CZ20004923A3 - Paroxetine salts - Google Patents

Abstract

Piperidine compounds, processes for preparing them, pharmaceutical compositions comprising them and their use in therapy are disclosed.

Description

Technical field

The present invention relates to novel compounds, processes for its preparation and its use in the treatment of internal disorders.

BACKGROUND OF THE INVENTION

Pharmaceutical products with antidepressant and antiparkinsonian properties are described in US-A-3 912 743 and US-A-4 007 196. Among the compounds described, paroxetine, the (-) - trans isomer is particularly important.

4- (4'-Fluorophenyl) -3- (3 ', 4'-methylenedioxyphenoxymethyl) piperidine. This compound is used in therapy as the hydrochloride salt for the treatment and prophylaxis of, inter alia, depression, obsessive compulsive disorder (OCD) and panic.

SUMMARY OF THE INVENTION

The present invention provides novel salts of paroxetine that can be used as an alternative to the hydrochloride currently on the market or as an intermediate for the preparation of the hydrochloride.

According to the present invention, there are provided salts of paroxetine with acids selected from the group consisting of:

2-methyl-3-phenylbutyric acid, tricyclo (10,2,2,2 (4,7)) octadeca-hexaene-9,10-dicarboxylic acid,

1-Pyreneacetic acid

2,4,6-trifluoro-cinnamic acid,

2-bromoisobutyric acid, cyclohexylsuccinic acid,

3,5-dichloro-2,6-dimethoxybenzoic acid,

5-ethoxy-2-hydroxybenzoic acid, trans-11-icosenoic acid,

3-bromopropionic acid,

3- [5- (4-bromophenyl) -2-furyl] acrylic acid,

2-Phenylacrylic acid

21-docosenoic acid, n- (p-amylcinnamoyl) anthranilic acid, (2'-methyl-4'-amino) phenylazonaphthylene-3,8-disulfonic acid,

7.7- dimethylikosadienoic acid,

2.5- dibromobenzenesulfonic acid,

5.7-icosadioic acid, nonadec-18-enoic acid,

3-methoxycyclohexanecarboxylic acid,

5-chloro-2-thiophenecarboxylic acid, β-naphthyl phosphate,

2- (1,4-Benzodioxan-2-yl) thiazole-4-carboxylic acid

2-methyl-1,6-naphthyrdrine-3-carboxylic acid, (10-ho-10-ph-4h-8-thia-7,10a-diazapentaleno (1,2-a) naphthalen-9-yl) acetic acid , fmoc-iso (hexahydropyridine-4-carboxylic acid),

4- [3- (2-fluoro-5-nitrophenyl) ureido] benzoic acid, n-ethylmaleinamic acid,

7-methoxycoumarin-4-acetic acid, trans-4-n-pentylcyclohexanecarboxylic acid,

2,4-dimethylcinnamic acid, (S) -3-methylnonanoic acid,

3-maleimimidobenzoic acid, acetoxyvalerenic acid,

7,12-Dimethylbenz (a) anthracene-5-carboxylic acid

4-chlorophthalic acid,

2- (carboxymethylamino) -6-chlorobenzoic acid,

3'-methoxyphthalanilic acid,

1- (+) - 2-amino-6-phosphonohexanoic acid, (L) -2,3-diacetoxy-n- [1- (1-naphthyl) ethyl] succinic acid diamide,

4-fluorophenoxydifluoroacetic acid,

3- (2-chloro-6-fluorophenyl) -5-methylisoxazole-4-carboxylic acid,

3- [4- (2-ethoxycarbonyl) -2,5-dimethoxyphenyl (propionic acid,

6- (6-hydroxy-3-oxo-3h-xanthen-9-yl) -3-cyclohexene-1-carboxylic acid, cis-n-tert-butylhexahydrophthalamic acid,

2.5- dihydroxycinnamic acid,

3-bromo-2- (bromomethyl) propionic acid,

3-ethyl-3-phenylglutaric acid, α- (2,4-dimethoxy-6-methylbenzylidene) hippuric acid,

5-phenylvaleric acid, (+/-) - 2-amino-3- [3- (carboxymethoxy) -5-methyl-4-isoxazolyl] propionic acid,

4-aminonicotinic acid, p-fluoro-α-acetamidicinnamic acid,

2.5-dihydroxybenzoic acid,

10- (1-pyrene) -10-ketodecanoic acid,

2-chloro-3,5-dinitrobenzoic acid, p-azoxybenzoic acid,

2-ethylthio-2,2-diphenylacetic acid,

4- (3-Cinnamoyl-2-thioureido) benzoic acid

2-hydroxydibenzofuran-3-carboxylic acid,

2- (3,5-dinitro-2-thienylamino) pentanoic acid,

2-Benzoylamino-cyclohexanecarboxylic acid

3-hydroxyhomophthalic acid,

2.5- dibromobenzoic acid,

4- (2-chloro-2-cyanoethyl) benzoic acid,

2-methylhydric cinnamic acid,

13-methylpentadecanoic acid,

3.4.5- trimethoxyphenylacetic acid,

D, L-2-hydroxy-4- (methylthio) butyric acid,

2-oxoadipic acid, bromoacetic acid,

1- (4-Isopropyl-3-methylphenyl) -5-oxo-pyrrolidine-3-carboxylic acid, perfluorazelaic acid, acetylsyringic acid,

3'-acetylphthalic acid, α-bromophenylacetic acid,

3- (3,4-diacetoxy-5-methylphenyl) acrylic acid, p-iodicinnamic acid,

4,4'-methylenebis (maleic acid),

3- (4-Trifluoromethylsulfanyl-phenylcarbamoyl) acrylic acid

3- [2- (2-pyrazyl) -1- [4- (trifluoromethyl) phenyl] ethoxy] propanoic acid,

2-Phenoxybutyric acid

2- [4-chloro (phenylsulfonyl) anilino] acetic acid, boc-D, L-3-aminobutyric acid,

3.5-dinitrobenzoic acid,

4-tert-butylcyclohexanecarboxylic acid, (R) -2,2-dimethyl-3-formyl-4-thiazolidinecarboxylic acid, (2S, 2S) - (-) - azetidine-2,4-dicarboxylic acid,

2- (4-nitrophenyl) -3-phenylacrylic acid,

3-nitrobenzoic acid,

10,11-dihydro-dibenzo (b, f) oxepine-4,6-dicarboxylic acid, (2-isopropyl-5-oxocyclohexyloxy) acetic acid,

(S) - (-) - N- (1-phenethyl) succinamic acid,

6- (2-bromobenzoyl (hexanoic acid, (lot, 3ot, 5β) -1,3,5-trimethyl-1,3,5-cyclohexanetricarboxylic acid),

2-methylpropanetricarboxylic acid,

5- (4-hydroxymethyl-3-methoxyphenoxy (valeric acid,

N- (3,4-dicyanophenyl) phthalamic acid,

5-fluorosalicylic acid, itaconic acid,

2,2-dimethylcyclobutane-1,3,3,3-tetracarboxylic acid,

8-hydroxy-5- (4-sulfophenylazo) -2-naphthalenesulfonic acid,

3- (4-chlorophenylthio)

N-benzylglutaramic acid,

3- (2,5-dimethoxybenzoyl) propionic acid,

4-Cyanocinnamic acid

2- (4-methoxyphenyl) -1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxylic acid,

2-hydroxyimino-pentanedioic acid,

6-methyl-1,3-benzodioxole-5-carboxylic acid,

2- (4-hydroxyphenoxy) propionic acid,

7H-dodecafluoroheptanoic acid,

3 ', 5'-dimethylmaleinanilic acid,

2-butyl-5-tert-butylisophthalic acid,

4-chloro-2-phthalimidobenzoic acid,

2-methyl-1,3-dithiolane-2-propionic acid,

4-chloro-2-nitrophenol-6-sulfonic acid, N-methyl-L-glutamic acid,

4,6,2 ', 4'-tetranitro-biphenyl-2-carboxylic acid, (R) - (-) - 2-amino-2-methylbutanedioic acid, - [2-C4-tert-butylphenoxy) -5- nitrophenyl (acrylic acid,

4- (trifluoromethylthio) phenylacetic acid, dithiodiglycolic acid,

N, N-bis (phosphonomethyl (glycine)

3- [10- (2-ethoxycarbonyl) anthracen-9-yl] propionic acid, cinnamic acid,

3,6-Dichloro-5-hydroxy-o-anisic acid

3,5-difluorophenylacetic acid,

2 '- (trifluoromethyl) succinanilic acid, cis-5,8,11,14,17-icosapentaenoic acid,

3,3 '- (dimethylsilylene) bispropionic acid,

1- (3-chloro-5-trifluoromethyl-2-pyridyl) pyrrole-2-carboxylic acid,

N- (4,6-dimethyl-2-pyrimidinyl) -4-aminobenzoic acid,

10,12-docodadiinedioic acid,

6,6-Dimethyl-3- (methylthio) -4,5,6,7-tetrahydrobenzo [c] -

-thiophen-4-one-1-carboxylic acid, gentisuric acid,

2-fluoro-4-heptyloxybenzoic acid,

2- (4-chloro-3-nitrobenzoyl) benzoic acid,

3- (4-bromo-2-thienyl) acrylic acid,

3,5-dimethoxycinnamic acid,

3 - [(2-ethoxycarbonyl) - (1,3,4) -2-thiadiazolylamino] propionic acid,

4-sulfoanthranilic acid,

D-pyroglutamic acid, (2,5-xylyl) phosphonic acid,

3-bromo-5-methoxybenzo (b) thiophene-2-carboxylic acid,

4.5.5.6.6.6-hexafluoro-4- (trifluoromethyl) -2-hexenoic acid,

2.3- difluorophenylacetic acid,

3.3.3-trifluoro-D, L-lactic acid,

3- [4- (4-methylphenylthio) -3-nitrophenyl] acrylic acid,

2,8-dimethoxydodecahydro-benzofuran-1-carboxylic acid,

4-cyclohexylbenzoic acid, boc-D-1,2,3,4-tetrahydronorharman-3-carboxylic acid,

2-Benzylcyclohexanecarboxylic acid

3 - [(4-fluorophenyl) - (toluene-4-sulfonyl) amino] propionic acid

acid,

3- (2,4,5-trimethylphenyl) butyric acid,

4- (1,3-dioxo-1,3-dihydroisoindol-2-yl) butyric acid, chelidamic acid,

4- [4- (1-methyl-1H-quinolin-4-ylidene) but-2-enylidenamino] benzoic acid,

8-carbamoylnaphthalene-1-carboxylic acid,

N- (m-tolyl) succinamic acid,

N- (1-naphthyl) phthalamic acid,

3- (3,4-dihydronaphthalen-1-yl) propionic acid,

4- (2-phenylsulfanylacetylamino) benzoic acid, perfluoroheptanoic acid,

4’-chloro-2'-methylphthalanic acid, diethylphosphonopentanoic acid,

2- (3-Methoxybenzylidene) pentanedioic acid

4,4'-biphenyldicarboxylic acid,

18-methylnonadecanoic acid,

4 '- (N-methylacetamido) glutaranilic acid, (+) - 3-methyladipic acid,

2-bromo-3-methoxythiophene-4-carboxylic acid, [5- (4-chlorophenyl) -4-pyrimidinylsulfanyl) acetic acid, glycyl-D-aspartic acid,

3- [N- (3,4-dichlorophenyl) carbamoyl] -5-norbornene-2-carboxylic acid,

N- (3-bromo-2,4,6-trimethylphenylcarbamoylmethyl) iminodiacetic acid,

1,2,3,4,5,6-cyclohexanehexacarboxylic acid, α- (phenylthio) phenylacetic acid, geranic acid,

5-hydroxy-2- (1-octynyl) -3-oxo-1-cyclopentene-1-heptanoic acid,

N-fmoc-2-aminoindan-2-carboxylic acid,

3- (9,10-Dioxo-9,10-dihydroanthracen-2-yl) -acrylic acid, ············· P-tolylacetic acid,

4- (4- (4-tolyl) butyl] phenylacetic acid,

2-methylcyclopropanecarboxylic acid,

4-chloro-α, α-dimethylphenylacetic acid, (2,4-dichloro-5-methylphenylthio) acetic acid,

3- (3,4-dichlorobenzylthio) thiophene-2-carboxylic acid, (+) - 3-methyl-2-phenylbutyric acid,

3-cyclopentenecarboxylic acid,

N-tris (hydroxymethyl) methyl-2-aminoethanesulfonic acid, (S) -5-oxotetrahydrofuran-2-carboxylic acid,

5-benzoylthiophene-2-acetic acid, p-toluenesulfonic acid,

3,6-dimethylcyclohex-4-ene-1,2-dicarboxylic acid,

3- (2-chlorophenyl) -5-methylisoxazole-4-carboxylic acid,

1- (4-acetylphenyl) iso (hexahydropyridine-4-carboxylic acid), phenyl-o-tolylphosphinic acid,

2- [1- / 2- (3,4-dimethoxyphenyl) ethyl] -5-ethyl-2-oxo-4-piperidinyljmalonic acid,

N- (4-methoxyphenyl) malonic acid, (+) - 3-pinanecarboxylic acid,

2- (2,4,5-trichlorophenoxy) propionic acid,

10-hydroxydecanoic acid,

5- (3-chlorophenyl) pentanoic acid,

4 - [[4 - [(4,6-dimethyl-2-pyrimidinyl) thio] phenyl] amino] -4-oxo-

- (2z) butenoic acid,

2-acetamido-3- (4'-chlorophenyl) acrylic acid,

2-hydroxy-6- [3- (trifluoromethyl) phenyl] -3,5-pyridinedicarboxylic acid,

9-hydroxyimino-9h-fluorene-4-carboxylic acid, mucochloric acid,

4-methyl-1-naphthoic acid,

2-naphthylacrylic acid,

4-hexylcyclohexanecarboxylic acid, • ♦ · · ·-------

4- (3,5-dimethylnaphthalen-2-yl) -3-methylpentanoic acid, Ν, Ν, ’,, N'-ethylenediaminotetra (methylenephosphonic acid),

6-heptinic acid,

2- (4-methoxybenzylidene) succinic acid, (R) - (+) - 2-chloropentanoic acid,

2- (3-chloro-4-methoxyphenylamino) benzoic acid,

3,5-bis (trifluoromethyl) cinnamic acid,

4-hexyloxybiphenyl-4'-carboxylic acid, (+/-) - 10-camphorsulfonic acid,

4,4'-oxybisbutanoic acid,

2-methyldecanoic acid,

4-Biphenylcarboxylic acid

3-chloro-n-butyric acid,

3-anthracen-2-ylacrylic acid, (S, S) - (+) - 2,3-diphenylsuccinic acid,

10-methyldodecanoic acid,

4'-fluorosuccinanilic acid,

2-bromo-3-methylbenzoic acid,

N- (4-trifluoromethoxyphenyl) malonamic acid,

3- (2-thienyl) acrylic acid,

3- (3-methoxyphenoxy) propionic acid,

2,3,6-trifluorocinnamic acid,

3-chloradamantane-1-carboxylic acid,

2,5-dichloro-α-methyl-3-thiophenacrylic acid,

2-ho-10-methanesulfonyl-9-oxa-tricyclo (6,2,1,0 (1,5)) undecane-4-carboxylic acid,

2,2-dichlorooctanoic acid,

7-chloro-6-fluoro-1-ethyl-4-oxoquinoline-3-carboxylic acid, acetoxy decanoic acid,

5-bromvaleric acid, meso-2,3-bis (benzylamino) succinic acid,

3,6-dimethyl-4,5-diphenylcyclohexa-3,5-diene-1,2-dicarboxylic acid

- 10 dodecafluoro-2-methyl-3-oxahexanoic acid,

D, L-2- (4-methoxyphenyl) butyric acid,

3- (N, N-diethylcarbamoyl) -5-norbornene-2-carboxylic acid, o-carboxyphenyl phosphate,

N-boc-2-aminoindan-2-carboxylic acid,

9-hydroxynonanoic acid,

3- (2,5-dimethoxyphenyl) propionic acid,

4 - [(2-hydroxy-3-nitrobenzylidene) amino] benzoic acid, fmoc-10-aminodecanoic acid, thiophene-2,5-dicarboxylic acid,

2-bromophenylacetic acid,

3- (3,4-methylenedioxyphenyl) propionic acid, (z) -styrylsulfonylpropionic acid,

2'-carboxymaleinanilic acid, gamma-oxo-1-naphthalene butyric acid,

11 - [(5-dimethylaminonaphthalene-1-sulfonyl) amino] undecanoic acid,

2- [[(4-chlorophenyl) sulfonyl] -3- (trifluoromethyl) anilino] acetic acid,

2-nonenoic acid,

2-formylphenoxyacetic acid,

2,4-pyridinedicarboxylic acid,

2-fluoro-6- (trifluoromethyl) phenylacetic acid, acenaphthalene-3-carboxylic acid,

2-fluoro-6-hydroxybenzoic acid,

4 - [(3-pyridylmethylene) amino] benzoic acid,

4-isobutylbenzoic acid, diheptylphosphinic acid,

3-chloropivalic acid,

2- [2-nitro-4- (trifluoromethyl) phenyl] acetic acid,

2,5-dichlorobenzoic acid,

4-Methoxy-3-methylbenzoic acid

2-fluoro-5-methoxybenzoic acid

14 (S), 15 (R) -epoxy- (5z, 8z, liz) -icosatrienoic acid, [2- (1-phenethyl) phenoxy] acetic acid,

4- (benzenesulfonamido) salicylic acid,

4-hydroxy-3-iodo-5-nitrophenylacetic acid,

2,6-dihydroxy-3,5-dimethylbenzoic acid,

2,4-dimethoxy-6-methylbenzoic acid,

N- (2-thiazolyl) succinamic acid,

7- (3,3-dimethyl-2,3-2H-benzo (b) -5-thienyl) -3-methyl-octa-

-2,4,6-trienoic acid

R-4-nitromanedioic acid, (IR) - (-) - 10-camphorsulfonic acid,

2-fluoro-4- (trifluoromethyl) cinnamic acid,

3- (4-tert-butylphenylsulfanyl) propionic acid,

2- (3,5-dinitro-2-thienylamino) succinic acid, [2 - [(3,4-dimethoxyphenyl) acetyl] -5-methoxyphenyl] acetic acid,

3.5-dijodalicylic acid,

2- (3-chlorophenoxy) propionic acid, erythro-9,10-dihydroxystearic acid, nitrous acid, shikimic acid,

2'-me-1,3,1 ', 3'-tetraoxo-1,3,2', 3'-4H-1'H- (2,5 ') biisoindolyl-5-carbaxylic acid, α3-chloro- 5,7-dimethyl-1,3-adamantanediacetic acid,

4- (4-pentylcyclohexyl) benzoic acid,

3-methyl-2- (toluene-4-sulfonylamino) butyric acid, (S) -1-amino- (3-methylbutane) phosphonic acid,

5-benzyloxy-4-methoxy-2-methylbenzoic acid,

4'-bromo-2'-chlorhexahydrophthalanic acid,

2-pentinoic acid,

2-Benzofurancarboxylic acid

3- (p-tolylthio) propionic acid,

2-cyano-3-ethoxyacrylic acid,

2- [3- (N'-octanoylhydrazino) -3-oxopropionylamino] benzoic acid,

4-hydroxy-3-nitroso-1-naphthalenesulfonic acid,

3-Iodo-4- (isopropylsulfonyl) -5- (methylthio) thiophene-2-carboxylic acid

N-boc-L-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid,

3- (1-naphthylthio) propionic acid,

2,4,6-trimethylbenzoic acid, bicyclo (2,2,1) heptane-3,4-dicarboxylic acid,

1,1'-ethylenebis (5-oxo-3-pyrrolidinecarboxylic acid), rhodanine-3-acetic acid, nitranilic acid, (R) - (-) - 2-hydroxy-2-phenylpropionic acid, methylthiohydantoin-D, L- aspartic acid,

6-methyl-2-pyridin-3-ylquinoline-4-carboxylic acid, citraconic acid,

N- (acetoacetyl) anthranilic acid,

N- (3-ethoxyphenyl) maleic acid,

2 ', 4'-difluorophthalanilic acid,

2,4-dimethoxycinnamic acid,

12-methicyclo (8,2,2,2 (4,7)) hexadeca-hexaene-5-carboxylic acid, [2- (propane-2-sulfonyl) acetylamino] acetic acid,

2-hydroxydecanoic acid, cis-N-benzylhexahydrophthalamic acid,

1,4-phenylenediacrylic acid, [2- (4-methoxyphenyl-6-oxocyclohex-1-enyl) acetic acid,

2- (5-fluoro-1-naphthoyl) benzoic acid, [2,2,2-trichloro-1- [3- (4-methoxycarbonyl-ph) thioureido / ethyl] carbamic acid,

2- [3- (N'-benzoylhydrazino) -3-oxopropionylamino] benzoic acid,

D, L-p-aminobenzylsuccinic acid,

2-isopropyl-2-phenylacetic acid, fmoc- (3S, 4S, 5S) -4-amino-3-hydroxy-5-methylheptanoic acid,

2-chlorisonicotinic acid,

3.4.4- trichloro-3-butenoic acid,

1- (4-chlorophenyl) -1-cyclobutanecarboxylic acid,

4- [4- (4-chlorophenoxy) benzenesulfonyl] benzoic acid, (4-acetylaminobenzenesulfonylsulfanyl) acetic acid,

N- (4-aminobenzoyl) -1-glutamic acid,

4- (3-Phenylureido) butyric acid

2'-fluoro-3,4,5,6-tetrachlorophthalic acid,

4-sulfobenzoic acid, ascorbyl palmitate, [4-chloro-6- (2,3-xylidino) -2-pyrimidinylthio] acetic acid,

2-amino-4-phenylthiazole-5-carboxylic acid,

4-hydroxy-5-methoxy-1-phenylnaphthalene-2-carboxylic acid,

3.4.5-trimethyl-1H-pyrrole-2-carboxylic acid,

3,3 ', 4,4'-benzophenontetracarboxylic acid,

4'-chloro-2 ', 5'-dimethoxyhexahydrophthalanic acid,

3- (4-ethoxybenzoyl) propionic acid,

4-chloro-2,6-dimethylnicotinic acid,

3- [2- (4-butoxybenzoylamino) -3- (4-methoxyphenyl) acryloylamino] propionic acid,

2-methylthiobenzimidazolesulfonic acid, phenaceturic acid, α, β-dibromocinnamic acid, o-trifluoromethyl-α-acetamidocinnamic acid, boc-Da-amino-gamma- (4-methylbenzylmercapto) butyric acid, N-α- (benzyloxycarbonyl) -D- aspartic acid,

2-fluoro-4-pentyloxybenzoic acid, boc- (3S, 4S) -4-amino-3-hydroxy-5-phenylpentanoic acid, pyruvic acid,

4- (2-chlorophenoxy) -3-nitro-cinnamic acid,

3- (aminocarbonylmethylthio) thiophene-2-carboxylic acid

chlorobenzoyl (4-) benzoic acid,

3-phenyl-2-p-tolylpropionic acid,

7-hydroxycoumarin-4-acetic acid,

2.3.4- Trifluorobenzoic acid

3-acetyl-2-phenyl-4-thiazolidinecarboxylic acid,

2- [3- (2,2,2-trichloro-1 - [(furan-2-carbonyl) amino] ethyl] thioureido (benzoic acid,

2- (3-chlorobenzoyl) benzoic acid,

N-phthaloyl-gly-D, L-α-amino-n-butyric acid,

2-naphthoic acid, cyclooctane-1,2-dicarboxylic acid,

4,4'-dicarboxydiphenylsulfone,

3- (4-n-heptyloxybenzoyl) propionic acid,

N- (4-methoxyphenyl) maleic acid,

3 - [(2-ethoxycarbonyl) - (6-methylbenzothiazol-2-yl) amino (propionic acid,

3,6-diphenylcyclohex-4-ene-1,2-dicarboxylic acid,

5- (3-bromobenzoyl) pentanoic acid, diisooctyldithiophosphinic acid,

5-bromo-2-pyroslizic acid,

1,2.3.4-tetrahydrophenanthren-1,2-dicarboxylic acid,

9-ethyl-3-carbazolphosphonic acid,

4- [2-hydroxy-6- (trimethylsilyl) -1-naphthylazo (benzoic acid, ethylmalonic acid, cyclobutylphenylglycolic acid,

3-bromophenylacetic acid,

N- (2-ethoxycarbonyl) iminodiacetic acid,

4- (tert-butyl) benzamidoacetic acid, fmoc-11-aminoundecanoic acid, fmoc-1-octahydroindole-2-carboxylic acid,

2- [3- / 4- (4,4-dicarboxybutyl) phenyl / propyl] malonic acid,

3- (4-Methylbenzamido) benzoic acid

1- (2-benzo [1,3] dioxol-5-yl-ethyl) -2- (2-carboxy-et) oxopyrrolidinecarboxylic acid,

4-hydroxy-3,5-diisopropylbenzoic acid,

3 - [(2-ethoxycarbonyl) phenylamino] propionic acid, p-phenylazomaleinanilic acid,

2-bromoacrylic acid,

2,3-bis- (4-chlorobenzylidene) succinic acid,

N- (4-methyl-3-nitrophenyl) glutaramic acid,

3-bromo-5-methoxy-2-propylbenzoic acid, oxamic acid,

2- (2-naphthoyl) benzoic acid,

2- (2-formamidothiazol-4-yl) -2-methoxyiminoacetic acid, (R) -tetrahydrofuran-2-carboxylic acid,

4-mercaptobenzoic acid, (S) -2-fluoro-2-methylpentanoic acid,

4-nitrophenoxyacetic acid, ac-D-ala-D-lactic acid,

2- (4-hydroxymethyl-3-methoxyphenoxy) butyric acid,

4- (3-nitrophenyl) -1,3-butadiene-1-carboxylic acid,

4-bromo-4,4-difluorobutyric acid,

3- (4-chloro-2-nitrophenyl) -2-oxopropionic acid,

20,20,20-trifluoroarachidonic acid, dibromofluoroacetic acid,

2-bromolauric acid, bis (4-chlorophenoxy) acetic acid,

4,4'-trimethylenebis (phenylacetic acid),

4-hydroxypyridine-3,5-dicarboxylic acid,

2-ethoxy-1-naphthoic acid,

3- (4,5-diphenyl-2-oxazolyl) propionic acid, tetrachlorophthalic acid, perchloric acid, [3- (methoxycarbonyl) -2-methyl-5-oxo-2-pyrrolin-4-yl] acetic acid,

3- [3- (1-butyrylamino-2,2,2-trichloroethyl) thioureido] benzoic acid,

3,4,9,10-perylentetracarboxylic acid,

3-fluoro-4-hydroxybenzoic acid,

D, L-α-hydroxyisovaleric acid,

3- (2-chloroethanesulfonyl) propionic acid, fmoc-1-pipecolic acid,

2-methyl-1,1-dioxo-2,3-dihydro-1H-benzo (b) thiophene-2-carboxylic acid,

3-acetylthiazolidine-2-carboxylic acid,

1-methyl-1-cyclohexanecarboxylic acid,

2- (3-benzyloxy-4-methoxybenzyl) -2-phenylmalonic acid,

N- [3- (triethoxysilyl) propyl] phthalamic acid,

2.2.5.5-tetramethyl-3-pyrroline-1-oxy-3-carboxylic acid, fmoc-8-aminocaprylic acid,

3-Methylthianaphthalene-2-acetic acid

3-bromocinnamic acid,

1-oxalyl-1,4-phenylenediamino-2-sulfonic acid, succinamic acid,

4 - [(di-n-propylamino) sulfonyl] benzoic acid, α-fluorocinnamic acid,

2,3-diphenyl-2-cyclopropene-1-carboxylic acid,

3.4-pyridinedicarboxylic acid, p-pentyloxybenzoic acid,

3- (1,3-dioxo-1H, 3H-benzo (d, e) isoquinolin-2-yl) benzoic acid,

3-tricyclo (8,2,2,2 (4,7)) hexadeca-hexaen-2-ylacrylic acid,

2- [1-methyl-2- (4-nitrophenyl) propoxy] benzoic acid,

2.4.5-trifluorophenylacetic acid,

3-chloro-3-p-tolylcarbamoylacrylic acid,

3,7-dihydroxy-2-naphthoic acid,

3-Methoxyphenylacetic acid, 44, 44, 44, 44, 44, 44

-Oylamino-3- (4-hydroxy-3-methoxyphenyl) propionic acid

3- (4-methylbenzoyl) acrylic acid,

N-cyclododecylmaleinamic acid,

11-hydroxyundecanoic acid,

3-bromo-2-methylbenzoic acid,

N- (2,3-dichlorophenyl) maleic acid,

2-fluoro-5-nitrobenzoic acid, hydroxy- (2,3,5,6-tetramethylphenyl) acetic acid,

2-isopropyl-2-phenylglycolic acid,

1-hydroxy-4- (4-nitrophenoxy) -2-naphthoic acid,

2-hydroxy-6- (3,4,5-trimethoxyphenyl) -3,5-pyridinedicarboxylic acid, (1-amino-1-phosphonoethyl) phosphonic acid,

N- (2,4-dichlorophenyl) maleic acid,

N, N'-terephthalylidenebis (4-aminosalicylic acid), trans-aconitic acid,

5'-chloro-2 ', 4'-dimethoxyphthalanilic acid, (R) -2-bromobutyric acid,

4-azido-2,3,5,6-tetrafluorobenzoic acid,

N- (3-methoxyphenyl) tetrachlorophthalamic acid,

5-fluoro-2- (trifluoromethyl) benzoic acid,

2.2-dimethyl-4-pentenoic acid, heptadecanoic acid,

3,5-pyridinedicarboxylic acid, β, β-dimethyl-1-pyrrolepropanoic acid,

2-chloro-3- (trifluoromethyl) benzoic acid,

2,3-dihydrobenzo (b) azepine-1-carboxylic acid,

4- (1-methylbutyl) benzoic acid, p- (β-bromoethyl) benzoic acid,

2,2-dichloropentanoic acid,

7- (dimethylaminosulfonyl) -2,3-dihydro-gamma-oxo-1- (1H) -indolbutanoic acid,

13 (S) -hydroxyoctadeca-9Z, HE-dienoic acid,

4-bromophenylacetic acid, (S) - (+) - o-acetylmandelic acid,

3-chloro-2-fluorobenzoic acid, camphorquinone-10-sulfonic acid,

3-nonenoic acid,

9-oxo-bicyclo (3,3,1) non-6-ene-3-carboxylic acid,

3'-chloro-2,3-dibromo-4'-methylsuccinanilic acid,

4-bromo-2-fluorobenzoic acid,

17-iodo-heptadecanoic acid,

1,2,3,4,6,7,8-heptachlor-tricyclo (4,2,0,0 (3,8)) oct-4-ene-2,7-dicarboxylic acid,

N-cbz-1-glutamic acid, carboxyphenyl-gamma-acid,

4-benzyloxy-3,5-dimethoxybenzoic acid,

4-cresidine-6-sulfonic acid,

2- (2,5-dichlorophenoxy) propionic acid, (2-bromo-4,5-dimethoxyphenyl) acetic acid,

2'-hydroxy-2-biphenylcarboxylic acid,

4,4,4-trifluoro-3- (trifluoromethyl) crotonic acid,

16-hydroxyhexadecanoic acid,

4-nitro-3- (octanoyloxy (benzoic acid,

1,3-diaminopropane-N, N, N ', N'-tetraacetic acid,

4-fluoro-2- (trifluoromethyl) cinnamic acid,

2.3- dichloroisobutyric acid,

3.4- Difluoro cinnamic acid

3- (3-adamantan-1-ylureido) propionic acid,

1,1-dimethylindan-4-carboxylic acid,

D - (-) - 2-amino-5-phosphonopentanoic acid, fmoc-5-aminovaleric acid,

3-methoxy-9-oxo-6,7,8,9-tetrahydro-5H-benzocycloheptene-6-carboxylic acid,

4,4-Dichloro-4-fluorobutanoic acid, · · · · · · · · · · · · · · · · · · · · · · · · · · · [4- (4-carboxymethylsulfanylbenzyl) phenylsulfanyl] acetic acid, trans-2- (2-thiophenecarbonyl) -1-cyclohexanecarboxylic acid,

3,5-dimethoxy-4-hydroxyphenylacetic acid,

1-Pyrenebutyric acid

N- (2,6-dimethylphenylcarbamoylmethyl) iminodiacetic acid,

4-nitrophenyloxamic acid,

3-ethylcyclohex-4-ene-1,2-dicarboxylic acid, (L) -menthylcarboxylic acid,

3,3,3-trimethylpyruvic acid,

1-methyl-2-phenylcyclopent-2-enecarboxylic acid, hexahydro-4'-sulfamoylphthalanilic acid,

2-methoxyphenylacetic acid,

3-carboxybenzaldehyde,

N-phenylethylated einamic acid, citrinine,

3-nitrophenoxyacetic acid,

8-hydroxyoctanoic acid, bis- (3-chlorophenyl) phosphinic acid,

2- (2-ethoxycarbonyl) -6,6-dimethyl-3-oxocyclohex-1-enecarboxylic acid, cis-8-methylnon-6-enoic acid, o- (methoxycarbonyl) salicylic acid,

3-Benzoyl-2- (3-chlorophenyl) propionic acid, [2- / 2- (5-methyl- (1,3,4) thiadiazol-2-ylsulfanyl) -α-amino / thiazol-4-yl] acetic acid acid, octahydro-3-methyl-1-pentalenecarboxylic acid, p-phenylhippuric acid,

N- (2,2-dichloroacetyl) -5-iodoanthranilic acid,

2-fluoro-4-nonyloxybenzoic acid,

3,5-dimethyl-p-anisic acid, ethylenediaminotetrapropionic acid,

2-amino-3,6-dimethyl-5-nitrobenzoic acid

4- (4-methoxybenzoyl) butyric acid, methoxyacetic acid,

5-benzo (1,3) dioxol-5-yl-8-hydroxynaphtho (2,3-d) (1,3) dioxole-6-carboxylic acid,

4-oxohexanoic acid,

2- (p-hydroxybenzoyl) benzoic acid,

2-hydroxyicosanoic acid, (R) -3-hydroxy-3-phenylpropanoic acid,

4-oxo-6-phenyl-5-hexenoic acid,

D-desthiobiotin,

7-oxo-6-oxa-bicyclo [3.2.1] octane-3-carboxylic acid,

2-hydroxy-3,5-dimethylbenzoic acid, (+) - cis-2-benzamidocyclohexanecarboxylic acid, anthracene-1,5-dicarboxylic acid, phenyl-n-propylphosphinic acid,

3-hydroxyundecanoic acid, (2-naphthalen-2-ylacetylamino) acetic acid, (5-cyano-6-hydroxy-4-methyl-2-oxo-2H-1-pyridyl) acetic acid,

2-Benzoylamino-3,3-dichloroacrylic acid

3-methylundecanoic acid,

4,4-bis- (3,5-dichloro-4-hydroxyphenyl) valeric acid, fmoc-D, L-2-aminohexanoic acid,

4-hexenoic acid, cyclobutanecarboxylic acid,

4,4,5,5,6,6,6-heptafluorohexanoic acid,

N, N-dimethylsuccinamic acid,

2'-carboxysuccinanilic acid,

2,5-dimethylbenzenesulfonic acid,

4-methyl-4-cyclohexene-1,2-dicarboxylic acid, (2-sec-butyl-3-chlorophenoxy) acetic acid,

3 ', 4'-dichloro-1,2,3,6-tetrahydrophthalanilic acid, (R) - (-) - (1-aminoethyl) phosphonic acid,

(S) - (+) - 2-oxo-4-phenyl-3-oxazolidineacetic acid,

4-hydroxymethylbenzoic acid,

3-hydroxy-4-methoxymandelic acid,

3-bromoanisic acid, (2-nitrobenzenesulfonyl) acetic acid,

3.3.3-trifluoro-2,2-dihydroxypropionic acid, n-α- (benzyloxycarbonyl) -gamma- (tert-butyl ester) -D-glutamic acid,

1- (+) - 2-amino-5-phosphonovaleric acid,

2-fluorobenzoic acid,

N- (3,3,5-trimethylcyclohexyl) dithiocarbamic acid,

1- (+) - Mandelic acid

5-fluoro-2- (trifluoromethyl) cinnamic acid,

2,6-dimethylbenzoic acid, (2-chloro-2-phenylvinyl) phosphonic acid,

3-benzoyl-2-benzylidenepropionic acid, aurintricarboxylic acid,

4- (2-naphthyl) butyric acid, cis-10-pentadecenoic acid (cl5: 1),

2-butynoic acid,

2,3-dibromo-N- (1-naphthyl) succinamic acid, p-chlorophenoxyacetic acid, (R) -3-phenylbutyric acid, (o-tolyl) phosphonic acid,

4'-bromo-3'-methylphthalanilic acid,

15-ketoicose-6E, 8Z, 11Z, 13E-tetranic acid, homoisocitric acid, p- (4-oxo-2-thioxothiazolidino) benzoic acid, trans-5-acetoxy-1,3-oxathiolane-2-carboxylic acid,

3-formyl-2,4,6-trimethylbenzoic acid, d-3-phenyl lactic acid,

4'-ethylphthalanilic acid,

2- [2- / 3-chloro-5- (trifluoromethyl) -2-pyridyl / carbohydrazonoyl] benzoic acid,

2'-methylglutaranilic acid,

4-nitropicolinic acid,

4-chloro-3,5-dinitrobenzenesulfonic acid,

2-cinnamic acid,

3-butoxy-4-nitrobenzoic acid, phosphorous acid, butyl malonic acid,

4-methoxycinnamic acid, thiophene-2-acetic acid, cycloundecanecarboxylic acid, 3'-hydroxyphthalanilic acid, (4-tert-butylphenoxy) acetic acid,

3- (4-n-Pentylbenzoyl) propionic acid,

5- (3,5-dichlorophenoxy) furan-2-carboxylic acid

2 - ((4,6-dimethoxy-2-pyrimidinyl) oxy] -6-methoxybenzoic acid, hydroxyphenyl-p-tolylacetic acid,

2-norbornene-2,3-dicarboxylic acid, (phenylthio) acetic acid,

5-keto-D-gluconic acid,

7-ho-1,3-dimethyl-2,4-dioxo-1,2,3,4-4H-pyrido (3,2-d) pyrimidine-6-carboxylic acid, m-hydroxymandelic acid, oxanilic acid, α - ethyl cinnamic acid,

3- (5- (4-methoxyphenyl) -2-furyl] acrylic acid,

2,5-dimethoxyphenylacetic acid, uvic acid,

2-hydroxyiminopropionic acid,

1,2,3-benzenetricarboxylic acid,

2,4-dimethylglutaric acid,

4-methylcyclohexaneacetic acid,

3- (2-chlorophenyl) -2-cyanopropionic acid, fmoc-L-norleucine,

1,4-benzodioxane-2-carboxylic acid,

3- (4-chloro-2-oxobenzothiazol-3-yl) propionic acid,

4,5,5,5-tetrafluoro-4- (trifluoromethoxy) pentanoic acid,

? 3-dimethylglutaric acid, heptafluorobutyric acid,

2-benzenesulfonyloxy-3-methoxybenzoic acid,

2'-carboxy-2-hydroxy-4-methoxybenzophenone,

7-methyl-2-phenylimidazo (1,2-a) pyridine-3-carboxylic acid,

5-hexenoic acid,

3'-chloro-2,3-dibromosuccinanilic acid,

2.2-dichlorohexanoic acid,

4 - [(pyridine-4-carbonyl) amino] butyric acid,

3.3- dichloropivalic acid,

2-imidazolidone-4-carboxylic acid, β-oxalylamino-D-alanine,

4'-ethoxy-3,4,5,6-tetrachlorophthalic acid, (2-benzothiazolylthio) acetic acid,

4-benzyloxyindole-2-carboxylic acid,

2-trans-benzoyl-5-trans-phenyl-1-cyclohexanecarboxylic acid,

12-nitrotricyclo (8,2,2,2 (4,7)) hexadeca-hexaene-5-carboxylic acid,

2-acetyl-3-thiophenecarboxylic acid,

4'-nitrosuccinanilic acid,

2-hydroxyisobutyric acid,

2.3-dimethylbenzoic acid, propylenediphosphonic acid,

2-cyclopentene-1-acetic acid,

4- (2-Pyridylacetyl) benzoic acid

4- [3- (3-chloro-4-fluorophenyl) ureido] benzoic acid,

4-nitrophenylglyoxylic acid,

pth-glutamic acid, (8R, 15S) -dihydroxy- (5Z, 9E, 11Z, 13E) -icosatetraenoic acid,

5-nitro-2-pyroslizic acid,

2-butyloctanoic acid,

N-formyl-4-nitroanthranilic acid,

2-methoxy-α-methylcinnamic acid,

2- (2-ethoxycarbonylacetylamino) benzoic acid,

2,3-dimethylphenoxyacetic acid,

3,5-dimethoxy-4-hydroxycinnamic acid,

3-chloro-4-nitrobenzenesulfonic acid,

D, L-α-aminopimelic acid, α-cyano-4-hydroxycinnamic acid,

3 - [(5-bromo-1,3-dioxo-1,3-dihydroisoindol-2-ylmethyl) amino] benzoic acid,

N-ethyl-L-aspartic acid,

N-α-fmoc-N-β-boc-d-diaminopropionic acid,

N-t-boc- (2S, 3R) -3-amino-2-hydroxy-4- (4-nitrophenyl) butyric acid,

2,6-pyridinedicarboxylic acid,

3-dibenzo (a, c) phenazin-11-ylacrylic acid, valerenic acid,

Nicotinic acid N-oxide,

5- (4-Benzyloxy-3-methoxyphenyl) penta-2,4-dienoic acid

4-chlorophenylcyclohexanecarboxylic acid,

4- (p-chlorophenoxy) butyric acid, n-tris (hydroxymethyl) methyl-4-aminobutanesulfonic acid, s-4-nitromanedioic acid,

4,5-dichloro-2-fluorobenzoic acid,

N- (2,3-xylyl) glutaramic acid,

4.5.5-trifluoro-4-pentenoic acid,

5-fluoro-2,6-dihydroxypyrimidine-4-carboxylic acid,

3-phenylsalicylic acid,

2- (2-hydroxy-5-methylbenzoyl) benzoic acid, cis-4-cyclohexene-1,2-dicarboxylic acid,

2-bromostearic acid,

1-trans-pyrrolidine-2,4-dicarboxylic acid

2-chloro-5-sulfobenzoic acid,

3-thiophenecarboxylic acid,

2 - [(3-methoxyphenyl) phenylmethylene] succinic acid,

3-chlorocinnamic acid,

4-phenyl cinnamic acid,

3- (3,5-dinitro-4-hydroxyphenyl) propionic acid,

7-acetoxycoumarin-3-carboxylic acid,

D-α-galacturonic acid,

3-bromo-2,5,6-trimethoxybenzoic acid,

3-tert-butyladipic acid,

2-methylnonanoic acid,

3-Hydroxy-4-methyl-2-nitrobenzoic acid

2,6-dihydroxy-4-methylbenzoic acid,

7- (3,3-dimethyl-2,3-dihydrobenzo-5-furyl) -3-methyl-octa-2,4,6-trienoic acid,

5-methoxy-2-propylisophthalic acid,

3- (3-benzyloxy-4,5-dimethoxyphenyl) propionic acid, (1S, 2S) - (+) - 1,2-cyclohexanedicarboxylic acid,

2- (amidinothio) ethanesulfonic acid,

D - (-) - s-Benzoyl-3-mercaptoisobutyric acid,

3-fluoro-5- (trifluoromethyl) benzoic acid,

2- (9H-fluoren-9-ylmethoxycarbonylamino) -3-hydroxybutyric acid,

2-bromo-4-nitrobenzoic acid, (S) -2-ethyldecanoic acid,

11-phenoxyundecanoic acid,

2-nitro-6- (2,4-pentadien-1-yloxy) benzoic acid,

5- (methanesulfonyl) thiophene-2-carboxylic acid,

2- (4-fluorobenzoyl) benzoic acid,

2-Benzoyl-3,6-dimethylbenzoic acid 4 4 4 4

2-ethoxycarbonylsyringic acid,

3,3 ', 4,4', 5,6-hexachlorophthalanilic acid,

3-methylthiopropionic acid, (+/-) - abscisic acid,

4-chloro-3-nitrophenylacetic acid,

2-octanoic acid,

3- (4-azidophenyl) propionic acid,

9,10-dihydro-9,10-ethanoanthracene-11-carboxylic acid, (2-hydroxyimino-propionylamino) acetic acid,

N- (4-ethoxycarbonylphenyl) phthalamic acid,

D, L-2-amino-3-phosphonopropionic acid,

2- (2-dibenzo (a, d) cyclohepten-5-ylidenethyl) malonic acid,

7-phenylheptanoic acid,

5-bromo-4,4,5,5-tetrafluoropentanoic acid,

8-benzoyloctanoic acid,

3-hydroxy-5- (1-hydroxy-1-methylethyl) -cyclohexanecarboxylic acid,

3-dodecenoic acid,

N- (1-naphthyl) -3,4,5,6-tetrachlorophthalamic acid,

4- (trifluoromethyl) phenylacetic acid, s-acetamidomethyl-3-mercaptopropionic acid, dihydroanthracene-9,10-dicarboxylic acid, meso-2,5-dibromadipic acid,

2,3-dibromo-2'-methoxy-5'-methylsuccinanilic acid,

3-chloro-4- (isopropylsulfonyl) -5- (methylthio) thiophene-2-carboxylic acid,

4-n-propylbenzoic acid,

2,3-dibromo-3- [2- (methoxycarbonyl) phenylcarbamoyl] propionic acid,

10-heptadecenoic acid,

3-methoxyphenoxyacetic acid,

4,4'-dimethylenebis (phenylacetic acid),

4-chloro-3,5-dinitrobenzoic acid,

Diethylphosphonoacetic acid, (1R) - (-) - (1-aminopropyl) phosphonic acid, (R) -3- (4-fluorophenyl) butanoic acid, phenazine-1,6-dicarboxylic acid [1R- (exo, exo)] - 3- (benzoyloxy) -8-azabicyclo (3,2,1) octane-23-carboxylic acid,

2'-fluorophthalanilic acid,

4-bromo-3-methylbenzoic acid,

3- (morpholine-4-carbothioylsulfanyl) propionic acid, (6-iodobenzo (1,3) dioxol-5-yl) acetic acid,

3'-fluoro-hexahydrophthalanic acid,

1-phenylsulfonyl-4,4-piperidinedicarboxylic acid,

2- (3,5-xylyl) acetic acid, β-chloro-lactic acid,

10,12-heptacosadiinic acid,

N-acetyl-L-thiazolidine-4-carboxylic acid,

6-hydroxy-2,5,7,8-tetramethylchroman-2-carboxylic acid, trans-15-octadecenoic acid,

2 '- (hydroxymethyl) -2-biphenylcarboxylic acid, coumarinic acid,

N- (2,4,6-trimethylphenylcarbamoylmethyl) iminodiacetic acid,

2- (3,4-dimethoxyphenyl) -3- (2-nitrophenyl) acrylic acid, suberic acid, heptadecanedioic acid,

2 ', 4', 6'-trimethylmaleanilic acid, uramil-N, N-diacetic acid, (2,3-xylyl) phosphonic acid,

6-chlorkynurenic acid,

8-iodo-1-naphthoic acid,

4- (1,1,2,2-tetrafluoroethoxy) benzoic acid,

3- [N- (4-methylphenyl) carbamoyl] -5-norbornene-2-carboxylic acid,

• * 4 * 4 «, -, -, -, -,,,,,,,,,,,,,,,,,,

Ν, Ν, Ν ', N'-1,4-phenylenediaminotetraacetic acid,

3- (3,4-dichlorobenzoyl) -2- (4-methylphenyl) propionic acid,

3-phenylpyrrolo (2,1,5-cd) indolizine-1,2-dicarboxylic acid, phenylglycine-o-carboxylic acid,

2,4-dimethyl-6- (2'-methylpropyl) benzene-1,2'-dicarboxylic acid,

4-Benzoylbutyric acid

Ν-α-Ν-β-di-Z-L-diaminopropionic acid,

4 - [(6-phenyl) -1,3,5-hexatrienyl] benzoic acid,

4- (2-chloroethyl) benzoic acid, (2,2-difluoradamantan-1-yl) acetic acid, trans-2-octenic acid, cis, cis-2,5-dimethylmuconic acid,

4- (fluorosulfonyl) benzoic acid,

2 - (/ (4-chlorophenyl) sulfonyl) - (2-pyridyl) amino] acetic acid, β-N-oxalylamino-L-alanine, octanoic acid,

1-dihydroorotic acid,

14-hydroxy-10,12-tetradecadioic acid,

4- (2,5-dimethylphenyl) butyric acid,

2,2-difluoro-2-phenoxyacetic acid,

N- [3- (trifluoromethyl) phenyl] maleinamic acid, n-carbamoyl-D, L-α-amino-n-butyric acid,

1- (m-sulfophenyl) -3-methyl-5-pyrazolone, acenaphthen-5-ylacetic acid, cis-15-octadecenoic acid, benzo (c) phenanthrene-6-carboxylic acid,

2-chloro-5-iodobenzoic acid,

1- (4-fluorophenyl) cyclopentanecarboxylic acid,

3-Heptenic acid, chromone-3-carboxylic acid, (S) - (-) - 2-chloropentanoic acid, · · · »» »»

3- (2,5-dimethylphenyl) -3-methylbutyric acid, (S) - (+) - 2-bromo-3-phenylpropionic acid, cyclohexylphenylacetic acid,

3,3 ', 3-nitrilotripropionic acid,

2-biphenylcarboxylic acid, (4-chloro-3,5-dimethylphenoxy) acetic acid,

4- (2-amino-5-bromo-3-ethylphenyl) -4-oxobutyric acid,

3,4-methylenedioxycinnamic acid,

5- (2-nitrophenyl) -2-pyroslizic acid,

4'-bromo-3'-methylsuccinanilic acid,

2,3-dihydrobenzofuran-7-carboxylic acid,

4- (2,4-di-tert-pentylphenoxy) butyric acid,

4- (3,4-dimethoxyphenyl) butyric acid,

2 - [(5-chloro-4,6-dimethoxy-2-pyrimidinyl) oxy] benzoic acid,

9-anthracenecarboxylic acid, (R) -3- (4-tert-butoxyphenyl) butanoic acid,

5,5'-methylenedisalicylic acid,

4-methylnonanoic acid,

2-fluoro-6-iodobenzoic acid,

L- (+) - s-acetyl-p-mercaptoisobutyric acid,

R - (+) - 2- (2,4-dichlorophenoxy) propionic acid, (+/-) - 5,6-epoxyicose-8Z, 11Z, 14Z-trienic acid,

1,6-naphthalenedicarboxylic acid,

3-isobutyrylamino-3-phenylpropionic acid, (Z) - (3) iodoacrylic acid,

1- (4'-Sulfophenyl) -3-carboxy-5-pyrazolone

4- (3-phenyl-2-thioureido) hippuric acid,

4- [2- (2-hydroxyphenoxy) acetylamino] benzoic acid, 1-ethyl-4-oxo-1,4-dihydroquinoline-3-carboxylic acid,

6- (trifluoromethyl) nicotinic acid,

5-norbornene-2-endo, 3-exo-dicarboxylic acid,

4'-bromo-2'-chlorosuccinanilic acid,

2-acetoxy-3-methylbenzoic acid,

4-chloro-3-nitro-cinnamic acid,

2- (benzenesulfonyl) ethylthioacetic acid, 11- (methoxycarbonylmethylthio) undecanoic acid, cis-3 ', 5'-dimethylhexahydrophthalanic acid,

