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EA201600442A1 - Мягкая фармацевтическая композиция на водной основе, содержащая тапентадол - Google Patents

Мягкая фармацевтическая композиция на водной основе, содержащая тапентадол

Info

Publication number
EA201600442A1
EA201600442A1 EA201600442A EA201600442A EA201600442A1 EA 201600442 A1 EA201600442 A1 EA 201600442A1 EA 201600442 A EA201600442 A EA 201600442A EA 201600442 A EA201600442 A EA 201600442A EA 201600442 A1 EA201600442 A1 EA 201600442A1
Authority
EA
Eurasian Patent Office
Prior art keywords
pharmaceutical composition
water basis
containing tapentadol
basis containing
soft pharmaceutical
Prior art date
Application number
EA201600442A
Other languages
English (en)
Other versions
EA033171B1 (ru
Inventor
Ульрих Райнхольд
Марк Шиллер
Эва Вульстен
Сабине Карине Катрин Ингхельбрехт
Роже Каролус Аугуста Эмбрехтс
Ульрих Файль
Original Assignee
Грюненталь Гмбх
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Грюненталь Гмбх filed Critical Грюненталь Гмбх
Publication of EA201600442A1 publication Critical patent/EA201600442A1/ru
Publication of EA033171B1 publication Critical patent/EA033171B1/ru

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/14—Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0014—Skin, i.e. galenical aspects of topical compositions
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/06—Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Engineering & Computer Science (AREA)
  • Dermatology (AREA)
  • Emergency Medicine (AREA)
  • Dispersion Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Rheumatology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)

Abstract

Изобретение относится к мягкой фармацевтической композиции на водной основе, содержащей тапентадол или его физиологически приемлемую соль.
EA201600442A 2011-03-04 2012-03-02 Полутвёрдая фармацевтическая композиция на водной основе, содержащая тапентадол EA033171B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201161449329P 2011-03-04 2011-03-04
EP11003603 2011-05-03

Publications (2)

Publication Number Publication Date
EA201600442A1 true EA201600442A1 (ru) 2017-02-28
EA033171B1 EA033171B1 (ru) 2019-09-30

Family

ID=44652117

Family Applications (2)

Application Number Title Priority Date Filing Date
EA201300988A EA025194B1 (ru) 2011-03-04 2012-03-02 Полутвёрдая фармацевтическая композиция на водной основе, содержащая тапентадол
EA201600442A EA033171B1 (ru) 2011-03-04 2012-03-02 Полутвёрдая фармацевтическая композиция на водной основе, содержащая тапентадол

Family Applications Before (1)

Application Number Title Priority Date Filing Date
EA201300988A EA025194B1 (ru) 2011-03-04 2012-03-02 Полутвёрдая фармацевтическая композиция на водной основе, содержащая тапентадол

Country Status (24)

Country Link
US (3) US9446008B2 (ru)
EP (3) EP3766489B1 (ru)
JP (3) JP6027549B2 (ru)
KR (2) KR101911362B1 (ru)
CN (1) CN103501774A (ru)
AU (2) AU2012224954C1 (ru)
BR (1) BR112013022556A8 (ru)
CA (1) CA2828637C (ru)
CY (1) CY1119725T1 (ru)
DK (1) DK2680834T3 (ru)
EA (2) EA025194B1 (ru)
ES (2) ES2654407T3 (ru)
HR (1) HRP20171836T1 (ru)
HU (1) HUE037491T2 (ru)
IL (2) IL227826B (ru)
LT (1) LT2680834T (ru)
MX (1) MX344473B (ru)
NO (1) NO2680834T3 (ru)
PL (1) PL2680834T3 (ru)
PT (2) PT3766489T (ru)
RS (1) RS56692B1 (ru)
SI (1) SI2680834T1 (ru)
WO (1) WO2012119729A1 (ru)
ZA (1) ZA201306480B (ru)

