HUP0103929A2 - Antibakteriális hatású heterociklil-amino-metil-oxazolidinonok és az ezeket tartalmazó gyógyszerkészítmények - Google Patents
Antibakteriális hatású heterociklil-amino-metil-oxazolidinonok és az ezeket tartalmazó gyógyszerkészítményekInfo
- Publication number
- HUP0103929A2 HUP0103929A2 HU0103929A HUP0103929A HUP0103929A2 HU P0103929 A2 HUP0103929 A2 HU P0103929A2 HU 0103929 A HU0103929 A HU 0103929A HU P0103929 A HUP0103929 A HU P0103929A HU P0103929 A2 HUP0103929 A2 HU P0103929A2
- Authority
- HU
- Hungary
- Prior art keywords
- methyloxazolidinones
- antibacterials
- same
- pharmaceutical compositions
- compositions containing
- Prior art date
Links
- -1 Heterocyclyl amino methyloxazolidinones Chemical class 0.000 title 1
- 230000000844 anti-bacterial effect Effects 0.000 title 1
- 229940088710 antibiotic agent Drugs 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
- C07F9/65583—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system each of the hetero rings containing nitrogen as ring hetero atom
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Oncology (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Communicable Diseases (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9821938.9A GB9821938D0 (en) | 1998-10-09 | 1998-10-09 | Chemical compounds |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| HUP0103929A2 true HUP0103929A2 (hu) | 2002-07-29 |
| HUP0103929A3 HUP0103929A3 (en) | 2002-08-28 |
Family
ID=10840200
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HU0103929A HUP0103929A3 (en) | 1998-10-09 | 1999-10-05 | Heterocyclyl amino methyloxazolidinones as antibacterials and pharmaceutical compositions containing the same |
Country Status (15)
| Country | Link |
|---|---|
| US (2) | US6734200B1 (hu) |
| EP (1) | EP1121358A1 (hu) |
| JP (1) | JP2002527439A (hu) |
| KR (1) | KR20010085887A (hu) |
| CN (1) | CN1165534C (hu) |
| AU (1) | AU754123B2 (hu) |
| BR (1) | BR9914379A (hu) |
| CA (1) | CA2342623A1 (hu) |
| GB (1) | GB9821938D0 (hu) |
| HU (1) | HUP0103929A3 (hu) |
| IL (1) | IL142420A0 (hu) |
| NO (1) | NO20011738L (hu) |
| NZ (1) | NZ510211A (hu) |
| WO (1) | WO2000021960A1 (hu) |
| ZA (1) | ZA200102659B (hu) |
Families Citing this family (41)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9821938D0 (en) * | 1998-10-09 | 1998-12-02 | Zeneca Ltd | Chemical compounds |
| GB9928568D0 (en) | 1999-12-03 | 2000-02-02 | Zeneca Ltd | Chemical compounds |
| US6642238B2 (en) | 2000-02-10 | 2003-11-04 | Pharmacia And Upjohn Company | Oxazolidinone thioamides with piperazine amide substituents |
| GB0009803D0 (en) * | 2000-04-25 | 2000-06-07 | Astrazeneca Ab | Chemical compounds |
| PE20030044A1 (es) | 2000-11-17 | 2003-02-09 | Upjohn Co | Isoxazolinonas biciclicas de formula i |
| PE20020689A1 (es) | 2000-11-17 | 2002-08-03 | Upjohn Co | Oxazolidinonas con un heterociclo de 6 o 7 miembros unidos con enlace anular al benceno |
| GB0108793D0 (en) * | 2001-04-07 | 2001-05-30 | Astrazeneca Ab | Chemical compounds |
| GB0113300D0 (en) * | 2001-06-01 | 2001-07-25 | Astrazeneca Ab | Purification process |
| GB0113299D0 (en) * | 2001-06-01 | 2001-07-25 | Astrazeneca Ab | Chemical process & intermediates |
| GB0113298D0 (en) * | 2001-06-01 | 2001-07-25 | Astrazeneca Ab | Purification process and intermediates |
| CA2459766A1 (en) | 2001-09-11 | 2003-03-20 | Astrazeneca Ab | Oxazolidinone and/or isoxazoline as antibacterial agents |