2,6- dichlorophenoxyacetic acid,

3-chloro-4-hydroxyphenylacetic acid,

7 - [(4-amino-3-sulfophenyl) amino] -4-hydroxy-2-naphthalenesulfonic acid, n-α- (benzyloxycarbonyl) -a- (tert-butyl ester) -1-glutamic acid,

6-ketoundecan-1,11-dioic acid,

6-amino-2- (2-ho-et) -1,3-dioxo-2,3-2H-1H-benzo (de) isoquinoline-5-sulfonic acid,

3-nitrophenylacetic acid,

5-methyl-2-thiophenecarboxylic acid, - [3 - C '- dodecanoylhydrazino) -3-oxopropionylamino] benzoic acid,

4'-nitrophthalanilic acid,

3-nitro-4-phenoxybenzenesulfonic acid,

1,2,3,4-butanetetracarboxylic acid, (1S) - (+) - (1-aminohexyl) phosphonic acid, (S) -3-phenylbutyric acid, diethylenetriaminopentaacetic acid, boc-D-2-aminobutyric acid,

3-bromo-4-chloropentafluorobutyric acid,

2.4.6- trinitrobenzoic acid,

2-nitrophenoxyacetic acid,

D, L-homocysteic acid, (4-ethylphenyl) phosphonic acid,

4- (4-nitrophenyl) butyric acid, cis-cyclobutane-1,2-dicarboxylic acid, thieno (3,2-b) thiophene-2-carboxylic acid, mesobutane-1,2,3,4-tetracarboxylic acid , pentafluorobenzenesulfonic acid, o-iodohippuric acid,

4,5,6,7-tetrafluoro-3-indole acetic acid,

2- (phenethylthio) acetic acid,

1-hydroxyethane-1,1-diphosphonic acid,

1- 2-Aminoadipic acid

6-oxoheptanoic acid,

2-formamido-3-thiophenecarboxylic acid,

14-methylpentadecanoic acid, bis- (4-bromophenyl) hydroxyacetic acid,

3-iodopropionic acid,

2,6-dioxo-4-piperidinecarboxylic acid, D-α-aminoadipic acid,

3-bromo-5-chloro-2,6-dimethoxybenzoic acid, orotic acid,

6- [2-acetylamino-3- (4-methoxyphenyl) acryloylamino] hexanoic acid,

3- (4-chlorobenzenesulfonyl) butyric acid,

2-bromoisophthalic acid,

3-amino-4-isopropenylbenzoic acid,

3-Phenoxypropionic acid

N- (2-chlorophenyl) glutaramic acid,

4 - [(E) -2- (5,6,7,8-tetrahydro-5,5,8,8-tetramethyl-2-naphthalenyl) -1-propenyl] benzoic acid,

3-chloro-2-methylbenzoic acid,

3- (3-ethoxyphenyl) propionic acid,

2'-chloro-6'-methylphthalanilic acid,

4- [[2-fluoro-5- (methylsulfonyl) phenyl] amino] -4-oxobutanoic acid,

3.6-dimethylsalicylic acid,

3- (2,6-dichlorobenzylthio) -2-thiophenecarboxylic acid, (S) - (-) - 2-guanidinoglutaric acid,

3.4-dinitrobenzoic acid, α-triryl-2-naphthalenepropionic acid,

3.4-dichlorophenylacetic acid, phenylbenzene-omega-phosphono-α-amino acid, n-methylhippuric acid, hydroquinone-o, o-diacetic acid,

3- (4-n-octylbenzoyl) propionic acid,

1-methyltridecanoic acid,

3-cyclohexylpropionic acid,

3,5-di-tert-butyl-4-hydroxybenzoic acid, [3-cyano-6- (4-methoxyphenyl) -3-methyl-2-oxocyclohexyl] acetic acid,

4-hydroxyisophthalic acid, di (cyclohexyl) phosphoric acid,

3-aminoadipic acid, (4-nitrobenzyl) phosphonic acid,

4- (4-Methoxyphenyl) -4-methylpentanoic acid

4- (2-hydroxybenzylideneamino) salicylic acid, n-hexadecylphosphonic acid, 1-methoxyphthalanilic acid,

1-Ho-8-imino-5-oxo-4- (4-sulfophenylamino) -5,8-2H-naphthalene-2-

-sulfonic acid, kainic acid, tetrahydrofuran-2,3,4,5-tetracarboxylic acid,

4-methyl-5-oxohexanoic acid,

12-0X0-12- (1-pyrenyl) dodecanoic acid, α-isoatropic acid,

4- (2-thienylmethyleneamino) salicylic acid, iodic acid,

2-fluorophenylacetic acid, (benzoylbenzylamino) acetic acid, cis-3-chloroacrylic acid,

3-pyrimidin-2-ylpropionic acid,

2- [2- (3,4-dimethylphenoxy) acetylamino] benzoic acid, malonamic acid, (S) - (+) - (1-aminoethyl) phosphonic acid,

6-methyl-2- (4-pyridyl) quinoline-4-carboxylic acid,

4,6-dimethylisophthalic acid, di-n-propyl phosphate, benzothiazol-2-yl-2- (2-aminothiazol-4-yl) acetic acid,

5- (4-fluorobenzoyl) thiophene-2-acetic acid,

2-Acetylaminobut-2-enoic acid

4-fluoro-2- (trifluoromethyl (benzoic acid,

8,11-icosadioic acid

N- (4-methylphenyl) tetrachlorophthalamic acid,

4'-butylhexahydrophthalanic acid, ethylxanthogenacetic acid, α-phenylcyclopentaneacetic acid, n-methyl-L-aspartic acid,

3-bromo-5-methoxy-2-methylbenzoic acid, isooctyl phosphate, -acid,

2- (2,2-dimethylpropionylamino) -4,5,6,7-4H-benzo (b) thiophene-3-

-carboxylic acid,

4-chloro-3-nitrobenzoylbenzoic acid,

N- (2-carboxyphenyl (malonamic acid,

2,5-norbornadine-2,3-dicarboxylic acid,

3-benzyloxy-4,5-dimethoxybenzoic acid,

4- (2-isopropylsulfanylacetylamino) benzoic acid,

5-fluoro-6-hydroxypyrimidine-4-carboxylic acid,

2- (3-nitrobenzylidene) pent-4-enoic acid, n-carbamoylmaleinamic acid,

4- (4-hydroxyphenoxy (benzoic acid, tetracosanedioic acid,

2-bromo-5-methoxybenzoic acid,

4-formyl cinnamic acid, (methylthio) acetic acid, •

4-oxo-4- [4- / 4- (ethoxycarbonyl) butyl / phenyl] butyric acid,

2,4- dichlorophenoxyacetic acid,

4 - ((1,3-dioxo-1,3-dihydroisoindol-2-ylmethyl) amino] benzoic acid,

3,4-dimethoxyphenylpyruvic acid, (S) -2-fluoro-2-methylheptanoic acid,

2-Benzoylamino-3- (4-benzyloxy-3-methoxyphenyl) acrylic acid

3-Naphthalen-1-ylpropinic acid

4.4- dinitroheptanedioic acid,

3-benzo (1,3) dioxol-5-ylpropinic acid, tetraacetylsulic acid, cis-hexahydro-N- (4-ethoxyphenyl) phthalamic acid,

3 - ((3,5-dimethoxyphenyl) - (toluene-4-sulfonyl) amino] propionic acid,

3- (4-n-Pentyloxybenzoyl) propionic acid,

2-chlorocinnamic acid,

N-cyclohexylglutaramic acid, (-) - cis-2-benzamidocyclohexanecarboxylic acid,

D, L-citramalic acid, 1H-pyrazole-3,4-dicarboxylic acid,

2-fluoro-4-hexyloxybenzoic acid,

N- (3-chloro-2-methylphenyl) glutaramic acid, trans-1,2-diaminocyclohexane-N, N, N ', N'-tetraacetic acid monohydrate,

2,2-dichlorooctadecanoic acid,

2-fluoro-6- (trifluoromethyl) cinnamic acid, boc-D-7-hydroxy-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid,

5- (3-methoxyphenyl) hexa-2,4-dienoic acid,

5- (4-hydroxy-3-methoxyphenyl) pentanoic acid,

5- (α-α-dimethyl-4-hydroxybenzyl) salicylic acid,

3-Decenoic acid, «

n-benzyliminodiacetic acid, n-α- (b enzyloxycarbonyl) L-glycyl-L-glycine, (4-ethoxyphenyl) phenylphosphinic acid, (4'-carboxymethylsulfanylbiphenyl-4-ylsulfanyl) acetic acid,

1-methylorotic acid,

3- (3,5-di-tert-butyl-benzoylamino) benzoic acid,

4- (2,5-dioxo-2,5-dihydropyrrol-1-yl) benzoic acid,

2 ', 5'-dimethoxymaleanilic acid, boc-α-aminobutyric acid, (3-nitrophenyl) phosphonic acid,

4- (2-acetylamino-3-phenylacryloylamino) butyric acid,

2-bis- (4-chlorophenyl) acetic acid,

1-α-glutamyl-L-α-glutamyl-L-glutamic acid,

4- (trifluoromethoxy) phenoxyacetic acid,

2-en-valproic acid,

N- (o-tolyl) phthalimide acid,

N- (2-ethylphenyl) glutaramic acid,

2,4,6-trihydroxybenzoic acid, cis-2-hydroxy-1-cyclopentanecarboxylic acid, diphenylphosphinic acid,

4- (4-methoxyphenyl) thiophene-2-carboxylic acid,

4- (4-methylbenzylideneamino) salicylic acid, [2,2,2-trichloro-1- (3-p-tolylthioureido) ethyl] carbamate, (S) - (+) - α-hydroxy-1,3-dioxo-2 -isoindolinebutyric acid,

2,2 '- (1,2-ethanediyl) -bis (5-aminobenzenesulfonic acid),

4'-nitromaleanilic acid,

3,5-diisopropoxybenzoic acid,

N- [4- (4-chlorophenoxy) phenyl] phthalamic acid, benzoylaminophenylacetic acid,

4-chloro-3-nitrobenzoic acid,

4-methylphthalic acid, *

β- (2-acetoxyphenyl) propionic acid, (3-fluorophenyl) phosphonic acid, (R, R) - (-) - 2,3-diphenylsuccinic acid,

2- (4-chlorophenyl) -1- [2- (3,4-dimethoxyphenyl) ethyl] -6-oxo-

-3-piperidinecarboxylic acid, ethoxyacetic acid,

3- [3- (2,4,5-trichlorophenyl) ureido] benzoic acid,

2- [3-oxo-3- (N'-tetradecanoylhydrazino) propionylamino] benzoic acid,

2- [2- (2-chlorophenyl) -4-phenyl-5-thiazolyl] acetic acid,

4- (benzylideneamino) benzoic acid, henicosanoic acid, cis-hexahydro-N- (3-nitrophenyl) phthalamic acid,

3- (N-cyclohexylcarbamoyl) -5-norbornene-2-carboxylic acid, cyclohexanecarboxylic acid,

3- (2-hydroxyphenyl) propionic acid,

3'-fluororglutaranilic acid, tetrafluorephthalic acid,

4-acetamido-3-fluorobenzoic acid, dihydroxyfumaric acid,

4-butoxyphenylacetic acid,

D, L-p-hydroxypalmitic acid,

13-ketooktadeca-9Z, HE-dienoic acid,

1-Propionylpyrrolidine-2-carboxylic acid

3 ', 5'-dichloro-2'-hydroxy-4'-methylmaleanilic acid,

3- (triphenylsilyl) propionic acid,

2-methyl-2-pentenoic acid, (3-chlorophenyl) phosphonic acid,

3- (3-thienylsulfanyl) thiophene-2-carboxylic acid,

3-fluoro-4-methoxybenzoic acid,

3- (4-biphenylyloxy) propionic acid, boc-gamma-amino butyric acid,

4,5-dimethoxy-2-nitrophenylacetic acid,

3- (2,4-dihydroxyphenyl) propionic acid,

2-Hexadecylcarbamoyl-4-nitrobenzoic acid

3-fluoro-4-hydroxyphenylacetic acid,

4- (tri fluoromethoxy) phenylacetic acid, benzoyl formic acid, camphoric acid,

5-Benzo (1,3) dioxol-5-ylpenta-2,4-dienoic acid

2,3,4-trimethoxyphenylacetic acid,

2- (3,5-dinitro-2-thienylamino) -3-methylbutyric acid,

3- (4-methoxyphenyl) -2- (1-phenylethylideneamino) acrylic acid,

1-ascorbic acid, methylsuccinic acid, (-) - isoborneol-3-acetic acid,

1,1,2-cyclopropanetricarboxylic acid, indole-6-carboxylic acid,

4- (hexadecylthio) benzenesulfonic acid, hexahydro-N- (2,3-xylyl) phthalamic acid, (R) - (+) - N- (1-phenethyl) succinamic acid,

2.6- naphthalenedicarboxylic acid,

5-chloro-2-iodobenzoic acid,

2- (4-bromobenzoyl) acrylic acid,

2-fluoro-3- (trifluoromethyl) cinnamic acid,

8,8'-diapocarotenedioic acid,

5.6-dichloroanilic acid,

3-hydroxytridecanoic acid,

2 - [[2- / 3-chloro-5- (trifluoromethyl) -2-pyridyl / hydrazino] carbonyl] benzoic acid,

2-methoxy-9-oxo-8,9-dihydro-7H-benzocycloheptene-6-carboxylic acid, cis-5,8,11-icosatrienoic acid,

3-hydroxybutyric acid,

2-nitro-4- (trifluoromethyl) phenylthioglycolic acid,

2,4-bis (trifluoromethyl) phenylacetic acid,

4-hydroxy-α-mercapto-3-methoxycinnamic acid,

4-chloro-nitrobenzenesulfonic acid,

4-methylumbellif erylphosphate,

2 ', 5'-dimethylphthalanilic acid,

3- (naphthalene-2-sulfonyl) propionic acid, ', 6'-diisopropylglutaranilic acid,

2- (3,4-dimethoxystyryl) glyoxylic acid,

6- [4- (3-carboxypropyl) phenyl] hexanoic acid, metavartaric acid, dodecafluorsubric acid, phenolsulfonic acid,

5-bromo-2,4-dihydroxybenzoic acid,

2- (9H-fluoren-9-ylmethoxycarbonylamino) -3-phenylpropionic acid,

4-butoxybiphenyl-4'-carboxylic acid, p-phenylazobenzenesulfonic acid,

4-methylsulfonylphenylacetic acid,

3-Benzyloxy-4-methoxy-2-nitrobenzoic acid

4,5-dihydro-4,5-dioxo-1H-pyrrolo (2,3-f) quinoline-2,7,9-tricarboxylic acid,

2 '- (trifluoromethyl) maleanilic acid,

2-benzoylbenzoic acid,

4-chloro-2- (2-thienylethyl) benzoic acid, (R) - (-) - hexahydromanedioic acid,

2,5-dichloro-4-methoxybenzoic acid, benzyloxycarbonyl-D-pyroglutamic acid,

N- (2-cyanoacetamido) -3,4,5,6-tetrachlorophthalamic acid, (R, S) -fmoc-1,3-dihydro-2H-isoindolecarboxylic acid, cis-1-amino-3- (2-phosphonoacetyl) ) cyclobutane-1-carboxylic acid, α- (2,4-dimethoxy-3-methylbenzylidene) hippuric acid,

5-fluoro-2-methylbenzoic acid,

• · · ·

1,3,3a, 4,7,7a-hexahydro-2-methyl-3-phenyl-1-oxo-3α-isoindolecarboxylic acid,

5 (S), 12 (S) -dihydroxyicose-6E, 8Z, 10E, 14Z-tetraenoic acid, 5 (S), 14 (R), 15 (S) -trihydroxyicose-6-trans-8-cis-10- trans-12-trans-tetraenoic acid,

4- [3- / 2,2,2-tri-Cl-1- (cyclopentanecarbonylamino) et thioureido] benzoic acid, dodecenylsuccinic acid, α-fluorophenylacetic acid mixture, [4-amino-5- (3-chlorophenyl) -2- pyrimidinylsulfanyl] acetic acid,

3- (3,4,5-trimethoxyphenyl) -2-thiopyruvic acid,

N-fmoc- (3S, 4S) -4-amino-3-hydroxy-5-cyclohexylpentanoic acid,

N-acetyl-D, L-glutamic acid,

2- (hexadecyloxy) benzoic acid,

3- (2,2-dimethylpropionylamino) -3-phenylpropionic acid,

4- (4'-n-heptylphenyl (benzoic acid,

3- (4-n-hexyloxybenzoyl) propionic acid, (+/-) - 1-amino-cis-3-phosphonocyclopentanecarboxylic acid,

D, L-pyroglutamic acid,

4- (2-carboxyacetylamino) benzoic acid,

8,11,14-icosatriic acid,

2.2- bis (hydroxymethyl (butyric acid,

1,10-phenanthroline-2,9-dicarboxylic acid,

2-carboxymethoxy-3-methoxybenzoic acid, (s) - (+) - 2,2-dimethyl-5-oxo-1,3-dioxolane-4-acetic acid,

1,2-diphenylcyclopropanecarboxylic acid,

D-glutamic acid, (4-isopropyl-2-methoxyphenoxy) acetic acid, (4-dimethylamino-6-methyl-2-pyrimidinylsulfanyl) acetic acid,

D, L-glyceric acid,

Ι-β-p-nitrophenyl lactic acid,

5-bromo-6-hydroxypyrimidine-4-carboxylic acid,

2- (2-chlorophenyl) -4-methylthiazole-5-carboxylic acid,

2-benzamido-3-methylcrotonic acid,

2-amino-4-trifluoromethylthiazole-5-carboxylic acid,

4,5,10,11-tetramethyltetradeca-2,4,10,12-tetraene-6,8-diindioic acid,

3-hydroxy-4,4,4-trifluorobutyric acid, '-fluoro-3'-nitroglutaranilic acid, (3,5-dimethoxyphenyl) acetic acid,

4-phenylphthalic acid,

2'-chlorhexahydro-5 '- (tri-fluoromethyl) phthalic acid,

N- (4,6-dimethyl-2-pyrimidinyl) -3-aminobenzoic acid,

4- (hexadecyloxy) -3-nitrobenzenesulfonic acid, (R) - (4-) -2-bromopentanoic acid, s-trans, trans-farnesylthiosalicylic acid, [4- (5,5-dimethylhexyl) phenoxy] acetic acid,

4- (2,4,5-trichlorophenoxy) butyric acid, (+/-) - 12-hydroxyicose-5Z, 8Z, 10E, 14Z-tetraenoic acid,

4- (octadecyloxy) benzoic acid,

4'-fluoro-3'-nitrohexahydrophthalanic acid,

4-bromophthalic acid, hydantoin-5-acetic acid, n-tert-butylphthalamic acid,

D - (-) - o-formyloxy-2-phenylacetic acid,

2,3-dichloropropionic acid,

2-dodecenedioic acid, isobutylacrylic acid,

3- (4-fluorothiophenoxy) propionic acid,

4- (2-benzoylacetamido) benzoic acid,

4-oxo-4-phenylamino-2-butenoic acid,

4-oxohepta-2,5-dienedioic acid, acetodiphosphonic acid, •

3.5.5- trimethylhexanoic acid,

3-ethyl-2-hexenoic acid,

3'-chloro-2'-methyl-1,2,3,6-tetrahydrophthalanilic acid,

3,4-diacetoxyphenylacetic acid, trans-1,4-cyclohexanedicarboxylic acid,

3- (3-hydroxyphenyl) -2-methylacrylic acid, boc-L-4-thiazolylalanine,

N- (5-chloro-2,4-dimethoxyphenyl) glutaramic acid,

16-methyloctadecanoic acid,

4-n-hexyloxybenzoic acid,

3- [N- (3,4-dimethylphenyl) carbamoyl] -5-norbornene-2-carboxylic acid,

2-dodecanoylaminobenzoic acid,

2-isopropoxybenzoic acid,

3- (2-ethoxycarbonyl) -6-chloro-1H-indole-2-carboxylic acid, β-phenylcinnamic acid, - N - (4-chlorophenyl) carbamoyl] -5-norbornene-2-carboxylic acid,

2- (3,4-dimethoxyphenyl) -3-phenylacrylic acid,

1.2.3.4-tetrahydro-2-naphthalenepropionic acid,

3- (3,5-dimethoxy-4-hydroxyphenyl) propionic acid,

3-bromo-4-methoxyphenylacetic acid, 1-acetoxy-2-naphthoic acid,

4-hydroxy-3- (p-diazophenylphosphorylcholine) phenylacetic acid,

6-nitrocaproic acid,

3-nitro-4- (4-chlorophenoxy) cinnamic acid, octadec-9-indioic acid,

N- (2-chlorophenyl) malonamic acid,

4'-ethoxyglutaranilic acid,

2.4.6- trihydroxybenzoic acid,

N-fmoc-1-homophenylalanine,

N- (4-acetamido-3-methoxyphenyl) phthalamic acid,

N- (4-piperidone) glutaramic acid

4- [1- [N- (2-chloro-5-nitrophenyl) carbamoyl] -3,3-dimethyl-2-oxobutoxy] benzoic acid,

1-naphthoxyacetic acid, benzyloxycarbonyl-1-pyroglutamic acid,

2-chlorisophthalic acid,

2-amino-3-bromo-5-iodobenzoic acid,

2,4,6-trifluorophenylacetic acid, fmoc- (3S, 4S) -4-amino-5-cyclohexyl-3-hydroxypentanoic acid,

3,3 ', 4,5,5', 6-hexachlorophthalanilic acid,

2,4,5-trifluoro-cinnamic acid,

2-bromo-5-fluoro-cinnamic acid,

3-hydroxy-α-mercapto-p-methylcinnamic acid,

3-Benzoyl-2- (4-chlorophenyl) propionic acid

1-homocysteic acid,

4- [3- (2,6-xylyl) ureido] benzoic acid,

N-4-tert-butylbenzoyl-N-phenylanthranilic acid, benzothiazole-2-sulfonic acid,

4-methyl-dec-4-en-8-ynoic acid,

4-methoxy-3-nitrobenzoic acid,

4- (3- (5-chloro-2-methoxyphenyl) ureido] benzoic acid,

3-bromo-2-methylacrylic acid,

D-borneolic acid, fmoc- (3S, 4S) -4-amino-3-hydroxy-6-methylthiohexanoic acid,

10,12-heptadecadiinic acid,

4- [[(4-chlorobenzenesulfonylimino) phenylmethyl] amino] benzoic acid,

13-cis-retinoic acid,

2- (carboxymethoxy) benzoic acid, cis-hexahydro-N- (4-methyl-3-nitrophenyl) phthalamic acid,

6-hydroxy-5-nitroso-2-naphthalenesulfonic acid,

3-chlorothiophene-2-carboxylic acid

3-benzyladipic acid,

- 43 2 ', 5'-dimethylsuccinanilic acid, bis (2-ethylhexyl) diphosphoric acid,

4-oxo-3-phenyl-2-thioxo-1-imidazolidinacetic acid, (1R, 2S) -1-hydroxy-1,2,3,4-tetrahydro-2-naphthoic acid,

5- (4-fluorophenyl) -2,3-dihydro-1H-pyrrolizine-6,7-dicarboxylic acid,

3- [N '- (2,4-dinitrophenyl) hydrazinocarbonyl] acrylic acid, N-chloroacetyl-D, L-α-aminobutyric acid,

2- (2-hydroxybenzoyl) benzoic acid,

3-Benzoylamino-3-phenylpropionic acid

4-Heptyloxybiphenyl-4'-carboxylic acid

4-nitrohippuric acid,

4'-iodosuccinanilic acid,

2-acetamidoisophthalic acid,

15-phenyl-3-methylpentadecanoic acid, trans-4-propylcyclohexanecarboxylic acid, dibutyl phosphate,

4 ', 4-sulfonyldimaleanilic acid, trans, trans-muconic acid,

2- (3,4-dimethoxyphenylthio) acetic acid,

4 - [(5-bromo-2-hydroxybenzylidene) amino] benzoic acid, (S) - (+) - 3- (benzyloxycarbonyl) -5-oxo-4-oxazolidineacetic acid, fmoc- (3S, 4S) -4-amino- 3-hydroxy-6-methylheptanoic acid,

3- (N-benzylcarbamoyl) -5-norbornene-2-carboxylic acid, (S) - (+) - 2- (benzyloxycarbonyl) -1,2,3,4-tetrahydro-3-isoquinolinecarboxylic acid, (2-phenoxyethylthio) )acetic acid,

1-nitroanthraquinone-2-carboxylic acid, D-homocysteinsulfinic acid,

3-methoxybutyric acid,

2-Iodobenzoic acid, and, 3-dibromo-1-adamantanacetic acid, • · · ······ · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · ···· · · · · · · ·

4- (2-Hydroxyethoxy) benzoic acid

4-Benzenesulfonyl-4-cyanoheptanedioic acid,

N-phthalyl-D, L-aspartic acid,

2- (1-cyclohexenyl) butyric acid,

3- (4-chlorobenzyloxy) thiophene-2-carboxylic acid,

4- (2-thiydroxyethylamino) -3-nitrobenzoic acid,

2,3-dichloro-6-fluorobenzoic acid,

6- (2-ethoxycarbonyl) -2,3-dimethoxybenzoic acid,

4.5- dibromo-2-fluorobenzoic acid, ethylchromotropic acid,

4-butylbenzoic acid, isothiocyanobenzylethylenediaminetetraacetic acid,

5.6-diamino-1,3-naphthalenedisulfonic acid,

11- (butylthio) undecanoic acid,

3- (2-ethylsulfanylbenzo-6-thiazolylcarbamoyl) acrylic acid,

5-nitrobenzofuran-2-carboxylic acid, (ethylenedithio) diacetic acid, o-isopropylbenzoic acid,

3- [3- (4-acetoxyphenyl) -2-benzoylaminoacryloylamino] propionic acid,

2.3.5.6- tetramethylbenzoic acid,

3.4-methylenedioxyphenylacetic acid,

2- ^for hydroxyamino-3-methylbutyric acid, trans, trans-2,4-hexadienoic acid,

3- (trifluoromethyl) benzoic acid,

1-naphthylamino-3,5,7-trisulfonic acid,

4-aminophenylsuccinic acid,

3- [benzyl (toluene-4-sulfonyl) amino] propionic acid,

II-methyldodecanoic acid,

3.5-Difluoromandelic acid

2, '4', 5'-trichlorosuccinanilic acid, (+/-) - jasmonic acid, ·

• ·

- 45 (+/-) - 2- (6-methoxy-2-naphthyl) propionic acid, nitrilotriacetic acid,

2-methoxy-3-methylbenzoic acid,

2- (4-chlorobenzoylamino) -3-hydroxypropionic acid,

3-Benzoyl-2-naphthoic acid

4 '- (trifluoromethyl) -2-biphenylcarboxylic acid,

4- (dodecylthio) butyric acid,

4- (trifluoromethyl) mandelic acid,

N-α-boc-N-gamma-fmoc-d-diaminobutyric acid,

4-formamidobenzoic acid, boc-11-aminoundecanoic acid,

4-fluoro-2-methylphenoxyacetic acid,

7-amino-1,3-naphthalenedisulfonic acid,

2,3-dibromo-3- (3,4-dimethoxyphenyl) propionic acid,

3 - (/ (4-chlorophenyl) sulfonyl / methyl) -4-nitrobenzoic acid, m-anisic acid,

2 ', 4'-dimethyl-3,4,5,6-tetrachlorophthalic acid,

3-bromothiophene-2-carboxylic acid,

2- (thiobenzoyl) thiol acetic acid, aminobenzylethylenediaminotetraacetic acid,

2,3-dibromo-2'-methyl-4'-nitrosuccinanilic acid, (1-carboxymethyl-3,3-dimethylcyclohexyl) acetic acid,

4'-ethyl-3,4,5,6-tetrachlorophthalanic acid, cis-1,2-cyclohexanedicarboxylic acid,

4-ureidobenzoic acid,

2-phenyl-5- (trifluoromethyl) oxazole-4-carboxylic acid,

5-chloro-2-hydroxybenzenesulfonic acid,

3-ethoxy-4-hydroxyphenylacetic acid,

3- (decyloxy) benzoic acid, n-acetyl-D, L-ethionine, icosa-5,8-dienoic acid,

2,5-dihydroxybenzene-1,4-disulfonic acid,

2-bromobenzoic acid,

• ·

2-chloromandelic acid, (R) -4-methoxymandelic acid,

3-chloro-3'-methyl-biphenyl-2,2'-dicarboxylic acid, p-nitro cinnamic acid,

6-bromo-2-pyridin-4-ylquinoline-4-carboxylic acid,

4-fluorophlutamic acid, benzo (c) phenanthrene-5,6-dicarboxylic acid,

3-Benzyloxythiophene-2-carboxylic acid

2- (4-methylbenzoyl) benzoic acid,

N- (phenethyl) succinamic acid, cyclohexane-1,1-bis- (3-mercaptopropionic acid),

2-iodo-5-methylbenzoic acid,

1- (4-fluorophenyl) cyclohexanecarboxylic acid, (adamantan-1-yloxy) acetic acid, fmoc-D-glutamic acid gamma-tert-butyl ester,

4- (tert-butoxycarbonylaminomethyl) benzoic acid,

9,10-dihydro-12-ethoxy-9,10-ethanoanthracene-11-carboxylic acid,

3-fluorophthalic acid, cis-hexahydro-N- (2-methoxy-5-methylphenyl) phthalamic acid,

2-bromo-5-iodobenzoic acid, α-methyllevulic acid,

2,6-dibromobenzoic acid,

N- (2,4-dichlorophenyl) malonamic acid, (+/-) - β-p-chlorophenylglutamic acid,

3-bromobenzoic acid, (+) - α-methyl-4-carboxyphenylglycine, boc-L-glutamic acid gamma-tert-butyl ester,

4- (2-benzoylamino-3-methyl-2-butenoylamino) butyric acid,

3- [N- (2,4,6-trimethylphenyl) carbamoyl] -5-norbornene-2-carboxylic acid,

1- (4-methoxyphenyl) -1-cyclopentanecarboxylic acid, n-α- (tert-butoxycarbonyl) -β- (1-adamantyl ester) 1-aspartic acid φ ft ·· * ·

acids,

3.4- difluorophenylacetic acid, chloric acid,

N - [(R) -1- (1-naphthyl) ethyl] phthalamic acid, hydroxy-2-naphthalenylmethylphosphonic acid,

3- (4-isopropylbenzoyl) acrylic acid, (3-methoxyphenyl) phosphonic acid,

2,4-difluorobenzoic acid,

2- (2,4,6-trimethylbenzoyl) benzoic acid, (3-chloro-1,4-dioxo-1,4-dihydronaphthalen-2-ylamino) acetic acid,

2-ethyl-2-hydroxybutyric acid, iminobis (methylphosphonic acid),

1- (aminocarbonyl) -1-cyclopropanecarboxylic acid, (R) - (+) - 3-hydroxy-1-cyclopentene-1-heptanoic acid,

2,3-dimethylsuccinic acid, di-n-propylmalonic acid,

4-dibenzo (a, d) cyclohepten-5-ylidenebutyric acid,

15 (S) -hydroxyicose-8Z, 11Z, 13E-trienic acid,

4-phosphonobenzoic acid, cis-2 ', 5'-dimethylhexahydrophthalanic acid, cis-N- (2,3-dichlorophenyl) hexahydrophthalamic acid,

3- (2-methoxybenzoylamino) benzoic acid, (+/-) - 1-aminocyclohexane-trans-1,2-dicarboxylic acid, n-benzoyl-D-aspartic acid,

2- (2-phenoxyacetylamino) -3-phenylpropionic acid, trans-2- (p-methylbenzoyl) -1-cyclohexanecarboxylic acid,

1-glutamic acid N-α- (benzyloxycarbonyl) -gamma- (benzyl ester),

4-bromobutyric acid, β- (3-acetoxyphenyl) propionic acid, α-chloro-3,5-dimethyl-1-adamantanacetic acid,

11-dodecenoic acid, · φ · Φ · Φ · Φ · Φ · ΦΦΦ · Φ · ΦΦΦ · ΦΦΦ ·

- 48 (S) -cbz-oxaproline, mosquelglyoxylic acid, cyclopentylacetic acid,

3-chlorosalicylic acid,

2-methylglutaric acid,

N-α- (9-fluorenylmethyloxycarbonyl) -1-norvaline,

1-α-glutamyl-1-aspartic acid,

N- (4,6-dimethyl-2-pyrimidinyl) -2-aminobenzoic acid,

6-heptadecyloxy-1-hydroxynaphthalene-2-carboxylic acid,

1,3-phenylenedipropionic acid,

4'-methyl-3'-nitromaleanilic acid, tricose-10,12-diindioic acid,

D, L-2- [4- (trifluoromethoxy) phenoxy] propionic acid,

N- (diphenylmethyl) glutaramic acid,

2-Benzoylpyridine-4-carboxylic acid

2.4.6- trichlorobenzoic acid,

2- (2,4-dimethylbenzyl) benzoic acid,

2,4-henicosadioic acid,

3-Methyl-2- (ortho-tolyl) butyric acid

2.3.4.5.6- pentachlorobenzoic acid,

3.4- dichloropentafluorobutyric acid,

3.4.4-trichloro-2-nitro-3-butenoic acid,

1.2.4-Benzenetricarboxylic acid

5-mercapto-tetrazole-1-propionic acid, lauric acid,

4-iodobutyric acid, cis-8,11,14-icosatrienoic acid,

3-carboxy-4-hydroxy-5-sulfoaniline,

2-furylthio pyruvic acid,

2-chloro-5-nitrobenzenesulfinic acid, n-α- (tert-butoxycarbonyl) -β- (2-adamantyl ester) 1-aspartic acid,

1-cis-pyrrolidine-2,4-dicarboxylic acid,

2-amino-5-cyano-3-ethylbenzoic acid,

1-Acetoxynaphthalene-6-sulfonic acid

5 (s) -hydroxyicose-6E, 8Z, 11Z, 14Z-tetraenoic acid, fmoc-D-norvaline,

4- [N- (3-chlorophenyl) carbamoyl] butyric acid,

3-Methyl-1,1-cyclohexanediacetic acid

6-nitro-1-diazo-2-naphthol-4-sulfonic acid,

2- (4-methoxyphenoxy) -5-nitrobenzoic acid, 4,4'-diaminodiphenylamino-2,2-disulfonic acid,

2-methyloctadecanoic acid,

2,6-difluoro cinnamic acid,

20-hydroxy- (5Z, 8Z, 11Z, 14Z) icosatetraenoic acid,

4-toluenesulfonylacetic acid,

5-bromo-3-methylsalicylic acid,

5-chlorvaleric acid,

5-benzyl-3,6-dioxo-2-piperazineacetic acid,

5-hydroxycyclohexane-1,3-dicarboxylic acid,

3-bromo-2-methoxy-5-methylbenzoic acid,

2-pyroslizic acid,

5- (2,5-dichlorophenylazo) -4-methylsalicylic acid,

4 - [(benzenesulfonyliminophenylmethyl) amino] benzoic acid,

1- Naphthylacetic acid

3 - [(furan-2-carbonyl) amino] benzoic acid, trans-2,4-pentadienoic acid,

3- [3- (2-chloro-6-methylphenyl) ureido] benzoic acid,

2 - ([3- / 2,2,2-trichloro-1- (2,2-di-propionylamino) et. Thioureido] benzoic acid,

5,5'-dithiobis (2-nitrobenzoic acid), cis-hexahydro-N- (3-chloro-4-methylphenyl) phthalamic acid, (Z) - [2- (formamido) thiazol-4-yl] (methoxyimino) acetic acid, pyridine-2-sulfonic acid,

4- (tetradecyloxy) benzoic acid,

4-cyclopentylnaphthalene-1-carboxylic acid

4- (4- (1-methyl-1H-quinolin-2-ylidene) -2-butenylidenamino] benzoic acid,

3-amino-2-naphthol-1,8-disulfonic acid,

5-nitroorotic acid,

4 '- (2-furoylamino) -3'-hydroxymalonanilic acid, (2-phenylcyclohexyl) acetic acid,

4-dodecyloxybenzoic acid,

15-methylhexadecanoic acid, (R) - (+) - 2-chlorobutanoic acid,

3-amino-1,5-naphthalenedisulfonic acid, isoindolin-1-one-2-acetic acid,

2- (3- / N '- (3-methylbutyryl) hydrazino) -3-oxopropionylamino] benzoic acid, (3,3-dimethyl-1-phenyl-1,3-dihydroisobenzo-1-furyl) acetic acid,

2-Methyl-4-naphthalen-1-ylbutyric acid

4- (chlorosulfonyl) benzoic acid,

3-carboxy-2-furanacetic acid,

3- (4- (4-bromophenylthio) -3-nitrophenyl) acrylic acid, bicyclo (2,2,1) heptane-1-carboxylic acid,

2'-ethoxymaleanilic acid,

3-nitro-5- (trifluoromethyl) benzoic acid, p- (benzylsulfonamido) benzoic acid,

3- (1-naphthyl) acrylic acid,

N-acetyl-8-hydroxy-2-naphthylamino-6-sulfonic acid, [biphenyl-2-yl (toluene-4-sulfonyl) amino] acetic acid,

N-acetylglycyl-D-glutamic acid,

3-ethylheptanoic acid,

7-chlorobenzofuran-2-carboxylic acid,

3,5-difluoro cinnamic acid,

3- (3,4-dimethylphenyl) -3-methylbutyric acid,

5,8,11,14,17-icosapentaenoic acid,

2,4,6-trinitrobenzenesulfonic acid,

- 51 nervonic acid,

5-methyl-2-phenyl-4-thiazolylacetic acid, (5,6-dimethoxy-3-oxo-1,3-dihydroisobenzo-1-furyl) acetic acid,

1-methylcyclopropane-1-carboxylic acid, dodecylbenzenesulfonic acid,

3-Ethylhexanoic acid

1- N- (1-carboxy-5-aminopentyl) iminodiacetic acid,

4-hydroxy-3-nitrobenzoic acid, di-n-butylphosphinic acid,

4'-octyloxy-4-biphenylcarboxylic acid,

2-diazo-1-naphthol-5-sulfonic acid,

4'-bromophthalanilic acid,

2,6-dinitrotoluene-4-sulfonic acid,

N-acetyl-6-chloranthranilic acid,

4- (2-acetylamino-4,5-dimethylphenyl) -4-oxobutyric acid,

2,4-dinitrobenzenesulfonic acid,

3- (2-chloro-3,4-dimethoxyphenyl) acrylic acid, p-heptyloxybenzoic acid,

4-chloro-3-hydroxybenzoic acid,

3- [ac- (5-nitro-1,3-dioxo-1,3-dihydro-2-isoindolylmethyl) amino] benzoic acid,

12-hydroxydodecanoic acid, trichloroacrylic acid, piperonyl acid,

4-Methoxy-α-methylcinnamic acid

5-benzyloxy-2-nitrophenylpyruvic acid,

2- (2-hydroxy-1-naphthylmethyleneamino) benzoic acid,

7-methoxy-2,2-diphenylbenzo (1,3) dioxole-5-carboxylic acid,

13-oxotetracosanoic acid, dipropylphosphinic acid, gibberic acid,

3'-chloro-4'-methylsuccinanilic acid, ·

1- hexadecenylsuccinic acid,

3-bromo-4-hydroxy-5-methoxyphenylacetic acid,

N- (2,4-dichlorobenzyl) -1,2,3,6-tetrahydrophthalamic acid,

2,4- heptadecadiinic acid, (+) - 4'-methyltartranilic acid,

3,5-dimethyl-4-formyl-2-pyrrolecarboxylic acid,

11 (R) -hydroxy- (5Z, 8Z, 12E, 14Z) icosatetraenoic acid,

N-formyl-4- (methylamino) benzoic acid, succinic acid,

2- (n-heptyloxy) butyric acid

2.3.4- Trifluoric acid,

3- (4-methoxy-2-methylphenyl) propionic acid, gamma-D-glutamyltaurine,

4-chloro-3-fluoro-cinnamic acid,

4- (5-indanylmethyleneamino) benzoic acid,

2.4- difluoromandelic acid,

5-oxoazelaic acid,

3- [3-chloro-5- (trifluoromethyl) -2-pyridyl (propanoic acid, trans-3- (4-methoxybenzoyl (acrylic acid,

N-α- (tert-butoxycarbonyl) -1-octahydroindole-2-carboxylic acid, (S) - (+) - hexahydromanedioic acid,

N- (3-chlorophenyl) phthalamic acid,

N- (1-naphthyl (maleic acid),

2- (4-tert-butylphenoxy) -2,2-difluoroacetic acid,

2-Ethylnonanoic acid

3- (5-bromo-2-ethoxyphenyl) acrylic acid, fmoc-6-aminohexanoic acid, chlorosuccinic acid, gamma-D-glutamylaminoethylphosphonic acid,

3-hydroxy-4,4,4-trichlorobutyric acid, acetyl-D-aminoheptylic acid,

3- (methoxycarbonylmethylthio) thiophene-2-carboxylic acid,

- 53 N- (1,1'-bis (hydroxymethyl) ethyl] -3,4,5,6-tetrachlorophthalamic acid,

1,1-cyclopropanedioic acid,

4-aminoacetanilide-2-sulfonic acid,

2- (4-hexylbenzoylamino) benzoic acid,

4,4 '- (carbonyldiimino) bisbenzoic acid,

3-isobutyrylamino-3- (4-methoxyphenyl) propionic acid, biphenyl-3,5-dicarboxylic acid,

3,3-dimethyl-4-oxovaleric acid, pinonic acid,

3-chloropentanedioic acid, gibberellic acid,

3- (nonylamido) benzoic acid,

4- (trifluoromethyl) benzoic acid,

3- (allylsulfanyl) -2-thiophenecarboxylic acid,

3 ', 4'-dibromophthalanilic acid,

3-hydroxynonic acid,

3- (4-oxo-3,4,5,6,7,8-6H-benzo (4,5) -thieno (2,3-d) pyrimidin-2-yl) -propionic acid,

4- (4-Phenoxybenzoyl) benzoic acid

5-diiodobenzoic acid,

3- [N- (2,4-difluorophenyl) carbamoyl] -5-norbornene-2-carboxylic acid, benzo (c) phenanthrene-3-carboxylic acid,

2-methyl-2- (7-methyl-4-indanyloxy) propionic acid, exo-2-bromo-5,5-ethylenedioxy-bicyclo (2,2,1] heptane-syn-7-carboxylic acid,

3-methoxy-2,4,5-trifluorobenzoic acid, (+) - 2- (1-naphthoxy) propionic acid,

2-dichloro-1-methylcyclopropanecarboxylic acid,

2-fluoro-4- (trifluoromethyl) phenylacetic acid, (+/-) - azetidin-2-one-4-carboxylic acid,

4- (3- (3,5-di-tert-butyl-4-hydroxyphenyl) -3-oxopropenyl)

- 54 benzoic acid, levulic acid, dimethylphosphate,

2.4- dinitrophenylacetic acid,

3.4-dichlorobenzenesulfonic acid, boc-3-aminobenzoic acid,

3,4-dimethylbenzoic acid,

2-fluoro-5-methylbenzoic acid, n-α- (9-fluorenylmethoxycarbonyl) -1-2-amino-5-ureido-n-valeric acid, o-nitrobenzoic acid,

2,3-dibromosuccinic acid, β- (S) - (4-methoxybenzylmercapto) isovaleric acid,

4-bromo-7-oxo-6-oxa-bicyclo (3.2.1) octane-2-carboxylic acid,

1-pentanesulfonic acid,

5-hydroxyisophthalic acid, (S) -4-chloromandelic acid,

1-hydroxy-2-oxo-1,2-dihydropyridine-3-carboxylic acid,

3-acetamido-3-methylbutyric acid,

3 '- (trifluoromethyl) succinanilic acid,

2-Meo-4-methyl-6- (2,2,2-trichloro-1-hydroxyethyl) cyclohexanecarboxylic acid

4-ethoxycinnamic acid,

5-bromoisophthalic acid,

2'-chloro-5'-nitropthalanilic acid,

2-methyl-3-p-tolylacrylic acid,

5,5,6,6,7,7,7-heptafluoro-4,4-bis (trifluoromethyl) -2-heptenic acid,

2 ', 4'-dimethylmaleanilic acid,

4-acetoxybenzoic acid,

3,6-disulfonaphthalene-1,8-dicarboxylic acid, (R) - (-) - citramalic acid,

• 44

1-octanesulfonic acid,

2-Methyl-2-phenylhexanedioic acid

3-noradamantanecarboxylic acid,

2-cyano-3- (3,4-dihydroxy-5-methoxyphenyl) acrylic acid,

3,5-dinitro-4-hydroxyphenylacetic acid,

2-chloro-3,4-dimethoxybenzoic acid,

5- (trifluoromethyl) thieno (3,2-b) pyridine-6-carboxylic acid,

9,9-dihydroxy-5-oxononanoic acid, diisoctylphosphinic acid, boc-hexahydropyridine-4-carboxylic acid,

3,4-dichloro-2-thiophenecarboxylic acid, Na-fmoc-N-gamma-aloc-1-diaminobutyric acid, cis-2- (tert-butoxycarbonylamino) -1-cyclopentanecarboxylic acid, boc-4-aminobenzoic acid, phosphatidic acid acid, cis-3 ', 4'-dimethylhexahydrophthalanic acid,

1,2.3-triazole-4,5-dicarboxylic acid,

N- (3-nitrophenyl) -1,2,5,6-tetrahydrophthalamic acid,

3 - [(2-ethoxycarbonyl) - (4-methylthiazol-2-yl) amino] propionic acid,

2.3.4- trimethylcyclobutanecarboxylic acid,

5- [2 '- (3'-chloro-5'-trifluoromethyl) pyridylamino] methyl-3,4-dihydroisoxazole-2-3- (n-ethylthiocarbamoylthio) propionic acid, na-boc-np-bromoacetyl-1-diaminopropionic acid acid, trans-1,2-cyclohexanediacetic acid,

6-difluoromandelic acid, cis-N- (2-chlorophenyl) hexahydrophthalamic acid,

2,6-dichloropyridine-4-carboxylic acid,

N- (1-naphthyl) -1,2,3,6-tetrahydrophthalamic acid,

3- (trifluoromethylthio) benzoic acid,

- 56 N- (2-bromophenyl) maleic acid, β-glutamic acid,

6-hydroxy-1-naphthoic acid,

4- (2-thienylmethyleneamino) benzoic acid,

N- (2,4-dinethoxyphenyl) phthalamic acid, heptafluoro-2-hexenoic acid, (4-benzyloxy-5-methoxy-2-nitrophenyl) acetic acid,

3- (4-chlorophenyl) propionic acid, boc-1-p-aminobutyric acid, (4-fluorophenylthio) acetic acid, (2-isopropylsulfanylacetylamino) acetic acid,

2- (3,5-dinitrothiophen-2-ylamino) pentanedioic acid,

3,3'-dichloropivalic acid, (2-butyrylphenoxy) acetic acid, styrene phosphonic acid,

1- (2-fluorophenyl) cyclopentanecarboxylic acid,

2- (2,3-dimethoxystyryl) glyoxylic acid,

3,5-di-tert-butylsalicylic acid,

2- (pentamethylbenzoyl) benzoic acid,

4-ethyl-2-pyridinecarboxylic acid,

N, N'-dodecamethylenebis (glutaramic acid),

N-cbz- (2R, 3R) -3-amino-2-hydroxy-4-phenylbutyric acid, carboxymethanesulfonylmethanesulfonylacetic acid,

3- (2,3,4-trimethoxyphenyl) propionic acid,

17- (p-toluenesulfonyloxy) heptadecanoic acid,

4 - [(2-hydroxy-5-nitrobenzylidene) amino] benzoic acid,

4 - [(naphthalen-1-ylmethylene) amino] benzoic acid,

3-benzoyl-3-benzylidenepropionic acid, valerylsalicylate,

3,4-diphenylcyclobutane-1,2-dicarboxylic acid,

2-chloro-5- (trifluoromethyl) benzoic acid,

3-pyridinepropionic acid,

4- [2,5-bis- (2,2-dimethylpropyl) phenoxybutyric acid, • *

3- (octadecyloxy) benzoic acid, (R) - (+) - 2-bromopropionic acid,

3,4-dihydro-6-methoxy-1-naphthoic acid,

2-nitro-4- (2,2,2-trifluoro-1-hydroxy-1-trifluoromethylethyl) benzoic acid, glycolic acid,

2-isoquinolin-1-ylmethylbenzoic acid,

3.4.4-trichloro-2-dichloromethylene-3-butenoic acid,

4-Methyl-2-phenyl-1,2,3-triazole-5-carboxylic acid

3-bromo-4-fluoro-cinnamic acid,

8-nitroquinoline-4-carboxylic acid,

3- (3-Me-5-oxo-4,5-dihydro-1-pyrazolyl) -2-phenylcarbamoylbenzenesulfonic acid,

4- (trifluoromethylthio (benzoic acid,

4- [3- (2-ethylphenyl (ureido) salicylic acid,

2'-ethylmaleanilic acid, p-xylene-2-sulfonic acid,

2,3,4,4,5,5,5-heptafluoro-2-pentenoic acid,

4-iodo-3-nitrobenzoic acid,

2-benzoylamino-3- (diethoxyphosphoryl) -3-phenylacrylic acid, 4,4'-dinitrostilbene-2,2'-disulfonic acid, trans-4-n-butylcyclohexanecarboxylic acid,

3,4-difluoro-5- (trifluoromethyl) phenylacetic acid,

2-nitro-α, α, α-trifluoro-p-toluylic acid,

2,4-dichloropyridine-5-carboxylic acid,

2- (morpholine-4-carbothioylsulfanyl) propionic acid, α-methyl-4-nitro-cinnamic acid,

6-methyl-2-phenylimidazo (1,2-a) pyridine-3-carboxylic acid, [1- / 2- (3,4-dimethoxyphenyl) ethyl] -5-ethyl-2-oxo-4-piperidin-4 -yl] acetic acid,

5-carboxyvanilic acid,

3-Benzylquinoline-4-carboxylic acid

3- (4-methylthiobenzoyl (propionic acid)

- 58 N- (2-benzylsulfanylbenzothiazol-6-yl) succinamic acid,

3- (8-benzyl-9-oxo-6,7,8,9-tetrahydro-5H-benzocyclohepten-8-yl) (propionic acid, succinanilic acid, n-tosyl-3-pyrrolecarboxylic acid,

2-ethyl-3- (4-methoxyphenyl (acrylic acid, butyric acid, (Ια, 2a, 3β, 4β) -2,4-bis (4-hydroxyphenyl) -1,3-cyclobutanedioic acid),

3,4-difluoro-5- (trifluoromethyl (benzoic acid,

2,3,5,6-tetrafluoro-p-toluic acid,

2-bromo-4,5-dimethoxybenzoic acid,

3- [2-benzoylamino-3- (4-methoxyphenyl (acryloylamino) propionic acid),

5-nitro-1,2,3,4-tetrahydro-1,4-ethenonaphthalene-2,3-dicarboxylic acid,

3- (4-n-heptylbenzoyl (propionic acid, (1-oxodecahydronaphthalen-2-yl) (acetic acid,

2- (carboxyhydroxymethyl) -6-hydroxy-4-methylcyclohexanecarboxylic acid,

N-furfurylphthalamic acid,

3- (2-furyl) -2-oximinopropionic acid,

10,11-dihydroxyundecanoic acid,

2-thioorotic acid,

2'-chloro-5'-nitroglutaranilic acid,

8-nonyonic acid, (R, S) -1-aminoindan-1,5-dicarboxylic acid,

4- (3,5-diisopropylbenzoylamino (benzoic acid,

2-butyl-3- (2-methoxyphenyl (acrylic acid, N-fmoc-1-aminocyclopropane-1-carboxylic acid, iminodiacetic acid, bis (p-nitrophenyl) phosphate),

