia, ansiedad, adicciones, epilepsia, dolor, enfermedades cardiacas, entre otras.
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