| US7022705B2 (en) | 2001-10-25 | 2006-04-04 | Astrazeneca Ab | Isoxazoline derivatives useful as antimicrobials |
| AR038536A1 (es) | 2002-02-25 | 2005-01-19 | Upjohn Co | N-aril-2-oxazolidinona-5- carboxamidas y sus derivados |
| US7141588B2 (en) | 2002-02-25 | 2006-11-28 | Pfizer, Inc. | N-aryl-2-oxazolidinone-5-carboxamides and their derivatives |
| BR0308018A (pt) | 2002-02-28 | 2005-01-04 | Astrazeneca Ab | Composto ou um seu sal farmaceuticamente aceitável ou um seu éster hidrolisável in vivo, pró-droga, método para produzir um efeito antibacteriano em um animal de sangue quente, uso de um composto ou um seu sal farmaceuticamente aceitável ou um seu éster hirolisável in vivo, composição farmacêutica, e, processo para a preparação de um composto ou um seu sal farmaceuticamente aceitável ou um seu éster hidrolisável in vivo |
| IL163688A0 (en) | 2002-02-28 | 2005-12-18 | Astrazeneca Ab | 3-Cyclyl-5-(nitrogen-containing 5-membered ring)methyl-oxazolidinone derivatives and theiruse as antibacterial agents |
| ES2258234T3 (es) | 2002-08-12 | 2006-08-16 | PHARMACIA & UPJOHN COMPANY LLC | N-aril-2-oxazolidinonas y sus derivados. |
| AR043050A1 (es) * | 2002-09-26 | 2005-07-13 | Rib X Pharmaceuticals Inc | Compuestos heterociclicos bifuncionales y metodos para preparar y usar los mismos |
| US6875784B2 (en) | 2002-10-09 | 2005-04-05 | Pharmacia & Upjohn Company | Antimibicrobial [3.1.0.] bicyclic oxazolidinone derivatives |
| JP2006509035A (ja) | 2002-11-21 | 2006-03-16 | ファルマシア・アンド・アップジョン・カンパニー・エルエルシー | 抗菌剤としてのｎ−（４−（ピペラジン−１−イル）−フェニル−２−オキサゾリジノン−５−カルボキサミド誘導体および関連化合物 |
| GB0227701D0 (en) * | 2002-11-28 | 2003-01-08 | Astrazeneca Ab | Chemical compounds |
| GB0229518D0 (en) * | 2002-12-19 | 2003-01-22 | Astrazeneca Ab | Chemical compounds |
| GB0229522D0 (en) * | 2002-12-19 | 2003-01-22 | Astrazeneca Ab | Chemical compounds |
| US7012088B2 (en) | 2003-02-24 | 2006-03-14 | Pharmacia & Upjohn Company | Indolone oxazolidinones and derivatives thereof |
| MXPA05010783A (es) | 2003-04-09 | 2005-12-12 | Pharmacia & Upjohn Co Llc | Derivados antimicrobianos de [3.1.0] biciclohexilfenil-oxazolidinona y analogos. |
| EP1625124A1 (en) * | 2003-05-06 | 2006-02-15 | Ranbaxy Laboratories, Ltd. | Oxazolidinone derivatives as antimicrobials |
| US8324398B2 (en) | 2003-06-03 | 2012-12-04 | Rib-X Pharmaceuticals, Inc. | Process for the synthesis of biaryl oxazolidinones |
| TWI378092B (en) | 2003-06-03 | 2012-12-01 | Rib X Pharmaceuticals Inc | Biaryl heterocyclic compounds and methods of making and using the same |
| WO2004113329A1 (en) * | 2003-06-20 | 2004-12-29 | Orchid Chemicals And Pharmaceuticals Ltd. | Oxazole derivatives as antibacterial agents |
| WO2005003087A2 (en) * | 2003-07-01 | 2005-01-13 | Orchid Chemicals And Pharmaceuticals Ltd. | Oxazole derivatives as antibacterial agents |
| US7687627B2 (en) * | 2003-09-08 | 2010-03-30 | Wockhardt Limited | Substituted piperidino phenyloxazolidinones having antimicrobial activity with improved in vivo efficacy |
| US7304050B2 (en) | 2003-09-16 | 2007-12-04 | Pfizer Inc. | Antibacterial agents |
| JP2007514782A (ja) | 2003-12-17 | 2007-06-07 | リブ−エックス ファーマシューティカルズ，インコーポレイテッド | ハロゲン化ビアリール複素環式化合物ならびにその作製方法および使用方法 |
| US8202843B2 (en) | 2004-02-27 | 2012-06-19 | Rib-X Pharmaceuticals, Inc. | Macrocyclic compounds and methods of making and using the same |