2-benzoylamino-3- (3,4-dimethoxyphenyl (propionic acid),

• · · ·

3- (3,5-dimethylnaphthalen-2-yl) -2-methylbutyric acid,

2-ethoxy-4-methoxybenzoic acid,

D, L-2-hydroxy-n-butyric acid, (2-carbamoylphenoxy) acetic acid,

5-acetylsalicylic acid,

N-benzylphthalamic acid,

N- (4-methylphenyl) maleic acid,

1-leucyl-1-glutamic acid, [4- (3-methylureido) benzoylamino] acetic acid, arabinic acid,

9-methylundecanoic acid,

2- (methylthio) benzoic acid, arachidonic acid,

2,4- dichlorophenylacetic acid,

2-Dibenzothiophenopropionic acid

3- (3,4-ethylenedioxybenzoyl) propionic acid,

2-methyl-2- (4-methyl-3-oxocyclohexyl) malonic acid,

8-cyanophthalene-1-sulfonic acid,

5- (methylthio) thiophene-2-carboxylic acid,

2-bromodecanoic acid,

2-Isopropylideneaminooxybutyric acid, allylmalonic acid

3,5-dimethoxy-4-methylbenzoic acid, α- (4-methoxy-1-naphthyl) -o-toluic acid,

3- (4-ethoxyphenyl) propionic acid,

3- (2-nitro-4-trifluoromethylphenoxy) -2-thiophenecarboxylic acid,

3- (2,6-dichlorophenyl) -2-methylacrylic acid,

4- (4-cyanophenoxy) benzoic acid, chlorenedic acid,

12-formyltricyclo (8,2,2,2 (4,7)) hexadeca-hexaene-5-carboxylic acid,

N- (2,6-dimethylphenyl) -1,2,3,6-tetrahydrophthalamic acid, poly-1-glutamic acid, (S) - (+) - ketopin aeid

3.4.5-trimethoxy-2-nitrobenzoic acid, homovanilic acid,

8-chloro-4-dibenzofurancarboxylic acid,

5,6a, 7,7a-tetrahydro-4H-cyclopropa (or Jacenaphthylene-7-carboxylic acid,

3- [N- (2,6-xylyl) carbamoyl] propionic acid, (4-methoxyphenyl) phenylphosphinic acid,

4-acetamidobutyric acid, trans-norpinic acid, fmoc- (3R, 4S) -4-amino-3-hydroxy-6-methylheptanoic acid,

3,4,5,6-tetrachloropyridine-2-carboxylic acid,

2'-methoxy-5'-methylmaleanilic acid,

3- (octane-1-sulfonyl) propionic acid,

2-chloropropionic acid,

4- [4- (1,3-dioxo-1,3-dihydroisobenzofuran-5-carbonyl] phenoxybenzoic acid,

12-methyltetradecanoic acid, triphenylacetic acid,

3-methyl-1-oxoisochroman-5-carboxylic acid, [4-phenyl-5-phenylamino-4H- (1,2,4) triazol-3-ylsulfanyl] acetic acid,

9-hydroxyimino-9,10-dihydroanthracene-1-carboxylic acid,

7-methoxy-1-methyl-4-oxo-2,3,4,5-tetrahydro-1H-benzo (d) azepine-2-carboxylic acid,

2,5-dichlorophenylthioglycolic acid,

1-Cyancyclopropanecarboxylic acid

2,6-dinitromesitylene-4-sulfonic acid,

3- (4-hydroxy-3-methoxyphenyl) -2-methylacrylic acid,

3- (4-cyclohexylbenzoyl) acrylic acid,

2-Cyano-2-methyl-3-phenylpropionic acid

2,3-dimethoxyphenylacetic acid,

η-α- (benzyloxycarbonyl) -gamma- (benzyl ester) d-glutamic acid,

N- (4-methoxyphenyl) tetrachlorophthalamic acid,

4-phenylbutyric acid,

3-nitrobenzaldehyde-4-sulfonic acid, n-octadecylsuccinic acid, pyridine-4-sulfonic acid,

2-hydroxy-2-trifluoromethylbutyric acid,

2.6- dimethyl terephthalic acid, terephthalic acid,

3,5-di-tert-butyl-4-hydroxycinnamic acid,

3-ethoxypropionic acid,

4-allyl-2-methoxyphenoxyacetic acid,

D - (-) - diisopropyl-d-tartaric acid,

4-bromomethylnaphthalene-1-carboxylic acid,

2'-chloro-6'-methylsuccinanilic acid,

2 ', 4'-dimethoxyhexahydrophthalanilic acid,

2,7-difluoro-9-oxo-4-fluorenecarboxylic acid,

2-Methoxy-6- (2,2-dimethylpropionamido) cyclohexanecarboxylic acid

3-hydroxyphenylacetic acid,

6-iodo-hexanoic acid,

3-bromo-2,6-dimethoxybenzoic acid,

3- (4-chlorophenyl) -2-phenylpropionic acid, (S) - (-) - 2-chloro-3-methylpentanoic acid, α-chloro-3- (trifluoromethyl) hydrocinnamic acid,

3- (hexadecane-1-sulfonyl) propionic acid,

12 (S) -hydroxy- (5Z, 8E, 10E) -heptadecatrienoic acid,

1.3.5-cyclohexanetricarboxylic acid,

3-hydroxy-4,5-dimethoxybenzoic acid,

4-bromo-1,2,3,4-tetrachloro-1,3-butadiene-1-carboxylic acid, (2,4-xylyl) phosphonic acid, • 4

4-bromo-3-methoxynaphthalene-2-carboxylic acid, (+/-) - threo-4-methylglutamic acid, levulic oxime, cis-13-octadecenoic acid,

4- (methylsulfonyl) benzoic acid, (3-methoxy-4-phenoxyphenyl) acetic acid, carboxypyrazolone-2,5-disulfonic acid,

5-methoxy-1-indanone-3-acetic acid, tnp-1-glutamic acid,

4-chlorobutyric acid,

1-naphthylamino-2,4,7-trisulfonic acid,

6-hydroxy-3-oxo-7α-propionyloktahydroindene-1-carboxylic acid, furan-2,5-dicarboxylic acid, α- (4-chlorophenyl) -4-nitro-cinnamic acid,

2-bromvaleric acid,

2.2- diethylbutyric acid,

D, L-glutamic acid,

4- (4-hydroxybenzylideneamino) salicylic acid, (S) - (+) - 2-methylbutyric acid,

Ν-α-Ν-β-bis-boc-1-diaminopropionic acid

2.2-diphenylpropionic acid,

1-hydroxycyclohexanecarboxylic acid, stearic acid,

2- (2-carboxyethylamino) succinic acid, coumarin-3-carboxylic acid,

4- (2- (4-tert-octylphenoxy) ethoxy] benzoic acid,

2- (2-chloro-4-fluorophenylthio) acetic acid,

5-bromo-2-methylbenzoic acid, myristic acid, cis-10-nonadecenoic acid,

2-bromo-4-fluoro-cinnamic acid,

1- (4-Methylbenzenesulfonyl) indole-3-acrylic acid

1-Et-6-fluoro-7-hydroxy-4-oxo-1,4-dihydro (1,8) naphthyridine-3-

-carboxylic acid,

3,4-diethoxyphenylacetic acid, (R) -hydroxy-16-heptadecinic acid,

4-chlorobenzenesulfinic acid, 11-bromoundec-10-ynoic acid,

3 - ((4,6-dimethoxy-2-pyrimidinyl) oxy] pyridine-2-carboxylic acid,

3.4.5- trimethoxybenzoic acid,

2-fluoro-4-octyloxybenzoic acid,

4-Methyl-2-thioxo-2,3-dihydrothiazole-5-carboxylic acid

4-methyl-2-pentenoic acid,

2-Methoxycarbonyl-2-methylcyclohexanecarboxylic acid

7-Hydroxy-4-methylcoumaron-3-ylacetic acid

1,5-pentanebisphosphonic acid, trans-3-furanacrylic acid,

3-acetamido-p-toluic acid,

3- (4- (methylsulfonyl) phenyl] - (2e) -propenoic acid,

4-fluoro-2,3,5,6-tetramethylbenzoic acid,

4-tricyclo (4,3,1,1 (3,8)) undecanecarboxylic acid,

2-methoxy-4-nitrobenzoic acid, vanilla acid,

N- (4-acetylphenyl) maleanilic acid, taurine-N, N-diacetic acid,

4.5.5-Tetrafluoro-4- (heptafluoropropoxy) pentanoic acid, diethylmalonic acid,

3- (3- / 3- (trifluoromethyl) phenyl / ureido] benzoic acid,

5-bromo-2-nitrobenzoic acid,

2- (4-cinnamoylphenoxy) acetic acid, adrenic acid, tetracosanoic acid,

3- (trifluoromethyl) anthranilic acid,

3- (2-o-tolyloxyacetylamino) benzoic acid,

N- (2,4,6-trimethylphenyl) glutaramic acid,

2 ', 4'-dichlorosuccinanilic acid,

2,3-dihydrobenzo (b) furan-5-carboxylic acid,

3- (2-chlorophenyl) propionic acid,

2-fluoropalmitic acid,

5- (4-methoxyphenyl) -2,3-dihydro-1H-pyrrolizine-6,7-dicarboxylic acid, [5-cyano-2- (4-methoxyphenyl) -6-oxocyclohex-1-enyl] acetic acid, glutathione sulfonic acid acid,

4- (4-acetamidophenylimino) -2,3-dichloro-2-butenoic acid, (4-benzyloxy-3-methoxyphenyl) acetic acid,

2-phenylhexanedioic acid,

4-Methyl-2-oxovaleric acid

2'-benzoyl-4'-chlorormaleanilic acid,

5,6-acenaphthenedicarboxylic acid,

5- [2-chloro-5- (trifluoromethyl) phenyl] -2-pyrosylic acid,

3- (2,4-dimethylbenzoyl (propionic acid,

2-fluoro-3- (trifluoromethyl) phenylacetic acid,

4,5-dihydro-1- (methylthio) benzo (c) thiophene-3-carboxylic acid, (2-methoxycarbonylcyclopropyl (acetic acid,

2- (butylcarbamoyl) benzoic acid,

3-allyloxypropionic acid,

2´-carbamoylbiphenyl-2-carboxylic acid,

6- (1,3-dioxo-1H, 3H-benzo (d, e) isoquinolin-2-yl) hexanoic acid,

3,5-diisopropylsalicylic acid,

4-ethylbenzenesulfonic acid, boc-1-pipecolic acid,

2,6-dichloro-4- (trifluoromethyl) phenylacetic acid,

3-thiophenmalonic acid,

3-Hydroxy-2-dimethyl-3-phenylpropionic acid, in the form of 3-hydroxy-2-dimethyl-3-phenylpropionic acid.

3- (9-methyl-9H-fluoren-9-yl) butyric acid,

2- (1,2,3,4,5-Pentahydroxypentyl) thiazolidine-4-carboxylic acid

D, L-Atromic acid,

N-t-boc- (2R, 3R) -3-amino-2-hydroxy-5-methylhexanoic acid,

2- (1-naphthoyl) benzoic acid,

1- [2- (3-chloro-5-trifluoromethylpyridyl) indole] -3-propenoic acid,

4'-butylmaleanilic acid,

4-fluoro-3,5-dimethylbenzoic acid,

4-chloro-3-fluorobenzoic acid, N-α-fmoc-N-gamma-boc-d-diaminobutyric acid, cyclohexa-2,4-dienyl- (2,3,5,6-tetramethylphenyl) acetic acid,

8- (4-methoxyphenyl) -6-methyl-8H- (1,3) dioxolo (4,5-g) chromene-7-carboxylic acid,

II- (4-chlorophenylsulfanyl) undecanoic acid,

1,3-dioxo-2-p-tolyl-2,3-dihydro-1H-isoindole-5-carboxylic acid, cis-2- (p-methylbenzoyl) -1-cyclohexanecarboxylic acid, mucic acid,

4 '- (methylthio) succinanilic acid,

3-ethoxy-2-butenoic acid, acetoxyacetic acid,

5-Methyl-2-nitrobenzoic acid

4-chloro-2-fluorobenzoic acid,

2,5-dimethoxycinnamic acid, (+/-) - β-phenylglutamic acid,

3-Methyl-2-oxobutyric acid

1-heptanesulfonic acid,

4-Methyl-3-nitrobenzoic acid

2-carcinnamic acid, α-methylcinnamic acid,

4- (3-hexadecyl-2-thioureido) benzoic acid, dehydroabietic acid, (2-nitrobenzenesulfonylamino) acetic acid, (3-benzyloxy-4-methoxyphenyl) acetic acid,

5-bromo-2-iodobenzoic acid,

1,1,3-trimethyl-3-phenylindan-4 ', 5-dicarboxylic acid, oxaleacetic acid,

2-aminoterephthalic acid, perfluorohexanoic acid,

6-dichlorophenylacetic acid,

6-Bromo-2-pyrid-3-yl-quinoline-4-carboxylic acid

4- (chloromethyl) benzoic acid,

2- (4-Isopropylbenzoyl) acrylic acid

5-iodferulic acid,

3- (1,2,3,4-tetrahydronaphthalen-1-yl) propionic acid,

2- [3-Oxo-3- (N'-tridecanoylhydrazino) propionylamino] benzoic acid,

2'-carbamoyl-3,4,5,6-tetrachlorophthalic acid,

4- (2,6-dibromo-1H-indol-3-yl) butyric acid, (4-bromobenzoylamino) acetic acid, diethylphosphonobutanoic acid,

4-aminobenzylsulfonic acid, N-benzoyl-8-hydroxy-2-naphthylamino-6-sulfonic acid,

6-dimethylphenoxyacetic acid, p-hydroxyhippuric acid,

N- [3- (trifluoromethyl) benzoyl] glycine, (2-phenoxyacetylamino) acetic acid,

8-methylnonanoic acid,

3- (3-methoxyphenyl) -2-methylacrylic acid,

2- (2,4-dibromophenoxy) propionic acid,

4-nitrosalicylic acid,

4- (3- (4-acetylphenyl) propyl) benzoic acid, (S) - (-) - 2-acetoxypropionic acid, · · ····

5- (phenylazo) salicylic acid,

5-carboxydehydroacetic acid, dimethyldianilinoterephthalic acid, phenylcyclohexyloxyacetic acid,

3.4- dichlorophenoxyacetic acid,

N- (2,6-diisopropylphenyl-carbamoylmethyl) iminodiacetic acid,

3- (4-n-propylbenzoyl) propionic acid, trans-3-hexenoic acid,

Ι-β-aminoadipic acid,

3- (4-chlorobenzylthio) thiophene-2-carboxylic acid,

3- (1,1,2,2-tetrafluoroethoxy) benzoic acid,

5-acetyl-4-hydroxy-3-methoxyfuran-2-carboxylic acid,

2,4-dihydroxy-5- (isobutylthio) benzenesulfonic acid,

3-acetoxycinnamic acid,

1-amino-2- (3-indolyl) ethanephosphonic acid,

2-fluoro-4-propoxybenzoic acid,

3- (4-chlorobenzoyl) -2- (4-isopropylphenyl) propionic acid,

2-acetyl-3,6-dimethylbenzoic acid,

2 ', 5'-dichlorosuccinanilic acid,

2-hydroxy-3 (S) - (N-tert-boc-amino) heptanoic acid, (-) - N- (phenylsulfonyl) glutamic acid, (Z-styrylthio) acetic acid, gamma-D-glutamylaminomethylsulfonic acid, dodecyloxyacetic acid acid,

4 '- (methylthio) -3,4,5,6-tetrachlorophthalic acid, α-methyl-2- (methylthio) -5-nitro-cinnamic acid,

1- (p-tolyl) -1-cyclopropanecarboxylic acid,

3- (hexadecylsulfonamido) propionic acid, (2S) -α-ethylglutamic acid, ethylene glycol bis (4-carboxyphenyl) ether, (+) - N-benzoylglutamic acid, α-ketovaleric acid,

2,3-diacetoxy-N- (1-naphthalen-1-ylethyl) succinamic acid,

5-methyl-1H- (1,2,3) triazole-4-carboxylic acid, dipivaloyl-D-tartaric acid,

3- (4-benzyloxy-3-methoxyphenyl) propynoic acid,

1- (4-bromobenzoyl) piperazine-2,3-dicarboxylic acid,

D, L-cyclopentylmandelic acid,

1- (4'-Sulfophenyl) -3-methyl-5-pyrazolone

2 ', 5'-dichloroglutaranilic acid, perfluoropentanoic acid,

4-hydroxymethyl-3-pyridinecarboxylic acid, n-boc-aminoheptanoic acid,

2.3.5- trichlorobenzoic acid,

2,2-dimethylsuccinic acid, benzoic acid,

D-isoascorbic acid,

D, L-phenylmercapturic acid, N-fmoc-1-aspartic acid β-benzyl ester,

2-chloro-4,5-difluorobenzoic acid, glyoxylic acid,

9-methyl-9H-fluorene-2-carboxylic acid, (2,3,4,5,6-pentahydroxyhexanoylamino) acetic acid,

4- (hexadecylthio) benzoic acid,

3- (5-hydroxy-4-methoxy-2-nitrophenyl) acrylic acid, trifluorothiol acetic acid,

N-formyl-D, L-2-amino-N-butyric acid,

4-ketopimelic acid,

3.4.5- trimethoxycinnamic acid,

2,5-dibromo-3,6-dichloro-terephthalic acid,

1-fluorenecarboxylic acid,

2- (2-chloro-1,1,2-trifluoroethylthio) benzoic acid,

11- (5-azido-1-naphthoxy) undecanoic acid,

2- (2,5-dimethoxybenzyl) benzoic acid,

3,8-dioxatricyclo (5,1,0,0 (2,4)) octane-5,6-dicarboxylic acid

acid,

2-cyclopentylhexanoic acid,

2- [4- (2,2-diethoxycarbonyl) -2,5-dimethoxybenzyl (malonic acid,

2-methyl-2-nonnoic acid, (4,4-dimethyl-3-oxocyclohexyl (acetic acid,

2-Methoxycarbonyl-5-methoxybenzoic acid, trans-4-hydroxy-4- (4-nitrophenyl) -2-butenoic acid,

3- (2,6-diethylphenylcarbamoyl (acrylic acid,

2- [2- (3-methoxyphenyl (acetylamino) -3-methylbutyric acid),

11,12-epoxy- (5Z, 8Z, 14Z) -icosatrienoic acid,

2-bromobutyric acid, phthalyl-D, L-glutamic acid,

4-nitro-2- (3-nitrophenoxy (benzoic acid,

4-methoxycyclohexanecarboxylic acid,

3-methyl-3- (3,4,5-trimethylphenyl (butyric acid,

2- (difluoromethoxy (benzoic acid,

N- (3,4-dichlorophenyl) malonamic acid, thiodisuccinic acid,

4-chlorophenylacetic acid,

5-chlorobenzo (b) thiophene-3-acetic acid,

4-benzyloxy-3-methoxycinnamic acid,

2-propylnonanoic acid, indazole-3-carboxylic acid, anthraquinone-2-carboxylic acid, boc-6-aminocaproic acid, fmoc-hexahydropyridine-4-carboxylic acid,

4 - [(2-hydroxy-5-methoxybenzylidene) amino (benzoic acid, hydroferulic acid, pth-D, L-cysteic acid, (+/-) - cis-1-amino-1-carboxycyclopentane-3-acetic acid,

1-Naphthol-3,6,8-trisulfonic acid,

3- (4-chlorobenzoyl) -2- (4-fluorophenyl) (propionic acid,

- 70 N-carbaitioyl-D, L-alanine, cis-hexahydro-N- (2-phenethyl) phthalamic acid, immobilized iminodiacetic acid, trans-2- (4-fluorobenzoyl) -1-cyclohexanecarboxylic acid,

2-pyridylacrylic acid,

4-tert-butyl-3-nitrobenzoic acid,

3- (4-Methyl-3-nitrophenylureido) benzoic acid,

2-Benzhydrylidene succinic acid

3-pentanoic acid,

2- (1-indenylidene) glycolic acid,

ΙΗ, ΙΗ, 2H, 2H-perfluordecanoic acid,

4- (3-chloro-1,4-dioxo-1,4-dihydronaphthalen-2-ylamino) butyric acid,

3- (3-bromo-4-hydroxyphenyl) propionic acid,

2-chloro-6-methylphenoxyacetic acid, α, β-dibromo-4-nitrohydrinnamic acid, α- (phenylthio) -o-toluic acid, heptacosanoic acid,

3,5-dibromo-2,4-dihydroxybenzoic acid,

5- (9,10-dioxo-9,10-dihydroanthracen-2-yl) penta-2,4-dienoic acid,

9-fluorenone-4-carboxylic acid, α, α, α ', α'-tetramethylheptanedioic acid, (+/-) - trans-2,3-piperidinedicarboxylic acid,

4,5-dichloroisothiazole-3-carboxylic acid,

2-iodophenylacetic acid,

4-iodophenoxyacetic acid,

1-amino-8-naphthol-3,6-disulfonic acid,

4 - [(4-chlorobenzylidene) amino] benzoic acid,

2-Cyano-3-methyl-2-butenoic acid

3 - [(adamantane-1-carbonyl) amino] benzoic acid,

5- (trifluoromethoxy) indole-2-carboxylic acid, meso-2,3-diphenylsuccinic acid,

Cyclopentanecarboxylic acid,

2-Fornylamino-2-phenylpropionic acid, gallic acid,

N- (2-butylsulfanylbenzothiazol-6-yl) succinamic acid,

3-nitro-α-phenylcinnamic acid,

4-Methoxyoxyphenoxyacetic acid

4-Hexanoic acid

5- (4-methoxybenzoyl) thiophene-2-acetic acid,

2-Methyl-5-phenylfuran-3-carboxylic acid

3 - [(5-nitro-1,3-dioxo-1,3-dihydroisoindol-2-ylmethyl) amino] benzoic acid,

N-ethyl-D-aspartic acid, D, L-p-hydroxycaproic acid,

3,5-dimethyl-2-iodobenzoic acid,

2-ethyl-2-methylhexanoic acid, diglycolic acid, glutaconic acid,

3-chloro-4-fluorobenzoic acid, tricyclo (8,2,2,2 (4,7)) hexadeca-1 (13), 4,6,10 (14), 11,15-hexaene-5-carboxylic acid ,

5-iodoanilic acid,

3-methylcinnamic acid,

2-bromooctanoic acid,

2-bromo-6-methoxybenzoic acid, boc-8-aminocaprylic acid,

1,8-naphthyridine-2-carboxylic acid,

3- (4-sulfamoylphenyl) acrylic acid,

2- (3- (2,4-xylyl) ureido {benzoic acid,

3- (3-thienyl) acrylic acid,

2,2-dimethyl-3-hydroxypropionic acid,

N, N-bis ((R) - (+) - 1-phenethyl) phthalamic acid,

1,3-phenylenediacrylic acid,

2- (2- (2-hydroxy-1-naphthoyl) vinyl {benzoic acid) ·

- 72 (1H) - erythro-4-methylglutamic acid,

7- (3-chloro-2-thienyl) -2,4-dimethylpyrrolo (1,2-a) pyrimidine-8-carboxylic acid,

4-chloro-3-iodobenzoic acid,

2- [2-chloro - [(4-fluorophenyl) sulfonyl / anilino] acetic acid, glycyl-1-aspartic acid,

5 - [(4-chlorophenyl) sulfanyl] -1,2,3-thiadiazole-4-carboxylic acid,

2-nitrobenzenesulfonic acid,

3- (1,1,4,6,7-Pentamethyl-5-indanyl) acrylic acid

2,5-dimethylphenoxyacetic acid, hypophosphoric acid, pyromellitic acid,

2-Methyl-2-phenylbutyric acid

3-hydroxy-2,4,6-tribromobenzoic acid,

1- (2-fluorophenyl) cyclohexanecarboxylic acid,

3.4-dimethylhippuric acid,

6,8-dichloro-2-hydroxy-4-quinolinecarboxylic acid,

Ν, Ν '- (1,3-phenylene) dimaleinamic acid,

1-butanesulfonic acid,

3-difluoric cinnamic acid, triphenylsilyl carboxylic acid, ethylphosphonic acid, chlorogenic acid, (IR, 2S, 3R) -1-hydroxy-3-hydroxymethyl-1,2,3,4-tetrahydronaphthalene-2-carboxylic acid, adamantan-2-ylacetic acid acid, α-methyl-2-furanacrylic acid,

4-oxatetradecanoic acid,

2 ', 5'-dimethyl-3,4,5,6-tetrachlorophthalic acid,

4,4-diphenyl-3-butenoic acid,

4-anisidine-2,5-disulfonic acid,

2 - [(3-allyl-2-hydroxybenzylidene) amino] -3- (1H-imidazol-4-yl) -

• propionic acid, benzylphosphonic acid, methanesulfonylacetic acid, • propionic acid, benzylphosphonic acid, methanesulfonylacetic acid,

4,4-bis- (4-hydroxy-3-nitrophenyl) valeric acid, acrylic acid,

1- (4-chlorophenyl) ethyliminoxyacetic acid,

2- (2-chloro-1,1,2-trifluoroethoxy) benzoic acid, cis-2- (p-chlorobenzoyl) -1-cyclohexanecarboxylic acid,

3-acetamidobenzoic acid,

2.4- bxs (trifluoromethyl) benzoic acid,

4-fluoro cinnamic acid, n-acetyl-D, L-homotryptophan, benzofurazan-5-carboxylic acid, cis-N- (5-chloro-2-methoxyphenyl) hexahydrophthalamic acid,

3- (3,4-dichlorophenyl) -2-methylacrylic acid,

4-chloro-2-iodobenzoic acid, n-phenylanthranilic acid, (+/-) - trans-2,5-piperidinedicarboxylic acid,

4-cyano-3,5-dimethyl-1H-pyrrole-2-carboxylic acid,

3 '- (trifluoromethyl) -1,2,3,6-tetrahydrophthalanilic acid,

3-anthracen-2-ylpropionic acid,

N, N '- (1,2-phenylene) dimaleinamic acid,

(R) - (-) - 4-Methylglutaric acid 1-monomethyl ester,

3-oxo-2-phenyl-1-cyclopentanecarboxylic acid,

1-homocysteinsulfinic acid,

2- (ortho-tolyl) heptanoic acid,

1- (-) - threo-3-hydroxyaspartic acid,

4-chloro-3-sulfamoylbenzoic acid,

3- (4-chlorophenyl) -3-isobutyrylaminopropionic acid, decanoic acid,

2-chloroethylphosphonic acid, β-d-aspartylaminomethylphosphonic acid,

3-n-propylglutaric acid, α-acetamidicinnamic acid, epsilon-N-oxalyl-D-α, epsilon-diaminohexanoic acid, d-camphoric acid,

3- (1H-indol-3-yl) -2- (toluene-4-sulfonylamino) propionic acid, α-methoxycinnamic acid, bone acid,

4-oxo-4- (2-oxocyclohexyl) butyric acid,

N- (2-methoxyphenyl) maleic acid,

4-ethoxycarboxy-3,5-dimethoxybenzoic acid,

2-Fluoren-9-ylidenemethylbenzoic acid

4-dipropylamino-3,5-dinitrobenzoic acid,

7,10,13,16,19-docosapentaenoic acid,

4- (3-chloro-5-trifluoromethyl-2-pyridyl) -4-phenylsulfonylbutanoic acid,

12- [N-methyl-N- (7-nitrobenz-2-oxa-1,3-diazol-4-yl)] aminododecanoic acid,

3,4,5-triethoxybenzoic acid,

2-Methoxyoxypropionic acid, (R) - (+) - 2-methylglutaric acid, boc-10-aminodecanoic acid, cis-aconitic acid,

N (a) -fmoc-N (β) -alloc-1-2,3-diaminopropionic acid,

3- (4-butoxybenzoylamino) benzoic acid,

4,6-Dihydroxy-5-methanesulfonyl-1-ph-3α, 6-methanoazulene-3-

-carboxylic acid,

2-bromangelic acid, dodecanedioic acid,

2,3,4-trifluorophenylacetic acid, (3-methoxystyryl) glyoxylic acid,

4- [[(3-hydroxy-2-naphthalenyl) carbonyl] amino] benzoic acid,

2-Benzyl-3-phenylpropionic acid

2-hydroxydodecanoic acid, · · «44 · ·

C · ···· · ·

2,3-dibromo-2-methylpropionic acid,

8-hydroxy-1-naphthylamino-4,6-disulfonic acid,

3.4- dihydroxyphenylacetic acid,

2,5-dimethyl-4- (ethoxycarbonyl) -3-pyroslizic acid,

4 - [(5-bromo-1,3-dioxo-1,3-dihydroisoindol-2-ylmethyl) amino] benzoic acid,

N-carbobenzyloxy-2-methylalanine, (3,4-dichlorobenzoylamino) acetic acid,

5-tert-butyl-2-pyroslizic acid,

2-hydroxy-3 (S) - (N-tert-boc-amino) hexanoic acid, cyclohexanepentanoic acid,

2'-nitrophthalanilic acid,

5-methoxy-3-methylphthalic acid, ricinlaidic acid,

2-oxo-6-pentyl-2H-pyran-3-carboxylic acid,

2-carboxyamino-3- (2-hydroxyphenyl) acrylic acid,

2-Acetamido-5-nitrobenzoic acid

3- (N-phenylcarbamoyl) -5-norbornene-2-carboxylic acid, D, L-mandelic acid,

3-fluoroanthen-1-ylacrylic acid,

2- (4-bromophenyl) -3- (4-chlorobenzoyl) propionic acid,

3-methyl-2-pyrosylic acid, (2-methylphenoxy) acetic acid, (4-methanesulfonyloxy-3-methoxyphenyl) acetic acid,

2-hydroxy-3-isopropyl-6-methylbenzoic acid,

4- (5,6,7,8-tetrahydronaphthalen-2-yl) butyric acid,

3-Benzoylacrylic acid

4-ethoxybenzoic acid, (4-hydroxy-3-methoxyphenyl) oxoacetic acid,

2 - [(5-bromo-1,3-dioxo-1,3-dihydroisoindol-2-ylmethyl) amino] benzoic acid,

3- [[(1-acetyl-2,3-dihydro- (1H) -indol-7-yl) amino] carbonyl] propanoic acid;

5-methyl-4-oxohexanoic acid, (8-ho-3-meo-1,5,9,9-tetra-me-4,12-dioxobenzocyclodecen-2-ylidene) acetic acid,

1- (4-fluoroanilino) -6-methyl-4-oxo-1,4-dihydro-3-pyridinecarboxylic acid,

N-α- (9-fluorenylmethyloxycarbonyl) - (3S) -1,2,3,4-tetrahydroisoquinoline-7-hydroxy-3-carboxylic acid,

2 - [(adamantane-1-carbonyl) amino] -3- (1H-indol-3-yl) propionic acid,

N-cbz-D, L-aspartic acid, methoxycarbonylmercaptosuccinic acid,

3-bromo-4,5-dimethoxybenzoic acid,

3.4- dichloradipic acid,

3'-bromophthalanilic acid,

6-methyl-3-pyridylacetic acid,

3,5,6-trichloroctafluorohexanoic acid,

3- [5- (4-chlorophenyl) -2-furyl] acrylic acid, epsilon-maleimido-caproic acid,

6- (acetoxymethyl) -3-methyl-3-cyclohexene-1-carboxylic acid, phenylsulfonylacetic acid,

2-methyl-2-phenyloctanoic acid,

2.5- dibromadipic acid,

1,1-cyclohexanedicarboxylic acid,

2-methyl-bicyclo (2,2,1) hept-5-ene-2-carboxylic acid,

2'-methyl-5'-nitromaleanilic acid,

2- [benzyl (toluene-4-sulfonyl) amino] benzoic acid, (carboxyphenylmethylsulfanyl) phenylacetic acid, indolizine-2-carboxylic acid, α-methylhydrinnamic acid,

10-methylundecanoic acid, α-cyano-β-methyl-2- (methylthio) cinnamic acid,

3-Hydroxypropanesulfonic acid, * * * * * * * * * * hydroxy hydroxy hydroxy hydroxy hydroxy hydroxy hydroxy hydroxy hydroxy hydroxy ··

2 - [[2- (2,4-dichlorophenyl) hydrazino / carbonyl] benzoic acid,

5-Iodoric acid, p-bromo-phenoxyacetic acid,

2-hexinoic acid,

2'-chloro-5 '- (trifluoromethyl) glutaranilic acid,

5-methyl-2-phenylimidazo (1,2-a) pyridine-3-carboxylic acid,

4- (3-chloropropoxy) benzoic acid,

4- (4,4-dimethyl-2-oxocyclohexyl) butyric acid,

2-methyl-5-nitro-3-pyroslizic acid, N-methyl-D-aspartic acid,

4-hydroxyphenoxyacetic acid, chloroacetic acid,

4'-nitroglutaranilic acid, (2S) -α-methylglutamic acid,

9 (S) -hydroxyoctadeca-10E, 12Z-dienoic acid,

2-sulfinobenzoic acid,

3- (difluoromethoxy) phenylacetic acid,

10-oxopalmitic acid,

3-benzamidobenzoic acid, hippuric acid, phenyl-s acid,

2,7-di-tert-butyl-9,9-dimethyl-4,5-xanthenedicarboxylic acid,

5-chloro-2-nitro-cinnamic acid, delta-N-oxalyl-D-a, delta-diaminopentanoic acid,

4'-pentylbiphenyl-4-carboxylic acid,

N- (1-naphthyl) glutaramic acid,

3'-Fluorophthalanilic acid, tricosanoic acid,

4-chloro-2,5-difluorobenzoic acid,

16-phenylhexadecanoic acid,

3 - [(R, S) -2-carboxypiperazin-4-yl] propyl-1-phosphonic acid,

2-Naphthalen-2-yl-1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxylic acid,

2-pyridin-2-ylquinoline-4-carboxylic acid,

2- (4-methylbenzoylamino) -3- (4-nitrophenyl) acrylic acid, dihydroxychicagic acid,

4-fluoro-3- (trifluoromethyl) phenylacetic acid,

2-Tolidine-3,3-disulfonic acid,

2 - [(2-hydroxy-5-methoxybenzylidene) amino] benzoic acid, 3 ', 4'-dichloroglutaranilic acid,

4- (3-dodecanoyl-2-thioureido) benzoic acid,

4-hydroxycyclohexanecarboxylic acid,

3,5-dihydroxy-4-methoxybenzoic acid, (S) - (t) -citramalic acid,

2-naphthylamino-3,6,8-trisulfonic acid,

3,5-diiodo-4-hydroxyphenylpropionic acid, (S) - (-) - 2-bromo-3-methylbutanoic acid, (R) - (-) - 2-phenylbutyric acid, fluorene-4-carboxylic acid,

N- (2-carboxyphenyl) glycine

2-methoxy-3,6-dichlorobenzoic acid,

7-bromkynurenic acid,

2-naphthylamino-3,6,8-trisulfonic acid, n-tert-butylsuccinamic acid, (4-ethyl-3,5-dimethyl-1H-pyrrol-2-yl) acetic acid, cyclopropylacetic acid,

5-chlorotetrazole-1-acetic acid, trans-2-hexenoic acid,

4-chloro-2-fluoro-cinnamic acid, terephthaloyl-bisacetic acid,

5- [4- (4-carboxybutyryl) phenyl] pentanoic acid,

3-bromo-4-methoxybenzoic acid, trans, trans-9-cyano-2-decalinecarboxylic acid, N- (5-chloro-2-methylphenyl) phthalamic acid,

1- (S) - (+) - endo-bromocapro-10-sulfonic acid,

2-cyano-3- (4-methoxyphenyl (acrylic acid, fmoc-1-amino-1-cyclohexanecarboxylic acid),

3- (3,4-dimethoxy-2-pyridyl (acrylic acid,

3-Methoxy-4-methylbenzoic acid

4- (2-phenylethenesulfonylamino) (butyric acid,

4-hydroxy-6- (trifluoromethoxy) quinoline-3-carboxylic acid,

3-hydroxymyristic acid,

3-methylthio-4-oxo-4,5,6,7-tetrahydrobenzo (c) thiophene-1-carboxylic acid,

2-Oxo-4-phenylpyrrolidine-3-carboxylic acid

3-chlorvaleric acid,

D - (-) - S-acetyl-β-mercaptoisobutyric acid, cis-parinaric acid,

2- (2,4-Diphenylthiazol-5-yl) acetic acid

3-acetylamino-3- (4-methoxyphenyl (propionic acid, (2S, 1'R, 2'S)) -2- (carboxycyclopropyl (glycine,

3- [phenyl (toluene-4-sulfonyl) amino (butyric acid,

4-chloro-α, β-diphenylacrylic acid,

5-chloro-2,4-dinitrobenzoic acid, kucuric acid,

2-decyldodecanoic acid, (R) -4-methylthiomandelic acid,

2- (9H-fluoren-2-ylmethyl (benzoic acid, tricyclo (12,2,2,2 (6,9)) icosa-1 (17), 6 (20), 7,9 (19), 14 ( 18), 15-hexaenylacetic acid,

4- [2- (methylsulfonamido) ethoxy] meta-anisic acid, fmoc-D-pipecolic acid, tiglic acid, fmoc-α, β-γβ1ιγάΓθ-2-3ΐηίηοιηέεβ1ηή acid,

N, N-diphenyloxalamic acid, dehydrothio-p-toluidine-7-sulfonic acid,

2-diazo-1-naphthol-4-sulfonic acid,

2-chloro-6-fluoro-cinnamic acid,

2-ethyldecanoic acid, terebic acid,

1-Benzoylpiperazine-2,3-dicarboxylic acid

3,5-bis (trifluoromethyl) hydro-cinnamic acid,

2 ', 4'-dimethoxymaleanilic acid,

5-amino-m-toluic acid,

2-chloro-α-methylcinnamic acid,

1,4-cyclohexanedicarboxylic acid, gamma-maleimide butyric acid, methylenediphosphonic acid,

N- (3-chlorophenyl) maleic acid, fmoc-2-aminobenzoic acid,

2 ', 4'-dichlorophthalic acid, o-sulfobenzoic acid, ethylenediaminotetraacetic acid,

1,4-benzodioxane-5-carboxylic acid, gamma-oxo-1-pyrene-butyric acid, n-fmoc- (2S, 3S) -3-amino-2-hydroxy-4-phenylbutyric acid,

2,4-dimethylbenzoic acid,

3-Oxo-1-phenyl-1-indaneacetic acid

2 - [[2- (2,4-difluorophenyl) hydrazino / carbonyl] benzoic acid,

(R) - (+) - 3-methylsuccinic acid 1-monomethyl ester,

2-chloromethylsulfanylbenzoic acid,

D, L-2-aminosubric acid,

4- (6-butoxynaphthalen-2-yl) butyric acid,

3- (2 ', 4'-difluorobenzoyl) propionic acid,

3'-nitromaleanilic acid,

2- (4-cyanophenoxy) -2-methylpropionic acid, hexahydrophthalic acid,

5.6-diphenyl-2,3-pyrazinedicarboxylic acid,

5- (4-carboxybenzoyl) benzene-1,2,4-tricarboxylic acid, (3R, 4S) - (-) - n-boc-4-amino-3-hydroxy-6-methylheptanoic acid,

3.4-dimethoxy-α-mercaptinnamic acid,

1-adamyltylmalonic acid,

3- (trifluoromethyl) butyric acid,

5-fluoro-2-nitrobenzoic acid,

2,3-dimethoxybenzoic acid,

3,5-diiodo-p-hydroxyphenylpyruvic acid,

4- (4-acetylphenyl) butyric acid, dicyclohexylacetic acid,

9-fluoro-1-oxo-ΙΗ, ΙΗ-pyrido (3,2,1-i, j) quinoline-2-carboxylic acid,

3-methyl-3-phenylglutaric acid, boc-D-2-aminoadipic acid,

7-amino-4-methyl-3-coumaronylacetic acid, homogentisic acid, coffee acid,

2-dimethylglutaric acid,

2- (4-chlorophenyl) -3- (3,4-dichlorobenzoyl) propionic acid,

4-pentinoic acid, (R) - (-) - 2-phenylpropionic acid, (2-propionylphenoxy) acetic acid,

N, N-diethyl-3,6-difluorophthalamic acid,

10,12-octadecadiic acid,

2-hydroxyphenylacetic acid,

2 ', 3'-dichlorosuccinanilic acid, sulfo-gamma-acid,

2- (2,4-dichlorophenoxy) propionic acid, (2-isopropylphenyl) phosphonic acid, cis-2'-ethylhexahydrophthalanic acid,

3-pentenoic acid,

3-hydroxy-3-methyl-N-valeric acid,

6-chloro-2- (4-methoxyphenylamino) -3-nitrobenzoic acid,

5,7-dichloro-4-hydroxyquinoline-3-carboxylic acid,

2- (2,5-dichlorophenylcarbamoyl) cyclohexanecarboxylic acid, atromic acid, dibenzofuran-2-sulfonic acid,

4-fluoro-3- (trifluoromethyl (benzoic acid, uracil-5-carboxylic acid,

2,3,6-trifluorophenylacetic acid,

1,3-dioxo-2-o-tolyl-2,3-dihydro-1H-isoindole-5-carboxylic acid,

4-chloro-p-methylhydrinnamic acid,

1- (meta-tolyl) -1-cyclopentanecarboxylic acid,

3-chlorophenoxyacetic acid,

2-chloro-5-methylbenzoic acid,

3- (phenylsulfonyl (propionic acid, angelic acid,

2-hydroxypalmitic acid,

4-methylcatechol-o, o-diacetic acid,

4- (6-methoxynaphthalen-1-yl) butyric acid,

2,4-dihydroxypyridine-5-carboxylic acid,

1-methionyl-1-glutamic acid,

3-methoxycarbonyl-1-methyl-1H-indole-2-carboxylic acid,

4- (3,4,5-trimethoxybenzoyl (butyric acid,

2- (p-anisyl) -3-phenylsuccinic acid,

2-methylsulfonylbenzoic acid,

15-methylheptadecanoic acid,

2-cyclohexylpropionic acid,

4- [phenyl (toluene-4-sulfonyl (amino) butyric acid, vinylacetic acid,

1,3-cyclohexanedicarboxylic acid,

3-Acetamino-6-bromobenzoic acid

2.3- dibenzylidene succinic acid,

2 ', 4', 6'-trimethylsuccinanilic acid,

N-phenylmaleinamic acid, (R) - (-) - 3-hydroxytetradecanoic acid, boc-1-glutamic acid, · · · ···· · · ···· · ··· ·······························

N-furfurylglutaramic acid, chromone-2-carboxylic acid,

2,6-bis- (1-trimethylsilanylvinyl) benzoic acid,

5-tert-butylisophthalic acid,

3- (3,4-dimethoxyphenyl) -2- (2,4-dimethoxyphenyl) acrylic acid,

N, N'-diglycylethylenediamino-N, N, N ', N'-tetraacetic acid,

5- (3-nitrophenyl) -2-pyroslizic acid,

2-methyl-1,8-naphthyridine-3-carboxylic acid,

5-methylfuran-3-carboxylic acid,

7-bromoheptanoic acid,

1-adamantanacetic acid, croconic acid,

2-hydroxytricosanoic acid, azelaic acid,

3-Methylnaphthalene-2-carboxylic acid

3- (hexadecylthio) benzoic acid,

11,14-icosadienoic acid, (+/-) - trans-epoxy antaric acid,

4'-bromo-3'-methyl-1,2,3,6-tetrahydrophthalanilic acid, (1S) - C -) - (1-amino-2-methylpropyl) phosphonic acid,

4- (methylthio) benzoic acid,

N- (4-nitrophenyl) iso (hexahydropyridine-4-carboxylic acid), o-anisic acid, benzophenone-4,4'-dicarboxylic acid, mono-methylsuccinate,

3-methoxy-9-oxo-8,9-dihydro-7H-benzocycloheptene-6-carboxylic acid,

5- (tert-butyl) -4-hydroxy-m-toluylic acid,

3- (5-phenyl-2,5-dihydro-2-furyl) acrylic acid,

16-bromo-hexadecanoic acid, cis-1,2-cyclopropanedioic acid, φφφφ · ·

* Φ · ΦΦΦ · · · * · * · · · • · φ · φ · · ·

2- (1-indolylcarbonyl) -3,4,5,6-tetrachlorobenzoic acid, (2-thioxobenzothiazol-3-yl) acetic acid,

4'-sulfamoylphthalanilic acid, ophthalmic acid, phthalic acid, gamma-linolenic acid,

1- (4-chlorophenyl) -1-cyclopropanecarboxylic acid, (R, S) -α-methyl-4-carboxyphenylglycine,

5- (2-nitrovinyl) benzoic acid,

5- (3-chlorophenyl) -2,3-dihydro-1H-pyrrolizine-6,7-dicarboxylic acid,

D, L-gamma-carboxyglutamic acid,

N-tert-butyl-3,4,5,6-tetrachlorophthalamic acid,

2-fluoro-4-methoxybenzoic acid,

3,5-dichlorosalicylic acid, bis (p-tolyl) acetic acid,

2- (4-hydroxyphenyl) isovaleric acid,

3- (cyanomethylthio) thiophene-2-carboxylic acid,

3-methylindene-2-carboxylic acid,

13-methyltetradecanoic acid,

2-propyloctanoic acid, hexahydro-N- [4- (methylthio) phenyl] phthalamic acid,

8-hydroxy-2-methylquinoline-5-sulfonic acid,

4- [2,4-bis- (2,2-dimethylpropyl) phenoxy] butyric acid,

4-chloroindole acetic acid,

2,3-dihydrobenzofuranoacetic acid,

5-octadecyloxylisophthalic acid,

4- (2-butylcarbamoylacetylamino) benzoic acid,

4-isopropylcyclohex-4-ene-1,2-dicarboxylic acid, fmoc-1-aspartic acid α-tert-butyl ester, N-α-fmoc-N-gamma-boc-1-diaminobutyric acid,

9-methyl-9H-fluorene-3-carboxylic acid, pentafluorobenzoic acid,

3-butene-1,2,3-tricarboxylic acid,

4-dibenzothiophenecarboxylic acid,

2,2-dimethylbutyric acid, m-toluic acid,

4- (4-Hydroxybenzenesulfonyl) benzoic acid,

2-dodecenoic acid,

4- (1- (2-mercapto-4,5-dihydro) imidazolo] benzoic acid,

5-chlorobicyclo (2,2,1] hept-2-ene-5-endo-carboxylic acid, cis-4- (phosphonomethyl) piperidine-2-carboxylic acid,

2-iodo-3-methylbenzoic acid,

2- (4-ethylphenyl) -1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxylic acid, dimethylmalonic acid, cumenesulfonic acid,

N-phthaloyl-gly-α-aminoisobutyric acid, tecloftalam,

3-benzoylamino-N-hexylcarbamoylmethylsuccinamic acid,

6,8-dibromocoumarin-3-carboxylic acid, boc-D-homophenylalanine,

2-fluorosuccinanilic acid,

2- (4-nitrophenyl) propionic acid,

4-trans-phenylcyclohexane-cis-1,2-dicarboxylic acid, o-sulfobenzaldehyde,

4-Bromocinnamic acid,

4- (2- (4-ethoxy-benzoylamino) -3-phenylacryloylamino) Butyric acid,

5-sulfosalicylic acid,

3'-Fluoraleanilic acid,

4- (tert-butoxy) benzoic acid,

2- (4- (4-cyanophenoxy) -ph) -1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxylic acid, cis-N- (4-acetylphenyl) hexahydrophthalamic acid, (S) -2-methyloctanoic acid,

• ·· · · · · · ·

9-hydroxyfluorene-9-carboxylic acid,

2-methyl-1-naphthylacetic acid,

2,4-dihydroxy-3,6-dimethylbenzoic acid,

2,2,5,7-tetramethylindan-1-one-4-carboxylic acid,

5- (dimethylaminosulfonyl) -2,3-dihydro-gamma-oxo-1- (1H) -indolbutanoic acid,

4-chlorophenylsulfonylacetic acid,

4- [2- (propane-2-sulfonyl) acetylamino (benzoic acid,

2- [2- (2-methoxyethoxy) ethoxy] acetic acid,

3,4,5-trichloro-2-thiophenecarboxylic acid,

4-carboxybenzaldehyde,

N-ethyl-N- (p-toluenesulfonyl) anthranilic acid, (S) - (+) - 2-hydroxy-2-phenylpropionic acid,

2-methoxycarbonyl-4,6-dimethoxybenzoic acid, Ν-α-Z-glycyl-1-glutamic acid,

4- (2-carbamoylphenylimino) -2,3-dichloro-2-butenoic acid,

4-methyl-2-heptenic acid,

2-carboxy-α-oxobenzeneacetic acid, (+/-) - 1-aminocyclopentane-cis-1,3-dicarboxylic acid, (-) - 1,2,3-trimethyl-2-cyclopentenacrylic acid,

2 ', 4'-difluorglutaranilic acid,

3-phenyl-1,3,5-pentanetricarboxylic acid, phthalylsulfacetamide,

4- (ethoxycarbonylmethoxy) -1-hydroxy-2-naphthoic acid,

2- (2-cyanophenylthio) benzoic acid,

3-chloro-5-iodobenzoic acid,

2- [3- (2,2,2-trichloro-1-isobutyrylaminoethyl) thioureido (benzoic acid,

10,12-nonacosadiic acid,

2-hydroxytetracosanoic acid,

2-phthalimidobenzoic acid,

4'-ethoxyphthalanilic acid,

4-iodoacetamidosalicylic acid,

4-Benzyl ester of N- (tert-butoxycarbonyl) -1-aspartic acid,

4-benzoylbenzoic acid,

4'-bromo-1,2,3,6-tetrahydrophthalanilic acid,

1-naphthylmethylphosphonic acid,

3-iodo-4-methylbenzoic acid, (S) -3-hydroxy-3-phenylpropanoic acid, (S) -2-ethyloctanoic acid,

N- (2-methyl-4-nitrophenyl) succinamic acid,

3-aminopropylphosphonic acid, (+) - 4'-chlorotartranilic acid, boc- (3S, 4S) -4-amino-3-hydroxy-6-methylheptanoic acid, D, Lp-hydroxylauric acid, (+/-) - 2 -hydroxypentadecanoic acid,

N-methylmaleinamic acid,

3-methylhippuric acid,

3-nitrocinnamic acid, mesaconic acid,

3-hydroxybenzoic acid,

2-bromo-4,5-dimethoxyhydricinnamic acid,

L-alanyl-L-aspartic acid,

4-Benzoyloxybenzoic acid

N-fmoc-L-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid,

3,4-diacetoxybenzoic acid,

1,2-dihydroxycyclobutanecarboxylic acid,

2 ', 3'-dimethylmaleanilic acid, 1-methyl-1H-indazole-3-carboxylic acid,

22-tricosenoic acid,

N-tert-boc-7-aminoheptanoic acid,

5-nitro-2- (phenylthio) benzenesulinic acid,

1- (3,4-dimethoxy-ph) -4-hydroxy-5,6,7-trimethoxy-naphthalene-2-carboxylic acid,

3- (3,4-dimethoxyphenyl) -3- (3,4,5-trimethoxyphenyl) propionic acid

acid, di (cyclohexyl) dithiophosphoric acid,

4-Methylphenoxyacetic acid

3- (trifluoromethyl) cinnamic acid, trimethylpyruvic acid,

N- (benzyl) -3,4,5,6-tetrachlorophthalamic acid,

2-ethyl-3- (4-nitrophenyl) acrylic acid,

5- (3-chloro-5-trifluoromethyl-2-pyridylmethyl) thiophene-2-sulfonic acid, boc-5-aminovaleric acid,