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EP3287123B1 (en) 2011-03-04 2020-04-22 Grünenthal GmbH Aqueous pharmaceutical formulation of tapentadol for oral administration
ES2654407T3 (es) * 2011-03-04 2018-02-13 Grünenthal GmbH Composición farmacéutica acuosa semisólida que contiene tapentadol
US9395306B2 (en) 2011-08-05 2016-07-19 Halliburton Energy Services, Inc. Methods for monitoring fluids within or produced from a subterranean formation during acidizing operations using opticoanalytical devices
US8997860B2 (en) 2011-08-05 2015-04-07 Halliburton Energy Services, Inc. Methods for monitoring the formation and transport of a fracturing fluid using opticoanalytical devices
US20140076550A1 (en) 2012-09-14 2014-03-20 Halliburton Energy Services, Inc. Systems and Methods for Detecting Microannulus Formation and Remediation
US8619256B1 (en) 2012-09-14 2013-12-31 Halliburton Energy Services, Inc. Systems and methods for monitoring the properties of a fluid cement composition in a flow path
US9228940B2 (en) 2012-09-14 2016-01-05 Halliburton Energy Services, Inc. Systems, methods, and apparatuses for in situ monitoring of cement fluid compositions and setting processes thereof
US20160136112A1 (en) * 2013-08-02 2016-05-19 Ratiopharm Gmbh Composition comprising tapentadol in a dissolved form
EP2845625A1 (en) 2013-09-04 2015-03-11 Grünenthal GmbH Tapentadol for use in the treatment of fibromyalgia and chronic fatigue syndrome
TW201642843A (zh) * 2015-03-27 2016-12-16 歌林達有限公司 他噴他多腸胃外給藥的穩定製劑
CA3037810A1 (en) * 2016-09-23 2018-03-29 Grunenthal Gmbh Stable formulation for parenteral administration of tapentadol
WO2020020879A1 (en) * 2018-07-24 2020-01-30 Dr. August Wolff Gmbh & Co. Kg Arzneimittel Topical emulsion of an anticholinergic compound

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Also Published As

Publication number Publication date
IL227826A0 (en) 2013-09-30
KR102039320B1 (ko) 2019-11-01
JP2014506900A (ja) 2014-03-20
CA2828637A1 (en) 2012-09-13
JP2017039756A (ja) 2017-02-23
BR112013022556A2 (pt) 2016-12-06
AU2017200040A1 (en) 2017-02-02
BR112013022556A8 (pt) 2018-01-16
CN103501774A (zh) 2014-01-08
EA025194B1 (ru) 2016-11-30
WO2012119729A1 (en) 2012-09-13
PT3766489T (pt) 2022-04-07
RS56692B1 (sr) 2018-03-30
AU2012224954B2 (en) 2016-10-20
IL227826B (en) 2018-04-30
SI2680834T1 (en) 2018-01-31
JP6027549B2 (ja) 2016-11-16
KR20180116463A (ko) 2018-10-24
AU2012224954C1 (en) 2017-04-06
EP2680834B1 (en) 2017-10-18
EP2680834A1 (en) 2014-01-08
EP3766489A1 (en) 2021-01-20
HUE037491T2 (hu) 2018-09-28
EP3290029A1 (en) 2018-03-07
LT2680834T (lt) 2018-01-10
ES2910085T3 (es) 2022-05-11
KR20140013020A (ko) 2014-02-04
HRP20171836T1 (hr) 2017-12-29
JP6259042B2 (ja) 2018-01-10
EP3766489B1 (en) 2022-03-16
IL258357A (en) 2018-05-31
CY1119725T1 (el) 2018-06-27
AU2017200040B2 (en) 2018-09-06
JP6670283B2 (ja) 2020-03-18
PL2680834T3 (pl) 2018-03-30
US20180133174A1 (en) 2018-05-17
KR101911362B1 (ko) 2018-10-25
MX2013010100A (es) 2013-10-01
US20160346229A1 (en) 2016-12-01
ZA201306480B (en) 2014-05-28
DK2680834T3 (en) 2017-12-04
MX344473B (es) 2016-12-16
PT2680834T (pt) 2018-01-25
US20120225950A1 (en) 2012-09-06
CA2828637C (en) 2019-06-11
EP3290029B1 (en) 2020-09-02
EA033171B1 (ru) 2019-09-30
AU2012224954A1 (en) 2013-09-19
JP2018065839A (ja) 2018-04-26
ES2654407T3 (es) 2018-02-13
US9446008B2 (en) 2016-09-20
NO2680834T3 (ru) 2018-03-17
EA201300988A1 (ru) 2014-06-30

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Legal Events

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MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): AM AZ BY KZ KG MD TJ TM

MM4A Lapse of a eurasian patent due to non-payment of renewal fees within the time limit in the following designated state(s)

Designated state(s): RU