| ATE496914T1 (de) | 2005-06-08 | 2011-02-15 | Rib X Pharmaceuticals Inc | Verfahren zur synthese von triazolen |
| US8278281B2 (en) | 2005-08-24 | 2012-10-02 | Rib-X Pharmaceuticals, Inc. | Triazole compounds and methods of making and using the same |
| CN101798302B (zh) | 2009-02-06 | 2014-11-05 | 上海盟科药业有限公司 | 抗生素类药物1-(邻-氟苯基)二氢吡啶酮的合成及生产的方法和工艺 |
| KR20130028703A (ko) * | 2009-11-04 | 2013-03-19 | 쓰촨 베이라이크 바이오테크놀로지 리미티드 라이어빌러티 컴퍼니 | 결정성 수화물, 이의 약학적 조성물 및 제조 방법 및 용도 |
| WO2013182070A1 (zh) * | 2012-06-08 | 2013-12-12 | 四川贝力克生物技术有限责任公司 | 一种用于预防或治疗分支杆菌疾病的药物 |
| ES2753244T3 (es) * | 2013-03-15 | 2020-04-07 | Univ Degli Studi Di Milano Bicocca | Compuestos novedosos 1,2,4 oxadiazol activos contra patógenos gram positivos |
| US9382276B2 (en) | 2014-02-21 | 2016-07-05 | Micurx Pharmaceuticals, Inc. | Water-soluble O-carbonyl phosphoramidate prodrugs for therapeutic administration |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES533097A0 (es) * | 1983-06-07 | 1985-08-01 | Du Pont | Un procedimiento para la preparacion de nuevos derivados del amino-metil-oxooxazolidinil-benzeno. |
| US4705799A (en) * | 1983-06-07 | 1987-11-10 | E. I. Du Pont De Nemours And Company | Aminomethyl oxooxazolidinyl benzenes useful as antibacterial agents |
| DE19604223A1 (de) * | 1996-02-06 | 1997-08-07 | Bayer Ag | Neue substituierte Oxazolidinone |
| GB9821938D0 (en) * | 1998-10-09 | 1998-12-02 | Zeneca Ltd | Chemical compounds |
-
1998
- 1998-10-09 GB GBGB9821938.9A patent/GB9821938D0/en not_active Ceased
-
1999
- 1999-10-05 BR BR9914379-8A patent/BR9914379A/pt not_active IP Right Cessation
- 1999-10-05 JP JP2000575866A patent/JP2002527439A/ja active Pending
- 1999-10-05 AU AU61131/99A patent/AU754123B2/en not_active Ceased
- 1999-10-05 WO PCT/GB1999/003299 patent/WO2000021960A1/en not_active Application Discontinuation
- 1999-10-05 KR KR1020017004351A patent/KR20010085887A/ko not_active Ceased
- 1999-10-05 US US09/807,113 patent/US6734200B1/en not_active Expired - Fee Related
- 1999-10-05 EP EP99947761A patent/EP1121358A1/en not_active Withdrawn
- 1999-10-05 HU HU0103929A patent/HUP0103929A3/hu unknown
- 1999-10-05 IL IL14242099A patent/IL142420A0/xx unknown
- 1999-10-05 CA CA002342623A patent/CA2342623A1/en not_active Abandoned
- 1999-10-05 NZ NZ510211A patent/NZ510211A/en unknown
- 1999-10-05 CN CNB998118346A patent/CN1165534C/zh not_active Expired - Fee Related
-
2001
- 2001-03-30 ZA ZA200102659A patent/ZA200102659B/en unknown
- 2001-04-06 NO NO20011738A patent/NO20011738L/no not_active Application Discontinuation
-
2003
- 2003-03-06 US US10/382,396 patent/US7087629B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| JP2002527439A (ja) | 2002-08-27 |
| NO20011738L (no) | 2001-06-07 |
| CN1165534C (zh) | 2004-09-08 |
| KR20010085887A (ko) | 2001-09-07 |
| NO20011738D0 (no) | 2001-04-06 |
| US20030207899A1 (en) | 2003-11-06 |
| AU6113199A (en) | 2000-05-01 |
| CN1322203A (zh) | 2001-11-14 |
| US6734200B1 (en) | 2004-05-11 |
| AU754123B2 (en) | 2002-11-07 |
| ZA200102659B (en) | 2002-07-01 |
| US7087629B2 (en) | 2006-08-08 |
| BR9914379A (pt) | 2001-08-07 |
| NZ510211A (en) | 2003-05-30 |
| EP1121358A1 (en) | 2001-08-08 |
| CA2342623A1 (en) | 2000-04-20 |
| GB9821938D0 (en) | 1998-12-02 |
| WO2000021960A1 (en) | 2000-04-20 |
| HUP0103929A3 (en) | 2002-08-28 |
| IL142420A0 (en) | 2002-03-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD9A | Lapse of provisional protection due to non-payment of fees |