3- p-tolyloxymethylbenzoic acid,

2-amino-1,5-naphthalenedisulfonic acid,

D, L-α-methoxyphenylacetic acid,

1-cyclopentenecarboxylic acid,

2-Methyl-1-naphthalenecarboxylic acid

2-fluoro-3-methylbenzoic acid, (R) -3-chloro-lactic acid,

2-phenoxybenzoic acid, (-) - 3-pinanecarboxylic acid,

5-methyl-2-pyroslizic acid,

2,3-dibromo-2'-methoxy-3'-nitrosuccinanilic acid, N-boc-L-aspartic acid β-cyclohexyl ester, (1-methylheptyl) phenylphosphinic acid,

3-iodo-4-methoxybenzoic acid, (+) - dimethyl 2,3-o-benzylidene-D-tartrate,

D, L-o-methoxymandelic acid,

2-chloro-para-anisic acid, (2-carboxyphenylimino) diacetic acid, meconic acid,

3-Methyl-1-oxo-1,2-dihydroisoquinoline-4-carboxylic acid

3- (4-Methylsulfanylphenyl) -3-oxopropionic acid

4- (diacetoxymethyl) benzoic acid,

3- [N- (2,5-xylyl) carbamoyl) -5-norbornene-2-carboxylic acid,

3- (4-chlorophenylamino) butyric acid,

3-acenaphthen-5-ylacrylic acid,

2,4-dimethylphenoxyacetic acid,

5.7- dodecadiindioic acid,

3,5-diphenylbenzoic acid, (2S, 4R) -4-methylglutamic acid, nitroterephthalic acid, cis-N-cyclohexylhexahydrophthalamic acid,

5-nitroindole-2-carboxylic acid,

D - (-) - 2-amino-6-phosphonohexanoic acid, (ethylthio) acetic acid,

4'-Brommaleanilic acid,

2- (p-tolylthio) acetic acid, thioacetic acid, (6-tert-butyl-1,1-dimethylindan-4-yl) acetic acid,

3-methyl-1,1-cyclopentanediacetic acid,

2- (carboxy-4-hydroxyphenyl) quinoline-4-carboxylic acid, dnp-L-aspartic acid,

2- (4-ethoxybenzoyl) acrylic acid,

1- (2,5-dichloro-4-sulfophenyl) -5-pyrazolone-3-carboxylic acid,

2- [3- (N'-nonanoylhydrazino) -3-oxopropionylamino] benzoic acid,

3-chloro-2- (toluene-4-sulfonylamino) benzoic acid,

2-Tridecenic acid

4.5.6.7-Tetrafluoro-2,3-dihydro-gamma-oxo-1- (1H) -indolbutanoic acid

3'-bromoglutaranilic acid,

3- (4-fluorobenzoyl) propionic acid,

3- [ac- (5-bromo-1,3-dioxo-1,3-dihydroisoindol-2-ylmethyl) amino] benzoic acid,

5- (chloroacetyl) thiophene-2-acetic acid, 9 · 9 * 9 · 9 · 9 · ··· ·· ··· ··

3- (phenylthio) acrylic acid, o-hydroxyhippuric acid,

4-isopropoxybenzoic acid, (R) - (-) - 2-chloro 3-phenylpropionic acid, 11-icosenoic acid, [(3-chlorophenyl) - (toluene-4-sulfonyl) amino] acetic acid,

4-isothiocyanatobenzenesulfonic acid,

4-chloro-5-nitro-o-toluenesulfonic acid,

2-chlorostearic acid,

3- (3,4-dimethoxyphenyl) propynoic acid,

3- [N- (3-nitrophenyl) carbamoyl] bicyclo (2,2,1) hept-5-ene-2-carboxylic acid, cyclohexylacetic acid,

5-norbornene-2-carboxylic acid, bromomaleic acid,

4-octyloxybenzoic acid, thymoxyacetic acid,

4- (4-chlorobenzenesulfonyl) phthalic acid,

2-difluoro succinic acid,

N-tert-boc-5-cyclohexylstatin, (+/-) - 3-exo-aminoticyclo [2.2.1.0 (2.6)] heptane-3-endo-7-anti-dicarboxylic acid, ( R) - (+) - 2-chlorohexanoic acid,

2- (3,4-dimethoxy-α-methylbenzyl) -6-methoxybenzoic acid, tridecafluoro-2-nonenoic acid,

3-Methyl-2- (ortho-tolyl) hexanoic acid

2-Methyl-7-oxononanoic acid

Ν-α-formyl-L-glutamic acid, (1-aminobutyl) phosphonic acid, exo-3,6-epoxy-1,2,3,6-tetrahydrophthalic acid,

N- (2,5-xylyl) glutaramic acid,

3-amino-2,6-naphthalenedisulfonic acid,

12 (R) —hydroxyicose-5Z, 8Z, 14Z-trienic acid, · · · · · · · · · · · ·, ·, · * ·, · · · · ·· · · ·

3-methyl-2-phenylhexanoic acid,

3-chloro-2,4,6-trimethylbenzoic acid,

6- (4-tert-butylphenyl) -4-oxo-5-hexenoic acid,

N-ethyl-D-glutamic acid,

D, L-tropic acid,

8-methylnon-6-enoic acid, α-chlorophenylacetic acid,

N-octadecylmaleinamic acid,

3- (3,4,5-trimethoxyphenyl (propionic acid,

1,3-dioxo-2-m-tolyl-2,3-dihydro-1H-isoindole-5-carboxylic acid, trans-2-decenoic acid,

3- (4-methylphenyl (propionic acid,

6-Methoxy-1-naphthoic acid

2- (4-acetoxy-3-tert-butylphenoxy) tetradecanoic acid,

2- [2-C1-4- (2-methyl-acryloylamino) phenylcarbamoyl] -3,3-dimethylbutyric acid,

2- [[(2,4-dichlorophenyl) sulfonyl] -3- (trifluoromethyl) anilino] acetic acid,

3-cyclohexenecarboxylic acid,

3-bromo-5-nitrobenzoic acid, bis (2-ethylhexyl (hydrogen phosphate,

3-succinimidopropionic acid,

2- (hydroxyphenylphosphinoyl (benzoic acid,

3- (4-chlorobenzoyl) -2- (4-methylphenyl (propionic acid,

4-bromo-2-chlorobenzoic acid,

2,4- dinitrobenzoic acid,

2,4,6-trimethylbenzenesulfinic acid, cyclopentenylacetic acid,

N-α-acetyl-N-gamma-boc-L-diaminobutyric acid,

3- (4-chlorophenyl) -3-phenylacetylaminopropionic acid,

2,3,4,5-tetrafluorobenzoic acid,

3- [4- (4-fluorobenzyloxy) phenyl] acrylic acid,

1-cyclopentene-1,2-dicarboxylic acid,

3-tert-butyl-5-methylsalicylic acid, pmp (p-mbzl),

3- (4-hydroxy-2-methylcyclohex-2-enyl) propionic acid,

1,3-dicyano-2,2-dimethylcyclobutane-1,3-dicarboxylic acid,

4,5-bis- (4-aminophenoxy) phthalic acid,

9-bromnonanoic acid,

7,7-dimethyl- (5Z, 8Z) -icosadienoic acid,

2,4,6-tri-tert-butylbenzoic acid,

2-Acrylamido-2-methylpropanesulfonic acid

N-methyl-D, L-glutamic acid,

1-hydroxy-4- (methoxycarbonylmethoxy) -2-naphthoic acid,

4-Ethylbenzoic acid

3- [2- (4-ethoxybenzoylamino) -3-phenylacryloylamino {propionic acid,

4- (bromomethyl) benzoic acid,

2-chloro-5-fluorobenzoic acid,

3- (4-chlorophenyl) glutaric acid, bis- (4-methoxyphenyl) phosphinic acid,

18-phenyloctadecanoic acid, (S) - (-) - α-methoxy-α- (trifluoromethyl) phenylacetic acid, (R) - (+) - citric acid,

4- (hydroxymethyl) phenoxyacetic acid,

4,5-dichloro-4,5,5-trifluoropentanoic acid,

4,4-bis-ethoxycarbonyl-heptanedioic acid, (S) - (-) - 2-bromopentanoic acid, 1H-imidazo (4,5-c) pyridine-2-sulfonic acid,

3- (2-hydroxy-5-methylbenzoyl {propionic acid, neononanoic acid,

4-Ho-6,7-dimethoxy-1- (3,4,5-trimethoxyphenyl) naphthalene-2-carboxylic acid,

L-2- (benzyloxycarbonylamino) -4-sulfamoylbutyric acid, cis-L-amino-3- (2-phosphono-1-hydroxyethyl) cyclobutane-1-carboxylic acid,

10-bromodecanoic acid,

3-nitrosalicylic acid,

Z-3- (2-benzimidazolylthio) propenoic acid,

4 '- (ethoxycarbonyl) maleanilic acid,

4'-fluoro-1,2,3,6-tetrahyropthalanilic acid,

6-hydroxycaproic acid, (R) - (-) - α-methoxyphenylacetic acid, dibromomaleic acid,

13-oxooctadecanoic acid,

1-Formyl-3-cyclohexene-1-propionic acid

2- (3,4-dichlorophenylcarbamoyl) cyclohexanecarboxylic acid,

2-methyl-3,3,3-triphenylpropionic acid, (8R, 15S) -dihydroxy- (5Z, 9E, 11Z, 13E) -icosatetraenoic acid,

3- (4-Methylsulfonylbenzoyl) propionic acid

D-glucuronic acid,

4 ', 6-dinitro-2'-methoxyphthalanilic acid,

5,8-dioxo-1,4,4a, 5,8,8a-hexahydro-1-naphthalenecarboxylic acid, hemimellitic acid,

4-Methyl-4-phenylhexanoic acid

N- (4-bromophenyl) glutaranilic acid, monofluorophosphoric acid,

2-ethylbutyric acid, boc- (3-aminomethyl) benzoic acid,

N- (2-pentylsulfanylbenzothiazol-6-yl) succinamic acid,

6-methoxysalicylic acid, α-mercapto-2-methoxy-p-methylcinnamic acid, cis-hexahydro-N- (2,4-dichlorophenyl) phthalamic acid,

2- [3- (1-butyrylamino-2,2,2-trichloroethyl) thioureido] benzoic acid,

2- [3- (N'-heptanoylhydrazino) -3-oxopropionylamino] benzoic acid, - (-) - cis-isoketopinic acid,

2-chloro-4,5-dimethoxybenzoic acid,

2-ethoxycinnamic acid,

5- (2-thienoyl) butyric acid,

3- (2,5-dimethylbenzoyl) propionic acid, pentachloro-cis-2,4-pentadienoic acid,

4 '- (2-hydroxyethyl) glutaranilic acid, N- (4-phenoxyphenyl) malonamic acid, (4-tert-butylphenylsulfanyl) acetic acid,

4- (tert-butyl) cinnamic acid,

N- (p-toluoyl) glycine, anthraquinone disulfonic acid,

4'-bromo-2'-methylglutaranilic acid,

2,2'-dithiodibenzoic acid,

2,4-difluorophenylacetic acid, trifluoromethanesulfonic acid,

4-Ethenyl-3-methyl-5- (methylthio) thiophene-2-carboxylic acid

2-bromohexanoic acid,

5- (2-carboxyphenylaminosulfo) -2-chlorobenzoic acid, p-nitrophenyl-β-D-galacturonide,

2-nitrotoluene-4-sulfonic acid,

3- (4-bromobenzoyl) -2- (4-chlorophenyl) propionic acid,

4-hydroxy-6-methoxy-1- (4-methoxyphenyl) naphthalene-2-carboxylic acid, (2-aminothiazol-4-yl) glyoxylic acid, (+/-) - 1-amino-trans-3-phosphonocyclohexanecarboxylic acid ,

N, N'-ethylenebis (succinamic acid),

2,2-diphenylbutyric acid, (S) -4,9-dihydro-1-methyl-3H-pyrido [3,4-b] indole-3-carboxylic acid,

3,4,5,6-tetrachloro-2 ', 4', 5'-trimethylphthalanilic acid,

5-bromo-2-methylpyrimidine-4-carboxylic acid,

(4-ho-4-ph-1,3,4,5-4H-2-thia-4a, 10-diazaindeno (2,1-a) inden-3-yl) acetic acid, (+/-) - 1-aminocyclohexane-cis-1,2-dicarboxylic acid,

2,3,4,5,6-pentafluoro cinnamic acid,

2- (3-chlorobenzoylamino) -3-hydroxypropionic acid, boc-2-aminoisobutyric acid,

N- (2-thiazolyl) glutaramic acid,

4- [ac- (5-bromo-1,3-dioxo-1,3-dihydroisoindol-2-ylmethyl) amino] benzoic acid,

2-cyano-3- (2-hydroxyphenyl) propionic acid, α- (ortho-tolyl) cyclohexaneacetic acid, [ethylenebis (oxyethylenennitrilo)] tetraacetic acid,

4-anthracen-2-yl-4-oxobutyric acid,

L - (-) - 3-phenyl-lactic acid,

N-chloroacetyldehydroalanine,

3- (4-fluorophenyl) propionic acid, boc-L-α-amino-gamma- (4-methylbenzylmercapto) butyric acid,

8-sulfo-2,4-quinolinedicarboxylic acid, cis-2- (2-thiophenecarbonyl) -1-cyclohexanecarboxylic acid,

5- [4- (3-methoxycarbonylpropyl) phenyl] -5-oxopentanoic acid, cis-hexahydro-N- (2-methylphenyl) phthalamic acid,

4-decyloxy-2-fluorobenzoic acid, fmoc-tranexamic acid,

4- (4-chlorobenzenesulfonyloxy) benzoic acid,

2,3-dibromo-4'-fluorosuccinanilic acid, stearolic acid, boc- (3S, 4S) -4-amino-3-hydroxy-5- (3-indolyl) pentanoic acid, docosahexaenoic acid,

3,5-dibromo-7-methyl-1-adamantanacetic acid,

3- [3- (2,2,2-trichloro-1-isobutyrylaminoethyl) thioureido] benzoic acid,

2-heptinic acid, dnp-D, L-α-aminocaprylic acid, (R) -2- (4-hydroxyphenoxy) propanoic acid,

3- (3- (2,2,2-trichloro-1 - [(furan-2-carbonyl) amino) et] thioureido] benzoic acid,

1-phenyl-1-cyclopentanecarboxylic acid,

D, L-thiacetic acid,

3-sulfophenyl-gamma-acid,

3-chloro-5-trifluoromethyl-2-pyridylthioacetic acid,

2,3-dimethyl-2-phenylsuccinic acid,

D - (-) - 2-amino-4-phosphonobutyric acid,

5-tert-butyl-2-methylfuran-3-carboxylic acid,

1-methionyl-1-aspartic acid, boc-D-thiazolidine-4-carboxylic acid, boc-D-thioproline,

S-4-methylmandelic acid,

4- (trifluoromethyl) cyclohexanecarboxylic acid,

2,4-dichloro-5-sulfamoylbenzoic acid,

5 (S), 6 (R), 15 (S) -trihydroxyicose-7E, 9E, 11Z, 13E-tetraenoic acid,

3- (5-oxo-4,5,6,7-tetrahydro-1H-pyrrolo (2,3-c) pyridin-3-yl) propionic acid, (4-octylphenoxy) acetic acid,

4-n-hexylbenzoic acid,

2- (4,5,6-trihydroxy-3-oxo-3H-xanthen-9-yl) benzoic acid, thymine-1-acetic acid,

4-chloro-3-nitrobenzenesulfonic acid, N-α-boc-N-β-dnp-L-diaminopropionic acid,

3-hydroxy-4-nitrobenzoic acid,

3- (3-trifluoromethylbenzylthio) thiophene-2-carboxylic acid, (R) - (-) - 5-oxo-2-tetrahydrofurancarboxylic acid,

2- (2- (4-chlorophenyl) -4-phenylthiazol-5-yl) acetic acid,

3- (4-tert-butylbenzyloxy) thiophene-2-carboxylic acid, resorcinol- (4-azo-1) -2-naphthol-4-sulfonic acid,

2-phenoxyphenylacetic acid,

4- (3-phenylureido) benzoic acid,

2- (3-fluorophenyl) -1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxylic acid,

3- (p-hydroxyphenyl) -2-phenylpropionic acid,

2- (dimethylthiocarbamoylthio) acetic acid,

5- (p-tosyl) mercaptoacetic acid,

2,3-bis- (3,4-dimethoxybenzylidene) succinic acid, (S) -2-amino-2-methyl-4-phosphonobutanoic acid,

2,3-dihydro-5- (methylsulfinyl) -gamma-oxo- (1H) -indolbutanoic acid,

5-bromothiophene-2-carboxylic acid,

4-amino-3-bromonaphthalene-1-sulfonic acid,

2- (methoxymethyl) succinic acid,

L-leucyl-L-aspartic acid,

4-aminoazobenzene-3,4'-disulfonic acid,

2-chloro-6-fluorophenylacetic acid,

2-cyclohexylidene-butyric acid,

2-methyloctanoic acid, n-octylphosphonic acid,

3-dimethylaminobenzoic acid,

3.4-thiophenedicarboxylic acid,

1-Hydroxy-4- (1-phenyl-1H-tetrazol-5-ylthio) -2-naphthoic acid

N-acetylneuraminic acid, (-) - dibenzoyl-L-tartaric acid,

2- (2-methyl-1-phenylpropyl) benzoic acid,

8-methyl-naphthalene-1-carboxylic acid,

4- (4-bromo-2,5-dimethoxyphenyl) butyric acid,

2-chloro-4-hydroxybenzoic acid,

2-chloro-3-methylbenzoic acid, (4,4-dimethyl-3,7-dioxo-2,3,4,5,6,7-hexahydro-1H-inden-1-yl) acetic acid, ··· ·· · · · · · · · · · · · · · · · · · · · ·

2,3-dihydro-4-ethoxyphthalic acid,

2- (trifluoromethyl) -1,6-naphthyridine-3-carboxylic acid,

1- Pyrenhexanoic acid

2-methoxy-4- (methylthio) benzoic acid, N-acetyl-L-glutamine,

2,4- pentadecadiic acid,

2- (2-Hydroxyiminopropionylamino) succinic acid

5-anthracen-9-ylpentanoic acid,

N- (2,3-dimethylphenyl) -1,2,3,6-tetrahydrophthalamic acid,

2-hydroxy-3 (S) - (N-tert-boc-amino) -4-phenylbutanoic acid,

3.3-dichloro-2-fluoropropionic acid,

5-bromo-2-methoxyphenylacetic acid,

2-aminoethylphosphonic acid,

4'-n-decyloxybiphenyl-4-carboxylic acid, cis-5-icosenoic acid,

2-hydroxyamino-4-methylpentanoic acid,

4-chloro-3,5-dinitrophenylacetic acid,

8- (3-oxo-4,5,6-trihydroxy-3H-xanthen-9-yl) -1-naphthoic acid,

N-acetyl-L-glutamic acid,

10,12-pentacosadioic acid, tricyclo [11,2,2,2 (5,8)] nonadecahexaene-7-carboxylic acid,

4-fluorophenoxyacetic acid,

2.3- diphenylacrylic acid,

N- (2,4-difluorophenyl) malonic acid,

5H-perfluoropentanoic acid, behenic acid,

4- (2-nitrophenylsulfanylamino) benzoic acid,

2-hexyldecanoic acid,

N-t-boc-L-α-aminoadipic acid, β-bromangelic acid,

4,5-dihydroxy-2-methylbenzoic acid, (-) - camphoric acid, · · · · · · · · · · · · · · · · · · · · · · · · ·

evernic acid,

5,6,7-trimethoxy-3,4-dihydronaphthalene-2-carboxylic acid,

2.4- nonadecadiic acid,

2- [3-oxo-3- (N'-pentanoylhydrazino) propionylamino] benzoic acid,

4- [3- (2-chloro-6-methylphenyl) ureido] salicylic acid,

3-o-tolylbut-2-enoic acid, α- (tert-butyl) hydro-cinnamic acid,

3,5-dimethyl-4-hydroxybenzoic acid,

3.4-dimethoxyphenylacetic acid,

3-hydroxypropionic acid, n-decylmaleinamic acid,

2- (2-methoxyphenyl) -1-methyl-6-oxo-3-piperidinecarboxylic acid,

5-aminoazelaic acid,

5-formyl-2-furancarboxylic acid,

4-allyl-2,3,5,6-tetrafluorobenzoic acid,

2 ', 5'-dichlorophthalanilic acid,

3'-hydroxyhexahydrophthalanic acid,

2-butoxy-3-nitrosalicylic acid,

4'-butylbiphenyl-4-carboxylic acid,

3-Benzo (1,3) dioxol-5-yl-2-benzoylaminopropionic acid

3.4-dimethoxyphthalic acid,

2-ketopimelic acid,

N ² -fmoc-N ⁴ -boc-1,2,4-diaminobutyric acid, pyrogallol-4-carboxylic acid,

4- (1-bromoethyl) benzoic acid,

5-hexynoic acid, trans-acetic acid,

3-Hydroxy-2-naphthoic acid

3.6-dichloro-2-hydroxybenzoic acid,

3- (4-Phenoxybenzoyl) propionic acid, Lecanic acid •

- 100 -

5- (4-fluorophenyl) valeric acid,

2- [4- (4-benzyloxy) phenylsulfonyl] phenoxybutyric acid,

3- (4-hydroxymethylphenoxy) propionic acid, pyridoxal-5-phosphate,

2- (2-methoxycarbonyl-ethylamino) benzoic acid,

3.4.5-trifluorobenzoic acid,

2,3-pyridinedicarboxylic acid,

6-dimethylterephthalamic acid,

4- [4- (3-methyl-3H-benzothiazol-2-ylidene) but-2-enylidamino] benzoic acid,

2-fluoro-4-isopropoxybenzoic acid, o-propionylbenzoic acid, tricyclo [16.2.2.2 (8.11)] tetracosahexaene-9-carboxylic acid, fmoc-trans-3-phenylazetidine-2-carboxylic acid, ( +/-) - 1-aminocyclopentane-trans-1,3-dicarboxylic acid, (R) - (+} - 2- (phenylcarbamoyloxy) propionic acid, benzoylsulfanylacetic acid, fmoc-D, L-aminobutyric acid,

1-aminocyclobutane-trans-1,3-dicarboxylic acid,

2,4-diphenylpyrimidine-5-carboxylic acid,

3- (3-hydroxyphenyl) propionic acid,

7-hydroxy-1,3-naphthalenedisulfonic acid, Ν-α-Ζ-4-aminobutyric acid,

2.3.5- trifluoro-cinnamic acid, β-hydroxypyruvic acid, phthalideneacetic acid,

2-Methylimidazole-4-carboxylic acid

9,10-dihydro-9,10-ethanoanthracene-11,12-dicarboxylic acid,

3,3-dichloro-2- (4-chlorobenzoylamino) acrylic acid,

3-bromo- [3- (4-chlorobenzoyl) propionic acid],

2- [4- / 3- (5-chloro-2,4-dimethoxyphenyl) ureido / phenylthio] acetic acid

- 101 acid,

3-Methyl-1-oxo-1H-isochromene-4-carboxylic acid

2 - [(4-methoxycarbonyl) phenoxymethyl (benzoic acid,

4-bromo-2,3,5,6-tetrafluorobenzoic acid,

2-methyl-3-butenoic acid, [(2-hydroxybenzylidene) amino] phenylacetic acid,

5-dimethylterephthalic acid, bis (hydroxymethyl) phosphinic acid,

5-iodosalicylic acid, (2,4-dimethoxyphenyl (acetic acid,

3- (4-chlorobenzoyl) -2- (4-chlorophenyl) (propionic acid,

4- (6-hexyloxynaphthalen-2-yl) (butyric acid, pth-aspartic acid,

2-amino-6-fluorobenzoic acid,

2,2 ', 2,2' - [1,2-ethanediylidene-tetrakis (thio)] - tetrakis-acetic acid,

N-acetyl-L-aspartic acid,

3- (hexadecyloxy) benzoic acid, fmoc-D-aminobutyric acid, 1-diazo-2-hydroxy-5-nitronaphthalene-4-sulfonic acid, Ν-α-chloroacetyl-L-glutamic acid,

1-phenyl-1-cyclopropanecarboxylic acid,

3,4-Difluorohydrinnamic acid, [3-ho-3-ph-2,3,5,6,7,8-6H-benzo (4,5) imidazo (2,1-b) thiazol-2-yl] acetic acid (R) -cbz-oxaproline, (1S, 3S) -1-aminocyclopentane-1,3-dicarboxylic acid, boc-tranexamic acid,

2,2-dichlorocyclopropanecarboxylic acid, (4-chlorophenyl) phosphonic acid,

2,5-dichloro-3-nitrobenzoic acid,

2-acetamidoacrylic acid,

1-glutamic acid, •

- 102 -

3- (4-bromobenzoyl) acrylic acid,

3,5-dibromo-4-methylbenzoic acid,

5-amino-N- (2,3-dihydroxy-1-propyl) isophthalamic acid,

3-Benzoyl-2-thiophenecarboxylic acid

D-homocysteic acid,

3,4-furanedicarboxylic acid,

2- (3,4-dimethoxyphenyl) -1-methyl-5-oxopyrrolidine-3-carboxylic acid, micyclo [8,2,2,2 (4,7)] hexadeca-1 (13), 4,6 , 10 (14), 11,15-hexaenecarboxylic acid,

L-phenylalanyl-L-glutamic acid,

6,6,7,7-tetrafluorobicyclo (3,2,0) heptane-2,4-dicarboxylic acid,

N-glycolylneuraminic acid,

6,15-dioxo-l, 20-icosanedioic acid,

1-Benzyl-5-oxo-3-pyrrolidinecarboxylic acid

2'-cyanglutaranilic acid, (Z) -3 - [(aminoiminomethyl) thio] prop-2-enoic acid, dicyclopentadiene dicarboxylic acid,

4-heptylbenzoic acid, o-ethylbenzoic acid, (1S, 3R) -1-aminocyclopentane-1,3-dicarboxylic acid,

5-phenyl-2,3-dihydro-1H-pyrrolizine-6,7-dicarboxylic acid, - (2-naphthylthio) propionic acid,

4 - [(2-hydroxybenzylidene) amino] benzoic acid,

2- (hexadecyloxy) cinnamic acid,

D, L-α-hydroxycaproic acid, tricarballylic acid,

3-methyl-4-oxo-2-pentenoic acid, [1,4-dioxa-spiro (4,5) dec-6-yl] acetic acid, phenylmalonic acid,

N- (4-ethoxyphenyl) maleic acid, thiazolidine-2,4-dicarboxylic acid,

- 103 -

4- (3-bromopropoxy) benzoic acid,

N- (3-acetylphenyl) glutaramic acid,

3-bromo-4-chlorobenzoic acid,

4-chloro-α-methylcinnamic acid,

2-benzamido-3-methoxy-3-phenylpropionic acid,

2-ethyl-3- (3-hydroxyphenyl) acrylic acid, cis-4,7,10,13,16,19-docosahexaenoic acid, (R) - (- t -) - 2-bromo-3-methylbutanoic acid,

2,6-dichloro-3-nitrobenzoic acid, (S) - (-) - N- (1-phenethyl) phthalamic acid,

2-fluoro-5- (trifluoromethyl) phenylacetic acid,

2,2-diphenylheptanoic acid,

4-amino-4'-methoxydiphenylamino-2-sulfonic acid,

6,6-dimethyl-3-oxobicyclo (2,2,2) octane-2-carboxylic acid, 2 '- (trifluoromethyl) phthalanilic acid,

2- (4-tert-butylbenzoylamino) benzoic acid, β-methyl-3-nitrohydroscinnamic acid,

7α-methanesulfonylacetyl-3,6-dioxooctahydroindene-1-carboxylic acid, α-chloro-2-norboraneacetic acid,

4- (3,4-dihydro-4-oxo-1,2,3-benzotriazin-3-yl) phenylacetic acid, fmoc-9-aminononanoic acid, diethylphosphonopropanoic acid, methyliminodiacetic acid,

3-Endo-aminobicyclo (2,2,1) hept-5-ene-2-endo-carboxylic acid

3-iodo-4-hydroxybenzoic acid,

ΙΗ-dibenz (a, kI) -7-anthracenone-13-carboxylic acid,

4,4,4-trifluoro-3- (4-methoxynaphthalen-1-yl) but-2-enoic acid,

3- (4-methoxyphenyl) -3- (4-methylbenzoylamino) propionic acid,

104

2-fluoro-4- (trifluoromethyl) benzoic acid,

3-Methyladipic acid

4- (2-methoxyphenyl) butyric acid,

4-Methylsalicylic acid

2-methoxy-2-phenylpropionic acid,

4- (2-chloro-1,1,2-trifluoroethoxy) benzoic acid,

2-oxo-1-phenylpyrrolidine-4-carboxylic acid, β-carboxyaspartic acid,

2- (1-phenyl-2,2,2-trifluoroethoxy) acetic acid,

1 - [(1,1-dimethylethoxy) carbonyl] -4-piperidineacetic acid,

11 (S), 12 (S) -epoxy-13 (S) -hydroxy-9Z-octadecenoic acid,

3-nitropropionic acid,

2- (2-hydroxyphenyl) thiazolidine-4-carboxylic acid,

3-carboxy-1,2,2-trimethylcyclopentanacrylic acid,

4- (2-hydroxyphenyl) butyric acid, phenylacetic acid,

9,10-dihydroxystearic acid,

7-dimethylaminocoumarin-4-acetic acid, (4-hydroxy-3-sulfophenylamino) acetic acid,

R-phthalimido-α-hydroxy-n-butyl acid,

N- (4-fluorophenyl) maleic acid,

4 - [[4 - [(4,6-dimethylpyrimidin-2-yl) oxy] phenyl] amino] -2-methyl-4-oxo- (2Z) -butenoic acid, (2-methoxyphenyl) phosphonic acid,

3'-nitrophthalic acid, indole-3-succinic acid,

D, L-2-amino-7-phosphonoheptanoic acid,

5-sulfoanthronilic acid,

3- (2-oxocyclododecyl) propionic acid,

19-methylicosanoic acid,

3- (3-methylphenyl) propionic acid,

7-ethyl-3-oxo-2-azabicyclo (2,2,2) octane-6-carboxylic acid, ·· ····

- 105 N- (1-cyclopropylethyl) -N-phenylsuccinamic acid, (R) -1-amino- (3-methylbutane) phosphonic acid,

3-Naphthalen-2-ylpropinic acid, propionic acid,

1- (4-methoxyphenyl) -1-cyclohexanecarboxylic acid, malonic acid, isodehydroacetic acid,

N-α- (benzyloxycarbonyl) -D-glutamic acid,

N- (3,4-xylyl) phthalamic acid,

8-amino-5- (4-hydroxyphenylamino) naphthalene-2-sulfonic acid, pentamethylbenzoic acid,

N-acetyl-8-hydroxy-1-naphthylamino-3,6-disulfonic acid,

2- (2-chloroacetamido) -4-thiazoleacetic acid, (4-ethylphenoxy) acetic acid,

3- (4-chlorobenzoyl) propionic acid, p-chlorophenylisovaleric acid,

3,3-dichlorocyclopropane-1,2-dicarboxylic acid,

N- (2-bromo-4-nitrophenyl) phthalamic acid,

L - (+) - 2-amino-4-phosphonobutyric acid, bicyclo (2,2,2) oct-5-ene-2,3-dicarboxylic acid,

2-chloro-5-nitro-cinnamic acid,

3- (3-benzyloxy-4,5-dimethoxyphenyl) acrylic acid,

5-bromo-2-methoxycinnamic acid,

3- (4-carboxyphenyl) propionic acid, methylphosphonic acid,

2-methyl-3-phenylsuccinic acid, boc- (3S, 4S) -4-amino-3-hydroxy-5- (4-benzyloxyphenyl) pentanoic acid,

N-α- (benzyloxycarbonyl) -a- (benzyl ester) -1-glutamic acid, (S) - (+) - 2- (4-biphenylyl) propionic acid,

4-hexadecyloxy-3-methoxycinnamic acid,

6-Benzoylhexanoic acid

3-nitro-4-trifluoromethylbenzoic acid,

- 106 -

3-vinylbenzoic acid, isopropylmalonic acid,

2,2-bis (trifluoromethyl) -2-hydroxyacetic acid,

R - (+) - 2- (4-chloro-2-methylphenoxy) propionic acid,

5- (3-methoxyphenyl) hexanoic acid,

4-Trifluoromethyl-2-aminobenzoic acid

4- (4-methoxyphenyl) butyric acid, tetrafluoroisophthalic acid,

2-anthracen-1-ylpropionic acid,

2.2-difluorobenzodioxole-5-carboxylic acid,

2- (3,5-dinitrothiophen-2-ylamino) -4-methylpentanoic acid, [2- (4-chlorobenzenesulfonyl) ethylthio] acetic acid,

3-methoxypropionic acid,

9,10-epithiooktadecanoic acid,

4- (2- (3,4-dimethylphenoxy) acetylamino] benzoic acid,

3-benzoylbenzoic acid,

4,4,5,5,6,6,7,7,8,8,9,9,9-tridecafluoroonanoic acid,

3-methylpentanoic acid,

6-methoxy-2-naphthalenic acid,

14-br-tricyclo [8,2,2,2 (4,7)] hexadeca-hexaene-5-carboxylic acid,

3- (4-methoxy-2,3-dimethylphenyl) propionic acid,

3- (2,2-dimethylpropionamido) benzoic acid,

3- (2,4,6-trimethylphenyl) acrylic acid, (2,4,6-trimethylphenyl) phosphonic acid, (+/-) - 5-hydroxyicose-6E, 8Z, 11Z, 14Z-tetraenoic acid,

5- (2-chloro-4- (trifluoromethyl) phenoxy] -2-nitrobenzoic acid,

5-fluoro-6-hydroxy-2-methylpyrimidine-4-carboxylic acid, N- (2-hydroxyethyl) iminodiacetic acid,

2- (benzoyloxymethyl) benzoic acid,

4- (3,4- (methylenedioxy) benzylideneamino] salicylic acid,

5- (2-bromobenzoyl) pentanoic acid,

• · ·

- 107 1,4,4a, 5,8,8a-hexahydro-5-hydroxy-8-oxo-1-naphthalenecarboxylic acid,

N- (1-naphthyl) -6-nitrophthaic acid,

3- (2,4,6-trimethylbenzoyl) -2-biphenylcarboxylic acid, (+/-) - erythro-3-methylglutamic acid,

5-methoxybenzofuran-2-carboxylic acid,

2-Imino-4-oxythiazole-5-acetic acid

2- (trifluoromethyl) -2-hydroxypropionic acid, bromopivalic acid, cyclopropanecarboxylic acid, cyclopropane-1,2,3-tricarboxylic acid,

7-oxo-8-nonenoic acid, nonacosanoic acid,

4- (4-bromobenzoyl) pentanoic acid, ', 4', 6'-trimethylphthalanilic acid,

1-methyl-2-oxo-1,2-dihydroquinoxaline-3-propionic acid, tribromoacetic acid, (3-acetyl-2-methyl-5-oxo-2-pyrrolin-4-yl) acetic acid,

4-tert-butylbenzoic acid, cis-N- (2-fluorophenyl) hexahydrophthalamic acid, fmoc-4-aminobenzoic acid,

2- (2-chloroacetamido) benzoic acid, acetyl-asp-glu-oh, lactobionic acid,

1-bromocyclohexanecarboxylic acid,

2-Methyl-2-naphthalen-1-ylmethylmalonic acid

2- (4-Isopropylbenzylidene) pent-4-enoic acid

2 ^{1-methoxy-3,4,5,5} ', 6-pentachlorftalanilová acid

2- (cinnamylidene) -2-phenylacetic acid, glycyl-L-glutamic acid,

3-phosphonopropionic acid,

2- (4-chlorophenoxy) -2-methylpropionic acid,

2,3-dichlorobenzoic acid,

108 (R) -2-methylhexanoic acid,

4'-Fluoro-glutaranilic acid,

2-tetradecenoic acid,

2-Methyl-5-nitrobenzoic acid

4-Hexadecyloxy-meta-anisic acid

L - (+) - 2-amino-7-phosphonoheptanoic acid, spirof 5,5) undecane-2,2-diacetic acid,

1-Acetylpiperidine-4-carboxylic acid

3-naphthalen-1-ylpropionic acid, p-propoxybenzoic acid, (IR) - (+) - (1-amino-2-methylpropyl) phosphonic acid,

3- (4-bromobenzoyl (propionic acid, α-L-glutamyl-L-tyrosine-L-glutamic acid),

3,3-diphenylpropionic acid,

2-dibenzofuransulfinic acid,

2- (difluoromethoxy) phenylacetic acid,

N-α-boc-N-β- (Z) -L-diaminopropionic acid,

D, L-2-amino-7-sulfoheptanoic acid,

3- (4-nitrophenoxy) -2-thiophenecarboxylic acid, D, L-2-methylglutamic acid,

R-2-chlorormanedioic acid,

N-boc-D, L-α-aminoadipic acid,

7- [4- (2-ethoxycarbonyl) phenyl] heptanoic acid,

1-sulfoanthraquinone,

4- [4-Chexadecyloxy) phenyl (butyric acid,

4-pentylbicyclo (2,2,2) octane-1-carboxylic acid, (biphenyl-4-yloxy) acetic acid,

6,12-dioxo-1,17-heptadecanedioic acid,

5-Benzoylamino-2-bromopentanoic acid

3-Cyclopentyloxy-4-methoxybenzoic acid, [2,2-dimethyl-5-oxo- (1,3) dioxolan-4-yl] acetic acid, (S) - (+) - 2-amino-6- (iodoacetamido) (hexanoic acid,

6- (2-nitrophenylsulfanylamino) hexanoic acid,

109 cis-2,5-piperidinedicarboxylic acid,

- (2,3-dimethoxyphenyl) -2-methylacrylic acid, tricyclo [10.2.2.2 (4.7)] octadecaheptaene-9-carboxylic acid,

4,6-heptadecadiinic acid, arteannuic acid,

5- (4-chlorophenyl) -2,3-dihydro-1H-pyrrolizine-6,7-dicarboxylic acid,

6,7,8,8a, 9,10-hexahydro-2-methoxyphenanthren-7,8-dicarboxylic acid,

2-benzylidenemalonic acid, benzo (b) thiophene-3-acetic acid,

2-acetylamino-3- (1H-imidazol-4-yl) acrylic acid, (9H-xanthen-9-ylsulfanyl) acetic acid,

3,3'-thiodipropionic acid, tetrafluorophthalic acid,

6-butylaminopyrimidine-4-carboxylic acid, n-dodecylphosphonic acid, m-tolylacetic acid, mycophenolic acid,

3-acetoxybenzoic acid,

1- (3,4-dichlorophenyl) -2-oxopyrrolidine-4-carboxylic acid, (2S, 5R) -fmoc-5-phenylpyrrolidine-2-carboxylic acid, hydrofluoric acid,

3-chloro-4- (isopropylsulfonyl) thiophene-2-carboxylic acid,

4-chlorosalicylic acid, p-methyl-4-nitrohydroscinnamic acid, trichloropyruvic acid,

3,5-di-tert-butylbenzoic acid,

3- (trifluoromethoxy) phenylacetic acid, bicyclo (2,2,2) octane-2-carboxylic acid,

2-phenylindole-3-acetic acid,

2,2'-biphenyldiacetic acid,

2-mesitylenesulfonic acid,

110 gamma-oxo-5-acenaphthenebutyric acid,

3-trifluoromethylphenoxydifluoroacetic acid,

S-2-chloroformic acid,

2-noninoic acid,

2,6-dichloro-3-methylbenzoic acid,

N, N '- (1,4-cyclohexylenedimethylene) dimaleinamic acid,

7-nitro-9-oxo-1-fluorenecarboxylic acid, icosanedioic acid,

12-methanesulfonyloxydodecanoic acid, thiosalicylic acid,

3-acetyl-2-naphthoic acid, poly (acrylic acid),

3-phenylbutyric acid,

1- (3,5-dimethylphenyl) -6-methyl-4-oxo-1,4-dihydro-3-pyridinecarboxylic acid,

2-bromo-4-chlorobenzoic acid,

N- (4-ethoxyphenyl) -1,2,3,6-tetrahydrophthalamic acid, phenylenedecanoic acid,

N-acetyl-S- (4-nitrophenyl) -L-cysteine,

3-acetylbenzoic acid, tert-butylphosphonic acid, cis-epoxysuccinic acid,

4-bromobenzoic acid, for-L-2-aminohexanoic acid,

4- (4'-nitrobiphenyl-4-sulfonyl) benzoic acid, crotonic acid,

15 (R) -hydroxyicose-5Z, 8Z, 11Z, 13E-tetraenoic acid,

3- [4-ΟΧΟ-5- (5-ph-2-furylmethylene) -2-thioxothiazolidin-3-yl] propionic acid, palmitic acid,

5-methoxy-2- (2,2,2-trifluoroethoxy) benzoic acid, α-chloro-3,5,7-trimethyl-1-adamantanacetic acid, (5,6,7,8-tetrahydroquinazolin-4-ylsulfanyl) acetic acid, · · · · · · · · · · · · · · · · · · · · ·

- 111 trans - (+) - chrysanthemic acid,

1,4-dihydro-1- (2-fluoroethyl) -4-oxo-6,7,8-trifluoro-3-quinolinecarboxylic acid,

3- (phenylthio) propionic acid,

2- (2-benzoyloxyphenoxy) acetic acid,

3- (4- / 6- (4- (2-methoxycarbonylethyl) phenyl) hexyl / phenyl] propionic acid,

4-hydroxyphthalic acid,

N-boc-aminovaleric acid,

2'-chlorophthalanilic acid,

3- (2-nonylsulfanylbenzothiazol-6-ylcarbamoyl) acrylic acid,

2- (trifluoromethyl) propenoic acid,

2-carboxy-3-indolebutyric acid,

13c, 16c-docosadienoic acid,

11-p-tolylsulfanylundecanoic acid, propiolic acid, p-methylbenzyl-3-thiopropionic acid,

13-icosinic acid,

2- (2,3-dichlorophenylthio) acetic acid, (+/-) - 12,13-epoxyoctadec-9Z-enoic acid,

3,5-dichloro-o-anisic acid,

3.5- dibromsalicylic acid,

3.4- (methylenedioxy) -6-nitro-cinnamic acid, cis-acetic acid,

4-nitrophenylsuccinic acid, p-chlorobenzoylacrylic acid,

3- (4-tert-butylphenyl) propionic acid,

2 ', 6'-dimethyl-3,4,5,6-tetrachlorophthalic acid,

11,14,17-icosatrienoic acid,

3- (2,4-dichlorobenzylthio) thiophene-2-carboxylic acid,

2- (2,6-dichlorophenylthio) acetic acid,

4,5-dimethoxy-iodobenzoic acid,

- 112 -

3,5,6-trichlorosalicylic acid,

6-bromo-1,3-dioxo-1H-benz (d, e) isoquinolin-2 (3H) -acetic acid,

3-bromo-4-fluorobenzoic acid, trichloroacetic acid, (+/-) - 1-amino-trans-3-phosphonocyclopentanecarboxylic acid,

2- [2- (2-aminoacetylamino) -4-carbamoylbutyrylamino] -3- (4-ho-ph) propionic acid,

2-cyano-2-hexenoic acid,

3.3- dimethylacrylic acid,

2-bromo-terephthalic acid,

8-phenyloctanoic acid,

3- (benzylthio) propionic acid,

2- (dodecyloxy) benzoic acid,

4,5-dibromothiophene-2-carboxylic acid, (N, N-diethylthiocarbamoylthio) acetic acid,

2- (4-methoxycarbonyl-ph) -1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxylic acid,

2.3-dimethoxycinnamic acid,

N-acetyl-D, L-methionine,

9-fluorenecarboxylic acid, (+/-) - threo-3-methylglutamic acid,

7c, 10c, 13c, 16c-docosatetraenoic acid,

3- (4-n-propoxybenzoyl) propionic acid, perfluoro- (4-methylpent-2-enoic acid),

4- (2-hydroxy-1-naphthylmethyleneamino) benzoic acid, ethylenediamine-Ν, Ν'-diacet-Ν, Ν'-dipropionic acid, cis-N-furfurylhexahydrophthalamic acid,

N- [3- (6-chloro) pyridazinyl] iso (hexahydropyridine-4-carboxylic acid),

1,2-dimethyl-4- (p-carboxyphenylazo) -5-hydroxybenzene,

N- (1-methyl-5-methylthio-1,2,4-triazol-3-yl) malonaitioic acid

- 113 (R) - (-) - 3-chloromandelic acid, (R) - (-) - o-acetylmandelic acid, β-methyl-1-pyrenepropionic acid,

4- (difluoromethoxy) phenylacetic acid, phenyl-4-D-glucuronide,

2-bromo-5-methylbenzoic acid,

N- (4-iodophenyl) glutaramic acid, m-ethylbenzoic acid,

2,2-bis- (4-benzyloxybutyl) malonic acid,

5-bromo-2-fluoro-cinnamic acid,

3,4-dihydro-2,2-dimethyl-4-oxo-2H-pyran-6-carboxylic acid,

7-nitrofluorene-1-carboxylic acid, boc-2-aminobenzoic acid,

3'-methylmaleanilic acid,

15- (3,4-dichlorophenyl) pentadecanoic acid,

4-vinylbenzoic acid,

2,3,6-trifluorobenzoic acid, tetrathiafulvalentetracarboxylic acid,

4 - [(pyridine-3-carbonyl) amino] butyric acid,

6-methoxy-2-naphthylacetic acid,

Z-L-2-aminohexanedioic acid, (+/-) - 13-hydroxyoctadeca-9Z, 1ΙΕ-dienoic acid,

1-hexanesulfonic acid, tnp-L-aspartic acid,

3- (2,4-dichlorobenzyloxy) thiopene-2-carboxylic acid, carbobenzyloxy-D-2-aminobutyric acid,

11-dodecylsulfanylndecanoic acid,

8- [3- (5-f-2-ho-phenyl) -3-oxopropenyl] -4H-benzo (1,3) dioxin-6-

-carboxylic acid,

4- (1,3-dioxo-ΙΗ, 3H-benzo (d, e) isoquinolin-2-yl) benzoic acid,

2- (2-chloroacetylamino) -3- (4-hydroxyphenyl) propionic acid,

- 114 -

3- (chloromethyl) benzoic acid,

7-ethoxybenzofuran-2-carboxylic acid, acetylsalicylic acid,

4- [3- (3-fluorophenyl) ureido] benzoic acid,

3-hydroxy-2-methylicosanoic acid,

2-Naphthalen-2-yl-benzoic acid

L-valyl-L-aspartic acid,

3.3-dimethylglutaric acid,

3,5-bis (trifluoromethyl) benzoic acid, (-) - 2- (4-methoxyphenyl) butyric acid, (S) -3- (4-fluorophenyl) butanoic acid,

2- (2-methyl-3-phenylpropionyl) benzoic acid,

4- (4-n-propylphenyl) benzoic acid,

5- or 6- or 7- or 8-nitro-2-anthraquinone carboxylic acid,

1,2-dihydro-3-methyl-2-oxo-4-quinolinecarboxylic acid,

1,8-naphthaldehyde acid,

1- (4-chlorophenyl) -1-cyclopentanecarboxylic acid,

2,5-dimethyl-2,4-hexadienedioic acid,

3- (4-fluorobenzyloxy) thiophene-2-carboxylic acid, (+/-) - trans-azetidine-2,4-dicarboxylic acid,

2- (4-nitrophenylthio) acetic acid, (3,5-xylyl) phosphonic acid,

3.4-dimethylphenoxyacetic acid,

2-ethylhexanoic acid, (+/-) - 2-hydroxynonanoic acid, adipic acid,

2- (4-isopropylbenzoyl) benzoic acid,

2- (6-bromo-2-naphthyloxy) propionic acid,

3,5-dibromo-2- (2-ethoxycarbonylacetylamino) benzoic acid,

N- (2,4,6-trimethylphenyl) maleic acid,

4-Morpholin-4-yl-4-oxobut-2-enoic acid

N- (2-allylsulfanylbenzothiazol-6-yl) succinamic acid,

115

4-Methylsulfonyl-3-nitrobenzoic acid

3.4- difluoromandelic acid,

3- (4-chlorophenyl) glutaramic acid,

3,5-dibromobenzoic acid, 1H-indene-2-carboxylic acid,

5- (-) - 2 - [(phenylamino) carbonyloxy] propionic acid, alizarin-5-sulfonic acid,

4-acetoxyphenylacetic acid,

2,4-dichlorobenzoic acid,

N- (2-thiazolyl) phthalamic acid, dibenzo (a, d) cyclohepten-5-ylideneacetic acid, thiophene-3-acetic acid,

3,3-dimethyl- (1,1 ', 3', 1) -terfenyl-2'-carboxylic acid,

5- (4-methoxyphenyl) pentanoic acid,

3-Oxo-1-indanecarboxylic acid

6-bromohexanoic acid, [4- (2-acetyl-3-oxocyclopent-1-enylamino) benzoylamino] acetic acid,

4- [4- (2-carboxybenzoyl) phenyl] butyric acid,

2-Dicyclohexylcarbamoylcyclohexanecarboxylic acid

13-oxopentadecanoic acid,

2,3,4,4a, 4b, 5,8,8a, 9,10-decahydro-8a-methyl-2-oxo-1-phenanthrenpropionic acid,

3- (7-methoxy-2,2-diphenylbenzo (1,3) dioxol-5-yl) propionic acid, phenylpyruvic acid,

4- [3- (2-Phenoxypropionyl) -2-thioureido] benzoic acid,

3- (4-ethylbenzoyl) propionic acid,

4-hydroxyazobenzene-4'-sulfonic acid,

2-Acetylamino-3- (1H-indol-3-yl) propionic acid,

2,3,4,6-tetramethylbenzoic acid, linoleic acid,

4- (2,6-dimethyl-4-hydroxyphenylazo) benzenesulfonic acid

- 116 -

3- (3-bromo-4-methoxyphenyl) propionic acid,

3 - [(4-methoxyphenyl) - (toluene-4-sulfonyl) amino] propionic acid,

5- (3-amino-4-chlorophenylsulfamoyl) isophthalic acid,

3-bromo-2,6-dimethoxy-5-nitrobenzoic acid, (+/-) - cis-2,3-piperidinedicarboxylic acid,

N-acetyl-N-n-butylanthranilic acid,

3,5-dimethylphenoxyacetic acid,

2-cyanobenzoic acid,

N-α-boc-N-gamma-aloc-L-diaminobutyric acid,

3,4-methylenedioxyphenylpyruvic acid,

6-hydroxy-2,5,7,8-tetramethylchroman-2-carboxylic acid,

1-benzylorotic acid, boc-L-7-hydroxy-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid, (3-methoxyphenyl) phenylphosphinic acid,

3- (3,6-dimethoxy-2-naphthoyl) propionic acid,

4- [3- (2,5-xylyl) ureido] benzoic acid,

D-α-hydroxyisovaleric acid,

5,5,6,6,7,7,7-heptafluoro-4,4-bis (trifluoromethyl) heptanoic acid,

2-chloro-4-fluoro-cinnamic acid, acetylenedicarboxylic acid,

N-acetyl-D, L-2-amino-n-butyric acid,

2-hydroxyvaleric acid,

5-difluoromandelic acid,

N-boc-L-1,2,3,4-tetrahydro-p-carboline-3-carboxylic acid,

5- (1-methylethoxy) -1,3-benzenedicarboxylic acid,

2 ', 4'-dichloroglutaranilic acid, thiopivalic acid,

5'-chloro-2 ', 4'-dimethoxymaleanilic acid, [4- / 3- (4-meophenyl) thioureido] -6-methylpyrimidin-2-ylsulfanyl] acetic acid,

117

2.2- dichloropropionic acid,

3-chloro-4-hydroxybenzoic acid,

4-ethoxy-2-hydroxybenzoic acid,

1,2,3,4-tetrahydro-2-naphthoic acid,

2- [1- (3-chlorobenzyl) -3-indolyl] acetic acid, trans-β-hydromuconic acid,

2- (3-chloro-1,4-dioxo-1,4-dihydronaphthalen-2-ylamino) succinic acid,

4-fluoro-3-hydroxybenzoic acid,

2-phenoxynicotinic acid,

6- (2-benzoylamino-3-phenylacryloylamino) hexanoic acid,

2-Methoxy-5-sulfamoylbenzoic acid

5-Oxotricyclo [2.2.1.0 (2.6)] heptane-2,3-dicarboxylic acid

2,2-bis- (4-carboxyphenyl) hexafluoropropane,

3- (trimethylsilyl) propynoic acid, (2S, 3S) -2-chloro-3-methyl-N-valeric acid,

6-nitro-3- (phenylacetamido) benzoic acid,

6- (2,3-dioxo-3-phenylpropyl) -2,3-dimethoxybenzoic acid,

5- (N-benzoylamino) -N-valeric acid, D, L-3-hydroxyglutamic acid,

13 (S) -hydroperoxyoctadeca-9Z, HE-dienoic acid, (2,4-di-tert-pentylphenoxy) acetic acid,

2-methylenedecanoic acid,

2-hydroxy-2-methylbutyric acid,

4'-methoxysuccinanilic acid,

2-anilinonaphthalene-6-sulfonic acid, (4'-carboxymethanesulfonylbiphenyl-4-sulfonyl) acetic acid, β-acetylmercaptoisobutyric acid,

3,5-diiodobenzoic acid,

4 - [(phenyl (toluene-4-sulfonylimino) methyl) amino] benzoic acid,

3- (4-methylbenzoyl) propionic acid,

2.2- dichlorotetradecanoic acid,

- 118 -

2- (2'-nitro-4 -trifluormethylfenylthio ¹ (benzoic acid,

2,8,14,20-docesatetrain-1,22-dioic acid, (2-bromo-4-methylphenoxy) acetic acid,

2-fluoro-4-nitrobenzoic acid, isostearic acid, (+/-) - 3-endo-aminotricyclo [2.2.1.0 (2.6) (heptane-3-endo-7-anti-dicarboxylic acid,

4-bromoisophthalic acid,

6-bromo-α-cyano-1,3-benzodioxole-5-acrylic acid,

1-ethoxycarbonylamino-7-naphthol-3-sulfonic acid,

6- [2-benzoylamino-3- (4-methoxyphenyl) acryloylamino (hexanoic acid,

2'-carboxy-2,5-dimethylbenzophenone,

2-methylbutyric acid,

3,3-bis (trifluoromethyl) -3-hydroxypropionic acid, α-phenyl-o-toluic acid,

6-oxotricosanoic acid,

3,6-dihydroxyphthalic acid,

4- (3,4,5-trihydroxy-6-hydroxymethyltetrahydropyran-2-ylamino) benzoic acid,

2-Bromo-hexadecanoic acid

6-acetoxy-2-naphthoic acid, octacosanoic acid,

3-carbamoyl-2,4-diphenylcyclobutanecarboxylic acid,

4'-bromo-2 ', 6'-dimethylphthalanilic acid,

3-acetyl-3-methylpentane-1,5-dicarboxylic acid, thiobenzoic acid,

2- [3-OXO-3- (N'-propionylhydrazino) propionylamino (benzoic acid, cis-1,4-cyclohexanedicarboxylic acid, tricyclo [11,2,2,2 (5,8) (nonadecane-7-carboxylic acid) , guanidinosuccinic acid,

2- (methoxycarbonylthio) benzoic acid and a 4 * 4 · 4 · 4 · 4 · · · ·

119

L - (+) - 2-amino-3-phosphonopropionic acid,

4- (4-bromobenzoyl) butyric acid,

3,5-dibromo-4-methoxybenzoic acid,

3-Iodobenzoic acid

4-bromo-4-methylpentanoic acid,

18,18,18-trifluorooctadecanoic acid,

4- (hexadecylsulfonyl) benzoic acid,

1- (2-chloro-6-fluorophenyl) cyclohexanecarboxylic acid,

2,3-dinitrobenzoic acid, (1R, 3R) -1-amino-1-carboxycyclopentane-3-acetic acid,

1,3-phenylenediacetic acid,

2 '- (morpholine-4-carbonyl) biphenyl-2-carboxylic acid,

N- (2,6-xylyl) phthalamic acid, agaric acid,

N-hexadecylmaleinamic acid, (S) -4-carboxyphenylglycine,

4'-fluoro-3'-nitropthalanilic acid,

3,3,3-trifluoropropionic acid,

4,5-dimethoxy-2-nitrobenzoic acid, (1R, 3S) -1-amino-1-carboxycyclopentane-3-acetic acid,

N- (2,6-diethylphenylcarbamoylmethyl) iminodiacetic acid, iodoacetic acid,

2- (trifluoromethylthio) phenylacetic acid,

4- [3- [2,2,2-trichloro-1- [(furan-2-carbonyl) amino] et] thioureido] benzoic acid, cyclopentylideneacetic acid,

2-fluoro-3- (trifluoromethyl) benzoic acid,

2,6-dioxo-5-ethyl-1- (3-methoxyphenyl) -1,2,3,6-tetrahydro-4-pyrimidinecarboxylic acid, fmoc-D-2-aminohexanoic acid,

2,6-dihydroxy-3- [3- (trifluoromethyl) phenylazo] benzoic acid,

5-oxoundecanoic acid,

120

5-acetylaminoisophthalic acid, - (trifluoromethoxy) benzoic acid,

2- (toluene-4-sulfonylamino) propionic acid,

2- (3,4-dimethylbenzoyl) benzoic acid, tetrahydro-3-pyroslizic acid,

1-erythro-4-fluoroflutamic acid,

6- (carbobenzyloxyamino) caproic acid,

3 ', 4'-dimethylsuccinanilic acid,

2- (2-nitro-4-trifluoromethylphenylamino) propionic acid,

4- (4-hydroxyphenylazo) benzoic acid,

9H-hexadecafluoronanoic acid,

2-fluorocinnamic acid,

3-chloro-6-fluorobenzo (b) thiophene-2-carboxylic acid,

2-furamido-4-nitrobenzoic acid,

2- [2 '- (3'-chloro-5'-trifluoromethyl) pyridylthio] nicotinic acid,

3,3'-methylenebis- (6-chlorobenzoic acid),

3- (4-n-hexylbenzoyl) propionic acid,

2-benzyloxyphenylacetic acid,

4- (3,4-ethylenedioxyphenyl) butyric acid,

3,6,9-trioxaundecanedioic acid,

2-methyl-6-nitrobenzoic acid,

6- (4-bromobenzoyl) hexanoic acid,

4-octylbenzoic acid,

2- (trifluoromethoxy) terephthalic acid,

10-undecinic acid, trans-13-octadecenoic acid,

2-phenyl-2-propylsuccinic acid,

5,7-octadecadiic acid, cystamine-s-phosphoric acid,

N-acetyl-D, L-alanine,

Ν-α-boc-L-norvaline, benzyloxyacetic acid,

- 121 -

3,5-dimethoxybenzoic acid,

D, L-α-bromoisocaproic acid, metaphosphoric acid,

4'-fluorophthalanilic acid,

4'-bromo-2'-chloro-1,2,3,6-tetrahydrophthalanilic acid, phenytoin-N-butyric acid, hydroxyiminophenylacetic acid, (+/-) - L-aminocyclohexane-trans-1,3-dicarboxylic acid,

D, L-2-amino-5-phosphonovaleric acid,

2-cyano-3- (5-naphthalen-1-yl-2-furyl {acrylic acid, trans-parinaric acid,

3- (2-benzothiazolylthio) propionic acid,

2- (1- (4-fluorobenzyl) -3-indolyl) acetic acid,

4- (4-methoxyphenyl) -2-oxopyrrolidine-3-carboxylic acid, comanoic acid,

4-chloro-2-nitrobenzoic acid, β-methyllevulinic acid,

1- (2- (3-chloro-5-trifluoromethyl {pyridyl) indole-3-acetic acid),

4-dibenzothiophen-2-yl-4-oxobutyric acid,

3.5-difluorobenzoic acid,

Ν-α-benzoylasparagine, cis-N- (3-chloro-2-methylphenyl {hexahydrophthalamic acid,

4-butoxy-2-fluorobenzoic acid, (+/-) - trans-2,4-piperidinedicarboxylic acid, cantaric acid,

D, L-α-hydroxyhexacosanoic acid,

4- (4-cyclopentylnaphthalen-1-yl) -4-oxobutyric acid,

1- (p-tolyl) -1-cyclohexanecarboxylic acid,

1-carboxy-3-cyclohexene-1-acetic acid, oleic acid,

N- (diphenylmethyl) phthalamic acid,

2-carboxybenzaldehyde,

- 122 tetrafluorosuccinic acid, isooctanoic acid,

3-Cyanocinnamic acid

2,3,5-trifluorophenylacetic acid, calcein blue,

4-ethoxy-3-methoxyphenylacetic acid,

1-amino-4-bromo-9,10-dioxo-9,10-dihydroanthracene-2-carboxylic acid, carboxymethoxymethylpentaoxabicyclo (15,3,1) henicosatriene-21-carboxylic acid,

3 - [(R) -2-carboxypiperazin-4-yl] propyl-1-phosphonic acid, tetraoxa-23-aza-tricyclo [17.3.1.1 (8.12)] tetracosahexaene-24-carboxylic acid, [4-oxo-5- (5-phenyl-2-furylmethylene) -2-thioxothiazolidin-3-yl] acetic acid,

2- (4- (3,5-dichloro-2-pyridyloxy) phenoxy] propionic acid,

2,6-dimethoxy-3-nitrobenzoic acid,

4-sulfophthalic acid,

15- (4-iodophenyl) pentadecanoic acid,

13-phenylsulfanyltridecanoic acid,

2-octyldodecanoic acid, cis-10-heptadecenoic acid,

N-ethyl-L-glutamic acid,

2'-chloro-5 '- (trifluoromethyl) succinanilic acid,

2,6-dichlorobenzoic acid, brassidic acid, naphthazin-8,8'-disulfonic acid,

8-carboxy-3-methylflavone,

1,6-dibromo-2-hydroxynaphthalene-3-carboxylic acid, α-bromoheptanoic acid, [4-methyl-5- (2,2,2-trichloroethyl) thiazol-2-ylsulfanyl] acetic acid,

D - (+) - threo-3-hydroxyaspartic acid, · * · · · re re re re re re re re re re re re ··· ·· ··· · ·

123

5- (methylthio) salicylic acid,

4-hydroxybenzoic acid,

2- [2- (4-fluorophenyl) hydrazino / carbonyl] benzoic acid,

3- (4-n-octyloxybenzoyl) propionic acid,

3-Phenylnaphthalene-2-carboxylic acid

4-methyloctanoic acid, phenanthrene-4-carboxylic acid, benzenepentacarboxylic acid,

9-Decenoic acid,

4,5-dihydro-3-methyl-5-oxo-1-phenylpyrazole-4-dithiocarboxylic acid,

3- [3- (3,4,5-trimethoxyphenyl) acryloylamino] benzoic acid,

4.5.5.5-Tetrafluoro-4-trifluoromethyl-2-pentenoic acid, phenyl (toluene-4-sulfonyl) acetic acid,

11-cyanundecanoic acid,

2.5-dibromo-terephthalic acid,

2-chloro-5- (trichloromethylthio) benzoic acid, (R, S) -1-amino-3- (phosphonomethylene) cyclobutanecarboxylic acid, (R) -1-amino- (1-phenyl) methanephosphonic acid, (+) - 4'-nitrotartranilic acid,

5-methoxy-1,3-benzenedicarboxylic acid, (S) -2-chloro-3-methylbutyric acid,

5-ethyl-2-methyl-1-oxyisonicotinic acid,

1.3.5-trimethyl-1,3,5-cyclohexanetricarboxylic acid,

5-hydroxy-2-methyl-4-nitrobenzoic acid,

2,6-dimethyl-4-hexadecyloxybenzenesulfonic acid, p- (trimethylsilyl) phenylacetic acid, boc-L-aspartic acid, isoindolin-1-one-2- (3-methyl-2-butyric acid),

3- (N'-phenylacetylhydrazinocarbonyl) propionic acid, glutaric acid,

2- (1,3-dioxo-1,3-dihydroisoindol-2-yl) -3-methylbutyric acid

- 124 acid,

3- (p-chlorophenoxy) propionic acid,

N-n-propyl-L-aspartic acid,

3-phosphonobenzoic acid, (Z) -5-fluoro-2-methyl-1- [[4- (methylsulfinyl) phenyl] methylene] -1H-indene-3-acetic acid, diphenylmethane-4-carboxylic acid, (+ / -) -) - 1,1'-binaphthyl-2,2'-dicarboxylic acid, (m-tolyl) phosphonic acid, chloromethylphosphonic acid,

2- (dibenzothiophen-2-ylcarbonyl) benzoic acid,

D - (-) - α- (4-ethyl-2,3-dioxopiperinyl) carboxamide-4-hydroxyphenylacetic acid,

2'-tert-butylbiphenyl-3-carboxylic acid, linolenlaic acid, sulfosuccinic acid,

5-methyl-2- (ortho-tolyl) hexanoic acid,

3-tert-butyl-4-hydroxybenzoic acid, n-butylphosphonic acid,

4-amino-2,7-naphthalenedisulfonic acid,

3- [4- / 6- (4- (2-ethoxycarbonyl) phenyl) -6-oxohexanoyl / phenyl] propionic acid,

1- (2-Cyanoethyl) -5-oxopyrrolidine-2-carboxylic acid

3- (2-Oxobenzothiazol-3-yl) -propionic acid

2-methylvaleric acid, β-azido-o-benzoyl lactic acid,

4- (2-hydroxyethoxy) salicylic acid,

2,4-dihydroxythiazole-5-acetic acid, Ν-α-fmoc-N-gamma-alloc-L-diaminobutyric acid, nitromethane trispropionic acid, trans-chrysanthemmonocarboxylic acid,

N- (2-methyl-4-nitrophenyl) phthalamic acid,

2-ethylenedecanoic acid,

• *

- 125 2 ', 6'-dichlorormaleanilic acid, dodecylsulfanylacetic acid,

1,2,3,4-cyclobutantetracarboxylic acid, trans-9,10-epoxystearic acid,

5-acetoxyisocaproic acid, tricycloph 9,2,2,1 (4,8)] hexadeca-1 (14), 4 (16), 5,7,11 (15), 12-hexaencarboxylic acid,

2-hydroxy-2-trifluoromethyl-docos-4-enoic acid,

4-tert-butylphenylacetic acid,

5-chloro-2-prop-2-yloxybenzoic acid,

3- (3,4-dimethoxyphenyl) propionic acid,

2-acetylamino-3- (3-nitrophenyl) acrylic acid,

2- [3- (2-phenylcyclopropyl) ureido (acetic acid,

4-methoxysalicylic acid,

2-hexadecenoic acid, o-iodo-benzoic acid, N- (3-acetylphenyl) (maleanilic acid, acetylneuraminic acid,

4-hydroxy-1-phenylnaphthalene-2-carboxylic acid,

4-Biphenylacetic acid

5-bromo-4-chloro-2-fluorobenzoic acid,

2'-methoxy-5'-methylsuccinanilic acid,

2-carbamoyl-2-phenylbutyric acid, [4-amino-5- (4-chlorophenyl) pyrimidin-2-ylsulfanyl] acetic acid,

2-bromo-5-nitrobenzoic acid, dichrostachinic acid, (S) -3- (4-tert-butoxyphenyl) butanoic acid,

9-fluoreneacetic acid,

N-butylmaleinamic acid,

4-bromo-1-naphthoic acid,

3-phenylglutaric acid,

4-bromo-2-methylbenzoic acid,

- 126 arachidic acid,

2- (p-tert-butylbenzoyl) acrylic acid, nitrilotris (methylene) triphosphonic acid, ketomalonic acid,

5-chlorosalicylic acid,

2,4,6-trichlorophenoxyacetic acid, (4-acetylaminophenyl) acetic acid,

4- [2- (1-methyl-1H-quinolin-4-ylidene) ethylideneamino] benzoic acid,

N- (4-chlorophenyl) malonamic acid,

2- (4-cyclohexylbenzoyl) acrylic acid, cis-hexahydro-N- [2- (trifluoromethyl) phenyl] phthalamic acid, fmoc-D-homophenylalanine,

1-phenyl-1-cyclohexanecarboxylic acid, dibenzylphosphinic acid, (2-hydroxyphenoxy) acetic acid, (2-bromophenyl) phosphonic acid,

3,4-dimethoxy-2,5-furanedicarboxylic acid, n-acetylmuramic acid, pentacosanoic acid,

5-fluoro-2-methoxyphenylacetic acid,

N- (2,6-dimethylphenyl) maleic acid,

3- (Pentamethylbenzoyl) acrylic acid

L-2-acetamidobutyric acid, trans-2- (p-chlorobenzoyl) -1-cyclohexanecarboxylic acid,

1,1-cyclohexanediacetic acid,

2- (1-octadecenyl) succinic acid,

N- (4-chlorophenyl) glutaramic acid, cis-11,14,17-icosatrienoic acid, anthracene-9,10-dicarboxylic acid,

2.3.4- triphenylbutyric acid,

4 '- (ethoxycarbonyl) glutaranilic acid,

1- (N-Cbz-amino) cyclopropanecarboxylic acid,

N- (chloroacetyl) -L-aspartic acid,

4-ethoxy-3-methoxycinnamic acid, dipivaloyl-L-tartaric acid,

2,6-bisphenoxymethylbenzoic acid,

4-acetamido-3-nitrobenzoic acid, omega-ketoheptanoic acid,

3,5-di-tert-butyl-4-hydroxyphenylpropionic acid,

8 (R) -hydroxy- (5Z, 9E, 11Z, 14Z) -icosatetraenoic acid,

3-anthracen-9-ylpropinic acid,

3- [4- (4-chlorophenylthio) -3-nitrophenyl] acrylic acid,

D, L-threo-4-fluoroflutamic acid,

N-p-toluenesulfonylimino-3,3'-dipropionic acid,

2 ', 5'-dichlorormaleanilic acid, o-tolylacetic acid, octafluoradipic acid,

3- [2,2,3,3,4,4,5,5-octafluoro-1- (trifluoromethyl) cyclopentyl] propanoic acid,

7-epi-jasmonic acid,

N-carbamoyl-D, L-aspartic acid,

3-cyano-5-methoxy-2-methylbenzoic acid, tetradecanedioic acid,

5.5-dimethyl-4-hydroxy-4- (4-phenoxyphenyl) -2-hexanoic acid,

4-phthalimidobenzoic acid,

4-fluorosulfonyl-1-hydroxy-2-naphthoic acid,

4- [2-chloro-5- (trifluoromethyl) phenylazo] -3-hydroxy-2-naphthoic acid, oxaluric acid, cis-2-benzoyl-1-cyclohexanecarboxylic acid,

4-oxo-4-phenanthren-2-ylbutyric acid,

15-phenylpentadecanoic acid, benzylisovanilic acid,

21-bromhenicosanoic acid,

6-hydroxypyrazine-2-carboxylic acid •

- 128 N- (2,4-dimethylphenyl) -1,2,3,6-tetrahydrophthalamic acid,

2- (2-nitrobenzylthio) acetic acid, neodecanoic acid,

4- (2-phenoxyethoxy) benzoic acid,

2- (6-methoxy-3-nitropyrid-2-ylthio) propionic acid,

12-hydroxystearic acid,

3-iodo-2-methylbenzoic acid, diphenolic acid,

3- (trifluoromethylthio) phenylacetic acid,

4-methyl-2- [4- (trifluoromethyl) phenyl] thiazole-5-carboxylic acid,

3-ethoxythiophene-2-carboxylic acid, (-) - 4'-chlorotartranilic acid,

2,5-diphenylfuran-3,4-dicarboxylic acid, methylmalonic acid, p-pentyloxycinnamic acid,

6-oxo-1,14-tetradecanedioic acid,

2- (methylaminomethyl) tartronic acid, [3-cyano-2-methoxycarbonylmethylene-6- (4-meo-ph) -3-methoxycyclohexyl] acetic acid,

2-Phenylpropionic acid

1-cyclohexenylacetic acid,

3- (4-hydroxyphenyl) -2 - [(naphthalen-2-ylmethylene) amino] propionic acid, [5-methoxycarbonylsulfanyl-2-thioxo- (1,3) dithiol-4-ylsulfanyl] acetic acid, α-cyano- 4-hydroxy-3-methoxycinnamic acid,

6-trifluoromethylthieno (3,2-b) pyridine-2-carboxylic acid, boc-L-α-tert-butylglycine, (5-ethyl-4-hydroxy-6-methylpyrimidin-2-ylsulfanyl) acetic acid,

3 - [(4-methoxyphenyl) - (toluene-4-sulfonyl) amino] butyric acid,

4-methoxythiophene-3-carboxylic acid,

4'-bromo-3'-methylhexahydrophthalanilic acid,

3- [2- (4-chlorophenylthio) -5-nitrophenyl] acrylic acid, cis-N- [4- (ethoxycarbonyl) phenyl] hexahydrophthalamic acid,

8-Oxobicyclo (3,2,1) oct-6-ene-3-carboxylic acid

2- (trifluoromethoxy) phenylacetic acid, N-boc-D, L-2-aminotetraline-2-carboxylic acid,

2- (3-chloro-5-trifluoromethyl-2-pyridylthio) -1-methylimidazole-5-carboxylate acid,

4- [2- (4,4-dimethylchroman-6-yl) propenyl] benzoic acid,

2-formyl-4-nitrophenoxyacetic acid,

2-chloro-5- (methylsulfamoyl) benzoic acid,

4-chloro-2- (2-cyanethylamino) benzoic acid, pentafluoropropionic acid, petroselaidic acid,

Ν-α-Z-glycyl-L-aspartic acid, N-acetylglycine, (+) - lich-ester-acid,

3-Hydroxyoctadecanoic acid

4'-ethylsuccinanilic acid,

3.4.5-trifluorophenylacetic acid, cis-hexahydro-N- (4-nitrophenyl) phthalamic acid, fmoc- (4-methoxycarbonyl) piperidine, (2-acetyl-4,5-dimethoxyphenyl) acetic acid,

2- (4-methoxy-1-naphthyl) -1-methyl-5-oxo-3-pyrrolidinecarboxylic acid,

3- (4-ethoxybenzoyl) acrylic acid, acetopyruvic acid, acenaphthene-5-carboxylic acid,

3-hydroxy-6-methoxyindane-1-carboxylic acid,

4- (2-cyclohexenyloxy) benzoic acid,

2-hydroxy-6-isopropyl-3-methylbenzoic acid,

3,5-dichloro-4-methoxybenzoic acid

130 nonanoic acid,

2-nitrophenylacetic acid,

4 - [(3-nitro-2-pyridyl) amino] butanoic acid,

3'-chloro-4'-methylmaleanilic acid,

3- (2-bromobenzoyl) propionic acid,

3-Fluoradamantane-1-carboxylic acid

2- (trifluoromethyl) benzoic acid,

17-octadecinic acid,

1- (4-Methoxyphenyl) -6-methyl-4-oxo-1,4-dihydro-3-pyridinecarboxylic acid,

3-fluoro-2,4,6-trimethylbenzoic acid,

4,4'-azobis- (4-cyanvalerianic acid),

5-aminoisophthalic acid,

6-methyl-2-phenyl-5,7b-diazacyclopenta (c, d) indene-3-carboxylic acid, α-ketoglutaric acid,

2-chloro-4-nitrobenzoic acid,

4-hydroxy-10-oxo-9-oxatricyclo [6.2.1.0 (1.5)] undecane-2-carboxylic acid,

N- (2-thienylmethylene) anthranilic acid,

N- (3-methoxyphenyl) maleic acid,

10-doxylstearic acid, 1-hydroxy-2-naphthoic acid,

3'-chloro-3,4,5,6-tetrachlorophthalic acid, pentane-1-phosphonic acid,

1-cysteinsulfinic acid,

3-phenyl-3-propylglutaric acid,

6-tert-butyl-1,1-dimethylindane-4-carboxylic acid,

3,5-diacetoxybenzoic acid,

3- (4-chlorophenyl) -3- (2,2-dimethylpropionylamino) propionic acid,

8a-Methylloctahydronaphthalene-4a-carboxylic acid, resorcinol-o, o'-diacetic acid, · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · ·· · • ·· · «··· ··

- 131 -

5-bromo-4-chloro-4,5,5-trifluoro-2-pentenoic acid, (1,1 ', 2', 1) -terfenyl-3 ', 5'-dicarboxylic acid, maleic acid,

2-amino-4-methoxybenzoic acid, N-boc-L-glutamic acid gamma-cyclohexyl ester,

4- (difluoromethoxy) benzoic acid,

3,4,5,6-tetrachloro-3 '- (trifluoromethyl) phthalic acid, phytanoic acid,

4-nitro-2-phosphonobenzoic acid,

3- [2- (4-methylphenylthio) -5-nitrophenyl] acrylic acid, imidazole-2-carboxylic acid,

4-iodobenzoic acid,

2- (4-fluorophenyl) acetic acid,

2,2-dimethylbut-3-enoic acid,

4'-acetoxybiphenyl-4-carboxylic acid,

2-bromo-5-fluorobenzoic acid,

N- (3,5-dimethylphenyl) -1,2,3,6-tetrahydrophthalamic acid,

2,3-dihydro-1- (1H) -indolpropanoic acid,

5-benzyloxycarbonylaminopentanoic acid, α-isopropylideneaminoxypropionic acid, α-bromo-1-adamantanacetic acid,

5-bromo-4-chloro-4,5,5-trifluoropentanoic acid,

4- (2,4-dimethylphenyl) butyric acid,

5- [4- / 4- (4-Carboxybutyl) benzyl / phenyl] pentanoic acid,

1,4-dihydro-2-methylbenzoic acid, diphenylacetic acid,

2,7-naphthalenedicarboxylic acid, phenyl-β-D-thioglucuronide, exo-2-chloro-5,5-ethylenedioxybicyclo (2,2,1) heptane-syn-7-carboxylic acid,

4- (3-butenyloxy) benzoic acid,

3- [2- (4-nitrophenyl) acetylamino] propionic acid,

3-chloro-6-methylbenzoic acid,

132

3-fluorobenzoic acid, hydroxy- (3) 2,4,5-trifluorobenzoic acid,

10-bromo-9-anthracenecarboxylic acid, diphenoic acid, p-anisic acid, (R) - (+) - 2-bromohexanoic acid,

3-bromo-6- (methoxycarbonylamino) -2-chlorobenzoic acid, n-methyl-D, L-aspartic acid, homophthalic acid, cinnamylideneacetic acid,

2.4.5-trifluorobenzoic acid, oxo- (1-oxo-1,2,3,4-tetrahydrophenanthren-2-yl) acetic acid,

12-nitrododecanoic acid, dichlorodianilinoterephthalic acid,

3-p-tolyladamantane-1-carboxylic acid,

3-methoxy-9-oxo-5,7,8,9-tetrahydrobenzocycloheptene-6,6-dicarboxylic acid,

4-chloro-3-nitrobenzenesulfinic acid,

4- (2-methylcarbamoylacetylamino) benzoic acid, asym-hydrazinediacetic acid, [4- (4-carboxymethanesulfonylphenylsulfanyl) benzenesulfonyl] acetic acid,

2-chloro-3-nitrobenzoic acid,

2-ethoxybenzoic acid,

2 - [(3-carboxypropyl) - (toluene-4-sulfonyl) amino] benzoic acid,

4'-bromohexahydrophthalanilic acid, (2-methoxycarbonylmethylcyclopropyl) acetic acid,

2- (4-Methylbenzylcarbamoyl) benzoic acid

2-hydroxyimino-3-phenylpropionic acid, aminomalonic acid,

2,5-bis (trifluoromethyl) hydro-cinnamic acid,

2.6- difluorobenzoic acid, • · φφφ

- 133 3,3'-dithiodipropionic acid,

9-oxo-1,2,4,5-tetrahydro-3H-10-oxo-2a-azaaceanthrylene-8-carboxylic acid,

2-hydroxy-1-naphthaleneacetic acid, aniline-2,5-disulfonic acid,

2-acetylbenzoic acid,

2-thiofenglyoxylic acid,

4'-methylglutaranilic acid,

3-chloro-4-methylbenzoic acid,

4-hydroxy-7-iodo-10-oxo-9-oxatricyclo [6.2.1.0 (1.5)] undecane-2-carboxylic acid, [3,5-dioxo-2,3,4,5] -tetrahydro (1,2,4) triazin-6-ylsulfanyl] acetic acid,

2,5-bis (trifluoromethyl) benzoic acid,

4-ethyl-3-methyl-2-pyrrolecarboxylic acid,

1,2-phenylenedioxydiacetic acid,

5-fluoro-2- (trifluoromethyl) phenylacetic acid,

4 - ((2,4-dihydroxybenzylidene) amino] benzoic acid,

2-methyl-1H-benzimidazole-5-carboxylic acid,

4- (1 ', 1'-dimethyl-1'-hydroxypropyl) phenoxyacetic acid,

11- (2-oxotetrahydrofuran-3-yl) undecanoic acid,

N- (4-phenoxyphenyl) glutaramic acid, linolenic acid,

2- (phenylthio) propionic acid,

2- (trifluoromethyl) -1,8-naphthyridine-3-carboxylic acid,

7-oxooctanoic acid,

2-chloro-3-methoxythiophene-4-carboxylic acid, benzilic acid, anti-3-oxotricyclo (2,2,1,02,6) heptane-7-carboxylic acid, tert-butylacetic acid, (3-benzyloxy- 4-methoxyphenyl) hydroxyacetic acid, hydroiodic acid,

4-hydroxyphenylacetic acid,

- 134 15-phenyl-3,3-dimethylpentadecanoic acid,

R-4-methylmandelic acid,

2- (4-fluorophenyl) -3- (3-methoxybenzoyl) propionic acid,

5- (4-carboxy-2-nitrophenoxy) isophthalic acid,

5-nitro-1, 10-phenanthroline-2,9-dicarboxylic acid,

3-bromo-5-iodobenzoic acid, tricyclo [8,2,2,2 (4,7)] hexadeca-hexaen-5,12-dicarboxylic acid,

7-methoxycoumarin-3-carboxylic acid, (+) - 4'-fluorotartranilic acid,

2- [4- (4-chlorobenzoyl) phenoxy] -2'-methylpropanoic acid,

5-fluorisophthalic acid,

3- [5- (2-carboxyethanesulfonyl) naphthalene-1-sulfonyl] propionic acid, salicylic acid, (S) -2- (4-fluorophenyl) -3-methylbutyric acid,

4-acetamidobenzoic acid, α, α-dimethylphenylacetic acid, cyclopropylphenylglycolic acid,

2-keto-D-galactonic acid,

2 - [[(4-methoxyphenyl) sulfonyl] - (2-pyridyl) amino] acetic acid,

5- (4-chloro-2-nitrophenyl) -2-pyroslizic acid, ethylenediamino-Ν, Ν'-bis (isopropylphosphonic acid) hydrate,

Z-L-2-aminohexanoic acid,

L-4-hydroxyproline-o-phosphoric acid,

2- (2-carboxyphenylsulfanyl) malonic acid, mellitic acid,

1-hydroxy-1-cyclopropanecarboxylic acid, (IR) - (-) - (1-aminohexyl) phosphonic acid, N-boc-D-glutamic acid gamma-benzyl ester,

4- (3-methoxybenzoylamino) benzoic acid,

4-hydrazobenzoic acid,

- 135 -

4-fluoro-1-naphthoic acid, benzoyl lactic acid,

3-Butyl-5- (2,6,6-trimethyl-1-cyclohexen-1-yl) -2,4-pentadienoic acid, fmoc-L-p-aminobutyric acid, (S) -3-hydroxybutyric acid,

N- (3,5-xylyl) glutaramic acid,

4,5-dichlorophthalic acid, (S) -1-amino- (1-phenyl) methanephosphonic acid,

6-amino-2,3-dimethoxybenzoic acid,

4- (trifluoromethyl) cinnamic acid, Ν-α-Ν-gamma-di-Z-L-diaminobutyric acid,

2,3-dibromobutyric acid,

5,5'-carbonylbis (trimellitic acid),

4- (2-bromobenzoyl) butyric acid,

6-hydroxypicolinic acid,

4- (3-hydroxypropylamino) -3-nitrobenzoic acid,

-toludine-2,5-disulfonic acid,

4-isopropylphenoxyacetic acid,

2-fluoro-6-methoxybenzoic acid,

13-phenyl-10,12-tridecadioic acid,

4-chlorocinnamic acid,

2-acetyl-3,5-dibromsalicylic acid, mesitylacetic acid,

4- [4- (3,4-dimethylbenzenesulfonyl) phenoxy] benzoic acid,

4-carcinnamic acid,

2-bromo-5-sulfobenzoic acid, cis-2- (4-bromobenzoyl) -1-cyclohexanecarboxylic acid,

4- (3,4-dimethoxyphenyl) -4-oxobutyric acid,

3- (2-thenoyl) propionic acid, cycloheptanecarboxylic acid, N-chloroacetyl-L-2-amino-N-butyric acid, L-tryptophyll-L-aspartic acid,

136

3- [N- (4-chloro-3-nitrophenyl) carbamoyl] -5-norbornene-2-carboxylic acid, hippuryl-D, L-phenyl lactic acid,

3-bromadamantane-1-carboxylic acid, (S) - (-) - citric acid,

1- (3,4-dimethoxyphenyl) -4-hydroxy-6,7-dimethoxynaphthalene-2-

-carboxylic acid, (S) -2-methylhexanoic acid,

4- (2,2,2-trichloroacetamido) salicylic acid,

1,2,3,4-tetrahydro-gamma-oxo-2-pyrido (4,3-b) (1,6 (naphthyridinobutanoic acid,

1,3-dioxo-2- (4-p-tolylcarbamoyl-ph) -2,3-dihydro-1H-isoindole-5-carboxylic acid,

3,4,5,6-tetrachlorophthalic acid,

N-benzoyl-L-glutamic acid, (S) - (-) - 4-oxo-2-azetidine carboxylic acid, dibromoacetic acid,

5.5.5-trifluoro-4,4-bis (trifluoromethyl (pentanoic acid,

3- [2- (2-carboxy-et) -1,1,3,3-tetraoxo-5-ph -, - (1,3) dithian-2-yl] propionic acid,

3-oxoadipic acid,

N- (o-tolyl) succinamic acid, (Z) -3-bromoacrylic acid,

2.5-dimethyladipic acid, fmoc-4-phenylpiperidine-4-carboxylic acid,

3.4- dichloro-α-methoxyphenylacetic acid,

2,2'-Bithiophene-5-carboxylic acid,

2'-chloro-3,4,5,6-tetrachlorophthalic acid,

5-chloro-3-methylbenzo (b) thiophene-2-acetic acid,

N- (2,4-dinitrophenyl) -L-2-aminobutyric acid,

2-nitrophenol-4-sulfonic acid,

3-imidazolacrylic acid,

2,3-dihydroxybenzoic acid, •

- 137 -

4 - [(4-dimethylaminobenzylidene) amino] benzoic acid,

4- (2,5-dimethylphenyl) pentanoic acid,

2 - [(2-chlorallyl) - (toluene-4-sulfonyl) amino] benzoic acid, bis- (2-methyl-5-nitrophenyl) phosphinic acid, cis, cis-1,3,5-tripropyl-1,3 5-cyclohexanetricarboxylic acid,

3-chloro-2-nitrobenzoic acid,

2 - [(4,6-dimethoxypyrimidin-2-yl) oxy] -3-methylbutanoic acid,

3,5-di-tert-butyl-4-hydroxyphenylacetic acid, tetrachloro-terephthalic acid, furylacetic acid,

3- [3- (2-methoxy-5-nitrophenyl) ureido] benzoic acid,

1,2-diarninocyclohexane-N, N, N ', N'-tetraacetic acid, phosphatidylglycerol, trans-2- (4-bromobenzoyl) -1-cyclohexanecarboxylic acid,

2- (2-bromobenzoylamino) -3-phenylpropionic acid,

3- (4-tert-butylbenzoyl) acrylic acid,

N-boc-D-glutamic acid, cis-hexahydro-N- (4-iodophenyl) phthalamic acid,

1,4-phenylenediacetic acid,

7-methyldecanoic acid,

4-nitrophthalic acid, p-toluic acid,

2 - [(4,6-dimethoxypyrimidin-2-yl) oxy] -3-methylpentanoic acid,

4'-acetylglutaranilic acid,

3-hydroxy-7-methoxy-2-naphthoic acid,

2- [4- (3,4-dimethylphenoxy) -ph] -1,3-dioxo-2,3-2H-1H-isoindole-5-carboxylic acid,

2,5-dimethoxy-3-nitrobenzoic acid, 1-methoxy-2-naphthoic acid, (2,4,6-trimethylphenoxy) acetic acid,

138

Ν, N-diethyl-4-sulfamoylbenzoic acid,

4-benzyloxy-3-methoxybenzoic acid,

3-chloroanthraquinone-2-carboxylic acid,

3- (imidazol-4-yl) propionic acid, (+/-) - pinoleic acid,

2,5-dihydroxy-1,4-benzenedioacetic acid, D, L-α-methylasparagic acid,

N- (2,6-xylyl) glutaramic acid,

3- [2- (1,3,3-trimethyl-1,3-dihydroindol-2-ylidene) ethylideneamino] benzoic acid,

4-anthracen-9-yl-4-oxo-butyric acid, perfluoro- (2-ethoxyethane) sulfonic acid,

3,5-diisothiocyanatobenzoic acid,

4-methoxy-1,7-dimethylindane-5-carboxylic acid, Ν, Ν-diethylmaleinamic acid,

2-undecenoic acid,

2-Methyl-3-o-tolylacrylic acid

4,4'-azobis- (4-cyanvaleric acid),

4- (4-chlorobenzoyl) phthalic acid,

D, L-α-aminoadipic acid,

4- (methylthio) phenylacetic acid, glycyl-D, L-aspartic acid, sulfoacetic acid, (+/-) - trans-1-amino-1-carboxycyclopentane-3-acetic acid,

3-hydroxy-2-methyl-3- (3-nitrophenyl) propionic acid,

4- [N-methyl (methylsulfonamido)] benzoic acid,

1,2,3-thiadiazole-4-carboxylic acid,

2-methylhexadecanoic acid,

3'-nitro-3,4,5,6-tetrachlorophthalanilic acid, psoric acid,

4-nonyloxybenzoic acid,

D-erythro-4-fluorophlutamic acid,

2 - [[2- (4-chlorophenyl) hydrazino] carbonyl] benzoic acid,

- 139 6b, 7,7a-trimethyl-7,7a-dihydro-6bh-cyclopropa (a) acenaphthylene-7-carboxylic acid,

3- (trifluoromethoxy) cinnamic acid,

2,6-diethoxybenzoic acid,

1- (tert-butoxycarbonyl) -4-hydroxy-2-pyrrolidinecarboxylic acid,

4-fluoro-α-methylphenylacetic acid,

3,3´-dithiobishydricinnamic acid,

2-Methyl-2-sulfooctadecanoic acid

2-chloro-4-methylthiobutanoic acid,

2-hydroxy-3- (2-hydroxybenzoyl) -6-trifluoromethylpyridine-5-carboxylic acid,

2-tert-butoxycarbonylamino-3- (4-hydroxyphenyl) propionic acid,

3- (4-chlorobenzoyl) -2- (4-ethylphenyl {propionic acid, (R) - (+) - α-methoxy-α- (trifluoromethyl) phenylacetic acid,

2-cyano-2- (2,3-dimethoxybenzylidene) acetic acid,

2- (4-carbamoylphenoxy) -2-methylpropionic acid,

2'-chlorormaleanilic acid,

2- (3,4-Dicyanophenyl) -1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxylic acid,

1,4-naphthalenedicarboxylic acid,

3- (2-methoxyphenyl) -3-methylbutyric acid,

D, L-2-amino-4-phosphonobutyric acid,

4-Isopropyl cinnamic acid

5- (4-methyl-2-nitrophenyl) -2-pyroslizic acid, trans-1,2-cyclohexanedicarboxylic acid,

3- (4-Methoxy-3-methylphenyl {propionic acid,

2- (4-bromophenylamino) malonic acid,

2-dibenzothiophenobutyric acid, polystyrenesulfonic acid, flavianic acid, p-methyl-α-phenylhydroscinnamic acid,

«• fc ·

- 140 -

1-Naphthol-3,6-disulfonic acid

5,6-dihydro- (1,4) -dioxine-2-carboxylic acid,

6- (3-bromobenzoyl) hexanoic acid,

2,6,2,6-tetramethyl- (1,1 ', 3', 1) terphenyl-2'-carboxylic acid,

3-chloro-3-phenylcarbamoylacrylic acid,

4-amino-1,7-naphthalenedisulfonic acid,

4-bromo-2-fluorocinnamic acid,

4,4'-dicarboxydiphenyl ether,

2- (4-chlorobenzoyl) benzoic acid, linoelaidic acid,

2-ethyl-5-methoxyisophthalic acid,

1.5-Naphthalenedisulphonic acid

4- (2,4-dichlorophenoxy) butyric acid, fmoc-12-aminododecanoic acid, pivalic acid, benzofuroxane-5-carboxylic acid,

4-amino-3- (trifluoromethoxy) benzoic acid,

3- (3-methylindol-1-yl) propionic acid,

2.5-dimethyl cinnamic acid,

6,7,8-trifluoro-4-oxo-1-propa-1,2-dienyl-1,4-dihydroquinoline-

-3-carboxylic acid,

2-chloro-5-maleiniinidobenzoic acid,

3-phenoxyphenylacetic acid, indazolone-4-carboxylic acid,

3- [N- (4-fluorophenyl) carbamoyl-5-norbornene-2-carboxylic acid,

4- (4-benzyloxybenzylideneamino) benzoic acid,

3'-acetyl-1,2,3,6-tetrahydrophthalanilic acid,

4-oxo-4,5,6,7-tetrahydrobenzo (b) furan-3-carboxylic acid,

3-bromo-3- (3-nitrophenyl) propionic acid,

3-methyl-2- (2-nitro-4-trifluoromethylphenylamino) butyric acid,

141 cis-8-icosenoic acid,

2,2'-iminodibenzoic acid,

4,4'-biphenyldisulfonic acid,

3.3.3- triphenylpropionic acid,

3- (dodecane-1-sulfonyl) propionic acid, hydroxyvalerenic acid,

3-quinolin-2-ylacrylic acid, cis-hexahydro-N- (3-methylphenyl) phthalamic acid,

1-benzyl-3-hydroxy-1,2,3,3a, 4,7-hexahydroinden-1,7a-dicarboxylic acid,

4-Methoxy-3-methylphenylacetic acid

N-formylanthranilic acid,

4- (3-phenylpropyl) benzoic acid, cyclopentylmalonic acid, α-hydroxypharnesylphosphonic acid,

3,5-dinitro-4-hydroxybenzoic acid,

4-Phenoxybutyric acid

3-isobutyrylaminobenzoic acid, cis-2 ', 6'-dimethylhexahydrophthalanic acid,

4- [4- / 4- (2-ethoxycarbonyl) benzyl / phenylbutyric acid,

4- [2- / 4-methyl-4H- (1,2,4) triazol-3-ylsulfanyl / acetylamino] benzoic acid,

N- (1,2-dimethylpropyl) phthalamic acid, icosa-5,8,11-trienic acid,

2,3-dibromo-3- (4-sulfamoylphenyl) (propionic acid, tridecanedioic acid,

3.5-dihydroxybenzoic acid, quinizarin-2-sulfonic acid,

4- (2,2-dimethylpropyl) benzenesulfinic acid,

4'-iodo-1,2,3,6-tetrahydrophthalanilic acid,

2 ', 4'-dimethylglutaranilic acid,

4-methyl-3-phenylpentanoic acid,

2- (3-hydroxy-4-methoxyphenyl) (glyoxylic acid)

142

3-carboxy-7-hydroxycoumarin, opianic acid,

4-Methyl-3- (2-nitroethyl) -2,5-pyrrole dicarboxylic acid

3- (2-hydroxy-1-naphthylmethyleneamino) benzoic acid,

2-fluoro-6-methoxyphenylacetic acid, petroselinic acid,

2 - [(5-oxotetrahydro-1H-2-pyrrolyl) sulfanyl] benzoic acid, (S) -2-chloro-4-methyl-N-valeric acid,

3-Methyl-2-thiophenecarboxylic acid

2,5-dimethylimidazo (1,2-a) pyridine-3-carboxylic acid

3- (p-nitrophenoxy) propionic acid,

2- (ortho-tolyl) valeric acid, bromosuccinic acid,

4,4'-dithio-butyric acid,

2- [3- (N'-decanoylhydrazino) -3-oxopropionylamino] benzoic acid, hexahydro-4-methylphthalic acid,

1.5-Naphthalenedisulphonic acid

2 - ((4,6-dimethoxypyrimidin-2-yl) oxy] benzoic acid,

3- (2-allylsulfanylbenzothiazol-6-ylcarbamoyl) acrylic acid,

5-phenylsalicylic acid,

3- (2-furyl) acrylic acid,

4-Methoxy-2- (3-methoxybenzoyl) benzoic acid

3-acetyl-2,2-dimethylthiazolidine-4-carboxylic acid,

6-bromo-1,3-benzodioxole-5-carboxylic acid,

1-cyclohexenecarboxylic acid,

3.4.5-trichloro-6-hydroxypyridine-2-carboxylic acid,

3- (4-methoxybenzoyl) propionic acid,

5-oxo-4-oxa-tricyclo [4.2.1.0 (3.7)] nonane-9-carboxylic acid,

2-oxo-4-phenylbut-3-enoic acid, [4- [1- (4-carboxymethoxy-3-methoxy) -1-methylethyl] -2-methyl

143 phenoxy (acetic acid,

2-benzoylamino-3-phenylacrylic acid, β, 5-dimethyl-2- (methylthio) cinnamic acid,

4- (4-octadecyl) -4-oxobenzenebutenoic acid,

4- (2-ethoxycarbonylacetylamino) benzoic acid,

4- (3-methoxy-5-methylphenyl) -4-oxobutyric acid,

3-hydroxypentadecanoic acid,

Z-styrene sulfonylacetic acid,

3- (4-methoxyphenoxy) propionic acid,

3 '- (trifluoromethyl (phtalanilic acid,

3,6-dioxaoctanedioic acid,

3'-chloro-4'-methylphthalanilic acid,

2- [2-chloro - [(2,5-dichlorophenyl) sulfonyl / anilino] acetic acid,

3-hydroxy-3- (2-oxo-1,2-dihydroindol-3-ylidene) (propionic acid,

6-phenylhexanoic acid,

3- (methylsulfonyloxy) -4-nitrobenzoic acid, (2-iodophenyl) phosphonic acid,

4-phenoxyphenylacetic acid, (1-aminopropyl) phosphonic acid, p-chlorobenzenesulfonic acid,

4,5-dibromocyclohexane-1,2-dicarboxylic acid, (-) - 2-oxo-4-thiazolidinecarboxylic acid,

4,6-dichloroindole-2-carboxylic acid,

2-chloro-6-nitrobenzoic acid, indole-3-acetyl-1-aspartic acid, cuminic acid,

9,12-octadecadiic acid,

2,2'-dimethoxy-5,5'-dimethylbiphenyl-3,3'-dicarboxylic acid,

6- (benzoylamino) -2-bromohexanoic acid,

3-Phenoxybenzoic acid, · · · · · · · · · · · · · · · · · · · · · · ·

144

3,4-dimethylcinnamic acid, (oxodi-pr-thioxoimidazolidinylidenethylidene) benzooxazolylpropionic acid,

7-formylnaphthalene-2-carboxylic acid, N-lauroyl-L-aspartic acid,

N- (4-chlorophenyl) maleic acid,

6-methoxycarbonyl-2,3-dihydroxybenzoic acid,

2-chloro-5- (methylthio) benzoic acid,

4-p-tolyl-1, 10-phenanthroline-2,9-dicarboxylic acid, homoquinoline acid,

5-sulfoisophthalic acid,

5- (4-Trifluoromethylphenyl) -2H-tetrazole-2-acetic acid

4'-octyl-4-biphenylcarboxylic acid,

1,3-dioxo-ih-benz (d, e) isoquinolin-2 (3H) -acetic acid,

3-Oxotetramethylperhydrophenanthro (2,3-d) (1,3) dioxole-4-propionic acid

4- (5-bromo-1,3-dioxo-1,3-dihydroisoindol-2-yl) benzoic acid, formimino-L-aspartic acid,

2- (4-ethylbenzoyl) benzoic acid, methylthiohydantoin-D, L-glutamic acid,

2- (4-aminophenyl) propionic acid,

2'-methyl-3'-nitro-3,4,5,6-tetrachlorophthalic acid,

4- n-octadecyloxycinnamic acid, diketopiperazine 1-aspartyl-L-phenylalanine,

N- (2,6-diethylphenyl) -3-nitrophthaic acid,

N-phthaloyl-D, L-phenylalanine, methanesulfonic acid,

1- (3-chlorobenzoyl) piperazine-2,3-dicarboxylic acid,

3,4-benzo-9-oxofluorene-1-carboxylic acid,

1-pyrenesulfonic acid, dehydroacetic acid,

2- (p-chlorophenyl) -3-methylbutyric acid,

5-Methyl-1,1-dioxotetrahydrothiophene-2-carboxylic acid

···· · · · · · ··· ·· ···

145

3-fluoro-5- (trifluoromethyl) cinnamic acid, α-benzyl ester N-boc-L-glutamic acid, n-hexylphosphonic acid,

2-acetamido-2-allylmalonic acid, diphenylmethane-4,4'-dicarboxylic acid,

Z - (-) - α-amino-4-phenylbutyric acid,

3,5-octadecadiic acid,

4-chloro-2,6-dinitrobenzenesulfonic acid,

N, N-bis [(S) - (-) - 1-phenethyl] phthatamic acid,

4- (3-bromobenzoyl) butyric acid,

8,10-henicosadiic acid,

4,4'-dithiobisbenzoic acid,

N- (4-carboxyphenyl) succinimide

3.4- dihydroxybenzoic acid,

5- [[(4-chlorophenyl) sulfonyl] amino] -5-oxopentanoic acid,

3,5-dichloro-4-hydroxybenzenesulfonic acid,

N- (2-hydroxybenzoyl) glutamic acid,

2-benzenesulfonyl-2-methyloctanoic acid,

2,3-diphenylpropionic acid,

3,4-dimethylthieno (2,3-b) thiophene-2,5-dicarboxylic acid,

4- [3- / 3- (trifluoromethyl) phenyl / ureido] benzoic acid,

2-methyl-3-nitrobenzoic acid,

2-Isopropyl malic acid

4- (2-phenylethenesulfonylamino) benzoic acid,

4-fluorophenylacetic acid, exo-2-chloro-5-oxobicyclo (2,2,1) heptane-syn-7-carboxylic acid,

2,5-dimethylphenylacetic acid,

3 ', 4'-dichlorophthalanilic acid, tricyclo [12,2,2,2 (6,9)] icosa-1 (16), 6 (20), 7,9 (19), 14,17-hexaendicarboxylic acid, (3,4,5,6-tetrahydroxytetrahydropyran-2-yl) acetic acid,

3'-chloro-2'-methylphthalanic acid,

- 146 -

3- (4- (3,4-dichlorobenzyloxy) phenyl] acrylic acid,

3-bromobutyric acid,

N- (4-Phenylphenyl) maleic acid, (+) - S-2-amino-6-iodoacetamidohexanoic acid,

2,4-dimethoxybenzoic acid,

3- (4- (hexadecyloxy) benzoyl] propionic acid, (R) - (-) - 2-bromo-3-phenylpropionic acid, (R) - (-) - camphor-10-sulfonic acid, antipyric acid,

2-indanylacetic acid,

N- (3,4-dimethylphenyl) maleic acid,

4-palmitamidobenzoic acid,

2- (1,6-naphthyridin-2-yl) benzoic acid,

2- (n-dodecylcarbamoylmethyl) -2-hydroxysuccinic acid,

4- (2-hydroxy-5-phenylanilino) -1-butanesulfonic acid,

14c-tricosenoic acid,

3- (toluene-4-sulfonyl) propionic acid, pentafluorophenylacetic acid, (+/-) - 1-aminocyclohexane-cis-1,3-dicarboxylic acid,

4-amino-4'-chlorodiphenylamino-2-sulfonic acid, pimelic acid,

2 - ((phenylsulfonyl) -3- (trifluoromethyl) anilino] acetic acid, (S) - (-) - 2-bromopropionic acid,

4- (2-phthalimidophenyl) butyric acid,

6-methylsulfanylpyrimidine-4-carboxylic acid,

3-Methyl-2-nitrobenzoic acid

3.4- dichlorobenzoic acid,

5-methylhexanoic acid,

4- (trifluoroacetyl) benzoic acid,

3- (3- / 2,2,2-trichloro-1- (2-fluoroacetylamino) ethyl / thioureido) benzoic acid,

4- (2-methoxyphenyl) pent-3-enoic acid,

2- (4-fluorophenyl) -1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxy

···· · · · · ·

- 147 glicic acid, bicyclo (3,3,1) nonane-1-carboxylic acid,

3,7-dimethyl-1-adamantaneacetic acid,

4-cyanobenzoic acid,

7-Isopropylidenebicyclo (2,2,1) hept-5-ene-2,3-dicarboxylic acid

2- (hexadecylthio) benzoic acid,

N- (3-carboxypropyl) phthalamic acid, α- (2,6-dimethoxybenzylidene) hippuric acid, trans-7-octadecenoic acid,

4-pentenoic acid,

5- (4-methylphenyl) -2,3-dihydro-1H-pyrrolizine-6,7-dicarboxylic acid,

4'-bromosuccinanilic acid,

4-acetyl-1-methylpyridine-2-carboxylic acid,

2- (1-naphthyl) -2-phenylacetic acid,

2'-hydroxy-5'-methylmaleanilic acid, cis-N- (4-fluorophenyl) hexahydrophthalamic acid,

4- (3- (piperidine-1-sulfonyl) benzoylamino) benzoic acid,

4'-bromo-2'-chlorophthalanic acid,

3,3 '- (carbonyldiimino) bisbenzoic acid, (7-methoxy-5,8-dioxo-1,4,5,8-tetrahydronaphthalen-1-yl) acetic acid,

2-phenylbutyric acid,

N-t-boc- (2S, 3R) -3-amino-2-hydroxy-4-phenylbutyric acid,

2- (4-fluorophenyl) -1-isoquinolone-4-carboxylic acid, 11c, 14c-icosadienoic acid, (4 (S) -trans] -4,5-dihydroxy-3-oxo-1-cyclohexene-1-carboxylic acid acid,

2- [N- (2,4,6-trimethylphenyl) carbamoyl] cyclohexanecarboxylic acid, β-hydroxyisovaleric acid,

N-benzoyl-N-phenylanthranilic acid,

148

3- (bromomethyl) crotonic acid, ethylene-acrylic acid copolymer, N-benzyl-D, L-aspartic acid, p- (naphthylmercapto) acetic acid, pentadecanedioic acid,

3,4-dimethyl-2,5-pyrrolo dicarboxylic acid,

2,3-bis- (3-methoxybenzylidene) succinic acid,

2- (2-hexylcarbamoylacetylamino) benzoic acid, n-octadecylphosphonic acid,

1- [2 '- (3'-chloro-5'-trifluoromethyl) pyridyl] piperid-4-onemethylenecarboxylic acid,

1,1,2-ethantricarboxylic acid,

D - (-) - 2-amino-3-phosphonopropionic acid,

5-bromo-N- (methoxycarbonyl) anthranilic acid,

16,17-dichlorheptadecanoic acid,

8-hydroxy-7-quinolinecarboxylic acid,

4- (4-fluorobenzoyl) butyric acid,

4.4.4-trifluoro-3- (trifluoromethyl) butyric acid,

2,4,6,8-decatetraenoic acid,

6- (3,4-dimethoxyphenyl) hexanoic acid,

2- [N- (2,5-dimethylbenzyl) carbamoyl] cyclohexanecarboxylic acid,

2- (1-methyl-2,2-diphenylethoxy) benzoic acid,

4,5-dicarboxy-gamma-pentadecanolactone,

6-heptenic acid, pentadec-14-enoic acid, d - (-) - quinic acid,

4,7-dioxo-7-phenylheptanoic acid,

3-hydroxypyridine-4-carboxylic acid, acetylsalicylsalicylic acid,

4- (bromomethyl) -3-nitrobenzoic acid,

2-methyl-4,4,4-trifluorobutyric acid,

N-t-boc- (2R, 3R) -3-amino-2-hydroxy-4-phenylbutyric acid,

149 α-hydroxyhippuric acid,

3- (methoxycarbonylaminomethyl) -4-hydroxybenzoic acid,

3- (4-ethoxyphenylcarbamoyl) propionic acid,

2-iodo-4,6-dibenzofuranedioic acid,

5-tert-butylsalicylic acid,

3- [3- (5-chloro-2,4-dimethoxyphenyl) ureido] benzoic acid,

4,5-dimethoxy-3-oxo-1,3-dihydroisobenzofuran-1-carboxylic acid,

4,4,4-trifluoro-3-methyl-2-butenoic acid,

2-methoxycinnamic acid, (1S, 3R) - (-) - camphoric acid,

3 ', 4'-dimethyl-1,2,3,6-tetrahydrophthalanilic acid, (R) -N- [1- (1-naphthyl) ethyl] succinamic acid,

4-nitrobenzenesulfonic acid,

3- (5,6,7,8-tetrahydronaphthalen-1-yl) propionic acid, pseudocumen-5-sulfonic acid, phenol disulfonic acid,

3- (2,4-dichlorobenzylideneamino) benzoic acid,

5-Benzoylpentanoic acid

4- (4-chlorobenzylideneamino) salicylic acid,

2 - [(1H-Indole-3-carbonyl) amino] benzoic acid,

5-methylsulfonamidoindole-2-carboxylic acid,

2,3-dichlorophenoxyacetic acid,

5-chloro-2-pyroslizic acid,

2-benzyloxybenzoic acid, p-chlorophenylpropiolic acid,

Ι-α-hydroxyisocaproic acid,

4'-chloro-2'-methoxyphthalanic acid, gamma-oxo-1-pyrrolidine butyric acid, trans-2,5-bis (trifluoromethyl) cinnamic acid,

2 - [(4,6-dimethoxypyrimidin-2-yl) oxy] -6-fluorobenzoic acid, d - (+) - 10-camphorsulfonic acid,

150

2.5-dichlorobenzenesulfonic acid,

2- [3- (N'-hexanoylhydrazino) -3-oxopropionylamino] benzoic acid,

3-methoxycinnamic acid,

N- (o-toluoyl) glycine,

2-naphthylamino-4,6,8-trisulfonic acid,

2-chloro-5-nitrobenzoic acid,

6-oxo-1,2-dihydro-6H-pyrrolo (3,2,1-ij) quinoline-5-carboxylic acid,

2-bromo-5-chlorobenzoic acid,

3- (2,6-dichlorophenyl) -5-methylisoxazole-4-carboxylic acid, 1-bromo-2-naphthoic acid,

D, L-p-hydroxycaprylic acid,

1- (2-chloro-6-fluorophenyl) cyclopentanecarboxylic acid,

2-chloro-5-nitrobenzenesulfonic acid,

4- (4-hydroxy-1-naphthylazo) benzenesulfonic acid,

2'-methoxy-5'-methylphthalanilic acid,

4-benzyloxyphenoxyacetic acid, β-butyl hydroscinnamic acid,

N- (4-nitrobenzoyl) anthranilic acid,

2-phenylmethanesulfinylbenzoic acid,

2- (trifluoromethyl) cinnamic acid,

5-hydroxylndole-3b-propionic acid, (2R, 3R) -2-benzyl-3-hydroxybutyric acid,

5- (3,4-dimethoxyphenyl) penta-2,4-dienoic acid,

4-nitro-2-phthalimidobenzoic acid, o-chlorophenoxyacetic acid, β-bromohydro-cinnamic acid,

2- (2-cyclohexen-1-yl) -2-methylmalonic acid,

2.5-dimethoxybenzoic acid, hydrocavic acid,

N- (2-ethylphenyl) phthalamic acid, (1R) - (+) - camphanoic acid,

- 151 -

4-chloro-6- (2,4-dihydroxyphenylazo) -1-hydroxybenzene-2-sulfonic acid,

1-cycloundecene-1-carboxylic acid, sulfosalicylic acid,

5,5'-dinitro-2,2'-biphenyldicarboxylic acid,

2-furanpropionic acid,

3- [4-ho-3-meo-6-oxodecahydro-4H-benzo (c) chromen-1-yl] propionic acid,

3 - [(2-methoxyphenyl) - (toluene-4-sulfonyl) amino] propionic acid, isoindolin-1-one-2- (3-phenyl-2-propionic acid),

4-bromo-4,4-difluoro-2-butenoic acid, p-nitrophenylpyruvic acid,

3-methyl-2-phenylvaleric acid, (S) - (-) - 2-bromohexanoic acid,

3,5-dibromo-2-anisic acid,

3-cyclopentylpropionic acid,

2.3.6- trichlorobenzoic acid,

2,6-difluorophenylacetic acid, cis-9,10-epoxystearic acid,

6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxylic acid,

3,5,7-trimethyladamantane-1-carboxylic acid,

3-Hexine-1,1,6,6-tetracarboxylic acid

3-hydroxy-4-methoxycinnamic acid,

4-tert-butyl-2,6-dimethylbenzoic acid,

3-Methylbenzofuran-2-carboxylic acid

2-hydroxyimino-3- (4-methoxyphenyl) propionic acid,

2,3,4-trimethylcyclopentanecarboxylic acid,

4-bromo-2- (phenoxy) benzoic acid,

4- (ethylthio) benzoic acid, (4-ethoxy-2-oxo-3-pyrrolin-1-yl) acetic acid,

2-naphthoxyacetic acid, (4,6-dihydroxy-5-phenylpyrimidin-2-ylsulfanyl) acetic acid,

- 152 -

11- (4-acetylphenoxy) undecanoic acid, cyanoacetic acid,

3-methylglutaric acid,

4,5-dimethoxy-2-methylbenzoic acid,

2-ethyl-2-methylsuccinic acid,

2-tert-butyl-5-pyridinesulfonic acid,

4- (trimethylsilyl) benzoic acid, boc-1-thiazolidine-4-carboxylic acid, (1S, 3R) -1-amino-1-carboxycyclopentane-3-acetic acid,

2- (3-phenylthioureido) benzoic acid,

2- (3-nitropyrid-2-ylthio) propionic acid,

4'-chloro-3'-nitroptalanilic acid,

3.4.5- triacetoxybenzoic acid, pyrazine-2,3-dicarboxylic acid monoamide,

3-ethoxycarbonyl-4,4-diphenylbut-3-enoic acid,

N- (3-methoxyphenyl) glutaramic acid, octenyl disuccinic acid,

3-Amino-2-chlorobenzoic acid

N-n-propyl-D-aspartic acid,

4-benzyloxy-3,5-dimethylbenzoic acid, (+/-) 9-hydroxyoctadeca-10E, 12Z-dienoic acid, (R) - (+) - indoline-2-carboxylic acid,

4-chlorobenzoic acid,

2- (2,2-dichloroethyl) -5-methoxybenzoic acid,

1,2-dihydro-6-methoxy-1-methyl-2-oxo-4-quinolinecarboxylic acid,

2.2- diisopropylmalonamic acid,

3-fluoro-4-methylbenzoic acid,

3-nitrobenzenesulfonic acid, N-p-nitrobenzoyl-L-glutamic acid,

5- (2-fluorobenzoyl) thiophene-2-acetic acid,

2-hydroxy-4-methoxybenzophenone-5-sulfonic acid, chromotropic acid, ········· · · ···

153

2- (trifluoromethylthio) benzoic acid, D, L-4-hydroxyphenyl lactic acid, (3-methyl-4-oxo-4,9-dihydropyrazolo (3,4-b) quinolin-1-yl) acetic acid,

3- (4-octyloxyphenyl) acrylic acid,

N-α-t-boc-5,5-dimethyl-D-thiazolidine-4-carboxylic acid,

2-methoxyisophthalic acid,

Ν-α-Z-L-alanyl-L-glutamic acid, Z-gamma-amino-β-hydroxybutyric acid,

4- (1,2,3,4-tetrahydronaphthalen-1-yl) butyric acid,

N- (4-nitrobenzoyl) -6-aminocaproic acid,

2-methoxycarbonylooctahydroindene-2-carboxylic acid, o-cresol-4-sulfonic acid,

2,3,3,4,4-pentachlorobutyric acid, trichloromethylphosphonic acid,

3-formyl-4-hydroxybenzoic acid, n-lauroyliminodiacetic acid,

2,3,5,6-tetrafluorobenzoic acid,

3-formylsalicylic acid,

4-bromo-2-chloro-5-fluorobenzoic acid,

3- (3-bromobenzoyl) propionic acid,

2-hydroxy-2-trifluoromethyllikos-4-enoic acid,

2 ', 3,4-benzophenone tricarboxylic acid,

2-hydroxyiminobutyric acid, naphtho (2,3-d) -1,3-dioxolene-2-carboxylic acid,

2- (8-chloro-1-naphthylthio) acetic acid, dihydronaphthalene-1,4-dicarboxylic acid, cyclobutane-1,2,3,4-tetracarboxylic acid, α-methyl-2,4,5-trimethoxycinnamic acid, p -tolylphosphonic acid, cis-3,4,4,4-tetrachlorotrotonic acid, α-ketoctanoic acid,

1,8-naphthalenedicarboxylic acid,

154

2,2-dimethylvaleric acid,

3-fluoro-2-methylbenzoic acid, (S) - (+) - 2-chloro-3-phenylpropionic acid,

3-chlorotetrafluoropropionic acid,

2.4- dibromobenzoic acid,

4- [5- (aminocarboxymethyl) thiophen-2-yl] butyric acid, p-cresidine-6-sulfonic acid, fmoc-D-aspartic acid β-tert-butyl ester,

3,4-diacetamidobenzoic acid,

2- (1-trimethylsilanylvinyl) benzoic acid,

N-formylglycine,

2,6-dimethoxybenzoic acid,

4-bromo-3-hydroxynaphthalene-2-carboxylic acid, cyclohexanediaminotetraacetic acid,

4-Pentylbenzoic acid

2-amino-4,5-dibromo-3,6-dimethylbenzoic acid,

2- (4-fluorophenyl) -2-adamantaneacetic acid,

2-cyclohexylglycolic acid,

4,5,5,5-tetrafluoro-4-trifluoromethoxy-2-pentenoic acid, β-hydroxyaspartic acid,

4- [2-benzoylamino-3- (4-methoxyphenyl) acryloylamino] butyric acid, cis-7-octadecenoic acid,

1-bromo-4,4-dichloro-1,3-butadiene-1-carboxylic acid,

4 ^1- ethylmaleanilic acid,

2-hydroxy-3-nitroacetanilide-5-sulfonic acid, (-) - diacetyl-1-tartaric acid,

4,4 '- (1,4-phenylene) bis (2-oxo-3-butenoic acid),

5-nitroisophthalic acid,

4-chloro-o-anisic acid,

2-amino-3- (4-carboxyphenyl) propionic acid,

5-Trityl-3-mercaptopropionic acid

5-bromo-3,4-dihydroxybenzoic acid,

- 155 3- (n-Propylcarbamoyl) -5-norbornene-2-carboxylic acid, (5S, 12S) -dihydroxy- (6E, 8E, 10E, 14Z) -icosatetraenoic acid, heptanoic acid, adamantan-1-ylbenzoylaminoacetic acid ,

3- (1H-imidazol-2-yl) -2- (4-methoxybenzoylamino) propionic acid,

N- [2- (3-chloro-5-trifluoromethyl) pyridylaminoethyl] maleic acid,

6-chloro-2- (1,3-dioxoindan-2-yl) quinoline-8-sulfonic acid,

3-phenylmethanesulfonylpropionic acid, (5,6,7,8-tetrahydronaphthalen-2-yl) acetic acid, [4- (3-phenylpropyl) phenyl] acetic acid,

2,3-dibromo-4 '- (ethoxycarbonyl) succinanilic acid,

3.4-diethoxybenzoic acid, fmoc-1-thiazolidine-4-carboxylic acid,

4- [6- (3-carboxy-propylamino) -5-nitro-2-pyridylamino] butyric acid,

2- (trifluoromethoxy) benzoic acid, [3-cyano-6- (4-methoxyphenyl) -2-oxocyclohexyl] acetic acid,

4-acetamido-4'-aminostilbene-2,2'-disulfonic acid,

2-bibenzylcarboxylic acid, tricyclo [12,2,2,2 (6,9)] icosa-1 (17), 6,8,14 (18), 15,19-hexaene-7-carboxylic acid,

4'-bromo-3'-methylglutaranilic acid,

4- [3- (3-nitrobenzoyl) -2-thioureido] benzoic acid,

5- (tert-butyl) -2-hydroxycyclohexanecarboxylic acid, cyclododecanecarboxylic acid,

5-hydroxymethyl-2,6-dimethylnicotinic acid,

3'-chloro-2'-methylsuccinanilic acid, boc-D-norleucine, tetraoxabicyclo (12,3,1) octadeca-1 (17), 14 (18), 15-triene-18-carboxylic acid,

2-methylimidazo (1,2-a) pyridine-3-carboxylic acid, 9 · 9 · 9 · 9 · * · * 4 ♦ 4 4 4 · ··· • · · · «« · ·

156

6-chloro-2H-1-benzopyran-3-carboxylic acid,

4- [2- (3,3-Dimethyl-2,3-dihydro-benzo (b) thiophen-5-yl) -propenyl] -benzoic acid,

3- [2-acetylamino-3- (4-methoxyphenyl) acryloylamino] propionic acid, stearidonic acid, (+/-) - 1-amino-cis-3-phosphonocyclohexanecarboxylic acid,

6-methylchromone-2-carboxylic acid,

4-acetoxyhydricinnamic acid,

3.4.5-tribromo-2-pyroslizic acid,

1- (p-tolyl) -1-cyclopentanecarboxylic acid,

5,7-bis (trifluoromethyl) -4-hydroxyquinoline-3-carboxylic acid,

N- (2-hydroxyethyl) ethylenediaminotriacetic acid, α-bromocinnamic acid,

2.3.4- trichlorglutaconic acid,

4-acetylphthalic acid,

3- (4-octadecyl) benzoylacrylic acid,

Ν-α-Ζ-Ν-β-boc-1-diaminopropionic acid,

N- (2-hydroxybenzoyl) -L-aspartic acid methyl [4-carboxy-2-nitrobenzoate],

4-amino-2-chloropyridine-5-carboxylic acid,

3,5-dihydroxy-2-naphthoic acid, p-coumaric acid,

9-hydroxydecanoic acid,

2- (3-chloro-1,4-dioxo-1,4-dihydronaphthalen-2-ylamino) hexanoic acid,

3- (2,4-dimethoxyphenyl) propionic acid,

4.4.4-trifluorobutyric acid, trans-2-phenyl-1-cyclopropanecarboxylic acid,

4-iodophenylacetic acid, [phenethyl (toluene-4-sulfonyl) amino] acetic acid,

2,3-dihydro-3-oxo- (1H) -isoindol-1-ylideneacetic acid,

157 boc-12-aminododecanoic acid,

2-acetyl-3,4,5,6-tetrachlorobenzoic acid, 1-benzoylpiperidine-4-carboxylic acid, (S) -2-methyldecanoic acid,

1-hydroxyaminocyclohexanecarboxylic acid,

8-chloromethyl-7-methoxy-4-oxo-4H-chromene-2-carboxylic acid,

2-bromo-3-nitrobenzoic acid,

3- (trifluoromethyl) phenylacetic acid,

3- (2-benzoylamino-3-phenylacryloylamino) (propionic acid,

N- (3,4-dimethoxyphenethyl (maleic acid,

4,6-dioxoheptanoic acid,

4-chloro-α-methylphenylacetic acid,

4'-methyl-2-biphenylcarboxylic acid, α-guanidinoglutaric acid,

N- (2,3-xylyl) phthalamic acid,

5-nitro-2- [4- (1,1,3,3-tetramethylbutyl) phenoxy (benzenesulfonic acid,

4-propoxybiphenyl-4'-carboxylic acid,

1- (4-chloroanilino) -6-methyl-4-oxo-1,4-dihydro-3-pyridinecarboxylic acid,

2-amino-4-methylthiazole-5-sulfonic acid,

3-chloro-4- (methylsulfonyl (thiophene-2-carbonyl chloride),

2- (2-o-tolyloxyacetylamino) benzoic acid,

3'-methylglutaranilic acid,

3-octylsulfanylpropionic acid,

2,3-dihydroxy-4-methoxybenzoic acid,

2-furanglyoxylic acid, chlordifluoroacetic acid,

1,3,3a, 6,7,7a-hexahydro-1-oxo-4,5,6-trimethyl-7-isobenzofurancarboxylic acid, (+) - benzylmethylphenylsilylacetic acid,

4,4'-stilbendicarboxylic acid;

- 158 -

4- (2-benzothiazolylthio) butyric acid,

2- (1-acetyl-2-naphthyloxy) propionic acid,

2-hydroxy-6-phenyl-3,5-pyridinedicarboxylic acid, o-benzamidoglycolic acid,

2-hydroxy-3-butynoic acid,

2-carboxy-4- (trifluoromethyl) diphenylsulfide, boc-L-homophenylalanine,

Ν-α-fmoc- (Ν-β-boc) diamonopropionic acid, (E) -10-hydroxy-2-decenoic acid,

2-Benzoylamino-3- (1H-imidazol-4-yl) acrylic acid

9-tetradecinic acid,

3 - [(2-ethoxycarbonyl) thiazol-2-ylamino] propionic acid,

5- [4- (4-methoxycarbonylbutyl) phenyl] -5-oxopentanoic acid,

2,3,4-trimethoxycinnamic acid,

4-dodecanoylaminobenzoic acid,

3-methyl picolinic acid,

2-chloro-n-butyric acid, fmoc-2-aminoindan-2-carboxylic acid, conjugated octadecadienoic acid,

3- (4-n-butoxybenzoyl) propionic acid, (2-methoxy-4-nitrophenyl) phosphonic acid,

2,4,6-octatrienoic acid,

5-chloro-2-nitrobenzoic acid,

3- (4-methoxyphenyl) propynoic acid,

2-chlorophenylacetic acid,

5- (4-morphilino) -2H-tetrazole-2-acetic acid,

6-methyl-4-oxo-1- (4-toluidino) -1,4-dihydro-3-pyridinecarboxylic acid, cbz-L-α-aminosubric acid,

3-adamantan-1-ylpropionic acid,

4- (6-butoxynaphthalen-2-yl) -4-oxobutyric acid,

4 - [(5,6,7,8-tetrahydro-5,5,8,8-tetramethyl-2-naphthalenyl) carboxamido] benzoic acid,

159

3.4- difluorobenzoic acid,

2-oxo-1-cyclohexanepropionic acid,

2 ', 4'-dichloro-1,2,3,6-tetrahydrophthalanilic acid,

3-bromomethylbenzoic acid, cis-hexahydro-N- (4-chlorophenyl) phthalamic acid, m-xylene-4-sulfonic acid,

2- (2-chloro-1,1,2-trifluoroethoxy) -β-anisic acid,

2- (1,2,3,4-tetrahydro-6-naphthylmethyl) benzoic acid,

3- (4-dimethylaminophenyl) -2-methylacrylic acid, boc-D, L-α-aminobutyric acid,

3 - [(4,6-dimethoxypyrimidin-2-yl) oxy] benzoic acid,

2.5-dinitrobenzoic acid, trans-12-octadecenoic acid,

2-Chloro-adamantane-2-carboxylic acid

3-fluoro-4-methoxyphenylacetic acid,

2,4,6-tribromobenzoic acid,

2- [[2- (4-methylphenyl) hydrazino / carbonyl] benzoic acid,

1- (3-fluorophenyl) cyclohexanecarboxylic acid, mesitylenesulfonic acid,

2.5- Difluoric cinnamic acid

3- (4-methoxyphenyl) propionic acid, methacrylic acid, D, L-s-acetyl-2-benzyl-3-mercaptopropionic acid,

2.5-difluorobenzoic acid,

2-nitroisophthalic acid,

2,3-difluoro-4- (trifluoromethyl) benzoic acid,

6- (2-hydroxybenzylideneamino) hexanoic acid, [IR- (Ια, 2β, 3a)] - (+) - 3-methyl-2- (nitromethyl) -5-oxocyclopentaneacetic acid,

4- (4'-methoxybenzylidene) amino-cinnamic acid,

4-bromo-3-nitrobenzoic acid,

9-benzoylnonanoic acid,

4'-acetamidosuccinanilic acid,

160 n-tosyl-L-glutamic acid,

2,4,6-triisopropylbenzoic acid,

5-azido-2-nitrobenzoic acid,

4-hexadecyloxybenzoic acid,

1,2-dihydroxyanthraquinone-3-sulfonic acid,

1.3- adamantanediacetic acid,

4- [2- (benzothiazol-2-ylsulfanyl) acetylamino] benzoic acid, phosphoglycolic acid, N-α-boc-N-β-aloc-1-diaminopropionic acid,

2-chloro-6-fluorobenzoic acid,

1- (4-methoxyphenyl) ethyliminoxyacetic acid,

4- [3- (1-butyrylatino-2,2,2-trichloroethyl (thioureido) benzoic acid), (+/-) - 5-iodo-3-isopropylpentanoic acid,

4-fluorofuranic acid, α-cyano-3-hydroxycinnamic acid,

5-Methoxy-2-nitrobenzoic acid

4-fluoro-2- (trifluoromethyl) phenylacetic acid, octane-2-sulfonic acid, cresolsic acid, aleuritic acid,

1- (2-chloro-5-sulfophenyl) -3-methyl-5-pyrazolone, pentadecafluorooctanoic acid,

N- (5-nitro-2-thiazolyl) phthalamic acid,

2- (2-chlorophenoxy) propionic acid,

1- gamma-carboxyglutamic acid, (R) - (-) - phenylsuccinic acid,

1,18-octadecanedioic acid,

3-amino-5-bromobenzoic acid,

5-chlorotricyclo [2.2.1.0 (2.6)] heptane-3-carboxylic acid,

2-hydroxydocosanoic acid,

4-methoxyphenylacetic acid, palmitoleic acid,

3-benzo (1,3) dioxol-5-yl-2-methylacrylic acid,

2 '- (piperidine-1-carbonyl) biphenyl-2-carboxylic acid,

3-benzoylamino-3- (4-chlorophenyl) propionic acid,

2-methylbenzylphosphonic acid, mucobromic acid,

2,3,6-trimethoxybenzoic acid,

2-Methylheptanoic acid

3-methyl-1-cyclohexanecarboxylic acid, phenyl- (2,4,6-trimethylphenyl) acetic acid,

2-thiophenecarboxylic acid,

3- [N- (4-ethoxyphenyl (carbamoyl) bicyclo (2,2,1) hept-5-ene-2-carboxylic acid),

2-methyl-4-phenylbutyric acid,

2- (3-methoxyphenyl (succinic acid, (S) -N- [1- (1-naphthyl) ethyl) succinamic acid),

2'-methoxy-5'-methyl-3,4,5,6-tetrachlorophthalic acid,

5-tert-butylsulfanylthiophene-2-carboxylic acid,

4- (octadecanamido) benzoic acid,

D - (-) - 2-Amino-7-phosphonoheptanoic acid,

4-methyl-1-cyclohexanecarboxylic acid,

3- (2,4-dichlorophenyl) -2-methylacrylic acid, boc-D-norvaline,

4- [5- (2,4-Dichlorophenyl) -2-furyl] thiazole-2-acetic acid,

3-hydroxy-3-methylglutaric acid,

3-hydroxy-4-methoxyphenylacetic acid, (S) - (+) - 2- (6-methoxy-2-naphthyl) propionic acid,

6-bromocoumarin-3-carboxylic acid,

3- (2-Butylsulfanyl-benzothiazol-6-ylcarbamoyl) -acrylic acid

2-naphthylamino-1,5,7-trisulfonic acid,

5- 3-chlorormanedioic acid, orsulic acid, ·

- 162 -

2- [2-οχο-2- / 4- (3-trifluoromethylphenyl) piperazin-1-yl / ethyl] malonic acid,

1,1-cycloheptanediacetic acid,

3-ethoxybenzoic acid,

2-methyl-1-cyclohexanecarboxylic acid,

5-methoxy-2-methylisophthalamic acid, n- (p-tosyl) anthranilic acid,

4-nitronaphthalene-1-carboxylic acid,

2-norboranacetic acid, benzyloxycarbonyl-1-norvaline,

3-Phenylcinoline-4-carboxylic acid

3-fluoro-4- (trifluoromethyl) phenylacetic acid,

4- (3-carboxypropionamido) benzoic acid,

2- (carbamoylmethylthio) benzoic acid,

2,4-dimethyl-5-oxohexanoic acid,

N- (2,5-dichlorophenyl) -1,2,3,6-tetrahydrophthalamic acid,

D, L-cyclohexylmandelic acid,

N-cyclohexylphthalamic acid,

4-phosphonobutyric acid,

5-fluoro-2-methoxybenzoic acid,

1,3-acetondicarboxylic acid,

4- (trifluoromethyl) hydrocinnamic acid,

4- (2-thienyl) butyric acid,

5- 4-methylthiomandelic acid,

3-Hydroxy-2-nitrobenzoic acid

3-hydroxycinnamic acid, ferulic acid,

3-bromo-4-oxo-4-thiophen-2-ylbutyric acid,

2,4,5-trimethylcinnamic acid,

4-Methyl-1,2,3-thiadiazole-5-carboxylic acid

2-butoxy-5-tert-octylbenzenesulfonic acid, β-gamma-aminobutyric acid,

1- (4-Methoxyphenyl) -2-oxopyrrolidine-4-carboxylic acid

163

5-chloro-2- (methylthio) pyrimidine-4-carboxylic acid,

N- (trifluoroacetyl) -D, L-aspartic acid,

2'-carbamoylglutaranilic acid,

2,6-dimethyl-4-oxopyran-3-carboxylic acid,

N-ethyl-5-sulfoanthranilic acid, cis-4'-ethylhexahydrophthalanic acid, (2R, 4R) - (+) - azetidine-2,4-dicarboxylic acid,

2-ethyl-2-methylbutanoic acid,

4-Aminosulfonyl-1-hydroxy-2-naphthoic acid

3- (3,4-dichlorophenyl) propionic acid,

2- (3-chloro-1,4-dioxo-1,4-dihydronaphthalen-2-ylamino) -4-methylpentanoic acid,

2,4-dihydroxy-3-methylbenzoic acid,

2-bromo-4,6-dimethyl-3-hydroxybenzoic acid,

3,5,7-trimethyl-1-adamantanacetic acid, α-hydroxybenzylphosphinic acid, [(2-hydroxy-5-nitrobenzylidene) amino] phenylacetic acid,

L-valyl-L-glutamic acid, ethacrynic acid,

9-fluorenone-2-carboxylic acid,

5- 4-methoxymandelic acid,

5-methylsalicylic acid,

4-acetoxyphenoxyacetic acid,

2- (o-chlorophenoxy) -2-methylpropionic acid,

4-hydroxythiobenzoic acid, ethanesulfonic acid,

2- [4-chloro / (4-chlorophenyl) sulfonyl / anilino] acetic acid, D, L-benzylsuccinic acid, (R) - (+) - gamma-butyrolactone-gamma-3-propionic acid,

5- (4-methoxybenzenesulfonyl) thiophene-2-carboxylic acid,

2-cyano-5-phenyl-2,4-pentadienoic acid, (-) - 4'-fluorotartranilic acid,

3,4-dichloro-2-pyroslizic acid, • «*

- 164 -

4- (2,4-dipentylphenoxy) butyric acid,

4,5,5-trifluoro-2,4-pentadienoic acid,

2'-methoxy-3,4,4 ', 5,6-pentachlorophthalic acid, erucic acid,

3-iodophthalic acid,

4'- (2-benzoylacetamido) succinanilic acid, (4-methoxybenzoylamino) acetic acid,

4-Phenylazobenzoic acid

3- (2-methylbenzothiazol-6-ylcarbamoyl) acrylic acid,

4-oxo-4H, 9H-1-thia-4α, 10-diazaindeno (1,2-a) indene-2-carboxylic acid,

N- (2-phenethyl) -3,4,5,6-tetrachlorophthalamic acid,

4-methyl-3-sulfobenzoic acid,

15-hydroxypentadecanoic acid,

4-hydroxy-3-methoxyphenylpyruvic acid,

2'-fluormaleanilic acid,

2-carbamoyl-2-propylvaleric acid, methylenebis (thioacetic acid),

4- (4-hydroxymethyl-3-methoxyphenoxy) butyric acid,

2-fluoro-5- (trifluoromethyl) cinnamic acid,

2-chlorobenzoic acid sulfonamide,

1,6-diaminohexane-N, N, N ', N'-tetraacetic acid,

4- (triphenylsilyl) benzoic acid,

5-chloro-2-methylimidazo (1,2-a) pyridine-3-carboxylic acid,

D, L-4-hydroxy-3-methoxymandelic acid,

2-Naphthylsulfonic acid,

1,1'-binaphthyl-8,8'-dicarboxylic acid, trans-3-chloroacrylic acid,

3- (4-chlorobenzoyl) -2- (2,4-dichlorophenyl) propionic acid,

3-benzo (1,3) dioxol-5-yl-2-ethylacrylic acid, indole-7-carboxylic acid,

11- [4- (methoxycarbonyl) phenoxy ]undecanoic acid,

4- (2,5-dimethylphenyl) -2-methylbutyric acid,

- 165 -

3- (4,5,6,6a-tetrahydro-fluoranthen-3-yl) -propionic acid, N- (4,6-dimethylpyrimidin-2-yl) -N-methyl-3-aminobenzoic acid,

N- (3,4-dicyanophenyl) -5-nitrophthaic acid, indazolone-4-carboxylic acid, (R) -2-chloro-3-methylbutyric acid,

2-methyl-3-naphthalen-1-ylacrylic acid, thionicotinic acid,

2-hydroxyoctanoic acid,

6- (4-chlorophenyl) -2-hydroxy-3,5-pyridinedicarboxylic acid,

2- (4-methyl-1-cyclohexylidene) acetic acid,

2-hydroxy-2- (2-aminothiazole) -4-acetic acid, (2-chloro-5-methylphenyl) phosphonic acid,

4-nitro-α- (ortho-tolyl) cinnamic acid, α-propyl-1-cyclopenten-1-acetic acid,

D, L-2-amino-6-phosphonohexanoic acid,

4- (3-hydroxyphenoxy) benzoic acid, (+/-) - 2-acetoxypropionic acid,

4- (3-methylureido) benzoic acid,

5-chloro-2-hydroxypyridine-3-carboxylic acid,

2,3,4,5-furantetracarboxylic acid,

2-bromo-3-phthalimidopropionic acid,

3-chloro-4-methoxybenzoic acid,

2,4,6-trifluorobenzoic acid,

5- (acetamido) -2-nitrobenzoic acid,

5- (4-nitrophenyl) -2-pyroslizic acid,

2-chloro-2- (3,4-dihydrophthalazin-4-on-1-yl) acetic acid, - (4-iodophenyl) propionic acid,

4-Phenyltetrahydropyran-4-carboxylic acid

3-phenyl-3- (toluene-4-sulfonylamino) propionic acid,

5,7-dioxooctanoic acid, (4-aminobenzyl) phosphonic acid,

4- (4-chloro-o-tolyloxybutyric acid),

166

N-boc-D, L-1-aminoindan-L-carboxylic acid,

N-phthaloyl-D, L-α-aminobutyric acid,

4-iodo-3-methylbenzoic acid,

2- [N- (1-naphthyl) carbamoyl] cyclohexanecarboxylic acid, bis (boc-3,5-diaminobenzoic acid), (D) -N-benzylglutamic acid,

4- (4-chloro-m-tolyloxy) butyric acid,

6-benzamidohexanoic acid,

11-bromundecanoic acid,

2- (2-carboxycyclohexa-2,5-dienylamino) -4-nitrobenzoic acid,

1,4-dioxo-2,5-methanopentalen-2,3a, 5,6a-tetracarboxylic acid,

3- (tetradecyloxy) benzoic acid, trifluoroacetic acid, cyclohexanebutyric acid,

5,5-dimethyl-2,4-thiazolidinedicarboxylic acid,

2,2,3,3-tetramethylcyclopropanecarboxylic acid, N-carbamoyl-L-leucine,

2-chloro-4-methylsulfonylbenzoic acid,

2- (1,8-naphthyridin-2-yl) benzoic acid,

5 - [[(4-methylphenyl) sulfonyl] amino] -5-oxopentanoic acid, trans-cyclobutane-1,2-dicarboxylic acid, exo-2-bromo-5-oxobicyclo (2,2,1) heptane-syn- 7-carboxylic acid, diamylacetic acid, (3-phosphonoadamantan-1-yl) phosphonic acid,

4- [3- / 2,2,2-trichloro-1- (2,2-di-methpropionylamino) -ethyl] thioureido] benzoic acid,

1H, 1H, 2H, 2H-perfluorooctanesulfonic acid, cis-2,4-piperidinedicarboxylic acid,

4- [3- (2,4-xylyl) ureido] benzoic acid,

3 ', 5'-dichlorophthalanilic acid,

- 167 -

2,4-dihydroxypyrimidine-5-carboxylic acid, cyclobutane-1,1,3,3-tetracarboxylic acid,

4-methyl-2- (ortho-tolyl) valeric acid, (S) - (+) - α-methoxyphenylacetic acid, (-) - 4'-methyltartranilic acid,

5- (2-hydroxy-3-methoxyphenyl) pentanoic acid, cis, cis-muconic acid,

2- (2,7-dichloro-6-hydroxy-3-oxo-2,3-dihydro-1H-xanthen-9-yl) benzoic acid, (E) -2-octadecenoic acid,

D, L-2-amino-4-methyl-5-phosphono-3-pentenoic acid,

5- (2,5-Dioxopyrrolidin-1-yl) -4-oxopentanoic acid

2,4-di (decyloxy) benzoic acid,

3,5-diiodo-4-hydroxybenzoic acid,

3- (4-chlorobenzoyl) -2- (3-chlorophenyl) propionic acid,

2- (2-benzothiazol-2-ylvinyl) benzoic acid,

11- (9-anthroyloxy) undecanoic acid,

1.3- adamantanedicarboxylic acid, myristoleic acid,

3- (2,2-difluoro-1,3-benzodioxol-5-yl) - (2E) propenoic acid, neooctanoic acid,

4- (2-benzoylamino-3-phenylacryloylamino) butyric acid,

2 - [(4,6-dimethoxypyrimidin-2-yl) thio] benzoic acid, N-boc-D-aspartic acid β-benzyl ester,

2-ethylsulfanyl-5-fluoro-6-hydroxypyrimidine-4-carboxylic acid,

N- (4-methoxyphenyl) -1,2,5,6-tetrahydrophthalamic acid,

1- (2-chloro-4-fluorophenyl) cyclopentanecarboxylic acid,

2-Methoxy-4-methylbenzoic acid

1-adamantanecarboxylic acid,

3- (2-nitrophenoxy) -2-thiophenecarboxylic acid,

3-chloro-2,6-dimethoxybenzoic acid,

2,3-dimethoxy-5-iodobenzoic acid, · · · · · · · · · · · · · · · · · · · · · · · · ·

- 168 -

2,4-dichloro-5-fluorobenzoic acid,

N- (3-chlorophenyl) -1,2,5,6-tetrahydrophthalamic acid,

2,3-diphenylbutyric acid,

3,5-dimethylbenzoic acid,

D, L-α-hydroxyisocaproic acid,

5- (4-chlorophenyl) -2-pyroslizic acid, (2-guanidinoethylmercapto) succinic acid,

7-nitro-4-fluorenecarboxylic acid, carbobenzyloxy-D, L-glutamic acid,

8-bromo-1-naphthoic acid,

12- [N- (7-nitrobenz-2-oxa-1,3-diazol-4-yl) amino] dodecanoic acid, n-hexadecylmalonic acid,

2.5- dichloro-terephthalic acid, hexacosanoic acid, heptagluconic acid,

2,3,5,6-tetrachlorobenzoic acid, p-4-methoxybenzylmercapto-p, β-cyclopentamethylenepropionic acid, glyphosate, cis-azetidine-2,4-dicarboxylic acid,

6-mercaptonicotinic acid,

2- [2- / 3-chloro-5- (trifluoromethyl) -2-pyridyl / hydrazono] acetic acid,

2- (2-methoxyethoxy) acetic acid,

N-cbz-D-norleucine,

2-chlorobenzoic acid,

N- (2,6-dinitro-4-trifluoromethyl) iso (hexahydropyridine-4-carboxylic acid),

2-hydroxyaminobutyric acid, bromo chloroacetic acid,

L-a-glutamyl-L-glutamic acid,

8-bromooctanoic acid,

- 169 -

3-fluorophenylacetic acid, tmoc-L-indoline-2-carboxylic acid,

2,3-dibromo-4'-ethoxysuccinanilic acid,

3- (4- (2,2-dimethylpropionyl) benzoyl] propionic acid,

2-nitrothiophene-4-carboxylic acid,

2-phenyl-2-adamantaneacetic acid,

7-phenyl-6,8-dioxa-spiro (3,5) nonane-2,2-dicarboxylic acid, 5,5'-thiodisalicylic acid, (S) - (-) - 2-chloropropionic acid,

7-nitro-9-oxo-4-fluorenecarboxylic acid,

Z - (+) - α-amino-4-phenylbutyric acid, α-cyano-3,4-dimethoxycinnamic acid, salicylsalicylic acid,

4-bromo-butyric acid,

2- (3-phenylureido) benzoic acid,

4- (isopropylsulfonyl) thiophene-2-carboxylic acid,

3-methyl-2-phenylacetylaminobutyric acid,

5-anthracen-2-ylpentanoic acid,

3- [1,2-dihydro-2-oxo-5- (trifluoromethyl) pyrid-1-yl] propionic acid,

3'-nitrosuccinanilic acid, fmoc-D, L-p-aminobutyric acid,

D, L-3,4-dihydroxymandelic acid, (2-benzylsulfanyl-6-methylpyrimidin-4-yloxy) acetic acid,

5-methyl-2- (trifluoromethyl) furan-3-carboxylic acid,

3-methyl-4-nitrobenzoic acid,

1-propanesulfonic acid,

5-indanacrylic acid,

3-acetamido-4-hexadecyloxybenzoic acid, sebacic acid, (10-methoxycarbonylanthracen-9-yl) acetic acid,

3- (4,5-dimethoxy-2-nitrophenyl) acrylic acid, pentadecanoic acid,

- 170 -

4-chloro-3-methylbenzoic acid,

N- (3-chlorophenyl) malonamic acid,

2-phosphonobutyric acid,

3- (3-Trifluoromethylbenzyloxy) thiophene-2-carboxylic acid

2-ketobutyric acid,

4-chloropicolinic acid,

4,4,4-trifluoro-3-phenylacetylaminobutyric acid,

4-acetamido-3,5-dichlorobenzoic acid, gamma- (2-pyridyl) butyric acid,

2-aminophenol-6-sulfonic acid,

3-oxo-1,8-octanedioic acid,

1-naphthoxy-lactic acid, (L) -N-benzylglutamic acid,

4-Methyl-2-phenylpentanoic acid, (5-hydroxy-5H-dibenzo (a, d) cyclohepten-5-yl) acetic acid,

2-pyridin-3-ylquinoline-4-carboxylic acid, di-p-toluoyl-L-tartaric acid,

2-hydroxycyclohexanecarboxylic acid,

4-nitroisophthalic acid,

3,3,3-tris (4-chlorophenyl) propionic acid,

6 - [(4-amino-3-sulfophenyl) amino] -4-hydroxy-2-naphthalenesulfonic acid, (chlorophosphonomethyl) phosphonic acid, (S) - (4 -) - 2-phenylbutyric acid, 1-oxypyridin-4- sulfonic acid,

4-chloro-2,5-dimethylthiophenoxyacetic acid, β-methyl-3-nitro-cinnamic acid,

D, L-2- (4-hydroxyphenyl) -2-phenylacetic acid,

4-methylthio-3-nitrobenzoic acid,

L-isoleucyl-L-glutamic acid,

3-chlorobenzoic acid,

6-bromo-3,4-methylenedioxycinnamic acid,

N- (4-bromo-2-chlorophenyl) maleic acid, ··········

171

1-carboxy-4- (trimethylsilyl) cyclohexaneacetic acid,

10,12-tricosadioic acid, (+/-) - 2-hydroxytridecanoic acid,

7-oxo-4,5,6,7-tetrahydrobenzofuran-3-carboxylic acid,

5-chloro-2-phenylimidazo (1,2-a) pyrimidine-3-carboxylic acid,

2- (ortho-tolyl) butyric acid,

4- (4-azidophenyl) butyric acid,

2- (4- (3-oxo-3-phenyl-1-propen-1-yl) phenoxy] acetic acid,

9-oxo-6,7,8,9-tetrahydro-5H-benzocycloheptene-6-carboxylic acid, (3-bromopropyl) phosphonic acid, (+ -) - 9-hydroxy- (5Z, 7E, 11Z, 14Z) -icosatetraenoic acid, o-crotylphenoxyacetic acid,

3-phenylacetylaminobenzoic acid,

2-Methoxy-4-nitro-cinnamic acid

1-indanylmalonic acid,

2,3,5-trifluorobenzoic acid,

5-bromorotic acid,

3-Methoxy-2-nitrobenzoic acid

2,3-dimethoxy-9-oxo-6,7,8,9-tetrahydro-5H-benzocyclohepten-

-5-carboxylic acid,

5- (4-chlorophenyl) -2-methylfuran-3-carboxylic acid, dibenzoyl-D-tartaric acid,

3- (difluoromethoxy) benzoic acid,

3-ureidopropionic acid, omega-3-arachidonic acid,

1.3-propanedisulfonic acid,

3- (toluene-4-sulfonylamino) propionic acid,

3- (4-methoxybenzo (1,3) dioxol-5-yl) acrylic acid,

4-hydroxymethyl-3-methoxyphenoxyacetic acid, cyclopropane-1,2-dicarboxylic acid,

4- [4- / 4- (2-ethoxycarbonyl) cyclohexylmethyl / cyclohexyl] butyric

172 acid,

17-bromheptadecanoic acid,

4- [3- (2,3-xylyl) ureido] benzoic acid, fmoc-α-methylalanine,

D, L-erythro-4-fluoroflutamic acid, trans-2-pentenoic acid,

3- (2-Benzoxazolin-2-one-3-yl) propionic acid

3.4.5-Trifluorinic acid, benzene-1,3,5-tricarboxylic acid

2- (azocan-1-carbothioylsulfanyl) -2-methylpropionic acid, cis-N- (dodecyl) hexahydrophthalamic acid,

3-cyanethylbenzoic acid,

4.5.5.5-Tetrafluoro-4- (trifluoromethyl) pentanoic acid

5- (3- (Trifluoromethyl) phenyl) -2-pyrosylic acid,

4- (2- (3-benzyloxy-4-methoxyphenyl) ethylcarbamoyl) butyric acid, α-methyl-2-thiopheneacetic acid,

3- [N- (m-tolyl) carbamoyl] -5-norbornene-2-carboxylic acid,

N-α- (tert-butoxycarbonyl) -a- (methyl ester) -1-glutamic acid,

2-methyl-3-pyroslizic acid,

2.4.5- trichlorophenoxyacetic acid, cyclohexylphosphonic acid, cis-chrysanthemmonocarboxylic acid,

12-methyltridecanoic acid,

4,10-dioxo-9-oxatricyclo [6.2.1.0 (1.5)] undecane-2-carboxylic acid,

4-acetoxycinnamic acid,

4- (tetradecanamido) benzoic acid, (S) - (+) - phenylsuccinic acid, o-toluic acid, (+) - di-p-toluoyl-D-tartaric acid, (S) - (-) - 2-bromobutyric acid acid, *, and acid; and " ", " "

- 173 2,2'-azoxydibenzoic acid,

N-formyl-L-2-aminobutyric acid,

N-fmoc-2-amino-4- (dimethoxyphosphono) butanoic acid,

3-amino-5- (trifluoromethyl (benzoic acid,

4,4 (methandiyl (bis (iminocarbonyl)) bisbenzoic acid,

3- (trifluoromethyl (hydro-cinnamic acid,

12-tridecenoic acid,

12,12,12-trifluorododecanoic acid, phosphonoacetic acid,

2,5-bis (2,2,2-trifluoroethoxy (benzoic acid, methanilsulfonylsalicylic acid,

3-fluorocinnamic acid,

5-ketogluconic acid,

12 (R) -hydroxyicose-5Z, 8Z, 10E, 14Z-tetraenoic acid, (+/-) - camphoric acid,

3-benzoylpropionic acid,

10,10,10-trifluorodecanoic acid,

1-methyl-2-oxocyclohexanepropionic acid, gamma-methylene-D, L-glutamic acid, pth-cysteic acid,

7-nitro-9-oxo-2-fluorenecarboxylic acid,

3- [N- (4-methoxyphenyl (carbamoyl) -5-norbornene-2-carboxylic acid), α, β-dibromo-2-nitrohydrinnamic acid,

4'-bromo-2'-methyl-12,3,6-tetrahydrophthalanilic acid, isophthalic acid, n-propylphosphonic acid,

14-methylhexadecanoic acid,

2-bromo-3-methylvaleric acid, trans-cinnamic acid,

2,4,6-trimethoxycinnamic acid,

2- (3,5-dinitrothiophen-2-ylamino) (propionic acid,

4-pyridinebutylic acid,

- 174 -

3- [4- (4-carboxybutyl) phenyl] pentanoic acid,

N- (4-bromophenyl) malonamic acid,

2,2'-dichlorobenzilic acid,

2,5-dimethylbenzene-1,3-disulfinic acid,

4,5-dibromo-2-hexenoic acid,

4-carboxyphenoxyacetic acid,

3- (octyloxy) propionic acid,

3'-chloro-4'-fluorophthalanic acid,

5-chloroanilic acid,

5.6-dehydroarachidonic acid,

3- (3-methoxyphenyl) propionic acid, nonylphenoxyacetic acid, (IS, 3S) -1-amino-1-carboxycyclopentane-3-acetic acid,

3- (2-fluoro-4-nitrophenoxy) -2-thiophenecarboxylic acid, α-bromodiethylacetic acid,

1-Isoleic acid (2-hydroxy-3-methylvaleric acid)

4-carboxy-1,1-cyclohexanediacetic acid, sulfanilide dicarboxylic acid,

6-acetamidohexanoic acid,

3-chlorophenylacetic acid,

2- (2-propynyl) malonic acid,

3-hydroxy-2-trifluoromethylpropionic acid, n-tetradecylphosphonic acid, trans-styrylacetic acid,

3- (methylthio) benzoic acid,

2- (3,5-dinitrothiophen-2-ylamino) -3-phenylpropionic acid,

4´-ethyl-4-biphenylcarboxylic acid,

2,2-bis (trifluoromethyl) propionic acid,

3-Benzoyl-2- (2,3-dichlorophenyl) propionic acid

2,4-dimethylthiazole-5-carboxylic acid,

4-phenyl-1,2,3-thiadiazole-5-carboxylic acid,

Ν-α-Z-L-alanyl-L-aspartic acid,

3- (pivaloylamino) thiophene-2-carboxylic acid,

175

11- (toluene-4-sulfonyl) undecanoic acid,

4-hydroxyphenylpyruvic acid,

5-chloro-6-hydroxy-2-methylpyrimidine-4-carboxylic acid,

1,1-cyclobutanedioic acid, tert-butyl- (1,2,2-trichlorvinyl) phosphinic acid,

2 ', 3'-dichlorophthalanilic acid,

3-methylenecyclopropane-trans-1,2-dicarboxylic acid,

1-α-hydroxyisovaleric acid, cis-hexahydro-N- (4-methoxyphenyl) phthalamic acid,

4-nitrobenzoic acid,

4-undecyloxybenzoic acid, biphenylenacrylic acid, methylphenylphosphinic acid,

4- (4'-N-hexylphenyl) benzoic acid, '-broin-2'-methylphthalanilic acid,

N- (4-methoxyphenyl) glutaramic acid,

3,5-diacetamidobenzoic acid,

2.4.5- trimethoxybenzoic acid,

2- (2-allylphenoxy) acetic acid,

2-Trifluoromethyl-α-acetamidocinnamic acid,

1-amino-trans-cyclobutane-1,3-dicarboxylic acid,

4- (2-anthranoyl) butyric acid,

16-doxylstearic acid,

4,8-dioxoadamantane-1,2,5,7-tetracarboxylic acid, trans-2-benzoyl-1-cyclohexanecarboxylic acid,

2- (4- (6-bromo-1-hydroxy-2-naphthylazo) phenoxy] acetic acid,

4-nitrophenylacetic acid,

3,5-dibromo-4-hydroxyphenoxyacetic acid,

2,3-difluoromandelic acid,

3,5-bis (trifluoromethyl) phenylacetic acid, benzenesulfinic acid, N-glutaryl-L-phenylalanine p-nitroanilide, (S) - (-) - bromosuccinic acid,

- 176 phenylethynylphosphonic acid,

N-allylmaleinamic acid,

3-Benzoylamino-3- (2-fluorophenyl) propionic acid

1-naphthalenesulfonic acid, xylenesulfonic acid, succinemialdehyde,

6- (4-benzylphenyl) hexanoic acid,

3'-chloro-4'-fluoroformalic acid, dnp-D, L-glutamic acid, cis-hexahydro-N- (4-chloro-3-nitrophenyl) phthalamic acid,

1,3,4,5,6,8,8-heptamethyl-7-oxobicyclo (2,2,2) octa-2,5-diene-2-carboxylic acid,

2,3-difluoro-4- (trifluoromethyl) phenylacetic acid,

N-boc-1-aminocyclopropane-1-carboxylic acid,

4-methoxy-3-oxoindane-1-carboxylic acid, (R) -2-hydroxy-4-phenylbutyric acid,

4- (trifluoromethyl) phthalic acid,

3,4,4-triphenylbut-3-enoic acid,

6-chloro-2-nitrophenol-4-sulfonic acid,

N-t-boc- (2S, 3R) -3-amino-2-hydroxy-5-methylhexanoic acid,

4-methoxy-p-methylcinnamic acid,

3.3-dichloro-2- (4-methylbenzoylamino) acrylic acid,

1- (4-chlorophenyl) -5-oxo-3-pyrrolidinecarboxylic acid,

4-hydroxyphenylmalonic acid,

4 - [[4 - [(4,6-dimethylpyrimidin-2-yl) oxy] phenyl] amino] -4-oxo-

- (2Z) -butenic acid,

9- (4-methylphenyl) benzisoxazole-6-propenoic acid, (+/-) - 1-aminocyclopentane-cis-1,2-dicarboxylic acid,

7-oxo-16-heptadecenoic acid, cis-N- (3-chlorophenyl) hexahydrophthalamic acid, diendo-3-benzoylbicyclo (2,2,1) heptane-2-carboxylic acid, hexaoxabicyclo (18,3,1) tetracose- l (23), 20 (24), 21-triene-24-carboxylic acid, 4 t, 1 t, 1 t, 1 t, 4 · r · »

177

2-methyl-3- (2,4,6-trimethyl-3,5-dinitrophenyl) acrylic acid, (+/-) - 1-aminocyclopentane-trans-1,2-dicarboxylic acid,

2-nitrocinnamic acid,

3-hydroxy-4-methoxybenzoic acid,

1-benzocyclobutenecarboxylic acid, didodecyl phosphate,

5-ethoxy-1,3-benzenedicarboxylic acid,

3- [N- (2-phenethyl) carbamoyl] -5-norbornene-2-carboxylic acid,

3-phenyl-spiro (5,5) undecane-3-carboxylic acid,

2,5-pyridinedicarboxylic acid, p-chlorophenyl (benzyl) acetic acid,

4-methyl-3b, 4,4a, 5-tetrahydrocyclopropa (a) phenalene-4-carboxylic acid, α-ethyl-m-nitro cinnamic acid,

3-amino-5-sulfosalicylic acid,

19-bromnonadecanoic acid,

1.2.3.4-tetrahydro-2-naphthalene butyric acid,

4-Benzyloxycinnamic acid

3-benzoyl-2-phenylpropionic acid,

4'-chlorosuccinanilic acid, meta-phenylenediamino-2-sulfonic acid,

1-Methyl-5-oxo-3-pyrrolidinecarboxylic acid

2- [4- (2-hydroxy-1-naphthylazo) phenoxy] acetic acid,

3,4-dimethoxy-2-hydroxybenzoic acid, n-phenylmalonamic acid,

1,6-naphthyridine-2-carboxylic acid,

3-ethoxycarbonylmethyl-1H-indole-2-carboxylic acid,

2'-ethoxyphthalanilic acid,

2,5-dibenzyloxyphenylacetic acid,

2 ', 4'-dimethylsuccinanilic acid,

N- (2-fluorophenyl) glutaramic acid, 4 9 9 9 9 9 9 9 9 9 9 9 9 9 9 · 9

9,999 * ·

9 ··· ··· 99 9 9 99999

- 178 -

1- (2,4-dimethylphenyl) -6-methyl-4-oxo-1,4-dihydro-3-pyridinecarboxylic acid, farnesylthioacetic acid,

3-hydroxy-4-methylbenzoic acid,

1-Methyl-4,9-dihydro-3H-3-carboline-3-carboxylic acid

4,4-dichloro-5,5,5-trifluoropentanoic acid,

5-bromosalicylic acid,

2-carbamoyl-6-nitrobenzoic acid,

4-Naphthalimidobutyric acid

9 (10) -bromstearic acid, glutaranilic acid,

3-trifluoromethyl-3-hydroxybutyric acid, fmoc-L-1,2,3,4-tetrahydronorharman-3-carboxylic acid,

2,4-pyridinedicarboxylic acid,

3- [3- (2,3-dichlorophenyl) ureido] benzoic acid,

3-deoxy-D-glycero-D-galacto-2-nonulosonic acid,

2- (4-chlorophenoxy) propionic acid, (+) - N-pinacolylphthalamic acid,

D-gamma-carboxyglutamic acid, (S) -1,4-benzodioxane-2-carboxylic acid, fmoc- (D, L) -2-aminotetraline-2-carboxylic acid, (S) -3-acetoxy-4-bromobutyric acid acid,

2-hexadecyloxy-5-sulfobenzoic acid, podocarpic acid, (-) - cis, trans-abscisic acid, fmoc-α-aminobutyric acid,

2- (3-nitrobenzylidene) tridec-12-enoic acid, [1- (4-hydroxyphenoxy) ethylidene] bisphosphonic acid,

3-ethoxyphenylacetic acid,

3- (hexadecanamido) benzoic acid, (4,5-dimethoxy-3-oxo-1,3-dihydroisobenzo-1-furyl) acetic acid,

2- (3-acetyl-4-hydroxyphenylcarbamoyl) cyclohex-1-enecarboxylic acid

- 179 acid,

4- (bromomethyl) phenylacetic acid,

2-butoxy-5-tert-pentylbenzenesulfonic acid, metaphosphoric acid, trans-4-hydroxy-2-butenoic acid,

1,3,5-pentanetricarboxylic acid,

4-aminobutylphosphonic acid,

3,4-dimethoxycinnamic acid,

N- (2-phenethyl) phthalamic acid,

2,6-heptadienoic acid,

6-oxo-1, 12-dodecanedioic acid,

2-chloro-3,5-dinitrobenzenesulfonic acid,

N-phthaloylglycine,

2-Naphthol-3,6,8-trisulfonic acid,

2,2,4,4,5,5,7,7,8,8,10,10,10-tridecafluoro-3,6,9-trioxadecanoic acid,

2,3: 4,6-di-o-isopropylidene-2-keto-L-gulonic acid, cis-2- (4-fluorobenzoyl) -1-cyclohexanecarboxylic acid, dichloromethylphosphonic acid, n-octylmaleinamic acid, phthalid-3- acetic acid,

2,3-dibromo-3 ', 4'-dichlorosuccinanilic acid,

2-acetamido-5-bromobenzoic acid, (2-bromo-4-methylphenyl) phosphonic acid,

2-hydroxy-4,6-dimethoxybenzoic acid, boc-iminodiacetic acid, methylene-bis (3-thiopropionic acid), dithioterephthalic acid, home acid,

3-Methylphenoxyacetic acid

2-methyl-3- (3-nitrophenyl) acrylic acid,

4-methyl-1,1-cyclohexanediacetic acid,

2-acetamido-4-fluorobenzoic acid,

- 180 -

1-Methyl-2-cyclohexene-1-carboxylic acid

4'-chlorophthalanilic acid,

3-formylphenoxyacetic acid, α-truxillic acid,

4- (2-nitrophenyl) butyric acid,

N-methylsuccinamic acid,

2'-benzylcarbamoylbiphenyl-2-carboxylic acid,

3- (1,3-dioxo-1,3-dihydroisoindol-2-yl) benzoic acid,

2-Methyl-5-norbornene-2-carboxylic acid

3-ethoxy-4-methoxybenzoic acid,

2- (fluoranthene-8-carbonyl) benzoic acid,

3- (2,3-dimethoxyphenyl) propionic acid,

R-4-bromomandelic acid,

4-acetamidicinnamic acid, (2-methoxyphenyl) phenylphosphinic acid,

6-hydroxy-2-naphthoic acid, (S) - (+) - N- [4 - [(aminoiminomethyl) amino] -1-carboxybutyl] -D-glutamic acid,

2,4,6-trimethoxyphenylacetic acid,

3-methylpyrazolo (3,4-b) quinoline-4-carboxylic acid,

3-aminomethylalizarin-N, N-diacetic acid,

N- (5-chloro-2-methylphenyl) maleic acid, dnp-L-glutamic acid,

2- (4-Biphenylyloxy) propionic acid

4-hydroxy-6- (trifluoromethyl) -3-quinolinecarboxylic acid, aniline-2,4-disulfonic acid, (S) - (-) - α-phenethylsulfamic acid, - (4-nitrophenyl) butyric acid,

4- (4-methoxy-2-methylphenyl) -4-oxobutyric acid,

3- (2-oxo-1,3,3-trimethylcyclohexyl) propionic acid,

4'-butyl-1,2,3,6-tetrahydrophthalanic acid, (R) -1,4-benzodioxane-2-carboxylic acid,

2- (2-ethoxyphenylcarbamoyl) cyclohexanecarboxylic acid,

181

6-hydroxy-3-oxo-3H-xanthene-9-carboxylic acid, phenylphosphinic acid,

4-methylcinnamic acid,

N-Naphthalen-1-ylsuccinamic acid

2-Methyl-5,6-dihydro (1,4) oxathiine-3-carboxylic acid

3-bromo-4-hydroxyphenylacetic acid, tricyclo [2.2.1.0 (2.6)] heptane-1-carboxylic acid,

3-methyl-3-phenylpentanoic acid,

1- (2-chlorobenzoyl) piperazine-2,3-dicarboxylic acid, ethylmandlate,

2-propyldecanoic acid, (R) - (+) - α-phenethylsulfamic acid,

3,5-dimethyl-1-cyclohexene-1,2-dicarboxylic acid,

3- (pyrrolidine-1-carbothioylsulfanyl) propionic acid,

2,2'-dithiodipropionic acid,

2- [3,5-bis (trifluoromethyl) benzoyl] benzoic acid,

4-fluorobenzoic acid,

2-fluorisophthalic acid,

3- (5- (2-chloro-5-trifluoromethylphenyl) -2-furyl] -2-cyanoacrylic acid,

5- (4-chlorophenylsulfanyl) furan-2-carboxylic acid, (S) - (-) - 2-chlorosuccinic acid,

S- (thiobenzoyl) thioglycolic acid,

5-hydroxy-2-nitrobenzoic acid, α-methyl-p- (2-thenoyl) phenylacetic acid, 3H-tetrafluoropropionic acid,

4-ethylthiobutyric acid,

3-fluoro-2,4-dimethylbenzoic acid, (2-methyl-4-nitrophenyl) phosphonic acid,

2-ethyl-3- (2-methoxyphenyl) acrylic acid,

3,5-dinitro-o-toluic acid,

2- (4-chlorophenyl) -3- (3-methylbenzoyl) propionic acid,

4-phenylvaleric acid,

- 182 (4-iodophenyl) phenylphosphinic acid, benzophenone-2,4'-dicarboxylic acid,

2-phthalimidoglutaranilic acid,

5-butylhydanoic acid, (2-hydroxynorboran-2-yl) phenylacetic acid,

2 - [(5-oxotetrahydro-1H-2-pyrrolyl) sulfanyl] acetic acid,

1,4-phenylenedipropionic acid,

N-furfurylmaleinamic acid,

4-methoxy-butyric acid, octahydro-6-oxo-6H-pyrido (3,2,1-j) carbazole-11b-propionic acid,

1-chloro-3-methylisoquinoline-4-carboxylic acid, benzyloxycarbonyl-L-aspartic acid β-benzyl ester,

2-chloroacrylic acid,

2,3-dimethylfuran-5-carboxylic acid,

2,6-dimethyl-3,5-pyridinedicarboxylic acid, cis-2,6-piperidinedicarboxylic acid, cis-hexahydro-N- [3- (trifluoromethyl) phenyl] phthalamic acid, trans-D, L-1,2-cyclopentanedioic acid,

2-hydroxy-3-isopropylbenzoic acid, phenoxyacetic acid,

N- (2-ethyl-6-methylphenyl) -3-nitrophthalamic acid,

2-iodo-5-nitrobenzoic acid,

5- (4-chloro-3-nitrophenylsulfamoyl) isophthalic acid,

6-methyl-2,3-pyridinedicarboxylic acid,

N-formyl-L-aspartic acid,

5-hydroxypyrazine-2-carboxylic acid,

2- (2,4-dimethylbenzoyl) benzoic acid,

5-bromo-2-chlorobenzoic acid,

2- (9H-xanthen-9-yl) malonic acid, cis-2 ', 4'-dimethylhexahydrophthalanic acid,

2,3,4,5-tetramethylbenzoic acid,

2- [7-oxo-7H-benz (d, e) anthracen-3-ylthio] acetic acid;

- 183 N- (p-tolyl) phthalamic acid,

4,4'-isopropylidenediphenoxyacetic acid, (IR, 2R) - (-) - 1,2-cyclohexanedicarboxylic acid,

4-fluoro-3- (trifluoromethyl) cinnamic acid, d-pantothenic acid,

4.5-imidazole dicarboxylic acid,

4- (2,4-dichlorobenzylideneamino) benzoic acid,

2-methylthio-5-benzothiazolesulfonic acid, benzo (b) thiophene-2-carboxylic acid,

5-benzoyl-7-bromo-2,3-dihydro-1H-pyrrolizine-1-carboxylic acid,

1- (3-fluorophenyl) cyclopentanecarboxylic acid, bromodichloroacetic acid, (+/-) - 2-hydroxyundecanoic acid,

2-butoxyacetic acid,

3-ethenesulfonylpropionic acid, pentafluorophenoxyacetic acid,

3-methyl-4-cyclohexene-cis-1,2-dicarboxylic acid, bicycio (2,2,1) heptane-2-carboxylic acid,

3- (4-methylsulfanylphenyl) acrylic acid,

5-norbornene-2-acrylic acid,

3,5-dimethyl-4-nitrobenzoic acid,

2-propylpentanoic acid,

1-cysteic acid, cinnamylidenemalonic acid,

5-formyl-2-thiophenecarboxylic acid, D, L-4-hydroxymandelic acid,

5- (hydroxyimino) azelaic acid,

2,3-naphthalenedicarboxylic acid, n-butylpyrophosphate, n-octadecylglutaramic acid, n-cyclohexylmaleinamic acid, dansyl-1-cysteic acid, c184 m-cresylgulutaric acid,

3-Hexadecyloxy-4-nitrobenzoic acid

5-nitro-2-propionamidobenzoic acid,

N, N-dibenzylhexahydrophthalamic acid,

4-methoxycarbonylsulfanyl-3-nitrobenzoic acid, ricinoleic acid, cis-12-octadecenoic acid,

3- (methylphosphinoyl) propionic acid, methylenebisthioglycolic acid,

2-methylcinnamic acid, (S) -2-chloro-n-butyric acid,

2-bromopropionic acid,

5-chloro-2-methoxybenzoic acid,

2-methylhexanoic acid,

2,6-bis (trifluoromethyl) benzoic acid,

4'-fluoro-3,4,5,6-tetrachlorophthalic acid,

3- (3,4-dichlorophenylamino) butyric acid, dimethylphosphinic acid,

2-hydroxy-3-butenoic acid,

2,3,4-trimethyl-5-nitrobenzoic acid,

2-hydroxy-3 (S) - (N-tert-boc-amino) -4-methoxybutanoic acid,

2- (3,4-dichlorobenzoyl) benzoic acid,

3,5-dibenzyloxybenzoic acid,

4- [4- (4-chlorobenzenesulfonyl) phenoxy] benzoic acid,

1-Naphthol-5-sulfonic acid

2-acetyl-3,6-difluorobenzoic acid, (R) - (+) - trolox ^(R) , cresolsulfonic acid,

2-oxo-1,1,3,3-cyclohexanetetrapropionic acid, (D, L) -2- (4-biphenylyl) propionic acid, palmitlaic acid, (10,11-dihydrodibenzo (a, d) cyclohepten-5-ylidene) 44)

185 acid,

5-bromo-2-methoxyisophthalic acid,

3-Methyl-4-p-tolylbutyric acid

2-anthracenecarboxylic acid,

4'-chloro-3,4,5,6-tetrachlorophthalic acid,

1-hydroxycycloheptanecarboxylic acid,

4-acetylphenoxyacetic acid,

3-fluoro-4- (trifluoromethyl) cinnamic acid, cis-hexahydro-N-phenylphthalamic acid, cis-13,16,19-docosatrienoic acid, hexacosanedioic acid,

2'-methyl-3,4,5,6-tetrachlorophthalanic acid,

4- (6-hydroxy-3-oxo-3H-xanthen-9-yl (benzoic acid, [4- (4-ethylphenoxy) phenoxy] acetic acid), (+/-) - cis-9,10-methylenoctadecanoic acid,

2-Benzoylamino-3- (ethoxyphenylphosphinoyl) -3-phenylacrylic acid

5- (4-chlorobenzoyl) thiophene-2-acetic acid,

9-anthracenepropionic acid,

4-Phenetidine-2-sulfonic acid

2- (bromomethyl) acrylic acid,

2-heptenic acid,

2,4-dibromophenoxyacetic acid, benzo (c) phenanthrene-5-carboxylic acid,

9- (10) -hydroxyphenylstearic acid,

R-4-chlorormanedioic acid,

5-fluoro-2,3-dihydro-gamma-oxo-1- (1H) -indolbutanoic acid, (S) -tetrahydrofuran-2-carboxylic acid, p-butoxybenzoic acid,

2- (4-nitrobenzoylamino) -3-phenylacrylic acid,

4-hydroxy-7-methoxy-1- (3-methoxyphenyl (naphthalene-2-carboxylic acid),

3- (4-Isopropylphenyl) -2-methylacrylic acid, ···········

- 186 difluoroacetic acid, cis, cis, cis, cis-1,2,3,4-cyclopentantetracarboxylic acid,

3-methyldecanoic acid, boc-D-pipecolic acid, (+/-) - 2-endo-aminobicyclo (2,2,1) heptane-2-exo-7-anti-dicarboxylic acid,

4'-fluoro-3,3 ', 4,5,6-pentachlorophthalic acid,

4-fluoro-3-nitrobenzoic acid,

2-Methyl-3,4,6-pyridine-tricarboxylic acid

3-Methylsulfonylbenzoic acid

2- (hexadecylsulfonyl) benzoic acid, isoindolin-1-one-2- (2-propionic acid), cis-5-norbornene-endo-2,3-dicarboxylic acid,

9-phenylnonanoic acid,

2-fluoro-5- (trifluoromethyl) benzoic acid,

2 '4', 5'-trichlorglutaranilic acid, meta-sulfophenyl-gamma-acid, α-methyl-2-thiophenacrylic acid, sulfuric acid,

6-amino-1,3-naphthalenedisulfonic acid,

6,9,12,15-octadecatetraenoic acid,

3- (2-ethoxyphenyl) propionic acid,

3-carboxy-1,4-dimethyl-1H-pyrrole-2-acetic acid, rhodanine-N-carboxylic acid, fmoc-3-abz-oh, 1-amino-9,10-dihydro-4-hydroxy-9, 10-dioxo-2-anthracenesulfonic acid,

4-bromo-1-hydroxy-2-naphthoic acid, chelidonic acid,

N- (2-cyanophenyl) tetrachlorophthalamic acid, (4-chlorophenylthio) acetic acid,

4-oxo-1,9-nonanedicarboxylic acid,

N- (3,4-dichlorophenyl) maleic acid,

187

4-Acetoxy-3-methoxybenzoic acid

2-Methoxy-5-methylbenzoic acid

5-Methyl-4-nitroisophthalic acid

5-chlorobenzofuran-2-carboxylic acid,

1- (4-chlorophenyl) -1-cyclohexanecarboxylic acid,

5-chloro-2-fluorobenzoic acid,

7-hydroxy-1,3,4-triazindolizine-5-carboxylic acid,

1-pyrendodecanoic acid,

3- (4-chlorobenzoyl) -2- (2-chloro-6-fluorophenyl) propionic acid,

2-chloro-6-methylbenzoic acid,

N- (4-bromo-2-methylphenyl) maleamic acid, vinylphosphonic acid,

4- (2-o-tolyloxyacetylamino) benzoic acid,

3-tert-butyl-6-methylsalicylic acid, carboxypyrazolone,

3-nitrophthalic acid,

2-bromo-4-hydroxy-5-methoxyphenylacetic acid, undecanoic acid,

1,3-diamino-2-hydroxypropane-N, N, N ', N'-tetraacetic acid, pent-3-enoylaminacetic acid,

2,3-dimethylbutyric acid, ', 4'-dimethyl-3,4,5,6-tetrachlorophthalanic acid,

2-hydroxyamino-3-methylpentanoic acid,

N- [4 '- (toluene-4-sulfonylamino) biphenyl-4-yl] succinamic acid,

4- [N '- / 2-oxo-1- (toluene-4-sulfonyl) propylidene / hydrazino] benzoic acid,

11- (phenylthio) undecanoic acid,

2-hydroxyamino-2-methylpropionic acid,

14,15-epoxy- (5Z, 8Z, 11Z) icosatrienoic acid,

2-phenoxymethylbenzoic acid, (3-ho-3-ph-4H-4H-1-thia-3α, 7-diaza-cyclopenta (a) pentalen-2)

188

-yl) acetic acid,

4'-sulfamoylglutaranilic acid, [[2- (3,4-dimethoxyphenyl) ethyl] - (toluene-4-sulfonyl) amino] acetic acid,

2- [4- (trifluoromethyl) phenylthio] acetic acid,

15-bromopentadecanoic acid,

2-hexyl-3- (2-methoxyphenyl) acrylic acid, (trimethylsilyl) acetic acid,

2- (4-hydroxyphenyl) propionic acid, pyrrole-3-carboxylic acid,

N- (3-indolylacetyl) -D, L-aspartic acid, phenyl- (3,5-xylyl) phosphinic acid,

3 ', 4'-dichlorosuccinanilic acid,

1,6-dihydro-6-oxo-1,2,5-trimethyl-3-pyridinecarboxylic acid,

1- (4-Isopropylphenyl) -6-methyl-4-oxo-1,4-dihydro-3-pyridinecarboxylic acid,

3-chloro-4-hydroxymandelic acid,

3- (methoxycarbonylthio) propionic acid,

3- (3,4-dimethoxyphenyl) -2-formylaminopropionic acid,

3- (p-methoxyphenyl) -2-phenylpropionic acid, cis-11-icosenoic acid,

4- [ac- (5-nitro-1,3-dioxo-1,3-dihydroisoindol-2-ylmethyl) amino] benzoic acid,

5'-isopropyl-2'-methyl-3,4,5,6-tetrachlorophthalanic acid,

5-bromo-2-fluorobenzoic acid, tetrahydro-2-pyroslizic acid, (R) - (-) -? - [[(4-ethyl-2,3-dioxo-1-piperazinyl) carbonyl] aminobenzeneacetic acid, (trans) , trans) -abscisic acid,

3-chloropropionic acid, (-) - menthoxyacetic acid,

- 189 4'-butylglutaranilic acid,

4'-hydroxyglutaranilic acid,

4-oxo-2,3,4-triphenylbutyric acid,

1,2.4-butantricarboxylic acid, cis-3-hexenoic acid, allo-gibberic acid,

2- (1,3-dioxo-1,2,3,4-tetrahydro-2-isoquinolyl) acetic acid,

4-Decyloxybenzoic acid, (3-et-9,10-dimethoxy-4-oxopyrido (2,1-a) isoquinolin-2-yl) acetic acid, (Z) -2- (2-chloroacetamido) -a- ( methoxylmino) -4-thiazoleacetic acid,

2-methoxy-9-oxo-6,7,8,9-tetrahydro-5H-benzocycloheptene-6-carboxylic acid,

4- [3- (2-Phenoxyacetyl) -2-thioureido] benzoic acid,

9,10-epoxyoctadecanoic acid,

D, L-p-phenyl lactic acid, imidazo (2,1-b) benzothiazole-2-carboxylic acid,

3-Methoxy-4-nitrobenzoic acid

2,4-diphenylfuran-3-carboxylic acid,

1,2-dihydro-2-methyl-1-oxo-3-isoquinoline butyric acid,

2- (cyclohexanecarbonylamino) benzoic acid,

2,3-diphenylsuccinic acid, cis-7,10,13,16,19-docosapentaenoic acid,

3,3'-tolidine-5-sulfonic acid,

2-Methoxy-1-naphthoic acid

3- (2-methoxyphenyl) propionic acid,

N- (4-fluorophenyl) malonamic acid, (-) - perilic acid, gamma-L-glutamyl-L-glutamic acid, tartronic acid,

4-Benzyloxyphenylacetic acid

N- (3,5,6-trimethylcyclohexyl) maleic acid,

• • •

190 (3,3-dimethyl-5-oxocyclohexylideneamino) acetic acid, D-threo-4-fluoroglutamic acid, (Z) -styrylthiopropionic acid, β-inaleinimidopropionic acid, chlorfumaric acid,

4-chloro-3-nitro-5-sulfonamidobenzoic acid, phenylphosphoric acid,

1.2-ethylenediphosphonic acid, fmoc- (3-aminomethyl) benzoic acid, boc-D-p-aminobutyric acid,

3- (4-hydroxyphenyl) propionic acid,

4,4 '- (trichloromethylmethylene) disalicylic acid, (4-formyl-3-methoxyphenoxy) acetic acid, (4-nitrophenyl) phosphonic acid, (1-R, S) -trans-permethric acid,

4-isobutyl cinnamic acid,

3.4- dibromobenzoic acid,

4'-methyl-3'-nitrosuccinanilic acid, phthalamic acid,

5-chlorosulfonyl-2-hydroxybenzoic acid,

3,4,5-tribromobenzoic acid,

2'-nitromaleanilic acid,

D - (-) - α-azidophenylacetic acid,

2,2-dihydroxy-3,3,3-trichloropropionic acid,

3 ', 4'-dimethylglutaranilic acid,

2,6-dichloro-cinnamic acid,

3-nitrohippuric acid,

3,4-dimethoxy-6-nitro-cinnamic acid, boc-1-indoline-2-carboxylic acid,

2-chloro-4-fluorobenzoic acid,

10-oxoundecanoic acid, (3-methyl-5-nitrophenyl) phosphonic acid,

3- (1,1,2,3,3,3-hexafluoropropyl) adamantane-1-carboxylic acid

191 acid, tricyclo [8,2,3,2 (4,7)] hexadeca-hexaene-2-carboxylic acid,

3,4-dimethoxybenzoic acid,

4-bromo-3,5-dihydroxybenzoic acid, o- (3,6-dichloroanilino) benzoic acid,

N-carbamoyl-α-anionic butyric acid, N-1-trityldeaminohistidine,

4-phenoxybenzoic acid, α-acetylmandelic acid,

3- (5-nitro-2-furyl) acrylic acid,

3 ', 5'-dimethoxymaleanilic acid,

3,5-dinitro-p-toluic acid,

4'-methyl-2'-nitromaleanilic acid,

2-bromophenoxyacetic acid,

2-chloroisobutyric acid,

3,5-dibromlevulinic acid, cis-13,16-docosadienoic acid,

4'-acetylphthalic acid,

2-chlorhippuric acid,

4- (4'-hydroxyphenyl) benzoic acid,

1-naphthoic acid,

12 (S) -hydroxy-16-heptadecinic acid, (2-cyclopenten-1-yl) malonic acid,

2'-methoxyphthalanilic acid,

3'-methyl-3,4,5,6-tetrachlorophthalic acid,

5-doxylstearic acid,

3,4-xylylphosphonic acid, (2-sec-butylphenoxy) acetic acid, adamantan-1-ylphosphonic acid, 1- (2,4-dichlorophenyl) -4-carboxytriazole acetic acid,

2,6-dichloro-5-fluoro-3-pyridinecarboxylic acid, tridecanoic acid, (2-ethylphenyl) phosphonic acid,

- 192 (S) -2-fluoro-2-methylhexanoic acid,

3-hydroxy-1-adamantanacetic acid,

3- (4-chlorobenzoyl) -2- (2,3-dichlorophenyl) propionic acid,

2 - [(3-carboxypropyl) - (toluene-4-sulfonyl) amino] -4-chlorobenzoic acid, (2,6-xylyl) phosphonic acid,

1-Aminoanthraquinone-2-sulfonic acid

5- (2,5-dimethoxyphenyl) -5-oxopentanoic acid,

4- (4-methyl-2,6-dinitrophenylamino) butyric acid,

3,5-dichlorobenzoic acid,

3-sulfobenzoic acid, bis (phenacyl) acetic acid, (3-benzylphenyl) acetic acid, (1R, 3S) -1-aminocyclopentane-1,3-dicarboxylic acid, cbz-D-1,2,3,4-tetrahydroisoquinoline -3-carboxylic acid, p-phenolsulfonic acid, perhydrocyclobutane (1,2: 3,4) dicyclopentene-2,5-dicarboxylic acid,

2- (2-oxo-1,2-dihydroindol-3-ylideneamino) benzoic acid, nonadecanoic acid,

4-aminophthalic acid,

4-acetylbutyric acid, chaulmogric acid,

3- (n-hexadecylcarbamoyl) -5-norbornene-2-carboxylic acid, phenylphosphonic acid, n-propylmaleinamic acid, benzyloxycarbonyl-2-aminobutanoic acid (L-Z-2-aminobutyric acid),

1- (4-methoxyphenyl) -1-cyclopropanecarboxylic acid,

3-chlorododecanedioic acid, (2-imino-4-oxothiazolidin-5-yl) acetic acid, ethylenediamino-N, N'-diacetyl-N, N'-di-α-propionic acid,

2-hydroxy-2-trifluoromethyldec-4-enoic acid,

- 193 -

3-nitro-5-sulfosalicylic acid,

9-hydroxy- 9H-fluorene-1-carboxylic acid

N-m-tolylphthalamic acid, phenylsuccinic acid, (S) - (-) - 2-methylglutaric acid,

4-fluoro-3-methoxybenzoic acid, ³ 15-pyrazole dicarboxylic acid,

2,3-dibromo-3- (p-chlorophenyl) propionic acid,

1,6-diphenyl-1,3,5-hexatriene-4'-acetic acid,

2H- (1,2,4) triazole-3-carboxylic acid

9,10-dihydro-9,10-dioxo-2,3-anthracenedicarboxylic acid,

4-Isopropylphenylacetic acid

2-bromotetradecanoic acid,

2- (3,5-di-tert-butylbenzoylamino) benzoic acid, valeric acid,

2-phenyl-1H-imidazole-4,5-dicarboxylic acid,

2-hydroxyoctadecanoic acid, bisacrylamidacetic acid,

4'-methyl-3'-nitrophthalanilic acid,

2-phosphonopropionic acid, chloroacetyl-L-gamma-glu-p-aminobenzoic acid,

3-ethoxycinnamic acid,

3-methyl-3H-imidazo (4,5-b) pyridine-2-sulfonic acid,

7-chloro-2,2,3,3,4,4,5,5,6,6,7,7-dodecafluoroheptanoic acid,

3,5-dichloro-4-hydroxybenzoic acid,

3- (3,5-dimethylphenyl) -3-methylbutyric acid,

3,5-dibromo-4-hydroxybenzoic acid, tricyclo [8,2,2,2 (4,7)] hexadeca-hexaen-5-ylacetic acid, α-cyanocinnamic acid,

2-bromisovaleric acid,

3-chlorobenzo (b) thiophene-2-carboxylic acid,

7-hydroxy-4-methylcoumarin-3-acetic acid,

194

N- (4,6-dimethylpyrimidin-2-yl) -N-methyl-4-aminobenzoic acid, methanedisulfonic acid, isatin-n-acetic acid, (2-benzyloxy-3-methoxyphenyl) acetic acid,

3-cyanobenzoic acid,

2.5-difluorophenylacetic acid, citric acid, ximeninic acid,

3-chloro-2,6-dimethoxy-5-nitrobenzoic acid,

3-methylsalicylic acid, diphosphoric acid, xanthene-9-carboxylic acid,

7-methoxybenzofuran-2-carboxylic acid,

2.4.5- trichlorobenzenesulfonic acid, m-iodophenylacetic acid,

2-benzoyl-3,4,5,6-tetrachlorobenzoic acid, phenylthiohydantic acid, myristlaic acid,

4 '- (ethoxycarbonyl) succinanilic acid, (R) - (-) - 2,2-dimethyl-5-oxo-1,3-dioxolane-4-acetic acid,

4-acetylbenzoic acid,

4-amino-2-nitrobenzoic acid,

2- (2,5-dimethylbenzoyl) acrylic acid, gamma-oxo-2-naphthalene butyric acid, 2-bromo-3-chlorobenzoic acid, p-toluenesulfinic acid,

1-benzyl-1,2,3-triazole-4,5-dicarboxylic acid,

12 (S), 20-dihydroxyicose-5Z, 8Z, 10E, 14Z-tetraenoic acid,

7-benzoylheptanoic acid,

2,6-dihydroxybenzoic acid,

4-chloro-2-methylbenzoic acid,

3'-nitroglutaranilic acid,

- 195 -

2,5-dimethyl-3-pyrosylic acid, (S) -2-methyldodecanoic acid,

L-boc-piperidine-4-carboxylic acid, dichloroacetic acid, α-phenyl cinnamic acid, benzyloxycarbonyl-L-glutamic acid gamma-tert-butyl ester, docosanedioic acid,

1- (2,4-dichlorophenyl) cyclopropanecarboxylic acid, m-nitrobenzoic acid sulfone, (R, S) -α-methoxy-α-trifluoromethylphenylacetic acid, N-phthaloyl-L-glutamic acid, [5- (1-ho- 2,2,6,6-tetramethyl-1,2,3,6-4H-pyridin-4-yl) -thiophen-2-yl) acetic acid,

3- (3-methoxybenzoyl) adipic acid,

3,6-epoxycyclohexane-1,2-dicarboxylic acid,

2-Bromo-1-naphthalenesulfonic acid

4- (trifluoromethoxy) benzoic acid,

N-α- (benzyloxycarbonyl) -a- (benzyl ester) -1-aspartic acid,

D, L-threo-3-hydroxyaspartic acid,

3- (2-Methylsulfanyl-benzothiazol-6-ylamino) -propionic acid

5-bromo-2,3-dihydrobenzofuran-7-carboxylic acid,

3- (2,3,5,6-tetramethylbenzoyl) acrylic acid,

2- (1,3-benzodioxol-5-yl) -1-methyl-5-oxo-3-pyrrolidinecarboxylic acid,

3- (2- (2-carboxybenzoylamino) ethyl) -5-chloro-1H-indole-2-carboxylic acid,

2.4- dihydroxybenzoic acid,

3- (4-fluorophenoxy) propionic acid,

6-oxo-1,11-undecanedicarboxylic acid,

2.4- Difluoric cinnamic acid, 9 9

9 9 9 9 999 · · ·

- 196 -

5-chloro-N- (2-chloroacetyl) anthranilic acid,

3- (4-nitro-1,3-dioxo-1,3-dihydroisoindol-2-yl) benzoic acid, quercetinsulfonic acid,

6-methyl-1- (3-methylphenyl) -4-oxo-1,4-dihydro-3-pyridinecarboxylic acid,

N- (4-carboxy-3-hydroxyphenyl) maleimide

2,3-dihydroxy-4-methoxycinnamic acid, fmoc-gamma-amino-butyric acid,

2- (2,4-dichlorophenylthio) acetic acid,

2,2'-oxydibenzoic acid,

1-Pyrenecarboxylic acid

9-fluorenone-1-carboxylic acid, (2-acetyl-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-1-yl) acetic acid,

3-n-propoxypicolinic acid,

S-benzylthioglycolic acid,

4- [4- / 3- (4-bromophenyl) -3-oxopropyl / phenyl] -4-oxobutyric acid,

N-benzylmaleinamic acid,

N- (4-chlorobenzoyl) aminoacetic acid, undecylenic acid,

2- (2,4-dimethylbenzoyl) -3-methylbenzoic acid,

2-acetylamino-4,5-dimethylthiophene-3-carboxylic acid, cyclohexane-1,1-bis (mercaptoacetic acid),

2- (3,4-dimethoxybenzoyl) benzoic acid,

2- (3-oxo-1-indanyl) acetic acid,

2-chloro-4-toluidine-6-sulfonic acid,

2- (1-ethoxycarbonylamino) benzoic acid,

N- (2,4-difluorophenyl) maleic acid,

1-aminocyclobutane-cis-1,3-dicarboxylic acid,

6,8-nonadecadiic acid,

3-Phenyl-7-fluoro-1-oxoindane-3-carboxylic acid, 3-carboxylic acid, 3-phenyl-7-fluoro-1-oxoindane-3-carboxylic acid «· · · ··· * · ·

197 boc-1-amino-1-cyclohexanecarboxylic acid,

3,3'-dithiobisbenzoic acid,

3-dodecanoylaminobenzoic acid,

4- [3- (2,2,2-trichloro-1-isobutyrylaminoethyl) thioureido (benzoic acid,

2-phenyllevulinic acid,

3-bromo-5-methoxybenzoic acid,

3-acetimidoylsulfanylpropane-1-sulfonic acid,

4-benzyloxybenzoic acid,

9,10,18-trihydroxyoctadecanoic acid,

3- [3,4- (trimethylenedioxy) benzoyl] propionic acid, (S) -2-benzylsuccinic acid, (2-oxobicyclopentyl-1'-en-1-yl) acetic acid,

4- [2- (4-chlorobenzoyl) acetamido (benzoic acid,

N-boc-D-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid,

4- (4-chlorophenylsulfonyl (benzoic acid, boc-L-2-aminosubric acid, farnesylic acid,

2-bromo-4,5-dimethoxycinnamic acid,

Ν-α-boc-glycyl-L-aspartic acid,

4,6-phenoxathiindicarboxylic acid,

3-nitro-4- (3-chlorophenoxy (cinnamic acid,

3-bromopyruvic acid, pentafluorophenylpropionic acid, lactone D, L-isocitronic acid,

3- [4- / 5- (4- (2-ethoxycarbonyl) phenyl) pentyl / phenyl (propionic acid,

2-methoxyphenoxyacetic acid,

1,2-ethanedisulfonic acid,

3,5-dinitro-2-fluorobenzoic acid,

2-ethoxyphenylacetic acid,

3-fluoro-4- (trifluoromethyl) benzoic acid,

3-p-tolylbutyric acid,

198

2- (5-nitro-1,3-dioxo-1,3-dihydroisoindol-2-yl) benzoic acid,

4-acetamidosalicylic acid,

7-doxylstearic acid,

2 ', 4'-dimethylphthalanilic acid,

Ν-α-fmoc-N-α'-boc-diaminoacetic acid, undecanedioic acid,

4-chloro-3-methoxybenzoic acid, (R) - (+) - 2-chloropropionic acid,

2,3-dibromo-2'-ethoxysuccinanilic acid,

3- [3- (2,5-dioxo-2,5-dihydropyrrol-1-yl) phenyl] acrylic acid,

3.3- tetramethyleneglutaric acid, (1S) - (+) - (1-aminopropyl) phosphonic acid,

4- (4-methoxyphenyl) but-2-enoic acid,

3-ethyladipic acid, meso-2,3-dimethylsuccinic acid,

3,4,5,6-tetrachloro-2 ', 4', 6'-trimethylphthalanilic acid,

2.4.5-trimethylbenzoic acid, free methyl-β-D-glucuronide acid monohydrate,

4-hydroxy-3-methyl- (α-aminoacetyl) benzoic acid, benzenesulfonic acid, phenylpropiolic acid,

2,5-dimethylbenzoic acid,

4,4,8,8-tetrafluoradamantane-1,3-dicarboxylic acid, N-fmoc-D-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid, (+/-) - trans-1-amino- 1-carboxycyclopentane-2-acetic acid,

11-benzenesulfonylundecanoic acid,

N - [(S) -1- (1-naphthyl) ethyl] phthalamic acid, (R) -3-hydroxybutyric acid,

19-phenylnonadecanoic acid,

2- [3- (N'-Butyrylhydrazino) -3-oxopropionylamino] benzoic acid

- 199 acid,

4-oxo-1-phenyl-1,4-dihydropyridine-2,6-dicarboxylic acid, chorismic acid,

N- (4-iodophenyl) phthalamic acid,

4-oxo-4H-1-thia-4α, 9-diazafluorene-2-carboxylic acid,

3-hydroxyphthalide-7-carboxylic acid,

5- (3-hydroxy-4-methoxyphenyl) pentanoic acid,

4 - ((4 - [(4,6-dimethylpyrimidin-2-yl) thio / phenyl] amino] -2-methyl-4-oxo- (2Z) -butenoic acid),

5,6-dichloro-3-indole acetic acid,

3- (2,5-dimethylbenzoyl) acrylic acid,

7-oxo-11-dodecenoic acid,

N, N'-dodecamethylenebis (maleic acid), threo-9,10-dihydroxystearic acid,

N-acetyl-D, L-aspartic acid,

1- pyroglutamic acid,

2-methyl-3-m-tolylacrylic acid, (2-acetylphenyl) acetic acid,

N-phenylacetyl-p-aminobenzoic acid,

12-bromododecanoic acid, chrysanthemmonocarboxylic acid, (1-benzoylamino-2,2-dichlorvinyl) phosphonic acid,

3-methyl-3- (5,6,7,8-tetrahydronaphthalen-2-yl) butyric acid,

4- (2-hydroxy-1-naphthylmethyleneamino) salicylic acid, (2-phenylethenesulfonylamino) acetic acid,

3-hydroxyadamantanecarboxylic acid,

5-bromo-2-benzofurancarboxylic acid,

4-acetoxy-3-methoxycinnamic acid, chicagic acid,

5-formylsalicylic acid,

3-ethyl-3-methylglutaric acid,

2- (3,5-di-tert-butyl-4-hydroxybenzylidene) malonic acid,

4- (2-hydroxyhexafluoroisopropyl) benzoic acid,

200 (R) - (+) - N- (1-phenethyl) phthalamic acid,

2-Acetylamino-4,5,6,7-tetrahydrobenzo (b) thiophene-3-carboxylic acid

2,5-diisothiocyanatobenzenesulfonic acid,

3- (dodecylthio) propionic acid,

10-Phenyldecanoic acid,

4-formylphenoxyacetic acid,

6-methyl-1- (3-nitroanilino) -4-oxo-1,4-dihydro-3-pyridinecarboxylic acid,

4-methyl-2- (2-nitro-4-trifluoromethylphenylamino) pentanoic acid,

2-chloro-6-methoxybenzoic acid,

4-hydroxy-3-iodo-5-nitrobenzoic acid,

5- C 4- (3-carboxypropyl) phenyl] -5-oxopentanoic acid,

3- (3,4-dimethoxy-6-nitrobenzoyl) propionic acid,

6-amino-2,3-dibromobenzoic acid,

2- (2,4,6-trichlorophenoxy) propionic acid,

3- (5-methylfuran-2-yl) acrylic acid, (2-fluorophenyl) phosphonic acid,

2- [2- (4-hydroxyphenyl) propyl] benzoic acid, cis-hexahydro-N- (4-methylphenyl) phthalamic acid,

4-Biphenylsulfonic acid

5-phenyl-2H-tetrazole-2-acetic acid, cis-2-methoxycinnamic acid,

4-methyldodecanoic acid,

3- (4-n-butylbenzoyl) propionic acid, (S) - (+) - 2-phenylpropionic acid,

12-doxylstearic acid, (1,2,3-triphenylcycloprop-2-enyl) acetic acid,

1- (4-chlorobenzoyl) piperazine-2,3-dicarboxylic acid,

17-methyloctadecanoic acid,

2,4-dichlorincinnamic acid,

2-bromo-6-chlorobenzoic acid, · β β • β β β β β β β β β brom brom brom brom ♦ brom

201

3-methoxy-5-methyl-4-oxo-2,5-hexadiene acid,

2.3- dibromopropionic acid,

3- [3- (2,4-dimethoxyphenyl) ureido] benzoic acid,

2 - [(2-ethoxycarbonyl) - (toluene-4-sulfonyl) amino] benzoic acid,

2,5-diamino-1,4-benzenedisulfonic acid,

2-bromomethylbenzoic acid, α- (bromomethyl) cinnamic acid,

3-benzoyl-2-pyridinecarboxylic acid, 2-phenyl-2-ethylbutyric acid,

4- [[(4,6-dimethyl-2-pyrimidinyl) amino] carbonyl] -5-methyl-3-isoxazolecarboxylic acid,

5- (3-hydroxyphenylvaleric acid),

8,9-epoxy- (5Z, 11Z, 14Z) icosatrienoic acid

3'-chloro-2'-methylmaleanilic acid, trans-4-methyl-1-cyclohexanecarboxylic acid, n-decylphosphonic acid, hexadecanedioic acid,

Ν-α-boc- (Ν-β-fmoc) diaminopropionic acid,

2-hydroxymyristic acid,

4,4'-dihydroxybiphenyl-2-carboxylic acid,

8-chloronaphthalene-1-sulfonic acid,

2,3-bis- (4-methoxybenzylidene) succinic acid,

3,5-dihydroxy-4-methylbenzoic acid, N-boc-L-aspartic acid α-benzyl ester,

4-carboxybenzenesulfonamide,

N-furfuryl-1,2,3,6-tetrahydrophthalamic acid,

2.5-dihydroxyterephthalic acid,

6 - [(4,5-di-meo-3-oxo-3H-isobenzofuran-1-ylidene) -home] -2,3-di-meobenzoic acid,

N- (1-ethoxycarbonyl-2-hydroxy-2-phenylethyl) succinamic acid,

2-methyl-4-pentenoic acid,

- 202 [(5-bromofuran-2-carbonyl) amino] acetic acid, α, α'-dibromo-1,3-adamantanediacetic acid,

D, L-4- (benzoylamino) -5- (dipropylamino) -5-oxopentanoic acid,

1- (2-chloro-4-fluorophenyl) cyclohexanecarboxylic acid,

3-methoxy-3-phenylpropionic acid, tert-butylperphthalic acid,

1-pyrendecanoic acid, trans-2- (2-methoxyphenyl) -5-oxotetrahydrofuran-3-carboxylic acid,

2-hydroxy-6- [4- (trifluoromethyl) phenyl] -3,5-pyridinedicarboxylic acid,

5-bromferulic acid,

3- (acetylmercapto) butyric acid,

4- [acetyl- (1,3-dioxo-1,3-dihydroisoindol-2-ylmethyl) amino] benzoic acid,

D, L-cysteic acid,

5,7-dimethoxy-1-oxo-2-indanecarboxylic acid,

4-hydroxy-3-methylbenzoic acid,

3- (3-chlorophenyl) -2-methylacrylic acid,

3- (o-tolylthio) propionic acid,

2-amino-6-sulfo-1-naphthalenemethanesulfonic acid,

N- (p-tosyl) -D-glutamic acid,

5-Norbornene-2,3-dicarboxylic acid

3-bromo-1-adamantaneacetic acid,

5- (5-indanylmethyleneamino) salicylic acid,

4- (4-benzyloxycarbonylaminobutyrylamino) butyric acid,

3- (dichloromethanesulfonyl) propionic acid, hydantic acid,

4-hydroxy-3-nitrophenylacetic acid,

3'-chloro-6'-methoxymaleanilic acid,

2-chloro-5- (fluorosulfonoyl) benzoic acid,

3-Methyl-2-oxovaleric acid, · * * * * * methyl methyl methyl methyl methyl methyl methyl methyl methyl

- 203 • · · ·

2-anilino-5-bromo-terephthalic acid, benzoic acid, cyclohexylidenecyanoacetic acid,

1,4-butanbis (thioglycolic acid),

2'-methoxy-4'-nitromaleanilic acid,

4- (3-methyl-4-hydroxyphenylazo) benzenesulfonic acid,

2- (3-carboxypropylamino) benzoic acid,

2- (bromomethyl) -2,3-dimethyl-4-oxocyclohexanecarboxylic acid,

11- [3- / 3- (trifluoromethyl) phenyl] ureido {undecanoic acid,

3- (3-benzyloxy-4-methoxyphenyl) propionic acid,

2.3.4- tribromobutyric acid, hexanoic acid,

4-fluoro-2-methoxybenzoic acid, benzylmalonic acid,

2-naphthylacetic acid,

D, L-2-amino-8-phosphonoctanoic acid,

2-bromo-5-chlorophenylacetic acid,

6-oxo-15-hexadecenoic acid,

1,2-phenylenediacetic acid, boc-L-norleucine, meso-2,3-dibromosuccinic acid,

3- (butane-1-sulfonyl) propionic acid, chlorosulfonic acid,

4-chloro-3,5-dihydroxybenzoic acid, isovaleric acid,

3- (3-fluoro-4-methoxybenzoyl) propionic acid, gamma-D-glutamylaminomethylphosphonic acid, 2-methyl-4-oxo-4-phenylbutyric acid,

N- (2,4-dichlorophenyl) -2,3-dihydroxysuccinamic acid, 2-anisidine-4-sulfonic acid,

2- (2'-pyridyl) ethylmalonic acid,

4-ethoxyphenylacetic acid, 4

- 204 -

3-pyroslizic acid,

4'-acetylbiphenyl-4-carboxylic acid, diisoctylthiophosphinic acid, (2,4-dinitrophenylimino) acetic acid, methylenebis (thiolactic acid), n-dodecylmaleinamic acid, n-acetylmuramic acid, benzenesulfonylaminoacetic acid,

1-methyl- [2-aminoterephthalate],

4-pentyloxybiphenyl-4'-carboxylic acid,

3- [2- (benzoyloxy) phenyl] propionic acid,

5-nitrothiophene-2-carboxylic acid,

4'-ethylglutaranilic acid,

4- (3-methylbenzoylamino) benzoic acid,

L-α-aspartyl-L-glutamic acid,

3,5-dimethylisoxazole-4-carboxylic acid, [4- (4-methoxycarbonylsulfanylphenoxy) phenylsulfanyl] acetic acid,

N- (4-adamantan-1-ylphenyl) phthalamic acid,

2-bromo-4-fluorobenzoic acid,

3-fluoro-4-n-octyloxybenzoic acid,

4-chloro-2,3,5,6-tetramethylbenzoic acid, p-chloromandelic acid,

2-methylbenzene-1,3,5-tricarboxylic acid, (+/-) - 10-methyloctadecanoic acid,

2-iodo-5-oxo-4-oxatricyclo [4.2.1.0 (3.7)] nonane-9-carboxylic acid,

2- (2,4-di-tert-pentylphenoxy) butyric acid,

5- 4-bromomandelic acid, cis-5-dodecenoic acid,

3-Acenaphthen-5-ylpropionic acid

2'-benzoyl-2-biphenylcarboxylic acid,

4-nitrotoluene-2-sulfonic acid,

- 205 -

4- (2-methoxyanilino) -4-oxo-2-butenoic acid,

Ν-α- (9-fluorenylmethyloxycarbonyl) -a- (tert-butyl ester) -L-glutamic acid,

11 (R), 12 (R) -epoxy-13 (S) -hydroxy-9Z-octadecenoic acid,

2-hydroxy-1-naphthoic acid,

3- (2-nitrophenyl) -2-o-tolylacrylic acid,

3.5-dinitrosalicylic acid,

4- (3- (2,6-xylyl) ureido] salicylic acid,

3-octenic acid, dehydrothio-4-toluidinedisulfonic acid,

5- (4-nitrophenyl) -2H-tetrazole-2-acetic acid, cyclohexanesulfamic acid,

2,3-norbornane dicarboxylic acid,

2-tridecinic acid,

R-4-hydroxymandelic acid,

3- (4-Butylbenzoylamino) benzoic acid

2-biphenylenecarboxylic acid,

2- (2-cyanethylamino) -3-methylbutyric acid,

3-aminophthalic acid,

3-hydroxy-o-toluic acid,

7-oxo-7H-benzo (e) pyrimidine-4-carboxylic acid,

3-bromo-4-hydroxybenzoic acid, [3- (4-bromo-2-fluorobenzyl) -4-oxo-3H-phthalazin-1-yl] acetic acid,

3- (1-cyanoethyl) benzoic acid,

N- (6-methyl-2-pyridyl) glutaramic acid,

N- (4-acetamidobenzylidene) anthranilic acid, quinoline-5-carboxylic acid,

4,5-dichloroaniline-2-sulfonic acid,

4-amino-3,5-dichlorobenzoic acid,

3- [N- (3-pyridyl) carbamoyl] -5-norbornene-2-carboxylic acid, o-naphthionic acid,

- 206 -

4-imidazolecarboxylic acid,

1-amino-8-naphthol-2,4-disulfonic acid, N- (5-nitro-3-pyridyl) phthalamic acid,

4-aminobenzoic acid,

3- (3-pyridyl) acrylic acid, nbd-aminohexanoic acid,

N- (5,7-dimethyl-1,8-naphthyridin-2-yl) succinamic acid,

5-amino-3-chloro-o-toluenesulfonic acid,

5-nitro-4-quinolinecarboxylic acid,

N- (2-naphthyl) -3,4,5,6-tetrachlorophthalamic acid,

2-amino-3-methoxybenzoic acid,

4-bromo-2,5-dimethylpyrrole-3-carboxylic acid,

4- (2-benzimidazolyl) benzenesulfonic acid,

2,6-diaminomesitylene-4-sulfonic acid,

4-pyridylacetic acid,

2-amino-3,4,5-trimethoxybenzoic acid, β-α-aminoisobutyric acid,

6-methylnicotinic acid,

6- (1,2,4-triazol-1-yl) nicotinic acid,

5-methylindole-2-carboxylic acid,

3- (N-methylanilino) -1-propanesulfonic acid,

2-amino-3,6-dimethylbenzoic acid,

2,3-dichloro-4- [2- / 3-chloro-5- (trifluoromethyl) -2-pyridyl] hydrazono] -2-butenoic acid,

8-amino-2-naphthalenesulfonic acid,

2-amino-5-methoxybenzoic acid,

5.6-dimethylmethanilic acid,

5-amino-2,4-xylenesulfonic acid, methanoic acid,

4- (butylamino) benzoic acid,

3-aminopyridine-4-carboxylic acid,

1,2-phenylenediamino-4-sulfonic acid,

2- (2,5-dimethoxyphenylthio) pyridine-3-carboxylic acid

- 207 N- [4 - [(aminoiminomethyl) amino] -1-carboxybutyl] -L-glutamic acid,

4H-1,2,4-triazole-3-carboxylic acid, 2-dimethylaminobenzoic acid,

N- (3-pyridyl (maleic acid),

2-propionyl-3-indole acetic acid,

6- (N-methylamino) -1-naphthol-3-sulfonic acid,

2- (2-pyridyl) ethanesulfonic acid,

N-methylsulfanilic acid, dnp-D, L-α-amino-n-butyric acid,

4- (hexadecyloxy) -3-nitro-cinnamic acid,

2- (4-chlorophenylthio) pyridine-3-carboxylic acid,

4-pyridoxic acid, dianilinoterephthalic acid,

2-hydroxyquinoline-4-carboxylic acid,

5- (aminomethyl) -4- (methoxycarbonyl) -1H-pyrrole-3-propanoic acid,

N- (3-nitrophenyl) (anthranilic acid,

3-amino-4-methoxybenzoic acid, monosodium salt of aniline-2,5-disulfonic acid,

7-amino-2-naphthalenesulfonic acid,

6-fluoro-7-morpholin-4-yl-4-oxo-1,4-dihydroquinoline-3-carboxylic acid,

3,5-diaminobenzoic acid,

8-hydroxyquinoline-2-carboxylic acid,

4- [3- (2,5-xylyl) ureido] salicylic acid,

5- (3-Amino-5-oxo-2-pyrazolin-1-yl) -2-phenoxybenzenesulfonic acid,

3-hydroxypicolinic acid,

4-hydroxyquinoline-2-carboxylic acid, p-toluidine-o-sulfonic acid, oxolinic acid,

3- (3-nitro-4-pyrrolidinophenyl (acrylic acid,

- 208 2-pyridylacetic acid,

2-chloronicotinic acid, meta-phenylenediamine-4,6-disulfonic acid,

3-pyridylacetic acid, 2-mercapto-4-methyl-5-thiazoleacetic acid, pyrrole-2-carboxylic acid,

4- (4-chlorophenyl) -6,8-dimethyl-1,9-diazaindene-3-carboxylic acid,

4-methylnicotinic acid,

1- (4-Methylphenyl) -4-hydroxy-6-pyridazinone carboxylic acid

1-indole acetic acid,

4,8-dihydroxyquinoline-2-carboxylic acid, benzoic acid,

2-naphtho-o-toluidine-3-phosphoric acid,

4-methoxy-2-quinolinecarboxylic acid,

2- (4-dimethylaminophenyl) thiazolidine-4-carboxylic acid,

1-methylpyrrole-2-carboxylic acid,

3-indole-lactic acid, phthalic acid,

5-benzyloxyindole-3-acetic acid, (Z) -2-amino-α- (1- (tert-butoxycarbonyl) -1-methylethoxyimino) -4-thiazoleacetic acid,

2- (4-chlorophenoxy) pyridine-3-carboxylic acid,

2-amino-1-naphthalenesulfonic acid,

5-amino-2- (p-aminoanilino) benzenesulfonic acid, α- (N-ethylanilino) -m-toluenesulfonic acid,

2-chloro-4-carboxyquinoline,

6- (p-toluidino) -2-naphthalenesulfonic acid,

N- [N'-methyl-N '- [2- (3-chloro-5-trifluoromethyl) pyridyl]] maleic acid,

3-amino-4-tert-butylbenzoic acid,

4-ethyl-5-formyl-3-methyl-2-pyrrolecarboxylic acid;

- 209 -

5-methylbenzo (1,2,5) thiadiazole-4-sulfonic acid, n-beta-gamma-aminobutyric acid,

6- (2,4,5-trichlorophenoxy) methanoic acid,

7-anilino-4-hydroxy-2-naphthalenesulfonic acid,

4-amino-3,5,6-trichloropicolinic acid,

3-hydroxyanthranilic acid,

2-methoxynicotinic acid,

N- (4-methyl-2-pyridyl) succinamic acid,

8-aminonaphthalene-1,3,6-trisulfonic acid,

4- (2,3-dihydro-2-thioxo-1-benzimidazolylmethylamino) benzoic acid,

2-formyl-4-methyl-3-pyrrolpropionic acid,

4-amidinobenzoic acid,

4-amino-5-chloro-m-toluenesulfonic acid,

2-amino-3,4,5,6-tetrafluorobenzoic acid,

5-formyl-4-methyl-3-pyrrolpropionic acid,

5- (2,5-dihydroxybenzylamino) -2-hydroxybenzoic acid,

2- (4-aminophenoxy) -2-methylpropionic acid,

1-methyl-3-indole acetic acid,

2-amino-3,5-dibromo-6-fluorobenzoic acid, picric acid,

2- (4-methylphenylthio) pyridine-3-carboxylic acid,

N- (3-pyridylmethyl) glutaramic acid, 1-methylindole-2-carboxylic acid,

6-dimethylamino-4-hydroxy-2-naphthalenesulfonic acid,

4-aminodiphenylamino-2-sulfonic acid,

1-isoquinolinecarboxylic acid,

3- (3-aminophenyl) propionic acid,

3-Acetamido-5-aminobenzoic acid

4-hydroxyquinoline-2-carboxylic acid,

1,4-dihydro-1-ethyl-7-methyl-4-oxo-1,8-naphthyridine-3-carboxylic acid, (2-benzimidazolylthio) acetic acid,

210

5-isoquinolinesulfonic acid,

4- (4-anilinophenylazo) benzenesulfonic acid,

4-dimethylaminonaphthalene-1-carboxylic acid, dinitrophenylpipecolic acid,

N- (2-pyridyl) -1,2,5,6-tetrahydrophthalamic acid, N-sulfanilylsulfanilic acid,

4-aminobenzenesulfonic acid,

5-aminosalicylic acid,

2-aminobenzoic acid 5-sulfamide, pyrazole-3-carboxylic acid,

2-amino-4-chlorophenol-6-sulfonic acid,

4,4'-diaminobiphenyl-2,2'-dicarboxylic acid,

8-amino-1,6-naphthalenedisulfonic acid,

N- (2,5-dichlorophenyl) anthranilic acid, phthalylsulfathiazole,

4-nitroanthranilic acid, indole-3-glyoxylic acid,

N- (2-nitrophenyl) anthranilic acid,

2,3-dimethyl-7-indolecarboxylic acid,

2- (p-chlorophenyl) quinoline-4-carboxylic acid,

1-naphthylamino-5-sulfonic acid,

2,4-diaminobenzoic acid, cis-hexahydro-N- (3-pyridylmethyl) phthalamic acid,

2-amino-3,4-dimethylbenzoic acid,

3-isothioureidopropionic acid,

N- [2- (N-methylanilino) ethyl] -1,2,3,6-tetrahydrophthalamic acid,

2-aminophenol-4-sulfonic acid, citrazic acid,

3-indolpropionic acid, α- [2-amino-4- (trifluoromethyl) phenyl] -4- (trifluoromethyl) cinnamic acid,

5- (pyrid-2-yl) thiophene-2-carboxylic acid;

• • • •

211

2-methyl-4-trifluoromethylthiazole-5-carboxylic acid,

2-amino-6-hydroxybenzenesulfonic acid,

5-chloro-6-hydroxynicotinic acid,

5-methyl-3-pyridinesulfonic acid,

5-amino-2-chlorobenzoic acid,

2-phenyl-4-quinolinecarboxylic acid, n-phenylglycine,

4-amino-2'-nitro-4'-sulfodiphenylamine,

8-hydroxyquinoline-5-sulfonic acid,

4,4'-diamino-5,5'-dimethyl-2,2'-biphenyldisulfonic acid,

N-ethylnaphthyl-2-amino-6-sulfonic acid,

2'-methyl-3,3 ', 4,5,6-pentachlorophthalanic acid, (Z) - (2-aminothiazol-4-yl) hydroxyiminoacetic acid, nicotinuric acid,

4- (veratrylideneamino) benzoic acid, quinaldic acid,

5-Methoxyindole-3-acetic acid

4-anisidine-2-sulfonic acid,

2- (n-methylamino) -8-hydroxynaphthalene-6-sulfonic acid, indole-5-carboxylic acid,

1- (3-Trifluoromethylphenyl) -4-hydroxy-6-pyridazinone carboxylic acid

4- (2,3-dihydro-2-thioxo-3-benzoxazolylmethylamino) salicylic acid,

8-amino-1-naphthol-3,6-disulfonic acid,

4-nitro-4'-aminodiphenylamino-2-sulfonic acid,

2- (4-sulfobutylamino) -4-chlorophenol

4-pyridylhydroxymethanesulfonic acid,

4- (2,3-dihydro-2-thioxo-1-benzimidazolylmethylamino) salicylic acid, acridone-10-acetic acid,

6-methoxy-2- (3-nitrophenyl) -4-quinolinecarboxylic acid, 1-amino-2-naphthol-4-sulfonic acid,

212

4-imidazolacrylic acid,

4-chloro-N-phenylanthranilic acid, anilino-4-hydroxy-2-naphthalenesulfonic acid,

2 - [(2-hydroxybenzylidene) amino] -3- (3H-imidazol-4-yl) propionic acid,

N- (6-methyl-2-pyridyl) -3,4,5,6-tetrachlorophthalamic acid,

1-Benzylindole-3-carboxylic acid

5-bromo-4-chloro-3-indolyl-β-D-glucuronic acid,

4'-anilinohexahydrophthalanic acid,

4- (ethoxycarbonylamino) anthranilic acid, indole-4-carboxylic acid,

4- (methylamino) benzoic acid,

2,5-diaminobenzoic acid,

2-amino-3-nitrobenzoic acid,

5-bromoindole-3-acetic acid,

N- (4-ethoxyphenyl) -4-nitroanthranilic acid,

5-nitro-3-phenylindole-2-carboxylic acid, (2-benzimidazolylmethylthio) acetic acid,

5-nitrochinaldic acid,

6-benzyloxy-5-methoxy-2-carboxyindole, indole-3-butyric acid,

6-methoxy-4-quinolinecarboxylic acid, (S) -2- (6-hydroxy-2-benzothiazolyl) -2-thiazolene-4-carboxylic acid,

N- (1-naphthyl) -5-nitroanthranilic acid,

4-amino-3,5-diiodosalicylic acid, quinoline-8-sulfonic acid, 1-methylbenzimidazole-2-sulfonic acid,

5-methyl-3-phenylisoxazole-4-carboxylic acid, indole-2-carboxylic acid, chloramben,

4-dimethylaminobenzoic acid,

1,3-dihydroxy-9-acridinecarboxylic acid; f · · · · ····· · V

213 cis-hexahydro-N- (4-methyl-2-pyridyl) phthalamic acid,

4- (ethylamino) benzoic acid, benzothiazole-6-carboxylic acid,

6-aminonicotinic acid,

5- (4-aminobenzamido) valeric acid,

N- (4-methyl-2-pyridyl) phthalamic acid,

2- (n-propylthio) nicotinic acid,

N- (3-pyridyl) glutaramic acid,

2,3,5,6-tetrachloro-4-pyridinecarboxylic acid,

2- (4-pyridyl) ethanesulfonic acid,

4-amino-2,3,5,6-tetrafluorobenzoic acid,

3-chloro-5-trifluoromethylpyridine-2-propenoic acid,

5- [3- (4-Chloro-phenyl) -4,5-dihydropyrazol-1-yl] -isophthalic acid,

N- (3-methyl-2-pyridyl) phthalamic acid,

4-Methylmethanilic acid

2-amino-6-chlorobenzoic acid,

N-ethylanthranilic acid,

4-thioureidobenzoic acid,

1-naphthylamino-6-sulfonic acid,

5-amino-2-p-toluidinobenzenesulfonic acid,

4- (di-n-hexylamino) benzoic acid,

4- (4-quinolylazo) benzenesulfonic acid,

2-fluoronicotinic acid,

2- [benzo (1,2,5) thiadiazole-4-sulfonylamino] -5-bromobenzoic acid,

5-fluoroindole-2-carboxylic acid, o-anisidine-5-sulfonic acid, dehydrothio-p-toluidine sulfonic acid,

3,5-diamino-2-methylbenzoic acid,

4 '- (dimethylamino) glutaranilic acid,

6- (1-imidazolyl) nicotinic acid,

2- (4-Hydroxyphenylazo) benzoic acid, K · K 9 · 0 · 0 · 0 · 0 · 0 · 0 · 0 · 0 · 0 · 0 · 0 · 0 · 0 · 0 * · · · · · 000 000

214

7-diethylaminocoumarin-3-carboxylic acid,

2 - [(2,3-dimethylphenyl) amino] benzoic acid,

2- [N- / 2- (N-methylanilino) ethyl / carbamoyl] cyclohexanecarboxylic acid,

2- (4-Isopropyl-4-methyl-5-oxo-2-imidazolin-2-yl) nicotinic acid

1- (2,4-dichlorophenyl) -4-hydroxy-6-pyridazinone carboxylic acid,

N, N-dimethyl-3-nitrosulfanilic acid,

8-anilino-1-naphthalenesulfonic acid,

5-amino-3-chloro-2,4-dihydroxybenzoic acid, N-4-dimethylmethanilic acid,

N- (2-thioxobenzothiazolin-3-ylmethyl) anthranilic acid,

2-chloro-6-methylnicotinic acid,

4-dimethylaminoazobenzene-4'-carboxylic acid,

2- (phenylthio) pyridine-3-carboxylic acid

5- (1-pyrrolidino) -2H-tetrazole-2-acetic acid

2,4-dichloro-3,5-dinitrobenzoic acid,

4'-methyl-2'-nitro-3,4,5,6-tetrachlorophthalic acid,

2- [4- (dibutylamino) -2-hydroxybenzoyl] benzoic acid,

3-pyridylacetic acid,

4-Aminoacetanilide-3-sulfonic acid

N-acetyl-D, L-tryptophan,

2 - ([2- (6-chloro-2-pyridyl) hydrazino / carbonyl] benzoic acid,

7-iodo-8-hydroxyquinoline-5-sulfonic acid,

4-amino-3-nitrobenzoic acid, 2-amino-5-methylbenzoic acid,

4- (diethylamino) benzoic acid,

4-chloroaniline-3-sulfonic acid, anthranilic acid, chloroacetyl-D, L-tryptophan,

1- (3-chlorophenyl) -4-hydroxy-6-pyridazinone-3-carboxylic acid

• ·

215 acid,

5-Butyl-2-pyridinecarboxylic acid,

N- (5-methyl-3-isoxazolyl) -3,4,5,5-tetrachlorophthalamic acid,

5- (phenylethynyl) pyridine-3-carboxylic acid,

2-methyl-2- (1,2,4-triazol-1-yl) propionic acid,

8-acetoxy-2-phenyl-4-quinolinecarboxylic acid,

4- [4- (dimethylamino) benzylideneamino] salicylic acid,

2- (4-tert-butylphenoxy) pyridine-3-carboxylic acid,

6- (trifluoroethoxy) pyridine-3-carboxylic acid,

D, L-α-bromo-β- (5-imidazolyl) propionic acid, 2-amino-3-bromo-5-methylbenzoic acid,

1-amino-8-naphthalenesulfonic acid,

5-chloroindole-2-carboxylic acid,

4- (4-methoxybenzylamino) benzoic acid,

4- [4- (diethylamino) benzylideneamino] salicylic acid,

2- (4-diethylamino-2-hydroxybenzoyl) benzoic acid,

2-carbamoylnicotinic acid, indoline-2-carboxylic acid, o-dianisidine,

N- (3-amino-4-hydroxyphenylsulfonyl) anthranilic acid,

3-methyl-5-pyrazolecarboxylic acid, trans-1-methyl-4-carboxy-5- (3-pyridyl) -2-pyrrolidinone, benzidine-3,3'-dicarboxylic acid,

2-aminonicotinic acid,

4- (2,5-Dimethyl-3-formyl-1-pyrrolyl) benzoic acid,

3-amino-4-hydroxybenzoic acid,

5-fluoroindole-3-acetic acid,

N- [2- (2-pyridyl) ethyl] -3,4,5,6-tetrachlorophthalamic acid, 1- (diethylmethyl) -1,2,3,4-tetrahydronorharman-3-carboxylic acid,

4-hydroxy-8- (trifluoromethyl) -3-quinolinecarboxylic acid,

N- (3-pyridyl) phthalamic acid, · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · · w · · · · · · ·

- 216

2- (n-amylthio) nicotinic acid,

2- (4-hydroxyphenyl) -6-methoxy-4-quinolinecarboxylic acid,

4- (4-methoxybenzylideneamino) benzoic acid, mercaptotetrazolylacetic acid,

6,6'-dithiodinicotinic acid,

6-amino-1-naphthol-3-sulfonic acid,

4-amino-2-chlorobenzoic acid, cis-hexahydro-N- (2-pyridyl) phthalamic acid,

2- [3 '- (1'-Phenylamino) thiazole] benzoic acid,

5- (methoxycarbonyl) pyridine-2-carboxylic acid,

2-amino-5-nitrobenzoic acid,

4- (trifluoromethyl) nicotinic acid,

8-hydroxyquinoline-4-carboxylic acid,

3-amino-2,4,6-tribromobenzoic acid,

3- (n-ethyl-3-hydroxy-4-nitrosoanilino) propanesulfonic acid,

2-amino-3,5-diiodobenzoic acid,

3-amino-2-methylbenzoic acid,

2 - [(2-hydroxy-3-nitrobenzylidene) amino] -3- (1H-imidazol-2-yl) propionic acid,

2- (2-furyl) -4-quinolinecarboxylic acid,

2,6-dichloronicotinic acid, p - [[(2-thioxobenzothiazolin-3-yl) methyl] amino] benzoic acid,

2'-methoxy-4-nitrodiphenylamino-2-sulfonic acid, N-methylanthranilic acid,

4'-methyl-3,3 ', 4,5,6-pentachlorophthalic acid,

6-amino-2-naphthalenesulfonic acid,

2-hydroxynicotinic acid,

1-dimethylaminonaphthalene-5-sulfonic acid,

3-anilino-1-propanesulfonic acid,

5-bromo-2- (ethoxycarbonyl) -3-indolebutyric acid,

2-Amino-3-methylbenzoic acid, ··· ···············

217

4-aminohippuric acid, indole-3-acetic acid,

3-methoxy-4-aminoazobenzenesulfonic acid,

2-amino-3,6-dichlorobenzoic acid,

N-Veratrylidenanthranilic acid,

N- (2-pyridyl) phthalamic acid, toluenesulfonic acid,

1,2,3,4-tetrahydroacridine-9-carboxylic acid,

2-amino-5-bromobenzoic acid,

Ι-β-imidazole-lactic acid,

9-fluoro-2-methyl-1-azaxanthan-3-carboxylic acid,

2-Methoxy-5-methylaniline-4-sulfonic acid

4-amino-3-methoxybenzoic acid,

N- (2,4-dinitrophenyl) -6-aminohexanoic acid,

5-ethyl-2-indolecarboxylic acid,

2,6-dimethylimidazo (1,2-a) pyridine-3-carboxylic acid,

3-hydroxy-2-methyl-4-quinolinecarboxylic acid,

N, N'-ethylenedianthranilic acid, 2-chloro-6-methoxypyridine-4-carboxylic acid, n-anilinosuccinamic acid,

6-methoxy-4-quinolinacrylic acid,

N- (2-amino-4-chlorophenyl) anthranilic acid,

5-nitro-N-phenylanthranilic acid,

L-tryptophyll-L-glutamic acid,

4-amino-5-methoxytoluene-2-sulfonic acid,

2-amino-4-fluorobenzoic acid,

5- (2,3-dihydro-2-thioxo-3-benzoxazolylmethylamino) salicylic acid, niflurnic acid,

3-aminophenylacetic acid,

2-chloroaniline-4-sulfonic acid,

4-nitroaniline-2-sulfonic acid, β-3-β-β-3-β-3-β-acid,

218 quinoline-8-carboxylic acid, quinoline-4-carboxylic acid,

3- (4-pyridyl) acrylic acid, methoxylidine-6-sulfonic acid,

5-benzimidazolecarboxylic acid,

4-aminoazobenzene-4-sulfonic acid,

2,6-toluylenediamino-4-sulfonic acid,

N- [2- (3-chloro-5-trifluoromethylpyridyl) -4-aminobutyric acid, imidazole-4-acetic acid,

1- (4- (4-methoxyphenyl) -1,3-thiazol-2-yl) -5- (trifluoromethyl) -1H-

-4-pyrazolecarboxylic acid, p-aminooxanilic acid,

2,3-dibromo-2'-methoxy-4'-nitrosuccinanilic acid,

9-chloro-2-methyl-1-azaxanthan-3-carboxylic acid,

4-amino-3-hydroxybenzoic acid,

2-chloroaniline-5-sulfonic acid,

5-Benzyloxyindole-2-carboxylic acid

4-chloro-N- (4-tolyl) anthranilic acid, 2-amino-5-chloro-p-toluenesulfonic acid,

2-ethoxynicotinic acid,

4-amino-3-methylbenzoic acid,

4-dimethylamino-3,5-dinitrobenzoic acid,

1- (4-ethoxyanilino) -2-anthraquinone carboxylic acid,

3-amino-4-methylbenzoic acid,

4- (1H-benzotriazol-1-ylmethylamino) benzoic acid,

7-chloro-6-fluoro-1-cyclopropyl-1,4-dihydro-4-oxoquinoline-3-carboxylic acid,

7-amino-1-naphthalenesulfonic acid,

N- (5-nitro-2-pyridyl) -3,4,5,6-tetrachlorophthalamic acid, diphenylamino sulfonic acid,

2-naphthylamine-5-sulfonic acid,

6-acetyl-N-phenylanthranilic acid,

219

3.5-dibromosulfanilic acid,

2-amino-3,5-dibromobenzoic acid,

3- (amidinothio) -1-propanesulfonic acid,

3- (2-Methyl-4-nitroimidazol-1-yl) propionic acid

4-nitro-2-aminophenol-6-sulfonic acid,

5.6- dichloronicotinic acid,

3,4-diaminobenzoic acid,

3- [N- (2-pyridyl) carbamoyl] -5-norbornene-2-carboxylic acid,

6-acetamido-3-pyridinesulfonic acid,

3- (4-chloro-2-nitroanilino) propionic acid, N-cyclohexylidene-anthranilic acid, 2-benzimidazolepropionic acid, cytosine-5-carboxylic acid,

6-acetylamino-2-aminophenol-4-sulfonic acid,

2,6-dimethylpyridine-3-sulfonic acid, dinitropyridyl-L-aspartic acid, 2-amino-3-chlorobenzoic acid,

8- (3-carboxypropyl) -1,3-dimethylxanthine, indole-3-pyruvic acid,

2,2'-bipyridine-4,4'-dicarboxylic acid,

2- (allylthio) nicotinic acid

2,3,4'-tribromosuccinanilic acid,

N- (6-methyl-2-pyridyl) phthalamic acid,

7-nitroindole-2-carboxylic acid,

4- (3-methyl-5-oxo-2-pyrazolin-1-yl) benzoic acid,

4- (n-hexylamino) benzoic acid, N-anilinoglutaramic acid,

3-anilinopropionic acid,

2-methoxyamino-2- (2-aminothiazol-4-yl) acetic acid, N- (4-methyl-2-pyridyl) glutaramic acid,

2-acetamidobenzoic acid,

2-pyrrolopyridine-5-carboxylic acid,

220

4,4'-dicarboxy-2,2'-quinoline,

3.4.5-trichloro-2-pyridinecarboxylic acid,

2.5-diaminobenzenesulfonic acid, aristolochic acid,

N- (4,6-disulfo-8-hydroxy-1-naphthyl) benzamide,

4-hydroxy-7- (trifluoromethyl) -3-quinolinecarboxylic acid,

2-amino-7-naphthalenesulfonic acid,

4-amino-2-methylcinnamic acid,

2- [2- (4-chlorobenzenesulfonyl) ethylthio] pyridine-3-carboxylic acid,

2-amino-3,4-dimethoxybenzoic acid,

4,6'-bianthranilic acid, nicotinic acid,

6-amino-4-hydroxy-2-naphthalenesulfonic acid,

2-amino-4,5-dimethoxybenzoic acid,

4-acetyl-3,5-dimethyl-2-pyrrolecarboxylic acid,

3-aminosalicylic acid,

3,3 ', 4,4'-tetramethyl- (2,2'-bipyrrolidinyl) -5,5 ^one dicarboxylic acid,

3-benzyloxythieno (1,2,3-b) pyridinecarboxylic acid,

4-amino-1-naphthalenesulfonic acid,

6-hydroxynicotinic acid,

3-amino-4-chlorobenzoic acid, m-toluidine-4-sulfonic acid,

2,3-dichloro-4- (2,4-dinitrophenylhydrazono) -2-butenoic acid,

4-nitropyrrole-2-carboxylic acid,

4- (dimethylamino) phenylacetic acid,

2- (2,6-dimethylmorpholino) -5-nitrobenzoic acid,

N- (4-chlorophenyl) maleimide

4-azidobenzoic acid, theophylline-7-acetic acid,

6-amino-3-pyridinesulfonic acid •

- 221 o-nitroaniline-p-sulphonic acid,

2- (3-amino-4-chlorobenzoyl) benzoic acid,

N- (2,4-dinitrophenyl) anthranilic acid,

4- (4-amino-m-tolylazo) -m-toluenesulfonic acid,

3- (3-hydroxy-4-nitroso-n-propylanilino) propanesulfonic acid,

3-amino-2,4,5-trifluorobenzoic acid,

4-amino-2-methoxycinnamic acid,

5-phenyl-2-pyrrolepropionic acid,

7-anilino-1-naphthol-3-sulfonic acid, pyridine-3-sulfonic acid,

2- [2- (benzenesulfonyl) ethylthio] pyridine-3-carboxylic acid,

2- (ethylthio) nicotinic acid

N- (3-methyl-2-pyridyl) glutaramic acid,

2-Amino-2-thiazoline-4-carboxylic acid

9-methyl-2-methyl-1-azaxanthon-3-carboxylic acid,

5-amino-2-nitrobenzoic acid,

3-nitro-2-pyridylthioacetic acid,

2,3-dibromo-4 ', 5'-dichloro-2'-methylsuccinanilic acid,

3,5-dichloranthranilic acid,

8-amino-1-naphthol-5-sulfonic acid,

N-ethyl-4-methylmethanilic acid,

2-aminobenzophenone-2'-carboxylic acid,

3-nitroaniline-4-sulfonic acid,

N- (1-naphthyl) anthranilic acid,

2- (2'-amino-4'-trifluoromethylphenylthio) benzoic acid,

6-methylpicolinic acid,

2- (pyrid-3-yl) thiazole-4-carboxylic acid,

2-hydroxy-3- (2'-aminophenylthio) -3- (4-methoxyphenyl) propionic acid,

1,2.5-trimethylpyrrole-3-carboxylic acid,

6-methoxycinchophen,

- 222 -

4-cinnamic acid,

4- [N- (2-amino-3-cyano-5-pyrimidinylmethyl) amino] benzoic acid,

5'-chloro-2,3-dibromo-2'-methoxysuccinanilic acid,

2-methyl-3-indole acetic acid, orthanilic acid,

3,5-dioxo-2,3,4,5-tetrahydro (1,2,4) triazine-6-sulfonic acid,

2-amino-4-phenyl-5-thiazolylacetic acid, indole-3-carboxylic acid,

8-methylpyrido (1,2-a) pyrimidin-4-one-3-carboxylic acid,

2- (4-methylphenoxy) pyridine-3-carboxylic acid,

8-hydroxyquinoline-7-sulfonic acid, 2-amino-4-chlorobenzoic acid,

N- (4-methoxybenzylidene) anthranilic acid,

5-bromonicotinic acid,

2-piperidinocinchoninic acid,

7-chlorkynurenic acid, (+/-) - 6-chloro-α-methylcarbazole-2-acetic acid,

N- (2,4,6-trinitrophenyl) -12-aminolauric acid,

2- (2-aminothiazol-4-yl) -2-methoxyiminoacetic acid,

11- (amidinothio (undecanoic acid,

4-amino-3,5-dibromobenzoic acid,

4- (1H-pyrrol-1-yl (benzoic acid,

N- (2-pyridyl) succinamic acid,

3-Indolacrylic acid

5 - [(3-ethyl-2 (3H) -benzoxazolylidene (ethylidene) -4-oxo-2-thioxo-

-3-thiazolidinacetic acid,

8-ethoxyquinoline-5-sulfonic acid, bromamine-acid,

N- (6-methyl-2-pyridyl) succinamic acid,

6-chloronicotinic acid,

4- (N, N-diethylamino) cinnamic acid •

223

3-Dimethylaminomethyl-1H-indole-2-carboxylic acid

2,2'-methylenebis (3,4-dimethyl-5-pyrrolecarboxylic acid),

2'-benzidinedisulfonic acid,

2 - [(2,3-dihydroindol-1-yl) imino] propanoic acid,

2,4-dinitro-4'-hydroxydiphenylamino-3'-sulfonic acid,

4-aminotoluene-3-sulfonic acid,

4- (4-aminophenyl (butyric acid,

N, N'-terephthalylidenedianthranilic acid,

2,2'-thiobis (5-aminobenzenesulfonic acid),

6-nitro-2-aminophenol-4-sulfonic acid, 2-methylnicotinic acid,

2- (5,6-dihydro-4H-1,3-oxazin-2-yl) (benzoic acid,

1-methyl-4- (2,4-dichlorobenzoyl) pyrrole-2-carboxylic acid,

2-amino-5-chlorobenzoic acid,

1-ethyl-3-methyl-1H-pyrazole-5-carboxylic acid,

4 '- (dimethylamino (-3,4,5,6-tetrachlorophthalic acid),

3-carboxy-4-hydroxy-6-methoxyquinoline

2-amino-6-chloro-3,5-dibromobenzoic acid, (4-pyridylthio) acetic acid,

2-pyridylhydroxymethanesulfonic acid,

2,6-dimethoxynicotinic acid,

2-chloro-6-methylpyridine-4-carboxylic acid,

4- (2,6-dichlorobenzylideneamino) benzoic acid, p-anisidine-2-sulfonic acid,

4- (4-amino-3-methylphenoxy) -1-butanesulfinic acid, (5,6-dimethyl-2-benzimidazolylthio),

4- (3-indolylmethylamino (benzoic acid,

4-amino-2-butoxybenzoic acid,

4-amino-3,5-diiodo-benzoic acid,

N-iodoacetyl-N '- (5-sulfo-1-naphthyl (ethylenediamine,

4,4'-diaminostilbene-2,2'-disulfonic acid, (2-amino-4-thiazolyl) acetic acid,

2-amino-5-hydroxybenzoic acid •

- 224 4'-anilinoglutaranilic acid,

2- (2-pyridylcarbonyl) benzoic acid,

N- (2-cyanethyl) anthranilic acid,

6-chloro-3-aminoethylbenzene-4-sulfonic acid,

1,3-phenylenediamino-4-sulfonic acid,

4'-amino-2'-hydroxysuccinanilic acid, amphonelic acid,

4-nitrodiphenylamino-2-sulfonic acid,

2,3-dihydro-5-oxothiazolo (3,2-a) pyrimidine-6-carboxylic acid,

2-amino-5-bromo-4-nitrobenzoic acid,

5-nitro-2- (3-phenylpropylamino) benzoic acid, isonicotinic acid,

2-hydroxy-6-methylpyridine-3-carboxylic acid,

6-chloro-2- (4-chlorophenyl) -4-quinolinecarboxylic acid,

4-amino-3,5-dinitrobenzoic acid,

2-methoxy-4-nitroaniline-5-sulfonic acid,

2-amino-3,5-dimethylbenzoic acid,

2- (1-imidazolylcarbonyl) benzoic acid,

5-hydroxyindole-2-carboxylic acid,

4,5-dibromanthranilic acid, (S) - (-) - indoline-2-carboxylic acid,

2-amino-4-methylbenzoic acid,

5-methoxy-2-methyl-3-indole acetic acid,

2.5-dichlorosulfanilic acid,

2-phenylbenzimidazole-5-sulfonic acid,

3-amino-2,5,6-trifluorobenzoic acid,

3-amino-5-nitrobenzoic acid, chloro-2-aminophenol-4-sulfonic acid,

4- (dimethylamino) cinnamic acid,

2 - [(3-chloro-2-methylphenyl) amino] benzoic acid,

5-dimethylamino-1-naphthalenesulfonic acid,

5-amino-1-naphthol-3-sulfonic acid, •

- 225 -

3- (4-aminophenyl) propionic acid, calconcarboxylic acid,

4-amino-5-chloro-2-methoxybenzoic acid, picolinic acid,

4'-anilinomaleanilic acid, p- [N, N-bis (2-chloroethyl) amino] benzoic acid, isoxazole-5-carboxylic acid,

7-chloro-4-hydroxyquinoline-3-carboxylic acid, [(3,5,6-trichloro-2-pyridyl) oxy] acetic acid,

7,8-dimethyl-4-hydroxy-3-quinolinecarboxylic acid,

2-naphthylamino-1,5-disulfonic acid,

5-methoxyindole-2-carboxylic acid,

3-aminobenzoic acid,

5,7-dichlorkynurenic acid,

4- (8-hydroxy-5-quinolylazo) -1-naphthalenesulfonic acid,

5-hydroxyindole-3-acetic acid,

2-Methyl-1-azanthon-3-carboxylic acid

5-acetamidoanthranilic acid,

4-amino-2-chlorotoluene-5-sulfonic acid,

1- (2 ', 5'-dichloro-4'-sulfophenyl) -3-methyl-5-pyrazolone,

4'-anilinosuccinanilic acid,

N- (2-thiazolyl) -1,2,3,6-tetrahydrophthalamic acid,

7-amino-4-methyl-3-coumarinylacetic acid,

2,5-dimethylpyrrole-3-carboxylic acid,

3-quinolinecarboxylic acid, imidazole-4-acrylic acid,

2-amino-6-methylbenzoic acid,

2-naphth-o-anisidide-3-phosphoric acid, β-n-indolpropionic acid,

1-Diazo-2-naphthol-4-sulfonic acid

3-hydroxy-2-phenylcinchoninic acid,

4 '- (dimethylamino) hexahydrophthalanic acid,

2-amino-α, β-dibromohydro-cinnamic acid,

226 (1,3-dimethyl-2,6-dioxo-2,3,6,7-tetrahydro-1H-purin-8-yl) acetic acid,

4,5-difluoroanthranilic acid,

3- (4-dimethylamino-1-naphthylazo) -4-methoxybenzenesulfonic acid,

2-amino-5-fluorobenzoic acid,

6-quinolinecarboxylic acid,

3-aminobenzylmethylamino-4-sulfonic acid, 2-nitroso-1-naphthol-4-sulfonic acid, 2-methylmercaptonicotinic acid,

N- (3-pyridyl) hexahydrophthalamic acid,

5- (2,3-dihydro-2-thioxo-1-benzimidazolylmethylamino) salicylic acid,

2-chloro-6-methylnicotinic acid,

2-amino-5-iodobenzoic acid,

5-methyl-4 - [[3- (trifluoromethyl) anilino / carbonyl] -3-isoxazolecarboxylic acid,

4-aminosalicylic acid,

5-bromoindole-2-carboxylic acid,

2-chloro-6-nitrophenol-4-sulfonic acid,

4- [bis (2-chloroethyl) amino] benzene butyric acid, (4-aminophenylthio) acetic acid,

N-benzylanthranilic acid,

3-pyridylhydroxymethanesulfonic acid,

4-chloro-N- (6-methoxy-3-pyridyl) anthranilic acid,

4-aminophenylacetic acid,

4-Benzothiazol-2-ylbutyric acid

2- (4-pyridyl) thiazole-4-carboxylic acid,

3- (4-diethylamino-2-hydroxyphenylazo) -4-hydroxybenzenesulfonic acid,

1-phenyl-4-hydroxy-6-pyridazinone carboxylic acid,

2-aminotoluene-5-sulfonic acid, pyrazol-1-ylacetic acid,

- 227 N- (3-pyridyl) succinamic acid,

5- (benzyloxycarbonyl) -2,4-dimethyl-3-pyrrolpropionic acid,

4-dimethylaminosalicylic acid, 3-chloro-2-toluidine-5-sulfonic acid,

2,4-dimethyl-5- (tert-butoxycarbonyl) -3-pyrrolpropionic acid,

5-amino-2-hydroxybenzenesulfonic acid a

3-Aminopyridine-2-carboxylic acid.

Hereinafter, the above set of acids is referred to as the set of acids.

If the acid selected from the group of acids is a polybasic acid, the paroxetine salts may contain varying amounts of paroxetine, depending on the number of acid groups that are associated with the paroxetine molecule. All such salts are within the scope of this invention.

In general, steric considerations are determined by the fact that in the case of a polyhydric acid having a functionality greater than two, the acidic anion will not be associated with more than two molecules of paroxetine.

Therefore, with respect to all of the acids of the set of acids in a particular aspect of the present invention, there is provided a paroxetine salt in which the (molar) ratio of paroxetine to acid is 1: 1.

With respect to the polyhydric acid of the set of acids in another aspect of the present invention, there is provided a paroxetine salt in which the (molar) ratio of paroxetine to paroxetine is in a molar ratio.

- 228 acid 2: 1.

In polyvalent acid salts, the acidic anion may be associated with a proton (hydrogen atom) in addition to paroxetine, or may be associated with another cation, for example an alkali metal or ammonium cation, to form a mixed salt.

When an acid of the acid group is present in enantiomeric forms, this invention includes salts with both D-acids and L-acids individually and as racemic mixtures of both salts as well as diastereoisomers.

In one aspect, the novel salts of the invention are provided in a non-crystalline form, which may be in the form of a solid or an oil. The oil is preferably absorbed onto a solid carrier, especially a carrier which is useful as a component of a pharmaceutical composition.

In another aspect, the novel salts of the invention are provided in crystalline form. Where a crystalline form exists in more than one polymorph, each polymorph forms another aspect of the invention.

Paroxetine salts can be prepared by contacting stoichiometric amounts of the acid and paroxetine free base. Preferably, the base is in solution, more preferably both the base and the acid are in solution. The acid may also be in solid (solid) form, provided that the resulting salt is not insoluble enough to form a coating on the added solid which hinders further reaction. Mixed salts may be prepared by forming a precursor of a 1: 1 salt in situ (or a 2: 1 salt for tribasic and higher acids), or may be used preformed and introduced into the mixture.

229 in solution with a solution containing a metal or ammonium ion.

Solvents such as toluene, alcohols such as methanol, ethanol, 2-propanol, esters such as ethyl acetate, ketones such as acetone or butanone, halogenated hydrocarbons such as dichloromethane and ethers are suitable for the mobility of the paroxetine free base. such as tetrahydrofuran and diethyl ether. The acid from the set of acids is preferably added as a solution, preferably an aqueous solution if it is water-soluble, optionally further diluted with a miscible organic solvent. The acid may also be added in the form of a soluble salt, for example, an ammonium salt, for example, ethylamine or diethylamine.

The concentration of paroxetine base is preferably in the range of from 50 to 50% (w / v), more preferably in the range of from 10 to 30% (w / v). The acid concentration is preferably in the range of 0.1- to 2 molar. Elevated temperatures can be used to increase solubility.

The salt may be isolated from its solution obtained according to the above process in solid form by conventional means. For example, a non-crystalline salt can be prepared by solution precipitation, spray drying and lyophilization of solutions, evaporation of the solution on glass or vacuum drying of oils, or solidification of molten substances obtained from the reaction of the free base and acid.

The crystalline salt may be prepared by direct crystallization from a solvent in which the product has limited solubility, or by trituration or other crystallization of the non-crystalline salt. General solvent systems that are •

230 suitable for preparing the paroxetine salt may also be used for recrystallization. The improved salt yield is achieved by evaporating some or all of the solvent or crystallization at elevated temperature followed by controlled cooling, preferably in stages. Careful clotting and seeding temperature control can be used to improve repeatability of the manufacturing process, particle size distribution and product form. The individual polymorphs are preferably crystallized directly from the salt solution, although recrystallization of a solution of one polymorph can also be performed using flakes of another polymorph.

An alternative method for preparing a paroxetine acid salt from an acid set is to start from a paroxetine salt with an organic acid such as acetic acid or maleic acid. The use of another salt of paroxetine as a starting material is suitable for preparing the crystalline salt or, if a volatile acid such as acetic acid is used, non-crystalline salts by methods which include evaporation (such as lyophilization or spray drying).

A salt can be obtained as a solvate if it is associated with the solvent in which it is dissolved during isolation from solution. Any such solvate forms form a further aspect of the invention. The solvates may be converted to the unsolvate salt by heating, for example by heating in an oven, or by exposure to a displacing solvent that does not form a solvate.

Prior to isolation of the paroxetine salt, water can be removed from the salt solution by azeotropic distillation to avoid formation of hydrates or to obtain the product in anhydrous form. In this case, suitable solvents for salt solutions are those that form an azeotrope with water.

231 such as toluene and 2-propanol. It should be noted that solvent mixtures may also be used to facilitate azeotropic removal of water.

The paroxetine free base may be prepared according to the procedures generally outlined in US Patent No. 4,007,196 and EP-B-0 223 403. The acids of the acid family are available commercially or are reported in the literature.

The compounds of the invention can be used to treat and prevent the following disorders:

alcoholism anxiety depression panic disorder obesity obsessive compulsive disorder chronic pain senile dementia anorexia migraine bulimia social phobia

premenstrual syndrome (PMS) adolescent depression

trichothilomania substance abuse dysthymia

These disorders are hereinafter referred to as disorders.

The present invention further provides a method of treating and / or preventing any or more disorders by administering an effective and / or prophylactic amount of a salt of the invention to a patient in need thereof.

The present invention further provides a pharmaceutical composition for use in the treatment and / or prevention of disorders comprising a mixture of a salt of the invention with a

- 232 a pharmaceutically acceptable carrier.

The present invention also provides the use of a salt of the invention for the treatment and / or prevention of disorders.

The present invention also provides the use of a salt of the invention for the manufacture of a medicament for the treatment and / or prevention of disorders.

Most preferably, the present invention is used in the treatment of depression, obsessive compulsive disorder (OCD) and panic.

The formulations of this invention are usually adapted for oral administration, but formulations for dilution for parenteral administration are also within the scope of the invention.

The formulation is usually presented as a dosage unit formulation containing from 1 to 200 mg of active ingredient, calculated on the basis of the free base, more usually from 5 to 100 mg, for example from 10 to 50 mg, such as 10, 12.5, 15, 20, 25 , 30 or 40 mg, as regards a human patient. Most preferably, the dosage unit contains 20 mg of active ingredient calculated on the free base basis. Such a formulation is usually used from 1 to 6 times a day, for example 2-, 3- or 4 times a day, so that the total amount of active ingredient administered is in the range of 5 to 400 mg of active ingredient, calculated on the basis of free base. Most preferably, the dosage unit is administered once per day.

Preferred dosage unit forms include tablets or capsules.

The compositions of the invention may be formulated.

233 by conventional mixing techniques such as mixing, filling and pressing.

Suitable carriers for use in the present invention include a diluent, binder, disintegrant, colorant, flavorant, and / or preservative. These agents may be used in a conventional manner, for example in a manner similar to that already used for marketed antidepressants.

Suitable pharmaceutical formulations include those described in EP-B-0 223 403 and US Patent No. 4,007,196 in which the products of the present invention can be used as active ingredients.

The following examples illustrate the present invention.

DETAILED DESCRIPTION OF THE INVENTION

Example 1

Folders 20mg tablet 30mg tablet Paroxetine salt 20,00 mg 30.0 mg (calculated as (calculated as free base) free base) Hydrogen phosphate Calcium (DCP) 83.34 mg 125.0 mg Microcrystalline cellulose 50.67 mg 76.0 mg Sodium starch glycolate 8.34 mg 12.5 mg Magnesium stearate 1,67 mg 2.5 mg

• ·

- 234 Commercial Source of Ingredients:

Calcium hydrogen phosphate - Emcompress or Ditab

Microcrystalline cellulose - Avicel PH 102

Natriumglykolat starch - Explotab * * Trademarks

Way

1) Calcium hydrogen phosphate is passed through a sieve and weighed into a planetary mixer.

2) Add 30 mesh of paroxetine salt to the pan.

3) Add Avicel and Explotab having a particle size of 0.833 mm (20 mesh) and mix all powders for 10 minutes.

4) Add magnesium stearate and mix for 5 minutes.

Tablets are made into pentagonal tablets using the following punches:

30 mg tablet 9.5 mm round

20mg tablet 8.25 mm round

The tablets are satisfactorily manufactured using a single punch or rotary press.

···· ··· ·· · · ·

235 Example 2

Ingredients 10mg tablet 20mg tablet 30mg tablet

Paroxetine salt 10 mg 20 mg 30 mg (calculated as (calculated as (counted free base) free base) free base Natriumglykolat starch 2,98 mg 5,95 mg 8.93 mg

Granular hydrogen phosphate

Calcium (DITAB) or Dicafos 158.88 mg 317.75 mg 476.63 mg Magnesium stearate 1.75 mg 3,50 mg 5,25 mg

Way

1) Sieve the paroxetine salt, sodium starch glycollate and dicalcium phosphate dihydrate in a suitable mixer (planetary, Cuble or high shear mixer).

2) Magnesium stearate is added and the mixture is compressed into a tablet using a single punch or rotary tabletting machine.

Claims (11)

PATENT CLAIMS A paroxetine salt with an acid selected from the group of acids. A salt according to claim 1, which is a salt with D-acid. The salt of claim 1, which is an L-acid salt. The paroxetine salt of claim 1, 2 or 3, wherein the ratio of paroxetine free base to acid is 1: 1 (indicated by molar). The paroxetine salt of claim 1, 2 or 3, wherein the ratio of paroxetine free base to acid is 2: 1 (indicated by molar). A compound according to claim 1, 2, 3, 4 or 5, which is in a non-crystalline form. The compound of claim 1, 2, 3, 4 or 5, which is in crystalline form. A process for preparing a compound according to claim 1, 2, 3, 4, 5 or 6, characterized in that it is prepared from a paroxetine salt solution, spray dried or lyophilized the paroxetine salt solution, evaporates the paroxetine salt solution on glass or dried the paroxetine salt oil under vacuum or the molten paroxetine salt is allowed to solidify. A process for the preparation of a compound according to claim 1, 2, 3, 4, 5, 6 or 7, characterized in that the paroxetine salt is crystallized or recrystallized from solution. A method according to claim 8 or 9, characterized in that the method is as follows: ························································· 237, wherein the solution, oil or melt of paroxetine salt is prepared by exposing paroxetine free base or its organic acid salt to an acid selected from the group of acids or its ammonium or amine salt. 11. A method of treating and / or preventing any or more of the disorders comprising administering an effective and / or prophylactic amount of a salt of paroxetine with an acid selected from the group of acids to a patient in need thereof.